indazoles has been researched along with Muscle Contraction in 43 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (6.98) | 18.7374 |
1990's | 29 (67.44) | 18.2507 |
2000's | 9 (20.93) | 29.6817 |
2010's | 2 (4.65) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Isselbacher, EM; Jaffer, FA; Jassar, AS; Kessinger, CW; Lindsay, ME; Lino Cardenas, CL; MacDonald, C | 1 |
Chen, YC; Du, GH; Fang, LH; Jiao, XZ; Li, L; Xie, P; Yuan, TY; Zhang, HF | 1 |
Cacanyiova, S; Gerova, M; Kristek, F | 1 |
García-Flores, M; García-Pascual, A; Sancho, M; Triguero, D | 1 |
Brioni, JD; Hsieh, GC; Moreland, RB; O'Neill, AB; Sullivan, JP | 1 |
Ertunc, M; Onur, R; Sara, Y | 1 |
Anctil, M; Pelletier, C; Poulain, I | 1 |
Behm, DJ; Bentley, R; Cui, H; Doe, CP; Dowdell, SE; Dul, E; Evans, C; Fries, HE; Gaitanopoulos, DE; Goodman, KB; Hu, E; Ivy, RL; Jolivette, LJ; Jung, DK; Khandekar, SS; Kirkpatrick, RB; Lee, D; Sehon, CA; Semus, SF; Smith, GK; Stavenger, RA; Viet, AQ; Wang, GZ; Wright, LL; Xu, W; Ye, G; Yi, T | 1 |
Gourgoulianis, KI; Hatziefthimiou, AA; Kitsiopoulou, E; Molyvdas, PA | 1 |
Allawi, HS; Bland-Ward, PA; Gaffen, Z; Moore, PK; Pitcher, A; Wallace, P | 1 |
Krasnopolsky, L; Lee, JG; Levin, RM; Longhurst, PA; Wein, AJ | 1 |
Buckner, CK; Conklin, R; Doran, O; Fishleder, RI; Graziano, FM; Will, JA | 1 |
Babbedge, RC; Gaffen, Z; Hart, SL; Moore, PK; Wallace, P | 1 |
Abram, TS; Cuthbert, NJ; Gardiner, PJ; Jennings, MA; Maxey, RJ; Norman, P; Thompson, AM; Tudhope, SR | 1 |
Abram, TS; Cuthbert, NJ; Gardiner, PJ; Norman, P; Tudhope, SR | 1 |
Bell, RL; Brooks, DW; Carter, GW; Malo, PE; Shaughnessy, TK; Summers, JB | 1 |
Bosnjak, ZJ; Coon, RL; Tudorić, N | 1 |
Bäck, M; Dahlén, SE; Jonsson, EW | 1 |
Nawrath, H; Wegener, JW | 1 |
Behar, J; Biancani, P; Jain, MK; Kim, N; Mangannan, V; Rich, H; Sohn, UD | 1 |
Etgen, GJ; Fryburg, DA; Gibbs, EM | 1 |
Hebeiss, K; Kilbinger, H | 1 |
Bloomquist, WE; Calligaro, DO; Cohen, ML; Schaus, JM; Susemichel, AD; Thompson, DC | 1 |
Endo, M; Hanaoka, K; Ikemoto, T; Kameya, S; Miyagoe, Y; Nabeshima, Y; Nonaka, I; Takeda, S | 1 |
Galle, J; Hatzelmann, A; Hübner, U; Schmidt, HH; Wagner, B; Wanner, C; Zabel, U | 1 |
Heinemann, A; Holzer, P | 1 |
Brien, JF; Marks, GS; McLaughlin, BE; Nakatsu, K; O'Reilly, DA | 1 |
Bredt, DS; Kobzik, L; Reid, MB; Stamler, JS | 1 |
Bäck, M; Cotgreave, IA; Dahlén, SE; Kumlin, M | 1 |
Fujimura, Y; Ikeda, Y; Iwasaki, T; Koide, T; Matsushita, H; Nagashima, R; Shindo, M; Shiraki, Y; Suzuki, S; Takano, N | 1 |
Falcone, RC; Krell, RD | 1 |
Ito, T; Kato, S; Omoya, H; Yoshida, N | 1 |
Itoh, Z; Iwanaga, Y; Mizumoto, A; Yoshida, N | 1 |
Itoh, Z; Iwanaga, Y; Mizumoto, A; Torii, K; Wakabayashi, K; Yoshida, N | 1 |
Ito, S | 1 |
Aharony, D; Fedyna, JS; Krell, RD; Redkar-Brown, D; Snyder, DW | 1 |
Moss, HE; Sanger, GJ | 1 |
Chen, HI | 1 |
Brown, FJ; Cronk, LA; Hebbel, KC; Krell, RD; Snyder, DW; Yee, YK | 1 |
Aharony, D; Hesp, B; Keith, RA; Krell, RD; Maduskuie, TP; Matassa, VG; Shapiro, HS; Snyder, DW | 1 |
Bermudez, J; Fake, CS; Joiner, GF; Joiner, KA; King, FD; Miner, WD; Sanger, GJ | 1 |
Aharony, D; Redkar-Brown, DG | 1 |
Buckner, CK; Castleman, WL; Saban, R; Will, JA | 1 |
43 other study(ies) available for indazoles and Muscle Contraction
Article | Year |
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Inhibition of the methyltranferase EZH2 improves aortic performance in experimental thoracic aortic aneurysm.
