imatinib mesylate has been researched along with Benign Neoplasms in 306 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 178 (58.17) | 29.6817 |
2010's | 102 (33.33) | 24.3611 |
2020's | 26 (8.50) | 2.80 |
Authors | Studies |
---|---|
Bharathi, EV; Dastagiri, D; Kamal, A; Pal-Bhadra, M; Pushpavalli, SN; Ramaiah, MJ; Reddy, JS; Reddy, MK; Reddy, TL; Sagar, MV | 1 |
Awadasseid, A; Jiang, SK; Liang, J; Sugiyama, H; Wu, YL; Xiong, XQ; Xu, L; Zhang, M; Zhang, W; Zhao, XY | 1 |
Johnson, GL; Ramos, AF; Rosner, MR; Yesilkanal, AE | 1 |
Chatelut, E; Clarke, WA; Fotoohi, AK; Larson, RA; Martin, JH; Mathijssen, RHJ; Salamone, SJ | 1 |
Fujii, T; Kitahara, S; Kobayashi, S; Matsui, T; Matsunaga, T; Ohno, N; Sahara, N; Sakamoto, N | 1 |
Bastos, M; Boechat, N; Dantas, R; Moura, S; Neto, J; Oliveira, A; Pimentel, L; Silva-Jr, F | 1 |
Bertoletti, L; Bin, V; Delavenne, X; Hodin, S; Lafaie, L; Saïb, S | 1 |
Li, CW; Lin, D; Mi, YC; Tian, Z; Wan, L; Wang, Z | 1 |
Attrill, E; Brown, LS; Cashion, JM; Courtney, JM; Foster, CG; Howells, DW; King, NE; Premilovac, D; Sutherland, BA | 1 |
Nathan, J; Palanivel, G; Shameera, R | 1 |
Dirkson, A; Gelderblom, H; Kraaij, W; van Oortmerssen, G; Verberne, S | 1 |
Anshu, A; Das, R; Jamwal, M; Lad, D; Rathore, S; Sreedharanunni, S; Virk, H | 1 |
Cho-Vega, JH; Loghavi, S | 1 |
Coltro, G; Santi, R | 1 |
Berry, A; Constantine, G; Khoury, P; Klion, AD; Kuang, FL; Lane, AA; Makiya, M; Maric, I; Pongdee, T; Rheinbay, E; Sun, X; Thumm, L; Wetzler, L; Yoon, P | 1 |
Agarbati, S; Benfaremo, D; Moroncini, G; Mozzicafreddo, M; Paolini, C; Svegliati Baroni, S | 1 |
Dal Cin, P; Ebert, BL; Grinshpun, DE; Hobbs, GS; Iafrate, AJ; Jan, M; Nardi, V; Sykes, DB; Villalba, JA | 1 |
Abbasnezhad, A; Abd El-Ghafar, OA; Abhilash, L; Abouzid, KAM; Achberger, AM; Ackerman, S; Akhatayeva, Z; Akin, D; Al-Kaysi, RO; Alakhdar, AA; Alame, M; Aleksic Sabo, V; Alinezhadbalalami, N; Allen, JD; Alonso, JM; Alqatani, S; Alsayed, B; Álvarez Larraondo, M; Alvarez, M; Amini, SB; An, Z; Anasir, MI; Anderson, GH; Andremont, A; Andrés, S; Angel, S; Anigboro, AA; Anini, Y; Antonides, CFJ; Arafa, K; Arafa, RK; Aryal, UK; Asbaghi, O; Assefa, MK; Atyah, M; Avwioroko, OJ; Ayora-Talavera, G; Azpilikueta, A; Azyazov, VN; Ba, YF; Bachmann, KF; Badoual, J; Bae, SJ; Baek, SH; Bahrami, B; Bai, J; Baid-Agrawal, S; Bailey, MR; Baillie, JK; Balani, N; Balcar, VJ; Banica, T; Banks, L; Barb, J; Bardeen, CJ; Barrett, HE; Bartnikowski, N; Bashir, R; Battaglia, M; Bautista-Hernández, V; Becker, B; Beekman, FJ; Benidir, M; Benjelloun, M; Bentley, RF; Bergé, J; Berger, D; Bernsen, MR; Berraondo, P; Bhattacharya, R; Bhayani, SB; Bi, W; Bi, X; Bi, YL; Bi, Z; Bian, K; Biesecker, LG; Billadeau, DD; Blaszczyk, R; Blum, JL; Boachie, R; Boelte, K; Bogers, AJJC; Boileau, I; Bonduelle, C; Bonny, O; Bonsu, JM; Boos, LA; Borges-Argáez, R; Bouchard, PA; Boudot, C; Bourgeade-Delmas, S; Boutet-Robinet, E; Boyle, AJ; Branigan, D; Briones, S; Broniowska, KA; Brossas, JY; Brown, WA; Brzezinska, J; Buitron, G; Burnier, M; Bursulaya, B; Burton, PR; Bush, AA; Busuttil, RW; Cabello-Aguilar, S; Cáceres-Farfán, M; Cacheux, V; Caffrey, PJ; Cai, B; Cai, Q; Cai, S; Cai, Y; Calders, P; Cammarota, G; Campbell, DA; Cancelli, C; Cao, Q; Cao, WH; Cao, X; Capet, M; Capoluongo, E; Carey, ME; Carnero, M; Carrasco, LI; Carreno, J; Carrillo-Reyes, J; Casini, I; Cassar, M; Catalan, G; Cattamanchi, A; Cazares-Granillo, M; Celie, B; Cen, YK; Cena, H; Cerbo, RM; Ceron, E; Cetina-Montejo, L; Chaâbane-Banaoues, R; Chabanet, C; Chace-Donahue, F; Chalfun-Júnior, A; Chan-Balan, R; Chang, CS; Chen, CS; Chen, D; Chen, J; Chen, L; Chen, PN; Chen, Q; Chen, S; Chen, W; Chen, WP; Chen, X; Chen, Z; Cheng, H; Cheng, J; Cheng, Q; Cheng, T; Chi, T; Chianelli, D; Chieppa, M; Child, CJ; Cho, JH; Cho, JY; Chogtu, B; Choi, GH; Choi, J; Choi, M; Choi, NG; Cholu, CO; Chow, ES; Chowdhury, AH; Chu, PC; Chu, Q; Chu, S; Chua, H; Chung, T; Chunyan, L; Church, JS; Civardi, E; Cobiella, J; Colinge, J; Collado, CJ; Collins, TJ; Cong, LM; Conkrite, KL; Cope, SJ; Corbett, JA; Cornet, M; Cornillot, E; Corvaisier, S; Costes-Martineau, V; Courtioux, B; Coussens, M; Covino, M; Criado, A; Cui, J; Cui, Y; Cunitz, BW; Curry, AE; Cussó, L; D'Urzo, AD; D'Urzo, KA; Dabbous, S; Dahlgren, RA; Dai, H; Dai, T; Dai, W; Dalinghaus, M; Dang, S; Davalos, RV; Davidson, H; de Andrea, CE; De Angelis, M; de Blois, E; de Carvalho, PA; De Clercq, E; De Giuseppe, R; de Jong, M; De Langhe, S; De Oliveira, L; de Souza Pinto Lemgruber, R; de Souza, LB; de Swart, J; De Wandele, I; de Woestijne, PCV; Delaney, S; Delorme, M; Delvenne, P; Deng, L; Deng, Z; Denkinger, CM; der Meulen, MHV; Deraeve, C; Desco, M; DeSilva, S; Destere, A; Dhali, A; Di Ciano, P; Dias-Santagata, D; Diskin, SJ; Djè, MK; Doddipatla, S; Doerr, AJ; Dokla, EME; Domiciano, D; Domingo, N; Dong, C; Dong, J; Dong, Q; Dong, S; Dong, X; Dong, Z; Douair, I; Douglas, TA; Doyle, SM; Drain, PK; Du, K; Du, L; Du, Q; Du, S; Duan, C; Duan, H; Duan, J; Duan, S; Duan, W; Dueluzeau, R; Dukic, L; Dunmire, BL; Duvauchelle, T; Dymek, B; Dzwonek, K; Earnest, A; Eckardt, KU; El Ghadraoui, L; El Massoudi, S; Elloumi, F; Elnour, IE; Embarak, S; Ende, M; England, K; Enikeev, D; Enyedy, I; Epple, R; Erickson, GE; Eriksson, J; Erndt-Marino, J; Errachidi, F; Etxeberria, I; Evan, AP; Fairlamb, AH; Falahi, E; Fan, CC; Fan, H; Fan, M; Fan, MZ; Fan, S; Fan, Y; Fang, CS; Fang, J; Fang, X; Fang, Z; Farmany, A; Farooqi, A; Farouk, HO; Fazelipour, S; Feng, D; Feng, J; Feng, JX; Feng, YL; Ferraz, SL; Ferreira, CR; Figenshau, RS; Finn, AV; Fiseha, T; Fleischer, AS; Fogleman, AD; Fontaine, O; Ford, CR; Fouladvand, F; Four, M; Fousteri, G; Francis, JR; Fraser, JF; Frazier, RP; Fu, H; Fu, P; Fu, YJ; Fujishima, A; Fuster, V; Gabilan, JC; Gagliani, N; Gai, QY; Galán-Arriola, C; Gale, P; Galimova, GR; Galkin, A; Gallo, A; Gallo, AA; Gang, DD; Ganschow, S; Gao, C; Gao, F; Gao, GP; Gao, H; Gao, K; Gao, M; Gao, MY; Gao, P; Gao, R; Gao, S; Gao, WJ; Gao, Y; Garbacz, P; García Ruiz, L; Garcia, EM; Garofoli, F; Gasbarrini, A; Gattinoni, L; Gaudig, M; Gbureck, U; Ge, X; Genko, N; Gentile, GL; George, MW; Gerety, GF; Gestwicki, JE; Geusens, PP; Ghassemi, M; Giardina, JD; Giebultowicz, JM; Gifford, CA; Gijsen, FJH; Gilfillan, R; Gilson, E; Gingl, K; Giuliano, C; Glybochko, P; Goessler, W; Gofflot, S; Golab, J; Goldstein, A; Golebiowski, A; Gómez, L; Gómez-Carballo, J; Gonçalves, PEO; Gonzales, R; Gonzalez-Cotto, M; González-Fernández, D; Gonzalez-Lopez de Turiso, F; Goodman, JM; Govinda Raju, S; Grimm, J; Gross, AJ; Gruenheid, S; Gu, C; Gu, FF; Gu, S; Gu, Z; Guest, RL; Gui, C; Gui, J; Guillem, A; Guo, G; Guo, L; Guo, Q; Guo, S; Guo, SW; Guo, W; Guo, Y; Guo, YG; Guo, Z; Guretzky, JA; Haenggi, M; Hahn, MS; Hakkola, J; Halim, AA; Hampel, D; Han, B; Han, BH; Han, D; Han, G; Han, J; Han, LZ; Han, R; Han, S; Han, X; Han, Z; Handley, MA; Hanke, I; Hannongbua, S; Hao, P; Happ, JT; Hara, M; Haraux, F; Hare, JL; Harper, JD; Hartley, AM; Harvey, E; Hashimoto, K; Hassan, HM; Hautajärvi, H; Hayton, TW; He, C; He, H; He, HJ; He, WP; He, Y; He, Z; Hedrick, V; Heffernan, JK; Hegrová, J; Heidarimoghadam, R; Helms, K; Hengphasatporn, K; Henry, D; Herrmann, TRW; Hesson, T; Himmelbauer, MK; Hindle, A; Hoffmann, R; Hogg, N; Hong, KB; Hong, SK; Honjol, Y; Hood, C; Hsi, RS; Hsu, JL; Hu, B; Hu, BC; Hu, D; Hu, H; Hu, J; Hu, K; Hu, M; Hu, MK; Hu, T; Hu, W; Hu, Y; Hu, Z; Hua, S; Huang, H; Huang, J; Huang, L; Huang, M; Huang, P; Huang, X; Huang, Y; Huang, Z; Hukkanen, J; Hung, MC; Huo, X; Hyötyläinen, T; Ianiro, G; Ibanez, B; Imran, M; Ireland, S; Irwin, MS; Ishiguro, H; Jackowski, K; Jackson, C; Jacob, SI; Jahromy, MH; Jakob, SM; Jang, J; Javvaji, PK; Jefferson, KK; Jena, P; Ji, H; Jiang, F; Jiang, GH; Jiang, H; Jiang, J; Jiang, X; Jiang, Z; Jiao, J; Jiménez, A; Jin, X; Jincai, W; Jintao, X; Jo, K; Jofra, T; Johari, Y; Johnson, ACM; Jones, JH; Josephine Fauci, A; Juhl, AK; Jun, S; Kaiser, RI; Kajioka, J; Kajiyama, H; Kalliyil, A; Kalthur, SG; Kamalanathan, M; Kamaldinov, T; Kanaani, L; Kang, D; Kang, J; Kang, S; Känsäkoski, P; Kaplan, DL; Karwan, M; Kasibhatla, S; Kaur, A; Kawazoe, Y; Ke, C; Keyser, J; Khalique, A; Khan, IT; Kharshoum, RM; Kher, R; Kherani, J; Ki, KK; Kikkawa, F; Kikkawa, R; Kim, BT; Kim, EH; Kim, GA; Kim, GD; Kim, HB; Kim, HG; Kim, JS; Kim, MJ; Kim, SI; Kim, SJ; Kim, Y; King, K; Kinyamu-Akunda, J; Kirkkala, T; Kjaer-Sorensen, K; Kleppinger, EL; Kloner, RA; Klopfenstein, TJ; Knappe, D; Knezevic, P; Kobos, LM; Kohli, M; Kolano, L; Kolodgie, FD; Kolte, AP; Koneru, B; Kong, D; Kong, F; Kong, X; Konggidinata, MI; Köpke, M; Koski, KG; Kotsis, F; Köttgen, A; Kouakou-Kouamé, CA; Kraemer, US; Krane, V; Krehbiel, CR; Krenning, BJ; Kretzschmar, D; Ku, KB; Kubota, Y; Kulich, P; Kumar, NG; Kupiec-Weglinski, JW; Lalani, SS; Lan, X; Landfeldt, E; Langenberg, E; Lapauw, B; Larkin, J; Lassoued, MA; Laukhtina, E; Laura Martinez, J; Laveillé, A; Lavela, P; Law, AD; Lazraq, A; Le Foll, B; Lee, BK; Lee, C; Lee, CS; Lee, EJ; Lee, EY; Lee, G; Lee, HY; Lee, JH; Lee, JJ; Lee, JO; Lee, JS; Lee, R; Lei, H; Lei, P; Lellouche, F; Lennerz, JK; Leong, W; Leslie, I; Lessem, E; Levin, M; Levinger, I; Li, C; Li, CW; Li, CX; Li, CY; Li, D; Li, H; Li, HM; Li, J; Li, L; Li, LM; Li, N; Li, S; Li, W; Li, X; Li, XX; Li, Y; Li, Z; Li, ZL; Li, ZX; Lian, Q; Liang, C; Liang, GH; Liang, H; Liang, J; Liang, X; Liao, CX; Liao, R; Ličbinský, R; Lim, YS; Lima, HK; Lin, JG; Lin, L; Lin, S; Lin, WP; Lin, Z; Liso, M; Liu, BX; Liu, C; Liu, H; Liu, J; Liu, M; Liu, Q; Liu, S; Liu, SF; Liu, SL; Liu, T; Liu, W; Liu, X; Liu, XB; Liu, Y; Liu, YY; Liu, Z; Liu, ZQ; Lobo, M; Loitzenbauer, M; López, F; Lopez, G; López, GJ; Lou, Z; Lu, IC; Lu, J; Lu, M; Lu, W; Lu, X; Lu, Y; Luhovyy, BL; Luna-Abanto, J; Luo, J; Luo, K; Luo, L; Luo, M; Luo, W; Luo, X; Luo, XM; Lv, Y; Lv, YQ; Lyu, HD; Lyu, J; Ma, C; Ma, G; Ma, L; Ma, Q; Ma, X; Ma, Y; Macha, SJ; MacLean, E; Mahalapbutr, P; Maina, T; Malfait, F; Malfertheiner, MV; Malzert-Fréon, A; Mansouri, E; Mao, C; Marcellin, E; Marchiori, PER; Marcotte, DJ; Maréchal, A; Maric, N; Maris, JM; Maron, L; Marti, CN; Martínez-Milla, J; Mateo, J; Mather, K; Mathison, CJN; Matthay, MA; Maxwell, CL; Mazier, D; Mazumder, D; Mazurkiewicz, M; Mazzucchelli, TG; McAuley, DF; Mccoy, K; McVicar, DW; Mebel, AM; Mech, A; Meester, EJ; Meiselbach, H; Melero, I; Ménard, G; Meng, X; Mengya, Y; Merle, G; Meunier, B; Mfarrej, B; Mi, K; Migueliz, I; Mikuška, P; Miladi, K; Miletich, R; Millar, JE; Mills, MR; Milne, R; Minute, L; Misiak, M; Mo, F; Modi, A; Mok, F; Molina, C; Mollen, CJ; Molteni, V; Montalto, M; Montet, D; Monti, MC; Moor, MB; Moravec, P; Morsiani, C; Murillo, E; Murugan, P; Muslem, R; Myers, RK; N'guessan, FK; Nabil, H; Nadal, J; Nadeem, M; Nafady, MM; Nafie, MS; Nair, HP; Nakano, R; Nance, J; Naren, N; Neil, CJ; Nelson, J; Nery, FC; Netsch, C; Nguyen, TH; Ni, L; Ni, YX; Nie, W; Nielsen, LK; Nigam, K; Nikolayev, AA; Nishiyama, M; Niu, LL; Niu, PP; Nock, BA; Noer, PR; Noll, G; Noll, S; Norenberg, JP; Nowicka, J; Nutho, B; O'Connor, M; Obonyo, NG; Ochiai, T; Ochoa, MC; Oh, BL; Oh, S; Olczak, J; Olivares, X; Ommurugan, B; Oosthuizen, MC; Operario, D; Orešič, M; Oshima, K; Otano, I; Ou, Y; Owen, TW; Oxvig, C; Pacey, V; Pai, M; Paik, H; Paiva, R; Palmieri, EM; Palpant, N; Pan, L; Pan, Q; Panahi, S; Pang, B; Pang, ZC; Pannecouque, C; Paris, L; Park, D; Park, DJ; Park, E; Park, EC; Park, IH; Park, JH; Park, JI; Park, S; Passmore, MR; Pattaranggoon, NC; Paun, M; Pedersen, S; Pedron, J; Peng, M; Peng, X; Penzhorn, BL; Pérez-Camargo, D; Perez-Maldonado, R; Pérez-Vicente, C; Pham, TD; Pickering, L; Pickersgill, NA; Pinault, E; Pinotsis, N; Plan, M; Pocino, K; Poh, CL; Pons, EDC; Popoff, MR; Porri, D; Pourmand, A; Pratviel, G; Prudente, DO; Qi, H; Qi, N; Qian, LY; Qiao, L; Qiao, Q; Qin, QP; Qiu, N; Qiu, SW; Qu, F; Quan, M; Quigg, A; Raee, E; Raibaud, P; Ramanitrahasimbola, D; Rapoport, L; Rasby, RJ; Rasoanirina, BNV; Raspini, B; Ratner, JR; Razafindrakoto, Z; Redd, MA; Ren, H; Ren, N; Rey, J; Reynolds, CP; Rich, PR; Richards, CJ; Rigol, M; Rimoldi, S; Robert, P; Rodrigues, AE; Roe, JH; Rohde, S; Rokita, JL; Roland, J; Rombaut, L; Ronkainen, J; Rothenberg, SM; Roy, SC; Ruan, Z; Rucker, PV; Rueda, D; Ruhwald, M; Rungrotmongkol, T; Rupert, AS; Rusjan, P; Ryabov, AD; Rysä, J; Saad, NES; Sabioni, P; Sadow, PM; Sahai, N; Salem, HF; Salinas, B; Salonurmi, T; Samé Guerra, D; Sánchez, J; Sanchez-González, J; Sanmamed, MF; Sansores-Peraza, P; Santoro, JC; Santschi, PH; Saritas, T; Sarkisova, Y; Savolainen, MJ; Scherberich, JE; Schlom, DG; Schmelz, EM; Schmid, MC; Schneider, MP; Schumacher, S; Schwartz, JC; Schwartzer, JJ; Schwehr, K; Schweitzer, DH; Scott, ME; Sedky, NK; See Hoe, L; Sejian, V; Selvaraju, S; Sen, SK; Seo, G; Šerý, O; Settles, JA; Sfar, S; Shaffer, J; Shan, GL; Shang, Q; Shannahan, JH; Shao, B; Shao, H; Shao, J; Shao, ZH; Shasha, Y; Shaw, K; Sheeba, V; Shekar, K; Shen, G; Shen, H; Shen, XD; Shen, Y; Sherrell, PC; Shete, PB; Shi, AX; Shi, J; Shi, JH; Shi, S; Shi, X; Shigeta, Y; Shimbo, A; Shin, E; Sikka, N; Silhavy, TJ; Simanon, N; Simard, S; Simon, J; Simon, M; Simpson, SD; Simundic, AM; Since, M; Singh, B; Singhroy, DN; Sinisterra, OT; Smith, EH; Sobreira, TJP; Solanes, N; Somasundar, Y; Sommerer, C; Sonei, A; Song, B; Song, E; Song, J; Song, M; Song, Y; Soo Lee, M; Sorensen, MD; Sournia-Saquet, A; Spaepen, E; Spirk, D; Srivastava, S; Stancill, JS; Stanczak, PS; Starenki, D; Starr, F; Step, DL; Steubl, D; Stigliani, JL; Stráská, J; Sträter, N; Su, ZZ; Sudano, I; Suen, JY; Suh, HJ; Sui, ZY; Suico, JG; Suleiman, K; Sumon, K; Sun, HB; Sun, J; Sun, L; Sun, LL; Sun, M; Sun, Q; Sun, W; Sun, X; Sun, XF; Sun, Y; Sun, YB; Sun, YH; Sun, YN; Sun, Z; Sunada, K; Suzuki, S; Sylvan, JB; Takala, J; Talla, D; Tamir, Z; Tan, SJ; Tanda, S; Tang, H; Tang, J; Tang, LF; Tang, SJ; Tang, Y; Tao, FB; Tappel, R; Taratkin, M; Teijeira, Á; Tellew, JE; Thomas, AM; Thomas, SG; Thomson, SR; Tian, J; Tie, Y; Tirado, JL; Tolonen, A; Tosato, G; Tronnet, A; Tsai, S; Turtoi, A; Turtoi, E; Tvrdoňová, M; Tyagi, A; Tzou, DT; Uddin Ahmad, Z; Urias, E; Usawachintachit, M; Ustriyana, P; Utsumi, F; Vacca, M; Vaculovič, T; Vaidya, SS; Valentin, A; Valgepea, K; van den Berg, P; van den Bergh, JP; van der Heiden, K; van Gaalen, K; Van Gemert, W; van Haard, PMM; van Hest, JCM; Vecchiarelli, E; Večeřa, Z; Venkatesh, R; Verhaeghe, P; Verhagen, HJ; Vetter, JM; Vieira, D; Vilchez-Tschischke, JP; Villena-Gutierrez, R; Villoslada Terrones, V; Vital-Jacome, M; Voelkl, J; Vogel, K; Vogrin, S; Volke, D; von Bahr, V; Vysloužil, J; Wade, TL; Wagner-Gillespie, M; Walsh, SW; Wan, LJ; Wan, SP; Wang, AL; Wang, B; Wang, BY; Wang, C; Wang, D; Wang, F; Wang, H; Wang, HR; Wang, HY; Wang, J; Wang, JY; Wang, K; Wang, L; Wang, LF; Wang, P; Wang, Q; Wang, R; Wang, SF; Wang, SP; Wang, SR; Wang, T; Wang, W; Wang, WP; Wang, X; Wang, XJ; Wang, Y; Wang, YL; Wang, YN; Wáng, YXJ; Wang, Z; Wang, ZF; Wang, ZY; Waning, B; Warner, JM; Washington, SL; Watson, AK; Wei, B; Wei, C; Wei, F; Wei, X; Wei, Y; Wemhoff, AP; Wen, Z; Weng, TT; Wesdemiotis, C; Wheeler, DA; Wildner, M; Wilson, BK; Wirth, LJ; Wissler, M; Wu, F; Wu, G; Wu, J; Wu, KH; Wu, MC; Wu, P; Wu, PK; Wu, S; Wu, W; Wu, X; Wu, XP; Wu, Y; Wyatt, E; Wyllie, S; Xia, Y; Xiao, BH; Xiao, SZ; Xiao, W; Xiao, X; Xiao, Z; Xie, D; Xie, K; Xie, X; Xie, Y; Xie, YF; Xin, S; Xin, Z; Xing, Q; Xing, WQ; Xiong, D; Xiong, X; Xu, C; Xu, D; Xu, F; Xu, G; Xu, H; Xu, J; Xu, JY; Xu, L; Xu, N; Xu, W; Xu, X; Xu, Y; Xu, YM; Xue, H; Xue, J; Xue, Z; Yan, R; Yan, SQ; Yan, W; Yan, X; Yan, Z; Yang, C; Yang, D; Yang, F; Yang, FC; Yang, G; Yang, J; Yang, M; Yang, P; Yang, Q; Yang, R; Yang, S; Yang, SJ; Yang, TWW; Yang, X; Yang, Y; Yang, Z; Yao, C; Yao, L; Yao, LP; Yao, M; Yao, T; Yao, W; Yao, Y; Yaseen, T; Yazdani, V; Ye, J; Ye, S; Yerys, BE; Yi, HWL; Yi, JL; Yin, F; Yin, J; Yin, Y; Yin, Z; Yong, ZP; Yongli, S; Yoo, JS; Yoshikawa, N; You, Q; Yu, B; Yu, CQ; Yu, H; Yu, HG; Yu, J; Yu, L; Yu, Q; Yu, X; Yu, Y; Yu, YK; Yu, Z; Yuan, Q; Yuan, R; Yuan, W; Yuan, X; Yuan, Y; Zager, RA; Zagozdzon, A; Zaller, N; Zang, YP; Zappi, ME; Zelikoff, JT; Zeman, T; Zhai, X; Zhan, P; Zhang, B; Zhang, C; Zhang, G; Zhang, H; Zhang, HB; Zhang, J; Zhang, JS; Zhang, L; Zhang, M; Zhang, Q; Zhang, RX; Zhang, S; Zhang, T; Zhang, W; Zhang, WH; Zhang, X; Zhang, XX; Zhang, Y; Zhang, YQ; Zhang, YW; Zhang, Z; Zhang, ZH; Zhao, D; Zhao, FL; Zhao, K; Zhao, L; Zhao, M; Zhao, R; Zhao, S; Zhao, W; Zhao, WG; Zhao, X; Zhao, Y; Zheng, G; Zheng, J; Zheng, S; Zheng, W; Zheng, Y; Zheng, YG; Zhong, Z; Zhou, C; Zhou, D; Zhou, H; Zhou, HY; Zhou, L; Zhou, Q; Zhou, X; Zhou, Y; Zhou, YL; Zhou, Z; Zhu, J; Zhu, L; Zhu, N; Zhu, X; Zhu, XF; Zhu, Y; Zhu, Z | 1 |
Blum, S; Brouland, JP; Chalandon, Y; Comoli, P; Comte, D; Du Pasquier, R; Dunet, V; Livio, F; Opota, O; Spertini, O; Tirefort, Y | 1 |
Chen, P; Liu, G; Liu, T; Ouyang, R; Shen, C; Zhou, L | 1 |
Triche, TJ | 1 |
Hoemberger, M; Kern, D; Pitsawong, W | 1 |
Byran, G; Lakshmanan, K | 1 |
Gota, V; Joshi, H; Patil, V; Ramaa, CS; Tilekar, K; Upadhyay, N | 1 |
Barkoh, BA; Bueso-Ramos, CE; Chen, W; Fang, H; Futreal, A; Gupta, SK; Jain, N; Khoury, JD; Loghavi, S; Luthra, R; Mao, X; Medeiros, LJ; Patel, KP; Routbort, M; Tang, G; Wang, SA; Yang, RK; Zhang, J | 1 |
Dholam, K; Gupta, L; Gurav, SV; Janghel, Y | 1 |
Bria, E; Cintoni, M; Gasbarrini, A; Mele, MC; Pompili, M; Ponziani, FR; Pozzo, C; Raoul, P; Rinninella, E; Strippoli, A; Tortora, G | 1 |
Allison, J; Bailey, A; Bass, A; Bean, S; Falchook, G; Fu, S; Hong, DS; Janku, F; Karp, D; Lim, J; Meric-Bernstam, F; Montez, S; Naing, A; Piha-Paul, S; Reilley, MJ; Sharma, P; Subbiah, V; Tsimberidou, A; Vence, L | 1 |
Burger, DM; Desar, IME; Kweekel, DM; Lankheet, NAG; Mulder, SF; van der Graaf, WTA; van Erp, NP; van Herpen, CML | 1 |
Naseer, MM; Rahman, MSU; Saeed, A; Shoaib, M | 1 |
Nair, P | 1 |
Cardoso, E; Csajka, C; Schneider, MP; Widmer, N | 1 |
Ahmed, G; Kim, SB; Shay, JW; Terman, JR; Yoon, J | 1 |
Allard, M; Bellesoeur, A; Blanchet, B; Cardoso, E; Rousseau, B | 1 |
Baker, SD; Jeon, JY; Sparreboom, A | 1 |
Boehm, JS; Hong, AL; Painter, CA; Sharifnia, T | 1 |
Burney, IA; Lakhtakia, R | 1 |
Asmis, T; Gilbert, S; Pysyk, CL | 1 |
Chang, JH; Choi, HG; Gautam, M; Jeong, JH; Jiang, L; Kim, JO; Ku, SK; Ou, W; Soe, ZC; Thapa, RK; Yong, CS | 1 |
Abouzid, KA; Fawzy, IM; Ismail, NS; Lasheen, DS; Youssef, KM | 1 |
Dusetzina, SB; Keating, NL; Rotenstein, LS | 1 |
Asami, Y; Crump, A; Ōmura, S | 1 |
Garcia-Gonzalez, P; Novakowski, AK; Stergachis, A; Wrigglesworth, M | 1 |
Bencze, J; Gergely, PA; Gombos, K; Hortobágyi, T; Kurucz, A; Murnyák, B; Varjas, T | 1 |
Tempero, M | 1 |
Abruzzese, E; Bernardi, S; Binotto, G; Bonifacio, M; Iurlo, A; Russo, D; Tiribelli, M; Zanaglio, C | 1 |
Cho, YS; Gwak, HS; Han, JM; Yee, J | 1 |
Kannan, N; Oruganty, K | 1 |
Buclin, T; Csajka, C; Gotta, V; Widmer, N | 1 |
Chatterjee, P | 1 |
Cook, SJ; Sale, MJ | 1 |
Despas, F; Laurent, G; Roche, H | 1 |
Coombs, J; Kruse, M; Parthan, A; Sasane, M; Taylor, D | 1 |
Lin, YL; Roux, B | 1 |
Adenis, A; Amela, EY; Blay, JY; Bui-Nguyen, B; Cassier, PA; Chauzit, E; Clisant, S; Fournier, C; Italiano, A; Molimard, M; Penel, N; Ray-Coquard, I; Tresch-Bruneel, E | 1 |
Beijnen, JH; Huitema, AD; Knapen, LM; Lankheet, NA; Schellens, JH; Steeghs, N | 1 |
Druker, BJ | 4 |
Waller, CF | 2 |
Brazzelli, V; Croci, G; Grasso, V; Vassallo, C | 1 |
Gravitz, L | 2 |
Bourzac, K | 1 |
Aittokallio, K; Alpay, K; Farshchian, M; Hietanen, S; Kähäri, VM; Kallio, M; Sandholm, J; Siljamäki, E; Tuomela, J | 1 |
Belmont, P; Mariaule, G | 1 |
Agafonov, RV; Buosi, V; Kern, D; Otten, R; Wilson, C | 1 |
Bonkobara, M | 1 |
Wissing, MD | 1 |
Huang, Z; Liu, P; Qian, J; Shu, Y; Wu, Y; Zhou, X; Zhu, W | 1 |
Abdi, M; Amini, S; Azadi, NA; Ghaderi, B; Salimizand, H | 1 |
Nishio, K; Togashi, Y | 1 |
Tanigawara, Y | 1 |
Brullo, C; Grossi, G; Musumeci, F; Sanna, M; Schenone, S | 1 |
Baruzzi, A; Berton, G; Chignola, R; Lorenzetto, E; Remelli, S; Sega, M | 1 |
Block, J; Meng, F; Wu, G | 1 |
Bower, M; Erbacher, I; Fortunak, J; Gotham, D; Hill, A; Levi, J; Martin, M; Meldrum, J; Powderly, WG; Shoman, H | 1 |
Amgoth, C; Dharmapuri, G; Kalle, AM; Paik, P | 1 |
Eckstein, N; Frötschl, R; Haas, B; Weber-Lassalle, K | 1 |
Bhattacharya, M; Chakraborty, C; Lee, SS; Patra, BC; Sharma, AR; Sharma, G | 1 |
Bedwell, C; Greystoke, B; McGregor, AK; Oakes, R; Wood, K | 1 |
Doroshow, JH; Parchment, RE | 1 |
Bonsignore, R; Gentile, C; Lauria, A; Martorana, A | 1 |
Tuma, RS | 1 |
Gasparini, G; Longo, R | 1 |
Becker, H; Berg, T; Binder, M; Dierks, C; Duque-Afonso, J; Hackanson, B; Lairmore, MD; Lübbert, M; Martens, U; Mertelsmann, R; Schäfer, HS; Schnitzler, M; Zeiser, R | 1 |
Dingermann, T; Laufer, S; Winckler, T | 1 |
Franke, RM; Sparreboom, A | 1 |
Sakai, H; Takeuchi, S | 1 |
Cogan, E; Roufosse, F | 1 |
Iwata, C; Kano, MR; Kataoka, K; Komuta, Y; Miyazono, K; Morishita, Y; Oka, M; Ouchi, Y; Shirai, YT | 1 |
Bird, R; Henden, A; Keane, C | 1 |
Adamson, PC | 1 |
Al Rashid, S; Bristow, RG; Choudhury, A; Jalali, F; Kiltie, AE; Ran, J; Supiot, S; Zhao, H | 1 |
Eck, MJ; Manley, PW | 1 |
Boderet, F; Bosq, J; Capdeville, R; Chatelut, E; Doz, F; Emile, JF; Frappaz, D; Geoerger, B; Geoffray, A; Hain, S; Kalifa, G; Le Deley, MC; Morland, B; Ndiaye, A; Opolon, P; Pichon, F; Vassal, G | 1 |
Bailey, S; Branson, M; Laird, G; Neuenschwander, B | 1 |
Ergolin, MJ | 1 |
Kapoor, S | 1 |
Belknap, SM; Bennett, CL; Boyle, S; Burdon, R; Djulbegovic, B; Dorr, DA; Edwards, BJ; Georgopoulos, C; Lagman, J; McKoy, JM; Sartor, O; Tallman, MS; Talpaz, M; Weitzman, SA; West, DP | 1 |
Decosterd, LA; Duchosal, MA; Haouala, A; Leyvraz, S; Montemurro, M; Ris, HB; Rochat, B; Widmer, N; Zaman, K; Zanolari, B | 1 |
Rochat, B | 2 |
Schiff, D; van den Bent, MJ; Wen, PY | 1 |
D'Incalci, M; Damia, G | 1 |
Lydon, N | 1 |
Sawyers, CL | 1 |
Chaput, N; Ménard, C; Tursz, T; Zitvogel, L; Zoubir, M | 1 |
Ashby, CR; Chen, A; Chen, X; Chen, ZS; Hopper-Borge, E; Kuang, YH; Lei, Y; Ouyang, J; Shen, T; Tiwari, AK; Zhou, Y | 1 |
Gauthier, H | 1 |
Marmorstein, R | 1 |
Wang, ZY | 1 |
De Greve, J; Decoster, L; Fontaine, C; Schallier, D; Trullemans, F | 1 |
Adrian, F; Berst, F; Cowan-Jacob, SW; Fabbro, D; Fendrich, G; Furet, P; Gray, NS; Grotzfeld, R; Jahnke, W; Liebetanz, J; Manley, PW; Marzinzik, A; Mestan, J; Pelle, X; Strauss, A; Szyttenholm, A; Warmuth, M; Zhang, J | 1 |
Aleksandrov, A; Simonson, T | 1 |
Dorsch, M; Sellers, WR; Stegmeier, F; Warmuth, M | 1 |
Golub, T | 1 |
Venkatraman, P | 1 |
Druker, B | 1 |
Brüggen, J; Conus, N; Cullinane, C; Hui, Y; Jackson, S; Manley, PW; McArthur, GA; Natoli, A | 1 |
Klein, S; Levitzki, A | 2 |
Blobe, GC; Dugan, E; Favaro, J; Fernando, NH; Hurwitz, HI; Meadows, KL; Morse, MA; Nixon, AB; Petros, WP; Truax, R | 1 |
Saijo, N | 1 |
Kong, D; Yamori, T | 1 |
Bernheim, A | 1 |
Agostino, NM; Chinchilli, VM; Drabick, JJ; Gingrich, R; Koszyk-Szewczyk, A; Lynch, CJ; Sivik, J | 1 |
Baker, LH; Chenevert, T; Chugh, R; Karantza, V; Mehnert, J; Moss, RA; Poplin, EA; Saraiya, B; Savkina, N; Stein, MN | 1 |
Harrop, R; Shingler, W | 1 |
Biollaz, J; Buclin, T; Decosterd, LA; Widmer, N | 1 |
Chaput, N; Flament, C; LeCesne, A; Marty, V; Pautier, P; Ribrag, V; Robert, C; Soria, JC; Viaud, S; Vielh, P; Zitvogel, L; Zoubir, M | 1 |
Chu, DT | 1 |
Angiolini, M | 1 |
Burris, H; Doss, H; Greco, FA; Hainsworth, J; Infante, J; Jones, S; Spigel, D; Thompson, D | 1 |
Bernstein, ML | 1 |
Chan, WL; Chang, JG; Chang, WH; Lee, CC; Lin, YH; Wu, YC | 1 |
Geoerger, B; Leblond, P | 1 |
Bandyopadhyay, S; Chile, S; Joshi, K; Monahar, S; Pal, BC; Sharma, S; Wagh, V | 1 |
Caponigro, F; Ciarmiello, A; Milano, A; Perri, F | 1 |
Schmidt, C | 1 |
Crane, K | 1 |
Bugnon, O; Jeanneret, LA; Lüthi, F; Schneider, MP; Troxler, S | 1 |
Croce, CM | 1 |
Demoulin, JB; Medves, S | 1 |
Beckeringh, JJ; Boven, E; Hugtenburg, JG; Timmers, L; van Herk-Sukel, MP | 1 |
Daw, HA; Peerzada, MM; Spiro, TP | 1 |
Adenis, A; Bay, JO; Bertucci, F; Blay, JY; Bouché, O; Cassier, P; Chevreau, C; Clisant, S; Collard, O; Fournier, C; Italiano, A; Kalbacher, E; Kramar, A; Penel, N | 1 |
Benesch, M; Burdach, S; Frühwald, M; Graf, N; Greulich, N; Grunewald, TG; Kontny, U; Kordes, U; Metzler, M; Mittler, U; Rutkowski, S; Scheurlen, W; Schmidt, W; Stachel, D | 1 |
Aitelhaj, M; Boutayeb, A; Boutayeb, S; Boutayeb, W; Errihani, H; Mesmoudi, M; Mrabti, H; Zakkouri, FZ | 1 |
Airley, R | 1 |
Balakrishnar, B; Clements, A; Gao, B; Gurney, H; Wong, M; Yeap, S | 1 |
Ho, WL; Wong, H; Yau, T | 1 |
Beumer, JH; Cotarla, I; Deeken, J; Egorin, MJ; Elston, B; Firozvi, K; Hartley, ML; He, AR; Hwang, J; Koh, EY; Liu, M; Malik, S; Marshall, JL; Pishvaian, MJ; Slack, R; Strychor, S | 1 |
Levitzki, A | 2 |
Blanc, J; Geney, R; Menet, C | 1 |
Branford, S | 1 |
Al-Saeedi, FJ; Luqmani, YA; Mathew, PM | 1 |
Hickman, JA; Lazo, JS | 1 |
Fabbro, D; Matter, A; Parkinson, D | 1 |
Blay, JY; Ray-Coquard, I | 1 |
Sugimura, T | 1 |
Couzin, J | 1 |
Scoazec, JY | 1 |
Garber, K | 3 |
Workman, P | 1 |
Britten, CD; Ma, BB; Siu, LL | 1 |
Buchdunger, E; Cowan-Jacob, SW; Fabbro, D; Fendrich, G; Furet, P; Manley, PW; Meyer, T; Zimmermann, J | 1 |
Akiyama, S | 4 |
Westwell, AD | 2 |
Schwartz, RS | 1 |
Hingorani, SR; Tuveson, DA | 1 |
Blasberg, RG; Tjuvajev, JG | 1 |
George, D | 1 |
Fischer, OM; Hart, S; Streit, S; Ullrich, A | 1 |
Kim, JA | 1 |
Abou-Jawde, R; Alemany, C; Choueiri, T; Mekhail, T | 1 |
Fleischer-Black, M; Strom, S | 1 |
Goldman, B | 1 |
Inui, A | 1 |
Shiotsu, Y | 1 |
Duhé, RJ; Mamoon, NM; Smith, JK | 1 |
Arteaga, CL; Roberts, RB; Threadgill, DW | 1 |
Haydon, RC; He, TC; Zhou, L | 1 |
Druker, BJ; Lydon, NB | 1 |
Kim, R; Toge, T | 1 |
Agarwal, NK; Arora, B; Gupta, SK; Kumar, L; Mathur, R; Velpandian, T | 1 |
Jones, RJ; Matsui, WH; Smith, BD | 1 |
Rowinsky, EK | 1 |
Fletcher, JA | 1 |
Pietras, K | 1 |
Nadal, E; Olavarria, E | 1 |
Ostman, A | 1 |
Abad, M; Astudillo, A; Balbín, M; Blay, P; Braña, A; Buesa, JM; Campo, E; Freije, JM; García-García, J; Lacave, A; Losa, R; Marco, V; Miquel, R; Sierra, M | 1 |
Ganesan, TS; Madhusudan, S | 1 |
Debiec-Rychter, M; Nasierowska-Guttmejer, A; Nowecki, Z; Ruka, W; Rutkowski, P | 1 |
Dillman, R; Oldham, R | 1 |
Mohindru, M; Verma, A | 1 |
Bhalla, K; Cheng, F; Cuenca, A; Horna, P; Sotomayor, EM; Wang, H; Zheng, Z | 1 |
Gastl, G; Hiddemann, W | 1 |
Bundi, M; Dimitrijevic, S; Dirnhofer, S; Kononen, J; Lugli, A; Mangialaio, S; Mirlacher, M; Sauter, G; Schraml, P; Simon, R; Went, PT | 1 |
Gahmberg, CG; Kervinen, J | 1 |
Cross, NC; Jones, AV | 1 |
Hirotab, S; Kitamura, Y | 1 |
Basile, M; Caponigro, F; de Rosa, V; Normanno, N | 1 |
Favaudon, V; Hennequin, C | 1 |
Attard, G; De Bono, J; Kaye, S; Vidal, L | 1 |
Barwisch, S; Duyster, J; Peschel, C; Speicher, MR; von Bubnoff, N | 1 |
Blay, JY | 2 |
Aulitzky, WE; Oetzel, C; Schwab, M; van der Kuip, H; Wohlbold, L | 1 |
Blum, HE; Geissler, M; Grimm, CF | 2 |
Bernards, R | 1 |
Brok, M; Burger, H; de Boeck, G; de Bruijn, EA; Guetens, G; Nooter, K; Sparreboom, A; van Tol, H; Verweij, J; Wiemer, EA | 1 |
Lin, C; Liu, ZR; Yang, L | 1 |
Armand, JP; Boige, V; Escudier, B; Le Cesne, A; Le Chevalier, T; Lhomme, C; Malka, D; Pautier, P; Robert, C; Soria, JC; Spatz, A; Wechsler, J | 1 |
Krause, DS; Van Etten, RA | 1 |
Heinemann, V; Hiddemann, W | 1 |
Blaise, D; Gaugler, B; Mohty, M; Olive, D | 1 |
Brownlow, N; Dibb, NJ; Domin, J; Taylor, JR | 1 |
Boros, LG; Serkova, N | 1 |
Frantz, S | 1 |
Roskoski, R | 1 |
Geoerger, B; Grill, J; Hartmann, O; Jubert, C; Vassal, G | 1 |
Christoffersen, T; Dajani, O; Guren, TK; Thoresen, GH; Tveit, KM; Wisløff, F | 1 |
Iwasa, Y | 1 |
Czerwenka, K; Handl, C; Hudelist, G; Kubista, E; Lamm, W; Mueller, R; Singer, CF | 1 |
Miki, Y; Nagasaki, K; Shimoji, T | 1 |
Sun, Y; Wang, Y | 1 |
Appleman, LJ; Demetri, GD; Desai, J; George, S; Manola, J; Paul Eder, J; Ryan, DP | 1 |
De Boeck, G; de Bruijn, EA; de Wever, I; Guetens, G; Highley, M; Prenen, H; van Oosterom, AT | 1 |
Jachimczak, P | 1 |
Dirnhofer, S; Went, P; Zimpfer, A | 1 |
Smyth, MJ | 1 |
Baselga, J | 1 |
Filov, VA; Gershanovich, ML; Imianitov, EN; Stukov, AN | 1 |
Jootar, S; Lassarat, S | 1 |
Ichinose, Y; Maehara, Y; Oda, S; Okamoto, T; Yamanaka, T | 1 |
Mann, DL | 1 |
Schultze, JL | 1 |
Fidler, IJ | 1 |
Fujii, S; Fujimoto, K; Hidaka, M; Kadowaki, N; Kawano, F; Konishi, N; Makita, N; Shimizu, K; Taniguchi, M; Uchiyama, T | 1 |
Curtiss, FR | 1 |
Abbott, LH; Michor, F | 1 |
Arslan, MA; Basaga, H; Kutuk, O | 1 |
Knuth, A; Pestalozzi, BC; Stenner-Liewen, F; Zippelius, A | 1 |
Ahmed, S; Andreoni, F; Boschelli, F; Cleris, L; Coluccia, AM; Donella-Deana, A; Formelli, F; Gambacorti-Passerini, C; Magistroni, V; Marchesi, E; Piazza, R; Puttini, M; Redaelli, S; Scapozza, L | 1 |
Necas, E; Sefc, L; Shchemelinin, I | 1 |
Kamb, A; Lengauer, C; Wee, S | 1 |
Chami, L; Lassau, N; Péronneau, P | 1 |
Kibble, A | 1 |
Corneo, G; Franceschino, A; Gambacorti, C; Gambacorti-Passerini, C; Piazza, R; Pogliani, E; Tornaghi, L | 1 |
Hatfield, A; Owen, S; Pilot, PR | 1 |
Atallah, E; Cortes, J; Kantarjian, H | 2 |
Baccarani, M; Martinelli, G; Rosti, G | 1 |
Adamson, PC; Bernstein, ML; Blaney, SM; Bond, M; Krailo, M; Pappo, A; Schultz, KR | 1 |
Alajez, NM; Bastianutto, C; Busson, P; Li, JH; Liu, FF; Lo, KW; Lunt, SJ; Milosevic, M; Mocanu, JD; Moriyama, EH; Shi, W; van Rooijen, N; Wilson, BC; Yip, KW | 1 |
Heldin, CH; Ostman, A | 1 |
Apperley, JF; Chaidos, A; Kanfer, E | 1 |
Altucci, L; Balducci, L; Irminger-Finger, I | 1 |
Daud, AI; Homsi, J | 1 |
Sparreboom, A | 1 |
Gross, WL; Hellmich, B; Holl-Ulrich, K | 1 |
Boyle, SN; Koleske, AJ | 1 |
Shah, NP | 1 |
Ali, Y; Egorin, MJ; Gharibo, MM; Gounder, MK; Lagattuta, TF; Lin, Y; Poplin, EA; Rubin, EH; Stein, MN | 1 |
Faivre, S; Le Tourneau, C; Raymond, E | 1 |
Biasco, G; Nannini, M; Pantaleo, MA; Saponara, M | 1 |
Bonmort, M; Chaperot, L; Chaput, N; Flament, C; Ménard, C; Mignot, G; Plumas, J; Terme, M; Ullrich, E; Zitvogel, L | 1 |
Grosdidier, A; Marull, M; Michielin, O; Rochat, B; von Grünigen, S; Zoete, V | 1 |
Alberti, L; Arifi, S; Blay, JY; Cassier, P; Decouvelaere, AV; Dufresne, A; El Sayadi, H; Fayette, J; Méeus, P; Ranchère, D; Ray-Coquard, I; Tabone-Eglinger, S | 1 |
Belani, CP; Doroshow, JH; Egorin, MJ; Grem, JL; Hamilton, A; Hayes, MJ; Ivy, SP; LoRusso, PA; Mulkerin, DL; Murgo, AJ; Peng, B; Potter, DM; Ramanathan, RK; Remick, SC; Takimoto, CH | 1 |
Egorin, MJ; Flick, SM; Fu, P; Gibbons, J; Grem, JL; Ivy, SP; Lagattuta, TF; Lenz, HJ; LoRusso, PA; Mani, S; Mulkerin, DL; Murgo, AJ; Parise, RA; Pavlick, A; Ramanathan, RK; Remick, SC; Reynolds, S; Shibata, S; Takimoto, CH; Wang, Y | 1 |
Beijnen, JH; Boss, DS; Olmos, RV; Schellens, JH; Sinaasappel, M | 1 |
Giordano, S; Petrelli, A | 1 |
Engelman, JA; Settleman, J | 1 |
Bentley, B; Shao, R; Yan, W | 1 |
Ohyashiki, JH; Ohyashiki, K; Tauchi, T | 1 |
Fojo, T | 1 |
Apperley, J; Corless, CL; Demetri, GD; Di Scala, L; Dirnhofer, S; Fletcher, JA; Harlow, A; Heinrich, MC; Herrmann, R; Joensuu, H; McArthur, AG; McKinley, A; Nikolova, Z; Seymour, J; Soulieres, D; Supple, SG; Town, A; van Oosterom, A | 1 |
Akutsu, M; Furukawa, Y; Honma, Y; Kano, Y; Mano, H; Sato, Y; Tsunoda, S | 1 |
Lemonick, MD; Park, A | 1 |
Stephenson, J | 1 |
Adams, J; Elliott, PJ | 1 |
Krystal, GW | 1 |
Sachsenmaier, C | 1 |
Goel, S; Mani, S; Perez-Soler, R | 1 |
Buser, C; Sepp-Lorenzino, L; Takaki, T | 1 |
Hochhaus, A | 1 |
Hess, JL | 1 |
Blanke, CD; Corless, CL; Druker, BJ; Heinrich, MC | 1 |
Abbott, A | 1 |
Hegedus, T; Kéri, G; Orfi, L; Sarkadi, B; Seprodi, A; Váradi, A | 1 |
134 review(s) available for imatinib mesylate and Benign Neoplasms
Article | Year |
---|---|
New strategies for targeting kinase networks in cancer.
Topics: Animals; Humans; Imatinib Mesylate; Neoplasm Proteins; Neoplasms; Protein Kinase Inhibitors; Protein Kinases | 2021 |
Therapeutic drug monitoring in oncology: International Association of Therapeutic Drug Monitoring and Clinical Toxicology consensus guidelines for imatinib therapy.
Topics: Consensus; Dose-Response Relationship, Drug; Drug Monitoring; Humans; Imatinib Mesylate; Medical Oncology; Neoplasms; Practice Guidelines as Topic; Protein Kinase Inhibitors; Toxicology; Voluntary Health Agencies | 2021 |
Myeloid Neoplasm with PCM1-PDGFRB Transcript Responded to Low-Dose Imatinib: One Case Report with Literature Review.
Topics: Humans; Imatinib Mesylate; In Situ Hybridization, Fluorescence; Myeloproliferative Disorders; Neoplasms; Oncogene Proteins, Fusion; Receptor, Platelet-Derived Growth Factor beta; Translocation, Genetic | 2022 |
Studying molecular signaling in major angiogenic diseases.
Topics: Angiogenesis Inhibitors; Bevacizumab; Cetuximab; Everolimus; Humans; Imatinib Mesylate; Neoplasms; Neovascularization, Pathologic; Sunitinib; Thalidomide; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors | 2022 |
Topics: A549 Cells; Acetylmuramyl-Alanyl-Isoglutamine; Acinetobacter baumannii; Acute Lung Injury; Adaptor Proteins, Signal Transducing; Adenine; Adenocarcinoma; Adipogenesis; Administration, Cutaneous; Administration, Ophthalmic; Adolescent; Adsorption; Adult; Aeromonas hydrophila; Aerosols; Aged; Aged, 80 and over; Aging; Agriculture; Air Pollutants; Air Pollution; Airway Remodeling; Alanine Transaminase; Albuminuria; Aldehyde Dehydrogenase 1 Family; Algorithms; AlkB Homolog 2, Alpha-Ketoglutarate-Dependent Dioxygenase; Alzheimer Disease; Amino Acid Sequence; Ammonia; Ammonium Compounds; Anaerobiosis; Anesthetics, Dissociative; Anesthetics, Inhalation; Animals; Anti-Bacterial Agents; Anti-HIV Agents; Anti-Infective Agents; Anti-Inflammatory Agents; Antibiotics, Antineoplastic; Antibodies, Antineutrophil Cytoplasmic; Antibodies, Monoclonal, Humanized; Antifungal Agents; Antigens, Bacterial; Antigens, CD; Antigens, Differentiation, Myelomonocytic; Antimetabolites, Antineoplastic; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Antioxidants; Antitubercular Agents; Antiviral Agents; Apolipoproteins E; Apoptosis; Arabidopsis; Arabidopsis Proteins; Arsenic; Arthritis, Rheumatoid; Asthma; Atherosclerosis; ATP-Dependent Proteases; Attitude of Health Personnel; Australia; Austria; Autophagy; Axitinib; Bacteria; Bacterial Outer Membrane Proteins; Bacterial Proteins; Bacterial Toxins; Bacterial Typing Techniques; Bariatric Surgery; Base Composition; Bayes Theorem; Benzoxazoles; Benzylamines; beta Catenin; Betacoronavirus; Betula; Binding Sites; Biological Availability; Biological Oxygen Demand Analysis; Biomarkers; Biomarkers, Tumor; Biopsy; Bioreactors; Biosensing Techniques; Birth Weight; Blindness; Blood Chemical Analysis; Blood Gas Analysis; Blood Glucose; Blood Pressure; Blood Pressure Monitoring, Ambulatory; Blood-Brain Barrier; Blotting, Western; Body Mass Index; Body Weight; Bone and Bones; Bone Density; Bone Resorption; Borates; Brain; Brain Infarction; Brain Injuries, Traumatic; Brain Neoplasms; Breakfast; Breast Milk Expression; Breast Neoplasms; Bronchi; Bronchoalveolar Lavage Fluid; Buffaloes; Cadherins; Calcification, Physiologic; Calcium Compounds; Calcium, Dietary; Cannula; Caprolactam; Carbon; Carbon Dioxide; Carboplatin; Carcinogenesis; Carcinoma, Ductal; Carcinoma, Ehrlich Tumor; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Pancreatic Ductal; Carcinoma, Renal Cell; Cardiovascular Diseases; Carps; Carrageenan; Case-Control Studies; Catalysis; Catalytic Domain; Cattle; CD8-Positive T-Lymphocytes; Cell Adhesion; Cell Cycle Proteins; Cell Death; Cell Differentiation; Cell Line; Cell Line, Tumor; Cell Movement; Cell Nucleus; Cell Phone Use; Cell Proliferation; Cell Survival; Cell Transformation, Neoplastic; Cell Transformation, Viral; Cells, Cultured; Cellulose; Chemical Phenomena; Chemoradiotherapy; Child; Child Development; Child, Preschool; China; Chitosan; Chlorocebus aethiops; Cholecalciferol; Chromatography, Liquid; Circadian Clocks; Circadian Rhythm; Circular Dichroism; Cisplatin; Citric Acid; Clinical Competence; Clinical Laboratory Techniques; Clinical Trials, Phase I as Topic; Clinical Trials, Phase II as Topic; Clostridioides difficile; Clostridium Infections; Coculture Techniques; Cohort Studies; Cold Temperature; Colitis; Collagen Type I; Collagen Type I, alpha 1 Chain; Collagen Type XI; Color; Connective Tissue Diseases; Copper; Coronary Angiography; Coronavirus 3C Proteases; Coronavirus Infections; Cost of Illness; Counselors; COVID-19; COVID-19 Testing; Creatine Kinase; Creatinine; Cross-Over Studies; Cross-Sectional Studies; Cryoelectron Microscopy; Cryosurgery; Crystallography, X-Ray; Cues; Cultural Competency; Cultural Diversity; Curriculum; Cyclic AMP Response Element-Binding Protein; Cyclin-Dependent Kinase Inhibitor p21; Cycloparaffins; Cysteine Endopeptidases; Cytokines; Cytoplasm; Cytoprotection; Databases, Factual; Denitrification; Deoxycytidine; Diabetes Complications; Diabetes Mellitus; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Diagnosis, Differential; Diatoms; Diet; Diet, High-Fat; Dietary Exposure; Diffusion Magnetic Resonance Imaging; Diketopiperazines; Dipeptidyl Peptidase 4; Dipeptidyl-Peptidase IV Inhibitors; Disease Models, Animal; Disease Progression; Disease-Free Survival; DNA; DNA Damage; DNA Glycosylases; DNA Repair; DNA-Binding Proteins; DNA, Bacterial; DNA, Viral; Docetaxel; Dose Fractionation, Radiation; Dose-Response Relationship, Drug; Down-Regulation; Doxorubicin; Drosophila; Drosophila melanogaster; Drug Carriers; Drug Delivery Systems; Drug Liberation; Drug Repositioning; Drug Resistance, Bacterial; Drug Resistance, Multiple, Bacterial; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Drug Synergism; Drug Therapy, Combination; Edema; Edible Grain; Education, Graduate; Education, Medical, Graduate; Education, Pharmacy; Ehlers-Danlos Syndrome; Electron Transport Complex III; Electron Transport Complex IV; Electronic Nicotine Delivery Systems; Emergency Service, Hospital; Empathy; Emulsions; Endothelial Cells; Endurance Training; Energy Intake; Enterovirus A, Human; Environment; Environmental Monitoring; Enzyme Assays; Enzyme Inhibitors; Epithelial Cells; Epithelial-Mesenchymal Transition; Epoxide Hydrolases; Epoxy Compounds; Erythrocyte Count; Erythrocytes; Escherichia coli; Escherichia coli Infections; Escherichia coli Proteins; Esophageal Neoplasms; Esophageal Squamous Cell Carcinoma; Esophagectomy; Estrogens; Etanercept; Ethiopia; Ethnicity; Ethylenes; Exanthema; Exercise; Exercise Test; Exercise Tolerance; Extracellular Matrix; Extracorporeal Membrane Oxygenation; Eye Infections, Fungal; False Negative Reactions; Fatty Acids; Fecal Microbiota Transplantation; Feces; Female; Femur Neck; Fermentation; Ferritins; Fetal Development; Fibroblast Growth Factor-23; Fibroblast Growth Factors; Fibroblasts; Fibroins; Fish Proteins; Flavanones; Flavonoids; Focus Groups; Follow-Up Studies; Food Handling; Food Supply; Food, Formulated; Forced Expiratory Volume; Forests; Fractures, Bone; Fruit and Vegetable Juices; Fusobacteria; G1 Phase Cell Cycle Checkpoints; G2 Phase Cell Cycle Checkpoints; Gamma Rays; Gastrectomy; Gastrointestinal Microbiome; Gastrointestinal Stromal Tumors; Gefitinib; Gels; Gemcitabine; Gene Amplification; Gene Expression; Gene Expression Regulation; Gene Expression Regulation, Bacterial; Gene Expression Regulation, Neoplastic; Gene Expression Regulation, Plant; Gene Knockdown Techniques; Gene-Environment Interaction; Genotype; Germany; Glioma; Glomerular Filtration Rate; Glucagon; Glucocorticoids; Glycemic Control; Glycerol; Glycogen Synthase Kinase 3 beta; Glycolipids; Glycolysis; Goblet Cells; Gram-Negative Bacterial Infections; Granulocyte Colony-Stimulating Factor; Graphite; Greenhouse Effect; Guanidines; Haemophilus influenzae; HCT116 Cells; Health Knowledge, Attitudes, Practice; Health Personnel; Health Services Accessibility; Health Services Needs and Demand; Health Status Disparities; Healthy Volunteers; Heart Failure; Heart Rate; Heart Transplantation; Heart-Assist Devices; HEK293 Cells; Heme; Heme Oxygenase-1; Hemolysis; Hemorrhage; Hepatitis B; Hepatitis B e Antigens; Hepatitis B Surface Antigens; Hepatitis B virus; Hepatitis B, Chronic; Hepatocytes; Hexoses; High-Throughput Nucleotide Sequencing; Hippo Signaling Pathway; Histamine; Histamine Agonists; Histidine; Histone Deacetylase 2; HIV Infections; HIV Reverse Transcriptase; HIV-1; Homebound Persons; Homeodomain Proteins; Homosexuality, Male; Hospice and Palliative Care Nursing; HSP70 Heat-Shock Proteins; Humans; Hyaluronan Receptors; Hydrogen; Hydrogen Peroxide; Hydrogen-Ion Concentration; Hydrolysis; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypoglycemia; Hypoglycemic Agents; Hypoxia; Idiopathic Interstitial Pneumonias; Imaging, Three-Dimensional; Imatinib Mesylate; Immunotherapy; Implementation Science; Incidence; INDEL Mutation; Induced Pluripotent Stem Cells; Industrial Waste; Infant; Infant, Newborn; Inflammation; Inflammation Mediators; Infliximab; Infusions, Intravenous; Inhibitory Concentration 50; Injections; Insecticides; Insulin-Like Growth Factor Binding Protein 5; Insulin-Secreting Cells; Interleukin-1; Interleukin-17; Interleukin-8; Internship and Residency; Intestines; Intracellular Signaling Peptides and Proteins; Ion Transport; Iridaceae; Iridoid Glucosides; Islets of Langerhans Transplantation; Isodon; Isoflurane; Isotopes; Italy; Joint Instability; Ketamine; Kidney; Kidney Failure, Chronic; Kidney Function Tests; Kidney Neoplasms; Kinetics; Klebsiella pneumoniae; Knee Joint; Kruppel-Like Factor 4; Kruppel-Like Transcription Factors; Lactate Dehydrogenase 5; Laparoscopy; Laser Therapy; Lasers, Semiconductor; Lasers, Solid-State; Laurates; Lead; Leukocyte L1 Antigen Complex; Leukocytes, Mononuclear; Light; Lipid Peroxidation; Lipopolysaccharides; Liposomes; Liver; Liver Cirrhosis; Liver Neoplasms; Liver Transplantation; Locomotion; Longitudinal Studies; Lopinavir; Lower Urinary Tract Symptoms; Lubricants; Lung; Lung Diseases, Interstitial; Lung Neoplasms; Lymphocyte Activation; Lymphocytes, Tumor-Infiltrating; Lymphoma, Mantle-Cell; Lysosomes; Macrophages; Male; Manganese Compounds; MAP Kinase Kinase 4; Mass Screening; Maternal Health; Medicine, Chinese Traditional; Melanoma, Experimental; Memantine; Membrane Glycoproteins; Membrane Proteins; Mesenchymal Stem Cell Transplantation; Metal Nanoparticles; Metalloendopeptidases; Metalloporphyrins; Methadone; Methane; Methicillin-Resistant Staphylococcus aureus; Mexico; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Inbred ICR; Mice, Knockout; Mice, Nude; Mice, SCID; Mice, Transgenic; Microarray Analysis; Microbial Sensitivity Tests; Microbiota; Micronutrients; MicroRNAs; Microscopy, Confocal; Microsomes, Liver; Middle Aged; Milk; Milk, Human; Minority Groups; Mitochondria; Mitochondrial Membranes; Mitochondrial Proteins; Models, Animal; Models, Molecular; Molecular Conformation; Molecular Docking Simulation; Molecular Dynamics Simulation; Molecular Epidemiology; Molecular Structure; Molecular Weight; Multilocus Sequence Typing; Multimodal Imaging; Muscle Strength; Muscle, Skeletal; Muscular Diseases; Mutation; Mycobacterium tuberculosis; Myocardial Stunning; Myristates; NAD(P)H Dehydrogenase (Quinone); Nanocomposites; Nanogels; Nanoparticles; Nanotechnology; Naphthalenes; Nasal Cavity; National Health Programs; Necrosis; Needs Assessment; Neoadjuvant Therapy; Neonicotinoids; Neoplasm Invasiveness; Neoplasm Metastasis; Neoplasm Proteins; Neoplasm Recurrence, Local; Neoplasm Staging; Neoplasm Transplantation; Neoplasms; Neoplastic Stem Cells; Netherlands; Neuroblastoma; Neuroprotective Agents; Neutrophils; NF-kappa B; NFATC Transcription Factors; Nicotiana; Nicotine; Nitrates; Nitrification; Nitrites; Nitro Compounds; Nitrogen; Nitrogen Dioxide; North Carolina; Nuclear Magnetic Resonance, Biomolecular; Nuclear Proteins; Nucleic Acid Hybridization; Nucleosomes; Nutrients; Obesity; Obesity, Morbid; Oceans and Seas; Oncogene Protein v-akt; Oncogenes; Oocytes; Open Reading Frames; Osteoclasts; Osteogenesis; Osteoporosis; Osteoporosis, Postmenopausal; Outpatients; Ovarian Neoplasms; Ovariectomy; Overweight; Oxazines; Oxidants; Oxidation-Reduction; Oxidative Stress; Oxides; Oxidoreductases; Oxygen; Oxygen Inhalation Therapy; Oxygenators, Membrane; Ozone; Paclitaxel; Paenibacillus; Pain Measurement; Palliative Care; Pancreatic Neoplasms; Pandemics; Parasympathetic Nervous System; Particulate Matter; Pasteurization; Patient Preference; Patient Satisfaction; Pediatric Obesity; Permeability; Peroxiredoxins; Peroxynitrous Acid; Pharmaceutical Services; Pharmacists; Pharmacy; Phaseolus; Phenotype; Phoeniceae; Phosphates; Phosphatidylinositol 3-Kinases; Phospholipid Transfer Proteins; Phospholipids; Phosphorus; Phosphorylation; Photoperiod; Photosynthesis; Phylogeny; Physical Endurance; Physicians; Pilot Projects; Piperidines; Pituitary Adenylate Cyclase-Activating Polypeptide; Plant Extracts; Plant Leaves; Plant Proteins; Plant Roots; Plaque, Atherosclerotic; Pneumonia; Pneumonia, Viral; Point-of-Care Testing; Polyethylene Glycols; Polymers; Polysorbates; Pore Forming Cytotoxic Proteins; Positron Emission Tomography Computed Tomography; Positron-Emission Tomography; Postprandial Period; Poverty; Pre-Exposure Prophylaxis; Prediabetic State; Predictive Value of Tests; Pregnancy; Pregnancy Trimester, First; Pregnancy, High-Risk; Prenatal Exposure Delayed Effects; Pressure; Prevalence; Primary Graft Dysfunction; Primary Health Care; Professional Role; Professionalism; Prognosis; Progression-Free Survival; Prolactin; Promoter Regions, Genetic; Proof of Concept Study; Proportional Hazards Models; Propylene Glycol; Prospective Studies; Prostate; Protein Binding; Protein Biosynthesis; Protein Isoforms; Protein Kinase Inhibitors; Protein Phosphatase 2; Protein Processing, Post-Translational; Protein Serine-Threonine Kinases; Protein Structure, Tertiary; Protein Transport; Proteoglycans; Proteome; Proto-Oncogene Proteins c-akt; Proto-Oncogene Proteins c-myc; Proto-Oncogene Proteins c-ret; Proto-Oncogene Proteins p21(ras); Proton Pumps; Protons; Protoporphyrins; Pseudomonas aeruginosa; Pseudomonas fluorescens; Pulmonary Artery; Pulmonary Disease, Chronic Obstructive; Pulmonary Gas Exchange; Pulmonary Veins; Pyrazoles; Pyridines; Pyrimidines; Qualitative Research; Quinoxalines; Rabbits; Random Allocation; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Histamine H3; Receptors, Immunologic; Receptors, Transferrin; Recombinant Proteins; Recurrence; Reference Values; Referral and Consultation; Regional Blood Flow; Registries; Regulon; Renal Insufficiency, Chronic; Reperfusion Injury; Repressor Proteins; Reproducibility of Results; Republic of Korea; Research Design; Resistance Training; Respiration, Artificial; Respiratory Distress Syndrome; Respiratory Insufficiency; Resuscitation; Retinal Dehydrogenase; Retreatment; Retrospective Studies; Reverse Transcriptase Inhibitors; Rhinitis, Allergic; Ribosomal Proteins; Ribosomes; Risk Assessment; Risk Factors; Ritonavir; Rivers; RNA Interference; RNA-Seq; RNA, Messenger; RNA, Ribosomal, 16S; RNA, Small Interfering; Rosuvastatin Calcium; Rural Population; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Salivary Ducts; Salivary Gland Neoplasms; San Francisco; SARS-CoV-2; Satiation; Satiety Response; Schools; Schools, Pharmacy; Seasons; Seawater; Selection, Genetic; Sequence Analysis, DNA; Serine-Threonine Kinase 3; Sewage; Sheep; Sheep, Domestic; Shock, Hemorrhagic; Signal Transduction; Silver; Silymarin; Single Photon Emission Computed Tomography Computed Tomography; Sirolimus; Sirtuin 1; Skin; Skin Neoplasms; Skin Physiological Phenomena; Sleep Initiation and Maintenance Disorders; Social Class; Social Participation; Social Support; Soil; Soil Microbiology; Solutions; Somatomedins; Soot; Specimen Handling; Spectrophotometry, Ultraviolet; Spectroscopy, Fourier Transform Infrared; Spectrum Analysis; Spinal Fractures; Spirometry; Staphylococcus aureus; STAT1 Transcription Factor; STAT3 Transcription Factor; Streptomyces coelicolor; Stress, Psychological; Stroke; Stroke Volume; Structure-Activity Relationship; Students, Medical; Students, Pharmacy; Substance Abuse Treatment Centers; Sulfur Dioxide; Surface Properties; Surface-Active Agents; Surveys and Questionnaires; Survival Analysis; Survival Rate; Survivin; Sweden; Swine; Swine, Miniature; Sympathetic Nervous System; T-Lymphocytes, Regulatory; Talaromyces; Tandem Mass Spectrometry; tau Proteins; Telemedicine; Telomerase; Telomere; Telomere Homeostasis; Temperature; Terminally Ill; Th1 Cells; Thiamethoxam; Thiazoles; Thiophenes; Thioredoxin Reductase 1; Thrombosis; Thulium; Thyroid Cancer, Papillary; Thyroid Carcinoma, Anaplastic; Thyroid Neoplasms; Time Factors; Titanium; Tomography, Emission-Computed, Single-Photon; Tomography, X-Ray Computed; TOR Serine-Threonine Kinases; Transcription Factor AP-1; Transcription Factors; Transcription, Genetic; Transcriptional Activation; Transcriptome; Transforming Growth Factor beta1; Transistors, Electronic; Translational Research, Biomedical; Transplantation Tolerance; Transplantation, Homologous; Transportation; Treatment Outcome; Tretinoin; Tuberculosis, Multidrug-Resistant; Tuberculosis, Pulmonary; Tubulin Modulators; Tumor Microenvironment; Tumor Necrosis Factor Inhibitors; Tumor Necrosis Factor-alpha; Twins; Ultrasonic Therapy; Ultrasonography; Ultraviolet Rays; United States; Up-Regulation; Uranium; Urethra; Urinary Bladder; Urodynamics; Uromodulin; Uveitis; Vasoconstrictor Agents; Ventricular Function, Left; Vero Cells; Vesicular Transport Proteins; Viral Nonstructural Proteins; Visual Acuity; Vital Capacity; Vitamin D; Vitamin D Deficiency; Vitamin K 2; Vitamins; Volatilization; Voriconazole; Waiting Lists; Waste Disposal, Fluid; Wastewater; Water Pollutants, Chemical; Whole Genome Sequencing; Wine; Wnt Signaling Pathway; Wound Healing; Wounds and Injuries; WW Domains; X-linked Nuclear Protein; X-Ray Diffraction; Xanthines; Xenograft Model Antitumor Assays; YAP-Signaling Proteins; Yogurt; Young Adult; Zebrafish; Zebrafish Proteins; Ziziphus | 2016 |
Prognostic value of skeletal muscle mass during tyrosine kinase inhibitor (TKI) therapy in cancer patients: a systematic review and meta-analysis.
Topics: Gefitinib; Humans; Imatinib Mesylate; Indazoles; Muscle, Skeletal; Neoplasms; Phenylurea Compounds; Prognosis; Pyrazoles; Pyridines; Pyrimidines; Quinolines; Sorafenib; Sulfonamides; Sunitinib; Survival Analysis | 2021 |
Emerging Opportunities for Target Discovery in Rare Cancers.
Topics: CRISPR-Cas Systems; Drug Discovery; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Precision Medicine; RNA Interference; Small Molecule Libraries | 2017 |
Staurosporine: new lease of life for parent compound of today's novel and highly successful anti-cancer drugs.
Topics: Anti-Bacterial Agents; Antineoplastic Agents; Bacteria; Bacterial Infections; Carbazoles; Drug Discovery; Furans; Humans; Imatinib Mesylate; Neoplasms; Protein Kinase Inhibitors; Staurosporine | 2018 |
Systematic review of population pharmacokinetic analyses of imatinib and relationships with treatment outcomes.
Topics: Animals; Antineoplastic Agents; Benzamides; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Population Surveillance; Pyrimidines; Randomized Controlled Trials as Topic; Treatment Outcome | 2013 |
That which does not kill me makes me stronger; combining ERK1/2 pathway inhibitors and BH3 mimetics to kill tumour cells and prevent acquired resistance.
Topics: Aniline Compounds; Animals; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Apoptosis Regulatory Proteins; Benzamides; Cell Cycle; Cell Line, Tumor; Down-Regulation; Drug Resistance, Neoplasm; Humans; Imatinib Mesylate; Indoles; MAP Kinase Kinase 1; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 3; Molecular Targeted Therapy; Neoplasms; Piperazines; Proto-Oncogene Proteins B-raf; Pyrimidines; Sulfonamides; Vemurafenib | 2013 |
[Anticancer drug adherence].
Topics: Administration, Oral; Age Factors; Antineoplastic Agents; Antineoplastic Agents, Hormonal; Benzamides; Breast Neoplasms; Female; Gastrointestinal Stromal Tumors; Humans; Imatinib Mesylate; Infusions, Intravenous; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lymphoma; Male; Medication Adherence; Neoplasms; Physician's Role; Piperazines; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Pyrimidines; Risk Factors; Socioeconomic Factors | 2013 |
Comparison of different adjuvant therapies for 9 resectable cancer types.
Topics: Antineoplastic Agents; Benzamides; Chemotherapy, Adjuvant; Disease-Free Survival; Humans; Imatinib Mesylate; Neoplasms; Numbers Needed To Treat; Piperazines; Pyrimidines; Randomized Controlled Trials as Topic; Survival Rate; Treatment Outcome | 2013 |
Imatinib mesylate.
Topics: Animals; Antineoplastic Agents; Benzamides; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Pyrimidines; Signal Transduction | 2014 |
Tyrosine kinase inhibitors: muco-cutaneous side effects at the microscope.
Topics: Antineoplastic Agents; Benzamides; Biopsy; Dasatinib; Exanthema; Humans; Imatinib Mesylate; Microscopy, Electron; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines; Thiazoles | 2014 |
Cyclin-dependent kinase inhibitors as marketed anticancer drugs: where are we now? A short survey.
Topics: Antineoplastic Agents; Benzamides; Cell Cycle; Cyclin-Dependent Kinases; Drug Design; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein Kinase Inhibitors; Pyrimidines | 2014 |
Dysregulation of tyrosine kinases and use of imatinib in small animal practice.
Topics: Animals; Antineoplastic Agents; Cat Diseases; Cats; Dog Diseases; Dogs; Imatinib Mesylate; Neoplasms; src-Family Kinases | 2015 |
Chemotherapy- and irradiation-induced bone loss in adults with solid tumors.
Topics: Adult; Antineoplastic Agents; Bone Resorption; Denosumab; Diphosphonates; Drug Therapy; Drug-Related Side Effects and Adverse Reactions; Humans; Imatinib Mesylate; Methotrexate; Neoplasms; Radioisotopes; Radiotherapy; Taxoids | 2015 |
Clinical efficacy of mTOR inhibitors in solid tumors: a systematic review.
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Combined Chemotherapy Protocols; Bevacizumab; Clinical Trials as Topic; Docetaxel; Erlotinib Hydrochloride; Everolimus; Gefitinib; Humans; Imatinib Mesylate; Neoplasms; Protein Kinase Inhibitors; Quinazolines; Signal Transduction; Sirolimus; Taxoids; TOR Serine-Threonine Kinases | 2015 |
[Kinase inhibitors and their resistance].
Topics: Antibodies, Monoclonal, Humanized; Benzamides; Biomarkers, Tumor; Crizotinib; Drug Discovery; Drug Resistance, Neoplasm; ErbB Receptors; Gefitinib; Humans; Imatinib Mesylate; Indoles; Molecular Targeted Therapy; Neoplasms; Niacinamide; Phenylurea Compounds; Piperazines; Protein Kinase Inhibitors; Protein Kinases; Pyrazoles; Pyridines; Pyrimidines; Quinazolines; Signal Transduction; Sorafenib; Sulfonamides; Trastuzumab; Vemurafenib | 2015 |
[Pharmacokinetic issues on cancer pharmacotherapy].
Topics: Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Drug Monitoring; Humans; Imatinib Mesylate; Molecular Targeted Therapy; Neoplasms; Piperazines; Precision Medicine; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Trastuzumab | 2015 |
Analogs, formulations and derivatives of imatinib: a patent review.
Topics: Animals; Antineoplastic Agents; Biological Availability; Chemistry, Pharmaceutical; Drug Design; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Nanoparticles; Neoplasms; Patents as Topic | 2015 |
Is sunitinib a Narrow Therapeutic Index Drug? - A systematic review and in vitro toxicology-analysis of Sunitinib vs. Imatinib in cells from different tissues.
Topics: Animals; Antineoplastic Agents; Apoptosis; Apoptosis Regulatory Proteins; Cell Line, Tumor; Cell Survival; Dose-Response Relationship, Drug; Drug and Narcotic Control; Drugs, Generic; Humans; Imatinib Mesylate; Indoles; Inhibitory Concentration 50; Neoplasms; Organ Specificity; Phosphorylation; Protein Kinase Inhibitors; Pyrroles; Risk Assessment; Signal Transduction; Sunitinib; Toxicity Tests | 2016 |
MicroRNAs mediated regulation of MAPK signaling pathways in chronic myeloid leukemia.
Topics: Animals; Cell Survival; Chromosome Mapping; Fusion Proteins, bcr-abl; Gene Expression Regulation, Leukemic; Humans; Imatinib Mesylate; K562 Cells; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; MAP Kinase Signaling System; Mice; MicroRNAs; Mitogen-Activated Protein Kinases; Neoplasms; Rats; Signal Transduction | 2016 |
Kinase Inhibitors in Multitargeted Cancer Therapy.
Topics: Anilides; Crizotinib; Humans; Imatinib Mesylate; Imidazoles; Indoles; Neoplasms; Niacinamide; Phenylurea Compounds; Piperidines; Protein Kinase Inhibitors; Pyrazoles; Pyridazines; Pyridines; Pyrroles; Quinazolines; Receptor Protein-Tyrosine Kinases; Sorafenib; Sunitinib | 2017 |
Anti-VEGF therapy: the search for clinical biomarkers.
Topics: Angiogenesis Inhibitors; Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Biomarkers, Tumor; Diagnostic Imaging; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Prognosis; Pyrimidines; Trastuzumab; Vascular Endothelial Growth Factor A | 2008 |
Imaging in early phase childhood cancer trials.
Topics: Benzamides; Child; Clinical Trials as Topic; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Positron-Emission Tomography; Protein Kinase Inhibitors; Pyrimidines; Signal Transduction; Tomography, X-Ray Computed | 2009 |
The interplay of structural information and functional studies in kinase drug design: insights from BCR-Abl.
Topics: Antineoplastic Agents; Benzamides; Drug Design; ErbB Receptors; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Models, Molecular; Molecular Structure; Neoplasms; Piperazines; Protein Conformation; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Proto-Oncogene Proteins B-raf; Pyrimidines | 2009 |
Importance of influx and efflux systems and xenobiotic metabolizing enzymes in intratumoral disposition of anticancer agents.
Topics: Antineoplastic Agents; Benzamides; Drug Resistance, Neoplasm; Drug Tolerance; Gene Expression Regulation, Neoplastic; Humans; Imatinib Mesylate; Inactivation, Metabolic; Membrane Transport Proteins; Models, Biological; Neoplasms; Piperazines; Pyrimidines; Tissue Distribution; Xenobiotics | 2009 |
Neurological adverse effects caused by cytotoxic and targeted therapies.
Topics: Angiogenesis Inhibitors; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Antineoplastic Agents, Alkylating; Benzamides; Bevacizumab; Boronic Acids; Bortezomib; Clinical Trials as Topic; Dacarbazine; Drug Approval; Epothilones; Humans; Imatinib Mesylate; Indoles; Neoplasms; Neurotoxicity Syndromes; Organoplatinum Compounds; Oxaliplatin; Piperazines; Pyrazines; Pyrimidines; Pyrroles; Sunitinib; Temozolomide; Tubulin Modulators; United States; United States Food and Drug Administration | 2009 |
Contemporary pre-clinical development of anticancer agents--what are the optimal preclinical models?
Topics: Angiogenesis Inhibitors; Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Disease Models, Animal; Drug Evaluation, Preclinical; ErbB Receptors; Genetic Engineering; Humans; Imatinib Mesylate; Mice; Neoplasm Transplantation; Neoplasms; Piperazines; Pyrimidines; Transplantation, Heterologous; Trastuzumab | 2009 |
Imatinib mesylate (Gleevec): targeted therapy against cancer with immune properties.
Topics: Animals; Antineoplastic Agents; Benzamides; Dendritic Cells; Humans; Imatinib Mesylate; Immunomodulation; Interferons; Killer Cells, Natural; Mutation; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines; T-Lymphocytes; T-Lymphocytes, Regulatory | 2010 |
[Positron emission tomography and evaluation of response to targeted therapies].
Topics: Antineoplastic Agents; Apoptosis; Benzamides; Cell Hypoxia; Cell Proliferation; Choline; ErbB Receptors; Fluorodeoxyglucose F18; Gastrointestinal Stromal Tumors; Humans; Imatinib Mesylate; Lipid Metabolism; Lung Neoplasms; Neoplasms; Neovascularization, Pathologic; Piperazines; Positron-Emission Tomography; Protein Biosynthesis; Protein Kinases; Pyrimidines; Radiopharmaceuticals; Receptors, Androgen; Receptors, Estrogen; TOR Serine-Threonine Kinases | 2009 |
[Bemusement and strategy on the efficacy of clinical application of targeted anticancer drugs].
Topics: Angiogenesis Inhibitors; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antimetabolites, Antineoplastic; Antineoplastic Agents; Benzamides; Benzenesulfonates; Bevacizumab; Carcinoma, Hepatocellular; Carcinoma, Renal Cell; Deoxycytidine; Drug Delivery Systems; Gastrointestinal Stromal Tumors; Gemcitabine; Humans; Imatinib Mesylate; Indoles; Neoplasms; Niacinamide; Pancreatic Neoplasms; Phenylurea Compounds; Piperazines; Pyridines; Pyrimidines; Pyrroles; Sirolimus; Sorafenib; Sunitinib | 2009 |
Imatinib mesylate.
Topics: Animals; Antineoplastic Agents; Benzamides; Clinical Trials as Topic; Disease Progression; Drug Resistance, Neoplasm; Gastrointestinal Stromal Tumors; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Piperazines; Protein Kinase Inhibitors; Pyrimidines | 2010 |
Targeted cancer therapies in the twenty-first century: lessons from imatinib.
Topics: Animals; Antineoplastic Agents; Benzamides; Drug Delivery Systems; Drug Therapy, Combination; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Pyrimidines | 2010 |
Specificity in the interaction of natural products with their target proteins--a biochemical and structural insight.
Topics: Antineoplastic Agents; Benzamides; Biological Products; Cyclohexanes; Epoxy Compounds; Fatty Acids, Unsaturated; Flavonoids; Humans; Imatinib Mesylate; Macrolides; Neoplasms; Piperazines; Piperidines; Proteins; Pyrimidines; Sesquiterpenes | 2010 |
Signal transduction therapy of cancer.
Topics: Animals; Antineoplastic Agents; Benzamides; Cancer Vaccines; Clinical Trials as Topic; Drug Discovery; Drug Evaluation, Preclinical; Drug Resistance, Neoplasm; Genetic Therapy; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Molecular Structure; Neoplasms; Piperazines; Proteasome Inhibitors; Protein Kinase Inhibitors; Pyrimidines; Signal Transduction | 2010 |
[Treatment with antiangiogenic drugs].
Topics: Angiogenesis Inhibitors; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Benzamides; Bevacizumab; Humans; Imatinib Mesylate; Indoles; Neoplasms; Piperazines; Pyrimidines; Pyrroles; Randomized Controlled Trials as Topic; Receptors, Vascular Endothelial Growth Factor; Sunitinib; Vascular Endothelial Growth Factor A | 2010 |
[Kinase inhibitors].
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antibodies, Monoclonal, Murine-Derived; Benzamides; Bevacizumab; Biomarkers, Tumor; Drug Design; ErbB Receptors; Fusion Proteins, bcr-abl; Genes, ras; Humans; Imatinib Mesylate; Mutation; Neoplasms; Phosphoinositide-3 Kinase Inhibitors; Phosphotransferases; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Proto-Oncogene Proteins B-raf; Pyrimidines; Rituximab; Signal Transduction | 2010 |
Cytogenomics of cancers: from chromosome to sequence.
Topics: Antineoplastic Agents; Base Sequence; Benzamides; Chromosome Aberrations; Chromosomes; Cytogenetics; Disease Progression; Genomics; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Piperazines; Protein Kinase Inhibitors; Pyrimidines | 2010 |
[Clinical manifestation of targeted drugs in individualized therapy of malignant tumors].
Topics: Antibodies, Monoclonal, Murine-Derived; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Cyclophosphamide; Doxorubicin; Drug Delivery Systems; ErbB Receptors; Gastrointestinal Stromal Tumors; Humans; Imatinib Mesylate; Indoles; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myeloid; Lymphoma, Large B-Cell, Diffuse; Mutation; Neoplasms; Piperazines; Prednisone; Pyrimidines; Pyrroles; Remission Induction; Rituximab; Sunitinib; Vincristine | 2010 |
Targeting the DFG-in kinase conformation: a new trend emerging from a patent analysis.
Topics: Benzamides; Dasatinib; Drug Discovery; Imatinib Mesylate; Inflammation; Models, Molecular; Molecular Conformation; Neoplasms; Patents as Topic; Phosphotransferases; Piperazines; Protein Binding; Protein Kinase Inhibitors; Pyrimidines; Signal Transduction; Thiazoles | 2011 |
Targeted therapy in pediatric and adolescent oncology.
Topics: Adolescent; Angiogenesis Inhibitors; Benzamides; Child; fms-Like Tyrosine Kinase 3; Gangliosides; Humans; Imatinib Mesylate; Molecular Targeted Therapy; Neoplasms; Pharmacokinetics; Piperazines; Pyrimidines; Young Adult | 2011 |
[Indications and current development of new targeted therapies in pediatric oncology].
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Benzenesulfonates; Bevacizumab; Child; Dasatinib; Erlotinib Hydrochloride; Hedgehog Proteins; Humans; Imatinib Mesylate; Indoles; Integrins; Molecular Targeted Therapy; Neoplasms; Niacinamide; Nifurtimox; Phenylurea Compounds; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyridines; Pyrimidines; Pyrroles; Quinazolines; Sorafenib; Sunitinib; Thiazoles; TOR Serine-Threonine Kinases | 2011 |
Targeted-therapy and imaging response: a new paradigm for clinical evaluation?
Topics: Antineoplastic Agents; Benzamides; Benzenesulfonates; Clinical Trials as Topic; Diagnostic Imaging; Fluorodeoxyglucose F18; Humans; Imatinib Mesylate; Neoplasms; Niacinamide; Phenylurea Compounds; Piperazines; Protein-Tyrosine Kinases; Pyridines; Pyrimidines; Radiopharmaceuticals; Receptors, Vascular Endothelial Growth Factor; Sorafenib | 2011 |
Tyrosine kinase gene fusions in cancer: translating mechanisms into targeted therapies.
Topics: Benzamides; Crizotinib; Fusion Proteins, bcr-abl; Gene Fusion; Humans; Imatinib Mesylate; MicroRNAs; Molecular Targeted Therapy; Neoplasms; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrazoles; Pyridines; Pyrimidines; Signal Transduction | 2012 |
Pulmonary toxicities of tyrosine kinase inhibitors.
Topics: Antineoplastic Agents; Benzamides; ErbB Receptors; Erlotinib Hydrochloride; Fusion Proteins, bcr-abl; Gefitinib; Humans; Imatinib Mesylate; Lung Diseases, Interstitial; Neoplasms; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Quinazolines | 2011 |
Targeted therapeutics in treatment of children and young adults with solid tumors: an expert survey and review of the literature.
Topics: Adolescent; Antibodies, Monoclonal, Humanized; Benzamides; Bevacizumab; Child; Delphi Technique; Humans; Imatinib Mesylate; Molecular Targeted Therapy; Neoplasms; Piperazines; Pyrimidines; Sirolimus; Young Adult | 2012 |
[Protein tyrosine kinase inhibitors in cancer therapy].
Topics: Antineoplastic Agents; Benzamides; Humans; Imatinib Mesylate; Molecular Targeted Therapy; Neoplasms; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Signal Transduction | 2012 |
Evidence for therapeutic drug monitoring of targeted anticancer therapies.
Topics: Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antibodies, Monoclonal, Murine-Derived; Antineoplastic Agents; Area Under Curve; Benzamides; Benzenesulfonates; Cetuximab; Dasatinib; Drug Monitoring; Everolimus; Evidence-Based Medicine; Half-Life; Humans; Imatinib Mesylate; Indoles; Injections, Intravenous; Molecular Targeted Therapy; Neoplasms; Niacinamide; Phenylurea Compounds; Piperazines; Pyridines; Pyrimidines; Pyrroles; Rituximab; Sirolimus; Sorafenib; Sunitinib; Thiazoles | 2012 |
The ophthalmological complications of targeted agents in cancer therapy: what do we need to know as ophthalmologists?
Topics: Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Bevacizumab; Cetuximab; Crizotinib; Erlotinib Hydrochloride; Eye Diseases; Humans; Imatinib Mesylate; Molecular Targeted Therapy; Neoplasms; Phosphorylcholine; Piperazines; Pyrazoles; Pyridines; Pyrimidines; Quinazolines; Trastuzumab | 2013 |
Tyrosine kinase inhibitors: views of selectivity, sensitivity, and clinical performance.
Topics: Animals; Benzamides; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines | 2013 |
Type II kinase inhibitors: an opportunity in cancer for rational design.
Topics: Animals; Antineoplastic Agents; Benzamides; Drug Design; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein Kinase Inhibitors; Pyrimidines | 2013 |
Monitoring after successful therapy for chronic myeloid leukemia.
Topics: Benzamides; Cell Line, Tumor; Cytogenetics; Drug Resistance, Neoplasm; Enzyme Inhibitors; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Medical Oncology; Medication Adherence; Neoplasms; Piperazines; Prevalence; Protein Kinase Inhibitors; Pyrimidines; Recurrence; Treatment Outcome | 2012 |
Protein tyrosine kinase inhibitors: new treatment modalities?
Topics: Animals; Benzamides; Clinical Trials as Topic; Drug Delivery Systems; Enzyme Inhibitors; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines | 2002 |
[The principles of cancer treatment--changes in chemotherapy].
Topics: ADP Ribose Transferases; Animals; Antineoplastic Agents; Benzamides; Cisplatin; Drug Combinations; Fluorouracil; Genes, ras; Humans; Imatinib Mesylate; Insect Proteins; Lung Neoplasms; Mice; Neoplasms; Neoplastic Syndromes, Hereditary; Oxonic Acid; Piperazines; Protein-Tyrosine Kinases; Pyridines; Pyrimidines; Signal Transduction; Tegafur; Tumor Cells, Cultured | 2002 |
[c-kit: an irresistible ascension from diagnostic marker to therapeutic].
Topics: Antineoplastic Agents; Benzamides; Biomarkers, Tumor; Enzyme Inhibitors; Humans; Imatinib Mesylate; Intestinal Neoplasms; Mutation; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-kit; Pyrimidines; Stomach Neoplasms | 2002 |
Cancer genome targets: RAF-ing up tumor cells to overcome oncogene addiction.
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Drug Therapy, Combination; Gefitinib; Genetic Therapy; Genome, Human; Humans; Imatinib Mesylate; Neoplasms; Oncogenes; Piperazines; Pyrimidines; Quinazolines; Signal Transduction; Trastuzumab | 2002 |
Clinical trial designs for targeted agents.
Topics: Animals; Antineoplastic Agents; Benzamides; Biomarkers; Biphenyl Compounds; Clinical Trials as Topic; Clinical Trials, Phase I as Topic; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Controlled Clinical Trials as Topic; Dose-Response Relationship, Drug; Double-Blind Method; Drug Design; Drug Screening Assays, Antitumor; Enzyme Inhibitors; Humans; Imatinib Mesylate; Matrix Metalloproteinase Inhibitors; Mice; Neoplasm Proteins; Neoplasms; Organic Chemicals; Outcome Assessment, Health Care; Patient Selection; Phenylbutyrates; Piperazines; Protein-Tyrosine Kinases; Pyrimidines; Randomized Controlled Trials as Topic; Rats | 2002 |
Imatinib: a selective tyrosine kinase inhibitor.
Topics: Adenosine Triphosphate; Antineoplastic Agents; Benzamides; Cell Communication; Drug Design; Enzyme Inhibitors; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Neoplasm Proteins; Neoplasms; Oncogene Proteins; Piperazines; Protein Binding; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-kit; Pyrimidines; Receptor, Platelet-Derived Growth Factor beta; Structure-Activity Relationship | 2002 |
Targeting oncogene dependence and resistance.
Topics: Alleles; Animals; Antineoplastic Agents; Benzamides; Cell Line, Tumor; Drug Resistance, Neoplasm; Enzyme Inhibitors; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Mutation; Neoplasms; Oncogenes; Piperazines; Pyrimidines | 2003 |
Molecular-genetic imaging: current and future perspectives.
Topics: Animals; Benzamides; Diagnostic Imaging; Gene Expression Regulation; Genes, Reporter; Genetic Techniques; Humans; Imatinib Mesylate; Models, Biological; Neoplasms; Piperazines; Pyrimidines; Time Factors; Tomography, Emission-Computed; Tumor Suppressor Protein p53 | 2003 |
Protein kinase inhibitors as a therapeutic modality.
Topics: Antineoplastic Agents; Benzamides; Drug Design; Enzyme Inhibitors; Humans; Imatinib Mesylate; Molecular Mimicry; Neoplasms; Piperazines; Protein Kinase Inhibitors; Protein Kinases; Pyrimidines; Signal Transduction | 2003 |
Targeting PDGF receptors in cancer--rationales and proof of concept clinical trials.
Topics: Benzamides; Clinical Trials as Topic; Enzyme Inhibitors; Humans; Imatinib Mesylate; Leukemia; Ligands; Male; Models, Biological; Mutation; Neoplasms; Neovascularization, Pathologic; Piperazines; Platelet-Derived Growth Factor; Prostatic Neoplasms; Protein-Tyrosine Kinases; Pyrimidines; Receptors, Platelet-Derived Growth Factor | 2003 |
Beyond Herceptin and Gleevec.
Topics: Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Cell Cycle; Drug Delivery Systems; Enzyme Inhibitors; ErbB Receptors; Humans; Imatinib Mesylate; Mitogen-Activated Protein Kinases; Neoplasms; Piperazines; Pyrimidines; Receptor Protein-Tyrosine Kinases; Receptor, ErbB-2; Receptors, Vascular Endothelial Growth Factor; Trastuzumab | 2003 |
Targeted therapies for the treatment of cancer.
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antibodies, Monoclonal, Murine-Derived; Antineoplastic Agents; Benzamides; Breast Neoplasms; Female; Humans; Imatinib Mesylate; Lymphoma, B-Cell; Male; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines; Rituximab; Trastuzumab | 2003 |
An overview of targeted treatments in cancer.
Topics: Antibodies, Monoclonal; Antineoplastic Agents; Benzamides; Cancer Vaccines; Drug Delivery Systems; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Pyrimidines; Tretinoin | 2003 |
[Current screening for molecular target therapy of cancer].
Topics: Angiogenesis Inhibitors; Animals; Antineoplastic Agents; Benzamides; Boronic Acids; Bortezomib; Drug Delivery Systems; Drug Screening Assays, Antitumor; Gefitinib; Heat-Shock Proteins; Humans; Imatinib Mesylate; Indoles; Lactones; Mice; Neoplasms; Phthalazines; Piperazines; Piperidines; Pyrazines; Pyridines; Pyrimidines; Pyrroles; Quinazolines; Sunitinib | 2003 |
Emerging roles of targeted small molecule protein-tyrosine kinase inhibitors in cancer therapy.
Topics: Angiogenesis Inhibitors; Benzamides; Enzyme Inhibitors; ErbB Receptors; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines | 2004 |
Modeling the cancer patient with genetically engineered mice: prediction of toxicity from molecule-targeted therapies.
Topics: Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Cardiomyoplasty; Colorectal Neoplasms; Cyclooxygenase 2; Disease Models, Animal; ErbB Receptors; Gastrointestinal Diseases; Genes, abl; Genetic Engineering; Humans; Imatinib Mesylate; Isoenzymes; Membrane Proteins; Mice; Mice, Transgenic; Neoplasms; Piperazines; Prostaglandin-Endoperoxide Synthases; Pyrimidines; Receptors, Platelet-Derived Growth Factor; Receptors, Transforming Growth Factor beta; Skin Abnormalities; Trastuzumab; Vascular Endothelial Growth Factor A | 2004 |
Lessons learned from the development of imatinib.
Topics: Benzamides; Drug Design; Drug Evaluation, Preclinical; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines; Structure-Activity Relationship | 2004 |
Changes in therapy for solid tumors: potential for overcoming drug resistance in vivo with molecular targeting agents.
Topics: Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Disease Progression; Drug Resistance, Neoplasm; Fusion Proteins, bcr-abl; Gefitinib; Humans; Imatinib Mesylate; Molecular Biology; Neoplasms; Paracrine Communication; Piperazines; Platelet-Derived Growth Factor; Protein-Tyrosine Kinases; Pyrimidines; Quinazolines; Receptor, ErbB-2; Signal Transduction; Trastuzumab | 2004 |
Cancer stem cells: are we missing the target?
Topics: Animals; Antineoplastic Agents; Benzamides; Drug Design; Drug Resistance, Neoplasm; Enzyme Inhibitors; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Neoplastic Stem Cells; Piperazines; Pyrimidines; Survival | 2004 |
Role of KIT and platelet-derived growth factor receptors as oncoproteins.
Topics: Antineoplastic Agents; Benzamides; Enzyme Inhibitors; Gene Expression Regulation, Neoplastic; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Platelet-Derived Growth Factor; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-kit; Pyrimidines; Receptor, Platelet-Derived Growth Factor alpha; Stem Cell Factor | 2004 |
Increasing tumor uptake of anticancer drugs with imatinib.
Topics: Animals; Antineoplastic Agents; Benzamides; Drug Delivery Systems; Enzyme Inhibitors; Extracellular Fluid; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Platelet-Derived Growth Factor; Protein-Tyrosine Kinases; Pyrimidines; Receptors, Platelet-Derived Growth Factor | 2004 |
Imatinib mesylate (Gleevec/Glivec) a molecular-targeted therapy for chronic myeloid leukaemia and other malignancies.
Topics: Antineoplastic Agents; Benzamides; Clinical Trials, Phase I as Topic; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Drug Resistance, Neoplasm; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Pilot Projects; Piperazines; Prognosis; Pyrimidines | 2004 |
PDGF receptors-mediators of autocrine tumor growth and regulators of tumor vasculature and stroma.
Topics: Animals; Benzamides; Biological Transport; DNA Mutational Analysis; Fibroblasts; Humans; Imatinib Mesylate; Models, Biological; Mutation; Neoplasms; Neovascularization, Pathologic; Piperazines; Platelet-Derived Growth Factor; Pyrimidines; Receptors, Platelet-Derived Growth Factor; Signal Transduction; Stromal Cells | 2004 |
Tyrosine kinase inhibitors in cancer therapy.
Topics: Benzamides; Clinical Trials as Topic; Forecasting; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Models, Biological; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines | 2004 |
[The mechanisms of the resistance to molecular targeting agents].
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Benzamides; Drug Delivery Systems; Drug Resistance, Neoplasm; Gefitinib; Humans; Imatinib Mesylate; In Vitro Techniques; Neoplasms; Piperazines; Pyrimidines; Quinazolines; Trastuzumab | 2004 |
Imatinib as a paradigm of targeted therapies.
Topics: Animals; Antineoplastic Agents; Benzamides; Clinical Trials as Topic; Drug Design; Drug Evaluation, Preclinical; Enzyme Inhibitors; Fusion Proteins, bcr-abl; Gastrointestinal Neoplasms; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Mice; Models, Molecular; Neoplasm Proteins; Neoplasms; Oncogenes; Patient Selection; Piperazines; Protein Conformation; Protein-Tyrosine Kinases; Pyrimidines | 2004 |
Kinase inhibitors translate lab discoveries into exciting new cures for cancers.
Topics: Antineoplastic Agents; Benzamides; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines | 2004 |
[Targeted anticancer drugs and their development].
Topics: Antineoplastic Agents; Benzamides; Cell Proliferation; Drug Delivery Systems; Female; Humans; Imatinib Mesylate; Male; Neoplasms; Neovascularization, Pathologic; Piperazines; Prognosis; Pyrimidines; Risk Factors; Treatment Outcome | 2004 |
Oncogenic derivatives of platelet-derived growth factor receptors.
Topics: Benzamides; Gene Deletion; Gene Expression Regulation, Developmental; Gene Expression Regulation, Neoplastic; Humans; Imatinib Mesylate; Ligands; Models, Biological; Models, Genetic; Mutation; Neoplasms; Piperazines; Point Mutation; Protein Isoforms; Protein Structure, Tertiary; Pyrimidines; Receptor, Platelet-Derived Growth Factor alpha; Receptor, Platelet-Derived Growth Factor beta; Receptors, Platelet-Derived Growth Factor; Signal Transduction; Translocation, Genetic | 2004 |
Kit as a human oncogenic tyrosine kinase.
Topics: Animals; Benzamides; Dimerization; Gastrointestinal Stromal Tumors; Homozygote; Humans; Imatinib Mesylate; Leukemia, Mast-Cell; Mice; Models, Biological; Mutation; Neoplasms; Neoplasms, Germ Cell and Embryonal; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines; Rats; Signal Transduction; Structure-Activity Relationship | 2004 |
Reversing resistance to targeted therapy.
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Antineoplastic Agents, Hormonal; Benzamides; Drug Delivery Systems; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Gefitinib; Humans; Imatinib Mesylate; Male; Neoplasms; Piperazines; Pyrimidines; Quinazolines; Risk Assessment; Sensitivity and Specificity; Trastuzumab | 2004 |
A cell-based screening strategy that predicts mutations in oncogenic tyrosine kinases: implications for clinical resistance in targeted cancer treatment.
Topics: Animals; Benzamides; Cell Line, Tumor; Cell Survival; Clinical Trials as Topic; Cloning, Molecular; DNA, Complementary; Drug Resistance; Drug Resistance, Neoplasm; Enzyme Inhibitors; Fusion Proteins, bcr-abl; Genetic Techniques; Humans; Imatinib Mesylate; In Situ Hybridization, Fluorescence; Mutagenesis; Mutation; Neoplasms; Piperazines; Protein Binding; Protein-Tyrosine Kinases; Pyrimidines | 2005 |
[Molecular target therapy for malignant tumors].
Topics: Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antibodies, Monoclonal, Murine-Derived; Antineoplastic Agents; Benzamides; Clinical Trials as Topic; ErbB Receptors; Fusion Proteins, bcr-abl; Gefitinib; Hematologic Neoplasms; Humans; Imatinib Mesylate; Intracellular Signaling Peptides and Proteins; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines; Quinazolines; Rituximab; Signal Transduction; Trastuzumab; Tretinoin | 2005 |
[Optimizing current drugs].
Topics: Antineoplastic Agents; Antineoplastic Agents, Phytogenic; Benzamides; Camptothecin; History, 20th Century; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Pyrimidines | 2005 |
Mechanisms of clinical resistance to small molecule tyrosine kinase inhibitors targeting oncogenic tyrosine kinases.
Topics: Animals; Benzamides; Drug Resistance, Neoplasm; Humans; Imatinib Mesylate; Mutation; Neoplasms; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines | 2005 |
Role of cytochrome P450 activity in the fate of anticancer agents and in drug resistance: focus on tamoxifen, paclitaxel and imatinib metabolism.
Topics: Antineoplastic Agents; Benzamides; Biotransformation; Cytochrome P-450 Enzyme System; Drug Interactions; Drug Monitoring; Drug Resistance, Neoplasm; Humans; Imatinib Mesylate; Isoenzymes; Neoplasms; Paclitaxel; Piperazines; Polymorphism, Genetic; Pyrimidines; Tamoxifen | 2005 |
[Tyrosine kinase inhibitors in tumor therapy--part 1. Molecular and genetic fundamentals].
Topics: Antibodies, Monoclonal; Antineoplastic Agents; Benzamides; Dimerization; Enzyme Activation; Growth Substances; Humans; Imatinib Mesylate; Neoplasms; Neovascularization, Pathologic; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Receptor Protein-Tyrosine Kinases; Receptors, Growth Factor; Receptors, Vascular Endothelial Growth Factor; Signal Transduction | 2005 |
[Tyrosine kinase inhibitors in tumor therapy--part 2. Current position and perspectives].
Topics: Angiogenesis Inhibitors; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Bevacizumab; Cetuximab; ErbB Receptors; Erlotinib Hydrochloride; Gefitinib; Genes, abl; Humans; Imatinib Mesylate; Neoplasms; Patient Selection; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Quinazolines; Trastuzumab; Vascular Endothelial Growth Factor A | 2005 |
Cutaneous side-effects of kinase inhibitors and blocking antibodies.
Topics: Antibodies, Blocking; Antineoplastic Agents; Benzamides; Benzenesulfonates; ErbB Receptors; Hair Diseases; Humans; Imatinib Mesylate; Nail Diseases; Neoplasms; Niacinamide; Phenylurea Compounds; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyridines; Pyrimidines; Skin Diseases; Sorafenib | 2005 |
Tyrosine kinases as targets for cancer therapy.
Topics: Antibodies, Monoclonal; Benzamides; Drug Resistance, Neoplasm; fms-Like Tyrosine Kinase 3; Gene Expression Regulation, Neoplastic; Hematologic Neoplasms; Humans; Imatinib Mesylate; Mutation; Neoplasms; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Pyrimidines; Receptor Protein-Tyrosine Kinases | 2005 |
[Current progress in therapy of malignant diseases].
Topics: Antibodies, Monoclonal; Antineoplastic Agents; Benzamides; Humans; Imatinib Mesylate; Leukemia; Lymphoma; Neoplasms; Piperazines; Pyrimidines | 2005 |
Detection of resistance to imatinib by metabolic profiling: clinical and drug development implications.
Topics: Animals; Antineoplastic Agents; Benzamides; Cell Line, Tumor; Drug Design; Drug Resistance, Neoplasm; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines | 2005 |
Structure and regulation of Kit protein-tyrosine kinase--the stem cell factor receptor.
Topics: Animals; Benzamides; Humans; Imatinib Mesylate; Mutation; Neoplasms; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines; Signal Transduction | 2005 |
[Genetic alterations and chemoresistance].
Topics: Antineoplastic Agents; ATP-Binding Cassette Transporters; Benzamides; Dihydrouracil Dehydrogenase (NADP); Drug Resistance, Neoplasm; Gefitinib; Gene Expression Profiling; Humans; Imatinib Mesylate; Mutation; Neoplasms; Oligonucleotide Array Sequence Analysis; Pharmacogenetics; Piperazines; Polymorphism, Genetic; Pyrimidines; Quinazolines; Thymidylate Synthase; Xeroderma Pigmentosum Group D Protein | 2005 |
[Targeted therapies in pediatric oncology: a new therapeutic approach?].
Topics: Antineoplastic Agents; Benzamides; Child; ErbB Receptors; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines; Receptor Protein-Tyrosine Kinases | 2006 |
[Antineoplastic agents targeting tyrosine kinases].
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Cetuximab; ErbB Receptors; Erlotinib Hydrochloride; Gastrointestinal Stromal Tumors; Gefitinib; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Quinazolines; Receptor Protein-Tyrosine Kinases; Receptors, Platelet-Derived Growth Factor; Signal Transduction; Trastuzumab | 2005 |
[Cancer initiation as mini-evolution].
Topics: Antineoplastic Agents; Benzamides; Cell Differentiation; Chromosomal Instability; Computational Biology; Epithelial Cells; Evolution, Molecular; Genes, Tumor Suppressor; Humans; Imatinib Mesylate; Intracellular Signaling Peptides and Proteins; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Models, Theoretical; Mutation; Neoplasms; Neoplastic Stem Cells; Piperazines; Pyrimidines | 2005 |
[Gene expression profiling for prediction of response to chemotherapy].
Topics: Antineoplastic Agents; Benzamides; Breast Neoplasms; Drug Screening Assays, Antitumor; Esophageal Neoplasms; Gene Expression Profiling; Gene Expression Regulation, Neoplastic; Gene Targeting; Genome, Human; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Oligonucleotide Array Sequence Analysis; Piperazines; Polymorphism, Single Nucleotide; Pyrimidines | 2006 |
[Problems in the current target therapy of malignancies].
Topics: Alemtuzumab; Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antibodies, Monoclonal, Murine-Derived; Antibodies, Neoplasm; Antineoplastic Agents; Azathioprine; Benzamides; Bevacizumab; Cetuximab; Erlotinib Hydrochloride; Gefitinib; Humans; Imatinib Mesylate; Neoplasms; Phthalazines; Piperazines; Pyridines; Pyrimidines; Quinazolines; Quinolones; Rituximab; Sesquiterpenes; Sesquiterpenes, Guaiane; Trastuzumab | 2005 |
Methodological aspects of current problems in target-based anticancer drug development.
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Drug Design; Gefitinib; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Quinazolines; Research Design; Trastuzumab | 2006 |
[Requirements for the development of molecularly defined targeted therapy in oncology].
Topics: Algorithms; Angiogenesis Inhibitors; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antimetabolites, Antineoplastic; Antineoplastic Agents; Benzamides; Bevacizumab; Biomedical Research; Biotechnology; Breast Neoplasms; Cetuximab; Clinical Trials, Phase I as Topic; Clinical Trials, Phase II as Topic; Computational Biology; Controlled Clinical Trials as Topic; Deoxycytidine; Drug Industry; Female; Gemcitabine; Genome, Human; Humans; Imatinib Mesylate; Medical Oncology; Molecular Biology; Multicenter Studies as Topic; Neoplasms; Phenotype; