Page last updated: 2024-08-21

indazoles and Abdominal Migraine

indazoles has been researched along with Abdominal Migraine in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (25.00)18.2507
2000's2 (25.00)29.6817
2010's3 (37.50)24.3611
2020's1 (12.50)2.80

Authors

AuthorsStudies
Ator, MA; Brown, AJH; Brown, J; Bucknell, SJ; Cansfield, AD; Cansfield, JE; Christopher, JA; Congreve, M; Cseke, G; Deflorian, F; Jones, CR; Mason, JS; O'Brien, MA; Ott, GR; Pickworth, M; Southall, SM1
Cantor, GH; Chaturvedula, PV; Conway, CM; Davis, C; Denton, R; Dubowchik, GM; Keavy, D; Macci, R; Macor, JE; Mathias, N; Mercer, SE; Moench, P; Pin, SS; Schartman, R; Signor, L; Thalody, G; Whiterock, V; Xu, C1
Chaturvedula, PV; Conway, CM; Cook, DA; Davis, CD; Degnan, AP; Denton, R; Dubowchik, GM; Han, X; Macci, R; Macor, JE; Mathias, NR; Moench, P; Pin, SS; Ren, SX; Schartman, R; Signor, LJ; Thalody, G; Widmann, KA; Xu, C1
Conway, CM; Dalterio, RA; Degnan, AP; Dubowchik, GM; Macci, R; Macor, JE; Mercer, SE; Schartman, R; Xu, C1
Fischer, MJ1
Allena, M; Amantea, D; Bolla, M; Greco, R; Mangione, AS; Meazza, C; Mizoguchi, H; Nappi, G; Sandrini, G; Tassorelli, C1
Clifford Rose, F; Couturier, EG; Foster, CA; Hering, R; Steiner, TJ1
Davis, A; Merrill, CF; Rowat, BM; South, V1

Reviews

1 review(s) available for indazoles and Abdominal Migraine

ArticleYear
Calcitonin gene-related peptide receptor antagonists for migraine.
    Expert opinion on investigational drugs, 2010, Volume: 19, Issue:7

    Topics: Animals; Azepines; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Clinical Trials as Topic; Dipeptides; Humans; Imidazoles; Indazoles; Migraine Disorders; Piperazines; Quinazolines; Quinazolinones; Treatment Outcome; Trigeminal Nerve

2010

Trials

2 trial(s) available for indazoles and Abdominal Migraine

ArticleYear
First clinical study of the selective 5-HT3 antagonist, granisetron (BRL 43694), in the acute treatment of migraine headache.
    Headache, 1991, Volume: 31, Issue:5

    Topics: Adult; Granisetron; Humans; Indazoles; Infusions, Intravenous; Middle Aged; Migraine Disorders; Serotonin Antagonists

1991
A double-blind comparison of granisetron and placebo for the treatment of acute migraine in the emergency department.
    Cephalalgia : an international journal of headache, 1991, Volume: 11, Issue:5

    Topics: Acute Disease; Adult; Double-Blind Method; Emergency Service, Hospital; Female; Granisetron; Humans; Indazoles; Male; Middle Aged; Migraine Disorders; Placebos; Serotonin Antagonists

1991

Other Studies

5 other study(ies) available for indazoles and Abdominal Migraine

ArticleYear
Structure-Based Drug Discovery of
    Journal of medicinal chemistry, 2020, 07-23, Volume: 63, Issue:14

    Topics: Animals; Binding Sites; Calcitonin Gene-Related Peptide Receptor Antagonists; Dogs; Drug Design; Humans; Indazoles; Macaca fascicularis; Migraine Disorders; Molecular Docking Simulation; Molecular Structure; Rats; Receptors, Calcitonin Gene-Related Peptide; Spiro Compounds; Structure-Activity Relationship

2020
Discovery of (R)-N-(3-(7-methyl-1H-indazol-5-yl)-1-(4-(1-methylpiperidin-4-yl)-1-oxopropan-2-yl)-4-(2-oxo-1,2-dihydroquinolin-3-yl)piperidine-1-carboxamide (BMS-742413): a potent human CGRP antagonist with superior safety profile for the treatment of migr
    Bioorganic & medicinal chemistry letters, 2013, Jun-01, Volume: 23, Issue:11

    Topics: Administration, Intranasal; Amides; Animals; Caco-2 Cells; Calcitonin Gene-Related Peptide Receptor Antagonists; Callithrix; Coronary Vessels; Drug Evaluation, Preclinical; Face; Humans; Indazoles; Migraine Disorders; Quinolones; Rabbits; Rats; Receptors, Calcitonin Gene-Related Peptide; Respiratory Mucosa

2013
Discovery of (R)-4-(8-fluoro-2-oxo-1,2-dihydroquinazolin-3(4H)-yl)-N-(3-(7-methyl-1H-indazol-5-yl)-1-oxo-1-(4-(piperidin-1-yl)piperidin-1-yl)propan-2-yl)piperidine-1-carboxamide (BMS-694153): a potent antagonist of the human calcitonin gene-related peptid
    Journal of medicinal chemistry, 2008, Aug-28, Volume: 51, Issue:16

    Topics: Administration, Intranasal; Animals; Biological Availability; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Callithrix; Coronary Vessels; Face; Humans; Indazoles; Migraine Disorders; Quinazolinones; Rabbits; Regional Blood Flow; Vasodilation

2008
Carbamates as potent calcitonin gene-related peptide antagonists with improved solution stability.
    Bioorganic & medicinal chemistry letters, 2009, Jul-01, Volume: 19, Issue:13

    Topics: Calcitonin Gene-Related Peptide Receptor Antagonists; Carbamates; Drug Stability; Humans; Indazoles; Migraine Disorders; Quinazolinones; Quinolones; Receptors, Calcitonin Gene-Related Peptide

2009
Temporal profile of vascular changes induced by systemic nitroglycerin in the meningeal and cortical districts.
    Cephalalgia : an international journal of headache, 2011, Volume: 31, Issue:2

    Topics: Animals; Blood Pressure; Cerebral Cortex; Cerebrovascular Circulation; Enzyme Inhibitors; Indazoles; Male; Meningeal Arteries; Meninges; Migraine Disorders; NG-Nitroarginine Methyl Ester; Nitroglycerin; Rats; Rats, Sprague-Dawley; Vasodilation; Vasodilator Agents

2011