Topics: Animals; Aorta, Thoracic; Aortic Aneurysm, Thoracic; Disease Models, Animal; DNA Methylation; Enhancer of Zeste Homolog 2 Protein; Epigenesis, Genetic; Fibrillin-1; Gene Knockout Techniques; Histones; Humans; Indazoles; Losartan; Marfan Syndrome; Mice; Mice, Knockout; Microfilament Proteins; Muscle Contraction; Muscle Proteins; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Pyridones; RNA, Small Interfering | 2018 |
DL0805-2, a novel indazole derivative, relaxes angiotensin II-induced contractions of rat aortic rings by inhibiting Rho kinase and calcium fluxes.
Topics: Actins; Angiotensin II; Angiotensin II Type 2 Receptor Blockers; Animals; Aorta, Thoracic; Calcium; In Vitro Techniques; Indazoles; Male; Molecular Docking Simulation; Muscle Contraction; Muscle Relaxation; Myocytes, Smooth Muscle; Myosin Light Chains; Phosphorylation; Protein Phosphatase 1; Rats, Sprague-Dawley; Reactive Oxygen Species; rho-Associated Kinases; Signal Transduction; Vasoconstrictor Agents; Vasodilator Agents | 2016 |
Hypotrophic effect of long-term neuronal NO-synthase inhibition on heart and conduit arteries of the Wistar rats.
Topics: Animals; Aorta, Thoracic; Blood Pressure; Body Weight; Carotid Arteries; Coronary Vessels; Dose-Response Relationship, Drug; In Vitro Techniques; Indazoles; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide Synthase Type I; Organ Size; Rats; Rats, Wistar; Time Factors | 2009 |
Presence of cyclic nucleotide-gated channels in the rat urethra and their involvement in nerve-mediated nitrergic relaxation.
Topics: Animals; Calcium Channel Blockers; Cyclic Nucleotide-Gated Cation Channels; Diltiazem; Enzyme Inhibitors; Female; Fluorescent Antibody Technique; Indazoles; Isometric Contraction; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Stereoisomerism; Urethra | 2009 |
YC-1 potentiates the nitric oxide/cyclic GMP pathway in corpus cavernosum and facilitates penile erection in rats.
Topics: Animals; Cells, Cultured; Cyclic GMP; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Guanylate Cyclase; In Vitro Techniques; Indazoles; Male; Muscle Contraction; Muscle, Smooth; Nitric Oxide; Nitroprusside; Oxadiazoles; Penile Erection; Penis; Phenylephrine; Quinoxalines; Rabbits; Rats; Rats, Wistar; Signal Transduction; Vasoconstrictor Agents; Vasodilator Agents | 2003 |
The role of nitric oxide on contractile impairment during endotoxemia in rat diaphragm muscle.
Topics: Animals; Caffeine; Diaphragm; Endotoxemia; Enzyme Inhibitors; Guanidines; In Vitro Techniques; Indazoles; Lipopolysaccharides; Male; Muscle Contraction; Neuromuscular Nondepolarizing Agents; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Oxadiazoles; Quinoxalines; Rats; Rats, Wistar; Ryanodine; Tubocurarine; Vasodilator Agents; Verapamil | 2004 |
Nitric oxide modulates peristaltic muscle activity associated with fluid circulation in the sea pansy Renilla koellikeri.
