Page last updated: 2024-08-21

isoxazoles and Anochlesia

isoxazoles has been researched along with Anochlesia in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19903 (23.08)18.7374
1990's4 (30.77)18.2507
2000's4 (30.77)29.6817
2010's2 (15.38)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barton, HA; Danhof, M; de Greef, R; Grimwood, S; Groothuis, GM; Johnson, M; Kozielska, M; Pilla Reddy, V; Proost, JH; Vermeulen, A1
Harada, Y; Koh, T; Nagino, K1
Cho, H; Cho, YS; Choi, KI; Jeong, D; Jung, JY; Jung, SH; Kim, GD; Koh, HY; Kong, JY; Lee, S; Pae, AN; Park, WK; Yun, CW1
Cha, MY; Cho, H; Choi, KI; Jeong, D; Koh, HY; Kong, JY; Lee, SJ; Pae, AN; Park, WK1
Brea, J; Cabrero-Castel, A; Castro, M; Dezi, C; Fernández-Espejo, E; Galán-Rodríguez, B; Loza, MI; Maldonado, R; Masaguer, CF; Pastor, M; Raviña, E; Robledo, P; Sanz, F1
Arnt, J; Christensen, AV1
Conway, PC; Corbett, R; Dunn, RW; Hartman, H; Helsley, GC; Kerman, LL; Strupczewski, JT; Woods, AT1
Hayakawa, H; Kawai, K; Kikumoto, O; Motohashi, N; Okamoto, Y; Yamawaki, S; Yokota, N1
Agut, J; Anglada, L; Bolós, J; De la Fuente, N; Gubert, S; Ortiz, JA; Planas, JM; Príncep, M; Sacristán, A1
Cadavid, MI; Carotti, A; Carrieri, A; Cid, J; Fontenla, JA; Loza, MI; Lozoya, E; Masaguer, CF; Negreira, J; Raviña, E; Rivas, ME; Rosa, E; Sanz, F; Tristán, H1
Cadavid, MI; Casariego, I; Demontis, GC; Enguix, MJ; Fontenla, JA; Loza, MI; Masaguer, CF; Montenegro, GY; Raviña, E; Rivas, ME; Villazon, M1
De Montis, GM; Mulas, G; Olianas, MC; Tagliamonte, A1
Catt, JD; Eison, MS; Lobeck, WG; Minielli, JL; New, JS; Riblet, LA; Smith, DW; Taylor, DP; Temple, DL; Yevich, JP1

Reviews

1 review(s) available for isoxazoles and Anochlesia

ArticleYear
[Pharmacological properties of paliperidone ER (INVEGA(®)) and results of its clinical studies].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 2011, Volume: 137, Issue:6

    Topics: Animals; Behavior, Animal; Catalepsy; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Double-Blind Method; Humans; Isoxazoles; Paliperidone Palmitate; Pyrimidines; Randomized Controlled Trials as Topic; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D2; Schizophrenia; Secondary Prevention

2011

Other Studies

12 other study(ies) available for isoxazoles and Anochlesia

ArticleYear
Dopamine D2 receptor occupancy as a predictor of catalepsy in rats: a pharmacokinetic-pharmacodynamic modeling approach.
    Pharmaceutical research, 2014, Volume: 31, Issue:10

    Topics: Animals; Antipsychotic Agents; Benzodiazepines; Brain; Catalepsy; Computer Simulation; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Humans; Isoxazoles; Markov Chains; Models, Biological; Olanzapine; Paliperidone Palmitate; Pyrimidines; Rats; Receptors, Dopamine D2; Risperidone; Severity of Illness Index

2014
Pharmacological actions of a novel and selective dopamine D3 receptor antagonist, KCH-1110.
    Pharmacological research, 2003, Volume: 48, Issue:6

    Topics: Animals; Antipsychotic Agents; Benzamides; Binding, Competitive; Body Temperature; Catalepsy; Cell Line; Clozapine; Cocaine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Haloperidol; Humans; Hypothermia; Isoxazoles; Male; Mice; Motor Activity; Prolactin; Psychomotor Performance; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes; Thiophenes; Tritium

2003
KKHA-761, a potent D3 receptor antagonist with high 5-HT1A receptor affinity, exhibits antipsychotic properties in animal models of schizophrenia.
    Pharmacology, biochemistry, and behavior, 2005, Volume: 82, Issue:2

    Topics: Animals; Antipsychotic Agents; Body Temperature; Catalepsy; Cell Line; Dopamine Uptake Inhibitors; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Ion Channels; Isoxazoles; Male; Mice; Mice, Inbred ICR; Piperazines; Postural Balance; Prolactin; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Receptors, Dopamine D1; Receptors, Dopamine D3; Receptors, Dopamine D4; Reflex, Startle; Schizophrenia; Schizophrenic Psychology; Serotonin Receptor Agonists; Spiperone; Swimming

2005
QF2004B, a potential antipsychotic butyrophenone derivative with similar pharmacological properties to clozapine.
    Neuropharmacology, 2006, Volume: 51, Issue:2

    Topics: Animals; Antipsychotic Agents; Butyrophenones; Carbazoles; Catalepsy; CHO Cells; Clozapine; Cricetinae; Cricetulus; Humans; In Vitro Techniques; Isoxazoles; Male; Mice; Models, Molecular; Motor Activity; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Histamine H1; Receptors, Muscarinic; Receptors, Serotonin; Reflex, Startle; Stereotyped Behavior

2006
Differential reversal by scopolamine and THIP of the antistereotypic and cataleptic effects of neuroleptics.
    European journal of pharmacology, 1981, Jan-05, Volume: 69, Issue:1

    Topics: Amphetamine; Animals; Antipsychotic Agents; Catalepsy; Humans; Isoxazoles; Male; Oxazoles; Rats; Scopolamine; Stereotyped Behavior

1981
Effects of atypical antipsychotic agents on social behavior in rodents.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 45, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Apomorphine; Benzazepines; Catalepsy; Chlorpromazine; Clozapine; Diazepam; Haloperidol; Isoxazoles; Male; Mice; Mice, Inbred Strains; Piperidines; Raclopride; Radioligand Assay; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Serotonin; Risperidone; Salicylamides; Social Behavior

1993
[Effects of risperidone on catalepsy and cerebral dopamine, serotonin and GABA metabolism in the rat: comparison with haloperidol].
    Yakubutsu, seishin, kodo = Japanese journal of psychopharmacology, 1993, Volume: 13, Issue:1

    Topics: Animals; Antipsychotic Agents; Brain; Catalepsy; Dopamine; gamma-Aminobutyric Acid; Haloperidol; Isoxazoles; Male; Piperidines; Rats; Rats, Wistar; Risperidone; Serotonin

1993
7-[3-(1-piperidinyl)propoxy]chromenones as potential atypical antipsychotics. 2. Pharmacological profile of 7-[3-[4-(6-fluoro-1, 2-benzisoxazol-3-yl)-piperidin-1-yl]propoxy]-3-(hydroxymeth yl)chromen -4-one (abaperidone, FI-8602).
    Journal of medicinal chemistry, 1998, Dec-31, Volume: 41, Issue:27

    Topics: Administration, Oral; Animals; Antipsychotic Agents; Brain; Catalepsy; Cell Line; Chromones; Drug Evaluation, Preclinical; Guinea Pigs; Humans; Isoxazoles; Male; Mice; Motor Activity; Prolactin; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Neurotransmitter; Stereotyped Behavior; Structure-Activity Relationship

1998
Conformationally constrained butyrophenones with mixed dopaminergic (D(2)) and serotoninergic (5-HT(2A), 5-HT(2C)) affinities: synthesis, pharmacology, 3D-QSAR, and molecular modeling of (aminoalkyl)benzo- and -thienocycloalkanones as putative atypical an
    Journal of medicinal chemistry, 1999, Jul-29, Volume: 42, Issue:15

    Topics: Animals; Antipsychotic Agents; Aorta, Thoracic; Brain; Catalepsy; Cattle; Dopamine Agents; In Vitro Techniques; Isoxazoles; Male; Mice; Models, Molecular; Motor Activity; Muscle Contraction; Muscle, Smooth, Vascular; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Dopamine D2; Receptors, Serotonin; Serotonin Agents; Structure-Activity Relationship; Thiophenes

1999
Conformationally constrained butyrophenones with affinity for dopamine (D(1), D(2), D(4)) and serotonin (5-HT(2A), 5-HT(2B), 5-HT(2C)) receptors: synthesis of aminomethylbenzo[b]furanones and their evaluation as antipsychotics.
    Journal of medicinal chemistry, 2000, Nov-30, Volume: 43, Issue:24

    Topics: Animals; Antipsychotic Agents; Behavior, Animal; Binding, Competitive; Butyrophenones; Catalepsy; Cattle; Corpus Striatum; Frontal Lobe; Humans; In Vitro Techniques; Isoxazoles; Male; Mice; Piperidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D4; Receptors, Serotonin; Retina

2000
The striatal dopaminergic function is mediated by the inhibition of a nigral, non-dopaminergic neuronal system via a strio-nigral GABAergic pathway.
    European journal of pharmacology, 1978, Jun-01, Volume: 49, Issue:3

    Topics: Aminobutyrates; Animals; Catalepsy; Corpus Striatum; Dopamine; Functional Laterality; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Isoxazoles; Male; Neural Inhibition; Neural Pathways; Picrotoxin; Rats; Stereotyped Behavior; Substantia Nigra

1978
Synthesis and biological evaluation of 1-(1,2-benzisothiazol-3-yl)- and (1,2-benzisoxazol-3-yl)piperazine derivatives as potential antipsychotic agents.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:3

    Topics: Animals; Antipsychotic Agents; Avoidance Learning; Binding, Competitive; Catalepsy; Cerebral Cortex; Corpus Striatum; Isoxazoles; Male; Models, Molecular; Norepinephrine; Oxazoles; Physostigmine; Piperazines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Serotonin; Sleep; Spiro Compounds; Stereotyped Behavior; Structure-Activity Relationship; Thiazoles

1986