Page last updated: 2024-08-17

indacrinone and Alzheimer Disease

indacrinone has been researched along with Alzheimer Disease in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's4 (50.00)24.3611
2020's4 (50.00)2.80

Authors

AuthorsStudies
Dai, Y; Fang, T; Jiang, T; Qiao, J; Xu, Y1
Bansal, R; Rana, P; Singh, R1
Abibiglue, YT; Bavili, A; Dastmalchi, S; Etemadi, A; Hamzeh-Mivehroud, M; Hemmati, S; Shahrivar-Gargari, M1
Albertini, C; Bartolini, M; Bolognesi, ML; de Sena Murteira Pinheiro, P; Di Pietri, F; Fato, R; Perone, R; Petralla, S; Pulkrabkova, L; Rizzardi, N; Soukup, O; Tramarin, A; Uliassi, E1
Huang, L; Li, X; Meng, F; Miao, H; Sun, Y1
Andrisano, V; Bartolini, M; Cavalli, A; Ceccarini, L; Gobbi, S; Piazzi, L; Rampa, A; Recanatini, M; Rizzo, S1
Huang, L; Li, XS; Mao, F; Meng, FC; Qin, F; Shan, WJ1
Gan, CS; Ge, JF; Nan, DD; Pan, J; Qiao, JP; Wang, CW; Zhou, JN1

Other Studies

8 other study(ies) available for indacrinone and Alzheimer Disease

ArticleYear
Multi-fluorine labeled indanone derivatives as potential MRI imaging probes for β-Amyloid plaques.
    Chemical biology & drug design, 2023, Volume: 101, Issue:3

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Brain; Fluorine; Humans; Indans; Magnetic Resonance Imaging; Mice; Mice, Transgenic; Plaque, Amyloid; Tissue Distribution

2023
Synthesis,
    Current computer-aided drug design, 2023, Volume: 19, Issue:2

    Topics: Alzheimer Disease; Animals; Indans; Lipopolysaccharides; Mice; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Rats; Structure-Activity Relationship

2023
Design, Synthesis, and Biological Evaluation of Novel Indanone Derivatives as Cholinesterase Inhibitors for Potential Use in Alzheimer's Disease.
    Chemistry & biodiversity, 2023, Volume: 20, Issue:8

    Topics: Acetylcholinesterase; Alzheimer Disease; Amines; Butyrylcholinesterase; Cholinesterase Inhibitors; Donepezil; Humans; Indans; Molecular Docking Simulation; Structure-Activity Relationship

2023
Turning Donepezil into a Multi-Target-Directed Ligand through a Merging Strategy.
    ChemMedChem, 2021, 01-08, Volume: 16, Issue:1

    Topics: Acetylcholinesterase; Alzheimer Disease; Amyloid beta-Peptides; Antioxidants; Blood-Brain Barrier; Cell Line, Tumor; Cell Survival; Cholinesterase Inhibitors; Donepezil; Drug Design; Humans; Indans; Ligands; Neuroprotective Agents; Oxidative Stress; Protein Aggregates; Structure-Activity Relationship

2021
Discovery of indanone derivatives as multi-target-directed ligands against Alzheimer's disease.
    European journal of medicinal chemistry, 2014, Nov-24, Volume: 87

    Topics: Acetylcholinesterase; Alzheimer Disease; Amyloid beta-Peptides; Antioxidants; Blood-Brain Barrier; Butyrylcholinesterase; Cholinesterase Inhibitors; Drug Design; Humans; Indans; Inhibitory Concentration 50; Ligands; Peptide Fragments; Permeability; Protein Aggregates

2014
Targeting Alzheimer's disease: Novel indanone hybrids bearing a pharmacophoric fragment of AP2238.
    Bioorganic & medicinal chemistry, 2010, Mar-01, Volume: 18, Issue:5

    Topics: Acetylcholinesterase; Alzheimer Disease; Amyloid beta-Peptides; Antineoplastic Combined Chemotherapy Protocols; Benzylamines; Binding Sites; Bleomycin; Cholinesterase Inhibitors; Computer Simulation; Coumarins; Donepezil; Humans; Indans; Lomustine; Methotrexate; Peptide Fragments; Piperidines; Recombinant Proteins; Stilbenes; Structure-Activity Relationship; Tetrahydronaphthalenes

2010
Design, synthesis, and evaluation of indanone derivatives as acetylcholinesterase inhibitors and metal-chelating agents.
    Bioorganic & medicinal chemistry letters, 2012, Jul-01, Volume: 22, Issue:13

    Topics: Acetylcholinesterase; Alzheimer Disease; Chelating Agents; Cholinesterase Inhibitors; Drug Design; Humans; Indans; Kinetics; Metals; Pyridines; Structure-Activity Relationship

2012
Novel indanone derivatives as potential imaging probes for β-amyloid plaques in the brain.
    Chembiochem : a European journal of chemical biology, 2012, Jul-23, Volume: 13, Issue:11

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Brain; Humans; Indans; Male; Mice; Mice, Inbred ICR; Molecular Imaging; Molecular Probes; Plaque, Amyloid; Radiopharmaceuticals; Tissue Distribution

2012