Topics: Animals; Anthozoa; Body Fluids; California; Guanidines; Immunohistochemistry; Indazoles; Muscle Contraction; Muscles; Neurites; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Oxadiazoles; Peristalsis; Phosphodiesterase Inhibitors; Purinones; Quinoxalines | 2005 |
Development of dihydropyridone indazole amides as selective Rho-kinase inhibitors.
Topics: Amides; Animals; Antihypertensive Agents; Aorta; Blood Pressure; In Vitro Techniques; Indazoles; Intracellular Signaling Peptides and Proteins; Models, Molecular; Muscle Contraction; Muscle, Smooth, Vascular; Protein Serine-Threonine Kinases; Pyridones; Pyrimidines; Rats; Rats, Inbred SHR; rho-Associated Kinases; Structure-Activity Relationship | 2007 |
Resting tension affects eNOS activity in a calcium-dependent way in airways.
Topics: Acetylcholine; Animals; Arginine; Calcium; Dose-Response Relationship, Drug; Drug Interactions; Female; Genistein; Hydroquinones; In Vitro Techniques; Indazoles; Male; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase Type II; Nitric Oxide Synthase Type III; Rabbits; Trachea | 2007 |
Effect of 7-nitro indazole on neurotransmission in the rat vas deferens: mechanisms unrelated to inhibition of nitric oxide synthase.
Topics: Adenosine Triphosphate; Amino Acid Oxidoreductases; Animals; Arginine; Electric Stimulation; In Vitro Techniques; Indazoles; Male; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Norepinephrine; Potassium Chloride; Propranolol; Rats; Rats, Wistar; Synaptic Transmission; Vas Deferens; Yohimbine | 1994 |
Effects of the peptide leukotriene receptor antagonist ICI 198,615 on the in vivo and in vitro changes in guinea pig bladder function which occur after sensitization with ovalbumin.
Topics: Animals; Female; Guinea Pigs; In Vitro Techniques; Indazoles; Indomethacin; Leukotriene Antagonists; Muscle Contraction; Ovalbumin; Pyrilamine; SRS-A; Urinary Bladder; Urodynamics | 1995 |
Pharmacologic modulation of the influence of the epithelium on immunologic- and nonimmunologic-induced histamine release and contraction in guinea pig superfused tracheal strips.
Topics: Animals; Epithelium; Female; Guinea Pigs; Histamine Release; Hydroxyurea; In Vitro Techniques; Indazoles; Indomethacin; Muscle Contraction; Ovalbumin; Pyrilamine; Trachea; Tubocurarine | 1993 |
Characterization of the novel nitric oxide synthase inhibitor 7-nitro indazole and related indazoles: antinociceptive and cardiovascular effects.
Topics: Amino Acid Oxidoreductases; Analgesics; Animals; Arginine; Blood Pressure; Cardiovascular Agents; Cerebellum; Enzyme Inhibitors; Formaldehyde; In Vitro Techniques; Indazoles; Male; Mice; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide Synthase; Pain Measurement; Rabbits; Rats | 1993 |
BAY u9773, a novel antagonist of cysteinyl-leukotrienes with activity against two receptor subtypes.
Topics: Animals; Binding, Competitive; Bronchi; Dicarboxylic Acids; Ferrets; Guinea Pigs; In Vitro Techniques; Indazoles; Leukotriene C4; Leukotriene D4; Lung; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Propionates; Quinolines; Rats; Rats, Wistar; Receptors, Immunologic; Sheep; Spleen; SRS-A; Trachea | 1994 |
Characterisation of leukotriene receptors on rat lung strip.
Topics: Animals; Dicarboxylic Acids; In Vitro Techniques; Indazoles; Leukotriene Antagonists; Leukotrienes; Lung; Male; Muscle Contraction; Muscle, Smooth; Potassium Chloride; Propionates; Quinolines; Rats; Rats, Wistar; Receptors, Leukotriene; SRS-A | 1994 |
The 5-lipoxygenase inhibitory activity of zileuton in in vitro and in vivo models of antigen-induced airway anaphylaxis.
Topics: Anaphylaxis; Animals; Anti-Inflammatory Agents, Non-Steroidal; Bronchoconstriction; Disease Models, Animal; Dose-Response Relationship, Drug; Female; Guinea Pigs; Humans; Hydroxyurea; Indazoles; Lipoxygenase Inhibitors; Male; Meclofenamic Acid; Muscle Contraction; Muscle, Smooth; Pyrilamine; SRS-A; Trachea | 1994 |
Phosphoramidon augments contraction of guinea pig tracheal smooth muscle induced by histamine and leukotriene-D4.
Topics: Anaphylaxis; Animals; Antigens; Dinoprost; Diphenhydramine; Glycopeptides; Guinea Pigs; Histamine; In Vitro Techniques; Indazoles; Leukotriene D4; Muscle Contraction; Muscle, Smooth; Neprilysin; Prostaglandin D2; SRS-A; Trachea | 1994 |
The cysteinyl-leukotriene receptor antagonist BAY u9773 is a competitive antagonist of leukotriene C4 in the guinea-pig ileum.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Female; Guinea Pigs; Ileum; In Vitro Techniques; Indazoles; Leukotriene Antagonists; Leukotriene C4; Leukotriene D4; Male; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Prostaglandin Endoperoxides, Synthetic; Receptors, Leukotriene; SRS-A; Thromboxane A2; Vasoconstrictor Agents | 1996 |
Differential effects of isoliquiritigenin and YC-1 in rat aortic smooth muscle.
Topics: Aldehyde Reductase; Animals; Carotid Arteries; Chalcone; Chalcones; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Guanylate Cyclase; Indazoles; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phosphodiesterase Inhibitors; Platelet Aggregation Inhibitors; Rats; Rats, Sprague-Dawley | 1997 |
Leukotrienes in acetylcholine-induced contraction of esophageal circular smooth muscle in experimental esophagitis.
Topics: Acetylcholine; Animals; Arachidonic Acid; Cats; Diglycerides; Drug Synergism; Esophagitis; Esophagus; Female; Indazoles; Leukotrienes; Male; Muscle Contraction; Muscle, Smooth; Phospholipases A; Phospholipases A2 | 1997 |
Nitric oxide stimulates skeletal muscle glucose transport through a calcium/contraction- and phosphatidylinositol-3-kinase-independent pathway.
Topics: 3-O-Methylglucose; Androstadienes; Animals; Calcium; Dantrolene; Dibutyryl Cyclic GMP; Enzyme Inhibitors; Female; Glucose; Indazoles; Muscle Contraction; Muscle, Skeletal; Nitric Oxide; Nitric Oxide Synthase; Nitroprusside; omega-N-Methylarginine; Phosphatidylinositol 3-Kinases; Rats; Rats, Sprague-Dawley; Sulfonamides; Wortmannin | 1997 |
Nitric oxide-sensitive guanylyl cyclase inhibits acetylcholine release and excitatory motor transmission in the guinea-pig ileum.
Topics: Acetylcholine; Animals; Depression, Chemical; Electric Stimulation; Enzyme Inhibitors; Female; Guanylate Cyclase; Guinea Pigs; Ileum; Indazoles; Male; Motor Neurons; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Oxadiazoles; Quinoxalines; Synaptic Transmission | 1998 |
Synthesis and structure-activity relationships of potent and orally active 5-HT4 receptor antagonists: indazole and benzimidazolone derivatives.
Topics: Adamantane; Administration, Oral; Adrenergic alpha-Antagonists; Animals; Aorta; Brain; Drug Evaluation, Preclinical; Esophagus; Guinea Pigs; Ileum; In Vitro Techniques; Indazoles; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, alpha-1; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Structure-Activity Relationship | 1998 |
alpha1-syntrophin gene disruption results in the absence of neuronal-type nitric-oxide synthase at the sarcolemma but does not induce muscle degeneration.
Topics: Animals; Base Sequence; Calcium-Binding Proteins; DNA Primers; Enzyme Inhibitors; Immunohistochemistry; Indazoles; Membrane Proteins; Mice; Mice, Inbred C3H; Mice, Inbred C57BL; Mice, Knockout; Muscle Contraction; Muscle Proteins; Muscle, Skeletal; NG-Nitroarginine Methyl Ester; Nitric Oxide Donors; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Nitroprusside; Sarcolemma | 1999 |
Effects of the soluble guanylyl cyclase activator, YC-1, on vascular tone, cyclic GMP levels and phosphodiesterase activity.
Topics: Animals; Aorta, Thoracic; Cyclic GMP; Enzyme Activation; Enzyme Inhibitors; Guanylate Cyclase; In Vitro Techniques; Indazoles; Isoenzymes; Kinetics; Muscle Contraction; Muscle Relaxation; Muscle Tonus; Muscle, Smooth, Vascular; Nitric Oxide Donors; Nitroprusside; Nitroso Compounds; Oxadiazoles; Phosphoric Diester Hydrolases; Quinoxalines; Rabbits; Vasodilator Agents | 1999 |
Intestinal motor depression by 7-nitroindazole through an action unrelated to nitric oxide synthase inhibition.
Topics: Animals; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Gastrointestinal Motility; Guinea Pigs; Imidazoles; In Vitro Techniques; Indazoles; Indomethacin; Intestine, Small; Male; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Peptide Fragments; Peristalsis; Sincalide; Substance P; Tetrodotoxin | 1999 |
YC-1 enhances the responsiveness of tolerant vascular smooth muscle to glyceryl trinitrate.
Topics: Animals; Aorta, Thoracic; Cyclic GMP; Drug Tolerance; Enzyme Activators; In Vitro Techniques; Indazoles; Isometric Contraction; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroglycerin; Rabbits; Vasodilator Agents | 2001 |
Nitric oxide modulates excitation-contraction coupling in the diaphragm.
Topics: Animals; Diaphragm; Enzyme Inhibitors; Guanidines; Hindlimb; Indazoles; Male; Muscle Contraction; Muscle, Skeletal; Nitrates; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type III; Nitrites; Nitroarginine; Rats; Rats, Sprague-Dawley | 1998 |
An alternative pathway for metabolism of leukotriene D(4): effects on contractions to cysteinyl-leukotrienes in the guinea-pig trachea.
Topics: Animals; Borates; Cysteine; Dicarboxylic Acids; Dose-Response Relationship, Drug; Glutathione; Guinea Pigs; In Vitro Techniques; Indazoles; Leukotriene Antagonists; Leukotriene C4; Leukotriene D4; Leukotriene E4; Leukotrienes; Male; Membrane Proteins; Muscle Contraction; Propionates; Quinolines; Receptors, Leukotriene; Serine; SRS-A; Trachea | 2001 |
Pharmacological studies on a new thymoleptic antidepressant, 1-[3-(dimethylamino)propyl]-5-methyl-3-phenyl-1H-indazole (FS-32).
Topics: Acetylcholine; Amphetamine; Animals; Antidepressive Agents; Barbiturates; Behavior, Animal; Biogenic Amines; Blood Pressure; Brain Chemistry; Catecholamines; Cats; Dogs; Electroencephalography; Female; Guinea Pigs; Haplorhini; In Vitro Techniques; Indazoles; Levodopa; Macaca fascicularis; Male; Mice; Muscle Contraction; Muscle, Smooth; Physostigmine; Pyrazoles; Rabbits; Rats; Reserpine; Tremorine | 1979 |
Guinea pig gall bladder contains a single peptide leukotriene receptor which resembles that present in human conducting airway smooth muscle.
Topics: Animals; Gallbladder; Guinea Pigs; Humans; Indazoles; Lung; Male; Muscle Contraction; Muscle, Smooth; Receptors, Immunologic; Receptors, Leukotriene; Signal Transduction; SRS-A | 1992 |
5-HT3 receptor antagonist effects of DAT-582, (R) enantiomer of AS-5370.
Topics: Animals; Azepines; Bradycardia; Cisplatin; Ferrets; Guinea Pigs; Ileum; In Vitro Techniques; Indazoles; Male; Muscle Contraction; Muscle, Smooth; Rats; Serotonin Antagonists; Stereoisomerism; Vomiting | 1992 |
Effects of 5-hydroxytryptamine 3 receptor antagonists on gastrointestinal motor activity in conscious dogs.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Digestion; Dogs; Dose-Response Relationship, Drug; Female; Gastrointestinal Motility; Granisetron; Imidazoles; Indazoles; Indoles; Infusions, Intravenous; Injections, Intravenous; Male; Motilin; Motor Activity; Muscle Contraction; Muscle, Smooth; Ondansetron; Serotonin Antagonists; Time Factors; Tropisetron | 1991 |
Involvement of 5-hydroxytryptamine 3 receptors in regulation of interdigestive gastric contractions by motilin in the dog.
Topics: Acetylcholine; Animals; Digestion; Dogs; Gastrointestinal Motility; Granisetron; Imidazoles; Indazoles; Motilin; Muscle Contraction; Muscle, Smooth; Ondansetron; Receptors, Serotonin; Serotonin Antagonists; Stomach | 1991 |
[Study on mechanism of interdigestive migrating contractions of a canine stomach].
Topics: Animals; Dogs; Fasting; Gastrointestinal Motility; Granisetron; Indazoles; Motilin; Muscle Contraction; Muscle, Smooth; Serotonin Antagonists; Stomach | 1990 |
Pharmacologic characterization of the contractile activity of peptide leukotrienes in guinea-pig pulmonary artery.
Topics: Acetophenones; Animals; Borates; Drug Synergism; Endothelium, Vascular; Guinea Pigs; In Vitro Techniques; Indazoles; Indomethacin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Pulmonary Artery; Receptors, Immunologic; Receptors, Leukotriene; Serine; SRS-A; Tetrazoles | 1990 |
The effects of granisetron, ICS 205-930 and ondansetron on the visceral pain reflex induced by duodenal distension.
Topics: Animals; Blood Pressure; Duodenum; Granisetron; Imidazoles; Indazoles; Indoles; Male; Morphine; Muscle Contraction; Muscle, Smooth; Ondansetron; Pain; Pyrazoles; Rats; Rats, Inbred Strains; Reflex; Serotonin Antagonists; Stomach; Tropisetron; Vagotomy | 1990 |
Evidence for the presynaptic action of 5-hydroxytryptamine and the involvement of purinergic innervation in the rabbit lower urinary tract.
Topics: Adenosine Triphosphate; Animals; Atropine; Electric Stimulation; Female; Granisetron; In Vitro Techniques; Indazoles; Indoles; Male; Muscle Contraction; Muscle, Smooth; Purines; Rabbits; Serotonin; Serotonin Antagonists; Synapses; Tropanes; Tropisetron; Urethra; Urinary Tract | 1990 |
Evolution of a series of peptidoleukotriene antagonists: synthesis and structure-activity relationships of 1,6-disubstituted indoles and indazoles.
Topics: Animals; Guinea Pigs; In Vitro Techniques; Indazoles; Indoles; Muscle Contraction; Pyrazoles; SRS-A; Structure-Activity Relationship | 1990 |
Evolution of a series of peptidoleukotriene antagonists: synthesis and structure/activity relationships of 1,3,5-substituted indoles and indazoles.
Topics: Animals; Dyspnea; Guinea Pigs; In Vitro Techniques; Indazoles; Indoles; Muscle Contraction; Pyrazoles; SRS-A; Structure-Activity Relationship | 1990 |
5-Hydroxytryptamine (5-HT3) receptor antagonists. 1. Indazole and indolizine-3-carboxylic acid derivatives.
Topics: Animals; Antiemetics; Carboxylic Acids; Ferrets; Guinea Pigs; Ileum; In Vitro Techniques; Indazoles; Indicators and Reagents; Indolizines; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Molecular Structure; Muscle Contraction; Muscle, Smooth; Pyrazoles; Rats; Receptors, Serotonin; Reflex; Serotonin; Serotonin Antagonists; Stereoisomerism; Structure-Activity Relationship | 1990 |
Inhibition of antigen-induced contraction of guinea pig trachea by ICI 198,615.
Topics: Animals; Antigens; Guinea Pigs; In Vitro Techniques; Indazoles; Indomethacin; Leukotrienes; Lipoxygenase Inhibitors; Male; Muscle Contraction; Muscle, Smooth; Ovalbumin; Phospholipid Ethers; Platelet Activating Factor; Pyrazoles; Pyrilamine; SRS-A; Trachea | 1989 |
Analysis of leukotriene receptor antagonists on isolated human intralobar airways.
Topics: Acetophenones; Azoles; Barium; Bronchi; Chromones; Humans; Indazoles; Muscle Contraction; Muscle, Smooth; Pyrazoles; Receptors, Leukotriene; Receptors, Prostaglandin; SRS-A; Tetrazoles | 1988 |