Page last updated: 2024-08-21

indazoles and Muscle Contraction

indazoles has been researched along with Muscle Contraction in 43 studies

Research

Studies (43)

TimeframeStudies, this research(%)All Research%
pre-19903 (6.98)18.7374
1990's29 (67.44)18.2507
2000's9 (20.93)29.6817
2010's2 (4.65)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Isselbacher, EM; Jaffer, FA; Jassar, AS; Kessinger, CW; Lindsay, ME; Lino Cardenas, CL; MacDonald, C1
Chen, YC; Du, GH; Fang, LH; Jiao, XZ; Li, L; Xie, P; Yuan, TY; Zhang, HF1
Cacanyiova, S; Gerova, M; Kristek, F1
García-Flores, M; García-Pascual, A; Sancho, M; Triguero, D1
Brioni, JD; Hsieh, GC; Moreland, RB; O'Neill, AB; Sullivan, JP1
Ertunc, M; Onur, R; Sara, Y1
Anctil, M; Pelletier, C; Poulain, I1
Behm, DJ; Bentley, R; Cui, H; Doe, CP; Dowdell, SE; Dul, E; Evans, C; Fries, HE; Gaitanopoulos, DE; Goodman, KB; Hu, E; Ivy, RL; Jolivette, LJ; Jung, DK; Khandekar, SS; Kirkpatrick, RB; Lee, D; Sehon, CA; Semus, SF; Smith, GK; Stavenger, RA; Viet, AQ; Wang, GZ; Wright, LL; Xu, W; Ye, G; Yi, T1
Gourgoulianis, KI; Hatziefthimiou, AA; Kitsiopoulou, E; Molyvdas, PA1
Allawi, HS; Bland-Ward, PA; Gaffen, Z; Moore, PK; Pitcher, A; Wallace, P1
Krasnopolsky, L; Lee, JG; Levin, RM; Longhurst, PA; Wein, AJ1
Buckner, CK; Conklin, R; Doran, O; Fishleder, RI; Graziano, FM; Will, JA1
Babbedge, RC; Gaffen, Z; Hart, SL; Moore, PK; Wallace, P1
Abram, TS; Cuthbert, NJ; Gardiner, PJ; Jennings, MA; Maxey, RJ; Norman, P; Thompson, AM; Tudhope, SR1
Abram, TS; Cuthbert, NJ; Gardiner, PJ; Norman, P; Tudhope, SR1
Bell, RL; Brooks, DW; Carter, GW; Malo, PE; Shaughnessy, TK; Summers, JB1
Bosnjak, ZJ; Coon, RL; Tudorić, N1
Bäck, M; Dahlén, SE; Jonsson, EW1
Nawrath, H; Wegener, JW1
Behar, J; Biancani, P; Jain, MK; Kim, N; Mangannan, V; Rich, H; Sohn, UD1
Etgen, GJ; Fryburg, DA; Gibbs, EM1
Hebeiss, K; Kilbinger, H1
Bloomquist, WE; Calligaro, DO; Cohen, ML; Schaus, JM; Susemichel, AD; Thompson, DC1
Endo, M; Hanaoka, K; Ikemoto, T; Kameya, S; Miyagoe, Y; Nabeshima, Y; Nonaka, I; Takeda, S1
Galle, J; Hatzelmann, A; Hübner, U; Schmidt, HH; Wagner, B; Wanner, C; Zabel, U1
Heinemann, A; Holzer, P1
Brien, JF; Marks, GS; McLaughlin, BE; Nakatsu, K; O'Reilly, DA1
Bredt, DS; Kobzik, L; Reid, MB; Stamler, JS1
Bäck, M; Cotgreave, IA; Dahlén, SE; Kumlin, M1
Fujimura, Y; Ikeda, Y; Iwasaki, T; Koide, T; Matsushita, H; Nagashima, R; Shindo, M; Shiraki, Y; Suzuki, S; Takano, N1
Falcone, RC; Krell, RD1
Ito, T; Kato, S; Omoya, H; Yoshida, N1
Itoh, Z; Iwanaga, Y; Mizumoto, A; Yoshida, N1
Itoh, Z; Iwanaga, Y; Mizumoto, A; Torii, K; Wakabayashi, K; Yoshida, N1
Ito, S1
Aharony, D; Fedyna, JS; Krell, RD; Redkar-Brown, D; Snyder, DW1
Moss, HE; Sanger, GJ1
Chen, HI1
Brown, FJ; Cronk, LA; Hebbel, KC; Krell, RD; Snyder, DW; Yee, YK1
Aharony, D; Hesp, B; Keith, RA; Krell, RD; Maduskuie, TP; Matassa, VG; Shapiro, HS; Snyder, DW1
Bermudez, J; Fake, CS; Joiner, GF; Joiner, KA; King, FD; Miner, WD; Sanger, GJ1
Aharony, D; Redkar-Brown, DG1
Buckner, CK; Castleman, WL; Saban, R; Will, JA1

Other Studies

43 other study(ies) available for indazoles and Muscle Contraction

ArticleYear
Inhibition of the methyltranferase EZH2 improves aortic performance in experimental thoracic aortic aneurysm.
    JCI insight, 2018, 03-08, Volume: 3, Issue:5

    Topics: Animals; Aorta, Thoracic; Aortic Aneurysm, Thoracic; Disease Models, Animal; DNA Methylation; Enhancer of Zeste Homolog 2 Protein; Epigenesis, Genetic; Fibrillin-1; Gene Knockout Techniques; Histones; Humans; Indazoles; Losartan; Marfan Syndrome; Mice; Mice, Knockout; Microfilament Proteins; Muscle Contraction; Muscle Proteins; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Pyridones; RNA, Small Interfering

2018
DL0805-2, a novel indazole derivative, relaxes angiotensin II-induced contractions of rat aortic rings by inhibiting Rho kinase and calcium fluxes.
    Acta pharmacologica Sinica, 2016, Volume: 37, Issue:5

    Topics: Actins; Angiotensin II; Angiotensin II Type 2 Receptor Blockers; Animals; Aorta, Thoracic; Calcium; In Vitro Techniques; Indazoles; Male; Molecular Docking Simulation; Muscle Contraction; Muscle Relaxation; Myocytes, Smooth Muscle; Myosin Light Chains; Phosphorylation; Protein Phosphatase 1; Rats, Sprague-Dawley; Reactive Oxygen Species; rho-Associated Kinases; Signal Transduction; Vasoconstrictor Agents; Vasodilator Agents

2016
Hypotrophic effect of long-term neuronal NO-synthase inhibition on heart and conduit arteries of the Wistar rats.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2009, Volume: 60, Issue:2

    Topics: Animals; Aorta, Thoracic; Blood Pressure; Body Weight; Carotid Arteries; Coronary Vessels; Dose-Response Relationship, Drug; In Vitro Techniques; Indazoles; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide Synthase Type I; Organ Size; Rats; Rats, Wistar; Time Factors

2009
Presence of cyclic nucleotide-gated channels in the rat urethra and their involvement in nerve-mediated nitrergic relaxation.
    American journal of physiology. Renal physiology, 2009, Volume: 297, Issue:5

    Topics: Animals; Calcium Channel Blockers; Cyclic Nucleotide-Gated Cation Channels; Diltiazem; Enzyme Inhibitors; Female; Fluorescent Antibody Technique; Indazoles; Isometric Contraction; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Stereoisomerism; Urethra

2009
YC-1 potentiates the nitric oxide/cyclic GMP pathway in corpus cavernosum and facilitates penile erection in rats.
    European journal of pharmacology, 2003, Jan-01, Volume: 458, Issue:1-2

    Topics: Animals; Cells, Cultured; Cyclic GMP; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Guanylate Cyclase; In Vitro Techniques; Indazoles; Male; Muscle Contraction; Muscle, Smooth; Nitric Oxide; Nitroprusside; Oxadiazoles; Penile Erection; Penis; Phenylephrine; Quinoxalines; Rabbits; Rats; Rats, Wistar; Signal Transduction; Vasoconstrictor Agents; Vasodilator Agents

2003
The role of nitric oxide on contractile impairment during endotoxemia in rat diaphragm muscle.
    European journal of pharmacology, 2004, Nov-28, Volume: 505, Issue:1-3

    Topics: Animals; Caffeine; Diaphragm; Endotoxemia; Enzyme Inhibitors; Guanidines; In Vitro Techniques; Indazoles; Lipopolysaccharides; Male; Muscle Contraction; Neuromuscular Nondepolarizing Agents; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Oxadiazoles; Quinoxalines; Rats; Rats, Wistar; Ryanodine; Tubocurarine; Vasodilator Agents; Verapamil

2004
Nitric oxide modulates peristaltic muscle activity associated with fluid circulation in the sea pansy Renilla koellikeri.
    The Journal of experimental biology, 2005, Volume: 208, Issue:Pt 10

    Topics: Animals; Anthozoa; Body Fluids; California; Guanidines; Immunohistochemistry; Indazoles; Muscle Contraction; Muscles; Neurites; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Oxadiazoles; Peristalsis; Phosphodiesterase Inhibitors; Purinones; Quinoxalines

2005
Development of dihydropyridone indazole amides as selective Rho-kinase inhibitors.
    Journal of medicinal chemistry, 2007, Jan-11, Volume: 50, Issue:1

    Topics: Amides; Animals; Antihypertensive Agents; Aorta; Blood Pressure; In Vitro Techniques; Indazoles; Intracellular Signaling Peptides and Proteins; Models, Molecular; Muscle Contraction; Muscle, Smooth, Vascular; Protein Serine-Threonine Kinases; Pyridones; Pyrimidines; Rats; Rats, Inbred SHR; rho-Associated Kinases; Structure-Activity Relationship

2007
Resting tension affects eNOS activity in a calcium-dependent way in airways.
    Mediators of inflammation, 2007, Volume: 2007

    Topics: Acetylcholine; Animals; Arginine; Calcium; Dose-Response Relationship, Drug; Drug Interactions; Female; Genistein; Hydroquinones; In Vitro Techniques; Indazoles; Male; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase Type II; Nitric Oxide Synthase Type III; Rabbits; Trachea

2007
Effect of 7-nitro indazole on neurotransmission in the rat vas deferens: mechanisms unrelated to inhibition of nitric oxide synthase.
    British journal of pharmacology, 1994, Volume: 113, Issue:1

    Topics: Adenosine Triphosphate; Amino Acid Oxidoreductases; Animals; Arginine; Electric Stimulation; In Vitro Techniques; Indazoles; Male; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Norepinephrine; Potassium Chloride; Propranolol; Rats; Rats, Wistar; Synaptic Transmission; Vas Deferens; Yohimbine

1994
Effects of the peptide leukotriene receptor antagonist ICI 198,615 on the in vivo and in vitro changes in guinea pig bladder function which occur after sensitization with ovalbumin.
    The Journal of urology, 1995, Volume: 154, Issue:3

    Topics: Animals; Female; Guinea Pigs; In Vitro Techniques; Indazoles; Indomethacin; Leukotriene Antagonists; Muscle Contraction; Ovalbumin; Pyrilamine; SRS-A; Urinary Bladder; Urodynamics

1995
Pharmacologic modulation of the influence of the epithelium on immunologic- and nonimmunologic-induced histamine release and contraction in guinea pig superfused tracheal strips.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:2

    Topics: Animals; Epithelium; Female; Guinea Pigs; Histamine Release; Hydroxyurea; In Vitro Techniques; Indazoles; Indomethacin; Muscle Contraction; Ovalbumin; Pyrilamine; Trachea; Tubocurarine

1993
Characterization of the novel nitric oxide synthase inhibitor 7-nitro indazole and related indazoles: antinociceptive and cardiovascular effects.
    British journal of pharmacology, 1993, Volume: 110, Issue:1

    Topics: Amino Acid Oxidoreductases; Analgesics; Animals; Arginine; Blood Pressure; Cardiovascular Agents; Cerebellum; Enzyme Inhibitors; Formaldehyde; In Vitro Techniques; Indazoles; Male; Mice; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide Synthase; Pain Measurement; Rabbits; Rats

1993
BAY u9773, a novel antagonist of cysteinyl-leukotrienes with activity against two receptor subtypes.
    European journal of pharmacology, 1994, Nov-03, Volume: 264, Issue:3

    Topics: Animals; Binding, Competitive; Bronchi; Dicarboxylic Acids; Ferrets; Guinea Pigs; In Vitro Techniques; Indazoles; Leukotriene C4; Leukotriene D4; Lung; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Propionates; Quinolines; Rats; Rats, Wistar; Receptors, Immunologic; Sheep; Spleen; SRS-A; Trachea

1994
Characterisation of leukotriene receptors on rat lung strip.
    European journal of pharmacology, 1994, Dec-12, Volume: 271, Issue:1

    Topics: Animals; Dicarboxylic Acids; In Vitro Techniques; Indazoles; Leukotriene Antagonists; Leukotrienes; Lung; Male; Muscle Contraction; Muscle, Smooth; Potassium Chloride; Propionates; Quinolines; Rats; Rats, Wistar; Receptors, Leukotriene; SRS-A

1994
The 5-lipoxygenase inhibitory activity of zileuton in in vitro and in vivo models of antigen-induced airway anaphylaxis.
    Pulmonary pharmacology, 1994, Volume: 7, Issue:2

    Topics: Anaphylaxis; Animals; Anti-Inflammatory Agents, Non-Steroidal; Bronchoconstriction; Disease Models, Animal; Dose-Response Relationship, Drug; Female; Guinea Pigs; Humans; Hydroxyurea; Indazoles; Lipoxygenase Inhibitors; Male; Meclofenamic Acid; Muscle Contraction; Muscle, Smooth; Pyrilamine; SRS-A; Trachea

1994
Phosphoramidon augments contraction of guinea pig tracheal smooth muscle induced by histamine and leukotriene-D4.
    International archives of allergy and immunology, 1994, Volume: 103, Issue:3

    Topics: Anaphylaxis; Animals; Antigens; Dinoprost; Diphenhydramine; Glycopeptides; Guinea Pigs; Histamine; In Vitro Techniques; Indazoles; Leukotriene D4; Muscle Contraction; Muscle, Smooth; Neprilysin; Prostaglandin D2; SRS-A; Trachea

1994
The cysteinyl-leukotriene receptor antagonist BAY u9773 is a competitive antagonist of leukotriene C4 in the guinea-pig ileum.
    European journal of pharmacology, 1996, Dec-12, Volume: 317, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Female; Guinea Pigs; Ileum; In Vitro Techniques; Indazoles; Leukotriene Antagonists; Leukotriene C4; Leukotriene D4; Male; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Prostaglandin Endoperoxides, Synthetic; Receptors, Leukotriene; SRS-A; Thromboxane A2; Vasoconstrictor Agents

1996
Differential effects of isoliquiritigenin and YC-1 in rat aortic smooth muscle.
    European journal of pharmacology, 1997, Mar-26, Volume: 323, Issue:1

    Topics: Aldehyde Reductase; Animals; Carotid Arteries; Chalcone; Chalcones; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Guanylate Cyclase; Indazoles; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phosphodiesterase Inhibitors; Platelet Aggregation Inhibitors; Rats; Rats, Sprague-Dawley

1997
Leukotrienes in acetylcholine-induced contraction of esophageal circular smooth muscle in experimental esophagitis.
    Gastroenterology, 1997, Volume: 112, Issue:5

    Topics: Acetylcholine; Animals; Arachidonic Acid; Cats; Diglycerides; Drug Synergism; Esophagitis; Esophagus; Female; Indazoles; Leukotrienes; Male; Muscle Contraction; Muscle, Smooth; Phospholipases A; Phospholipases A2

1997
Nitric oxide stimulates skeletal muscle glucose transport through a calcium/contraction- and phosphatidylinositol-3-kinase-independent pathway.
    Diabetes, 1997, Volume: 46, Issue:11

    Topics: 3-O-Methylglucose; Androstadienes; Animals; Calcium; Dantrolene; Dibutyryl Cyclic GMP; Enzyme Inhibitors; Female; Glucose; Indazoles; Muscle Contraction; Muscle, Skeletal; Nitric Oxide; Nitric Oxide Synthase; Nitroprusside; omega-N-Methylarginine; Phosphatidylinositol 3-Kinases; Rats; Rats, Sprague-Dawley; Sulfonamides; Wortmannin

1997
Nitric oxide-sensitive guanylyl cyclase inhibits acetylcholine release and excitatory motor transmission in the guinea-pig ileum.
    Neuroscience, 1998, Volume: 82, Issue:2

    Topics: Acetylcholine; Animals; Depression, Chemical; Electric Stimulation; Enzyme Inhibitors; Female; Guanylate Cyclase; Guinea Pigs; Ileum; Indazoles; Male; Motor Neurons; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Oxadiazoles; Quinoxalines; Synaptic Transmission

1998
Synthesis and structure-activity relationships of potent and orally active 5-HT4 receptor antagonists: indazole and benzimidazolone derivatives.
    Journal of medicinal chemistry, 1998, May-21, Volume: 41, Issue:11

    Topics: Adamantane; Administration, Oral; Adrenergic alpha-Antagonists; Animals; Aorta; Brain; Drug Evaluation, Preclinical; Esophagus; Guinea Pigs; Ileum; In Vitro Techniques; Indazoles; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, alpha-1; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Structure-Activity Relationship

1998
alpha1-syntrophin gene disruption results in the absence of neuronal-type nitric-oxide synthase at the sarcolemma but does not induce muscle degeneration.
    The Journal of biological chemistry, 1999, Jan-22, Volume: 274, Issue:4

    Topics: Animals; Base Sequence; Calcium-Binding Proteins; DNA Primers; Enzyme Inhibitors; Immunohistochemistry; Indazoles; Membrane Proteins; Mice; Mice, Inbred C3H; Mice, Inbred C57BL; Mice, Knockout; Muscle Contraction; Muscle Proteins; Muscle, Skeletal; NG-Nitroarginine Methyl Ester; Nitric Oxide Donors; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Nitroprusside; Sarcolemma

1999
Effects of the soluble guanylyl cyclase activator, YC-1, on vascular tone, cyclic GMP levels and phosphodiesterase activity.
    British journal of pharmacology, 1999, Volume: 127, Issue:1

    Topics: Animals; Aorta, Thoracic; Cyclic GMP; Enzyme Activation; Enzyme Inhibitors; Guanylate Cyclase; In Vitro Techniques; Indazoles; Isoenzymes; Kinetics; Muscle Contraction; Muscle Relaxation; Muscle Tonus; Muscle, Smooth, Vascular; Nitric Oxide Donors; Nitroprusside; Nitroso Compounds; Oxadiazoles; Phosphoric Diester Hydrolases; Quinoxalines; Rabbits; Vasodilator Agents

1999
Intestinal motor depression by 7-nitroindazole through an action unrelated to nitric oxide synthase inhibition.
    Pharmacology, 1999, Volume: 59, Issue:6

    Topics: Animals; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Gastrointestinal Motility; Guinea Pigs; Imidazoles; In Vitro Techniques; Indazoles; Indomethacin; Intestine, Small; Male; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Peptide Fragments; Peristalsis; Sincalide; Substance P; Tetrodotoxin

1999
YC-1 enhances the responsiveness of tolerant vascular smooth muscle to glyceryl trinitrate.
    Canadian journal of physiology and pharmacology, 2001, Volume: 79, Issue:1

    Topics: Animals; Aorta, Thoracic; Cyclic GMP; Drug Tolerance; Enzyme Activators; In Vitro Techniques; Indazoles; Isometric Contraction; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroglycerin; Rabbits; Vasodilator Agents

2001
Nitric oxide modulates excitation-contraction coupling in the diaphragm.
    Comparative biochemistry and physiology. Part A, Molecular & integrative physiology, 1998, Volume: 119, Issue:1

    Topics: Animals; Diaphragm; Enzyme Inhibitors; Guanidines; Hindlimb; Indazoles; Male; Muscle Contraction; Muscle, Skeletal; Nitrates; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type III; Nitrites; Nitroarginine; Rats; Rats, Sprague-Dawley

1998
An alternative pathway for metabolism of leukotriene D(4): effects on contractions to cysteinyl-leukotrienes in the guinea-pig trachea.
    British journal of pharmacology, 2001, Volume: 133, Issue:7

    Topics: Animals; Borates; Cysteine; Dicarboxylic Acids; Dose-Response Relationship, Drug; Glutathione; Guinea Pigs; In Vitro Techniques; Indazoles; Leukotriene Antagonists; Leukotriene C4; Leukotriene D4; Leukotriene E4; Leukotrienes; Male; Membrane Proteins; Muscle Contraction; Propionates; Quinolines; Receptors, Leukotriene; Serine; SRS-A; Trachea

2001
Pharmacological studies on a new thymoleptic antidepressant, 1-[3-(dimethylamino)propyl]-5-methyl-3-phenyl-1H-indazole (FS-32).
    Arzneimittel-Forschung, 1979, Volume: 29, Issue:3

    Topics: Acetylcholine; Amphetamine; Animals; Antidepressive Agents; Barbiturates; Behavior, Animal; Biogenic Amines; Blood Pressure; Brain Chemistry; Catecholamines; Cats; Dogs; Electroencephalography; Female; Guinea Pigs; Haplorhini; In Vitro Techniques; Indazoles; Levodopa; Macaca fascicularis; Male; Mice; Muscle Contraction; Muscle, Smooth; Physostigmine; Pyrazoles; Rabbits; Rats; Reserpine; Tremorine

1979
Guinea pig gall bladder contains a single peptide leukotriene receptor which resembles that present in human conducting airway smooth muscle.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:3

    Topics: Animals; Gallbladder; Guinea Pigs; Humans; Indazoles; Lung; Male; Muscle Contraction; Muscle, Smooth; Receptors, Immunologic; Receptors, Leukotriene; Signal Transduction; SRS-A

1992
5-HT3 receptor antagonist effects of DAT-582, (R) enantiomer of AS-5370.
    European journal of pharmacology, 1992, Jun-17, Volume: 216, Issue:3

    Topics: Animals; Azepines; Bradycardia; Cisplatin; Ferrets; Guinea Pigs; Ileum; In Vitro Techniques; Indazoles; Male; Muscle Contraction; Muscle, Smooth; Rats; Serotonin Antagonists; Stereoisomerism; Vomiting

1992
Effects of 5-hydroxytryptamine 3 receptor antagonists on gastrointestinal motor activity in conscious dogs.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:1

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Digestion; Dogs; Dose-Response Relationship, Drug; Female; Gastrointestinal Motility; Granisetron; Imidazoles; Indazoles; Indoles; Infusions, Intravenous; Injections, Intravenous; Male; Motilin; Motor Activity; Muscle Contraction; Muscle, Smooth; Ondansetron; Serotonin Antagonists; Time Factors; Tropisetron

1991
Involvement of 5-hydroxytryptamine 3 receptors in regulation of interdigestive gastric contractions by motilin in the dog.
    Gastroenterology, 1991, Volume: 100, Issue:4

    Topics: Acetylcholine; Animals; Digestion; Dogs; Gastrointestinal Motility; Granisetron; Imidazoles; Indazoles; Motilin; Muscle Contraction; Muscle, Smooth; Ondansetron; Receptors, Serotonin; Serotonin Antagonists; Stomach

1991
[Study on mechanism of interdigestive migrating contractions of a canine stomach].
    Nihon Heikatsukin Gakkai zasshi, 1990, Volume: 26, Issue:5

    Topics: Animals; Dogs; Fasting; Gastrointestinal Motility; Granisetron; Indazoles; Motilin; Muscle Contraction; Muscle, Smooth; Serotonin Antagonists; Stomach

1990
Pharmacologic characterization of the contractile activity of peptide leukotrienes in guinea-pig pulmonary artery.
    Prostaglandins, 1990, Volume: 39, Issue:5

    Topics: Acetophenones; Animals; Borates; Drug Synergism; Endothelium, Vascular; Guinea Pigs; In Vitro Techniques; Indazoles; Indomethacin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Pulmonary Artery; Receptors, Immunologic; Receptors, Leukotriene; Serine; SRS-A; Tetrazoles

1990
The effects of granisetron, ICS 205-930 and ondansetron on the visceral pain reflex induced by duodenal distension.
    British journal of pharmacology, 1990, Volume: 100, Issue:3

    Topics: Animals; Blood Pressure; Duodenum; Granisetron; Imidazoles; Indazoles; Indoles; Male; Morphine; Muscle Contraction; Muscle, Smooth; Ondansetron; Pain; Pyrazoles; Rats; Rats, Inbred Strains; Reflex; Serotonin Antagonists; Stomach; Tropisetron; Vagotomy

1990
Evidence for the presynaptic action of 5-hydroxytryptamine and the involvement of purinergic innervation in the rabbit lower urinary tract.
    British journal of pharmacology, 1990, Volume: 101, Issue:1

    Topics: Adenosine Triphosphate; Animals; Atropine; Electric Stimulation; Female; Granisetron; In Vitro Techniques; Indazoles; Indoles; Male; Muscle Contraction; Muscle, Smooth; Purines; Rabbits; Serotonin; Serotonin Antagonists; Synapses; Tropanes; Tropisetron; Urethra; Urinary Tract

1990
Evolution of a series of peptidoleukotriene antagonists: synthesis and structure-activity relationships of 1,6-disubstituted indoles and indazoles.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:6

    Topics: Animals; Guinea Pigs; In Vitro Techniques; Indazoles; Indoles; Muscle Contraction; Pyrazoles; SRS-A; Structure-Activity Relationship

1990
Evolution of a series of peptidoleukotriene antagonists: synthesis and structure/activity relationships of 1,3,5-substituted indoles and indazoles.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:6

    Topics: Animals; Dyspnea; Guinea Pigs; In Vitro Techniques; Indazoles; Indoles; Muscle Contraction; Pyrazoles; SRS-A; Structure-Activity Relationship

1990
5-Hydroxytryptamine (5-HT3) receptor antagonists. 1. Indazole and indolizine-3-carboxylic acid derivatives.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:7

    Topics: Animals; Antiemetics; Carboxylic Acids; Ferrets; Guinea Pigs; Ileum; In Vitro Techniques; Indazoles; Indicators and Reagents; Indolizines; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Molecular Structure; Muscle Contraction; Muscle, Smooth; Pyrazoles; Rats; Receptors, Serotonin; Reflex; Serotonin; Serotonin Antagonists; Stereoisomerism; Structure-Activity Relationship

1990
Inhibition of antigen-induced contraction of guinea pig trachea by ICI 198,615.
    European journal of pharmacology, 1989, Jun-08, Volume: 165, Issue:1

    Topics: Animals; Antigens; Guinea Pigs; In Vitro Techniques; Indazoles; Indomethacin; Leukotrienes; Lipoxygenase Inhibitors; Male; Muscle Contraction; Muscle, Smooth; Ovalbumin; Phospholipid Ethers; Platelet Activating Factor; Pyrazoles; Pyrilamine; SRS-A; Trachea

1989
Analysis of leukotriene receptor antagonists on isolated human intralobar airways.
    Annals of the New York Academy of Sciences, 1988, Volume: 524

    Topics: Acetophenones; Azoles; Barium; Bronchi; Chromones; Humans; Indazoles; Muscle Contraction; Muscle, Smooth; Pyrazoles; Receptors, Leukotriene; Receptors, Prostaglandin; SRS-A; Tetrazoles

1988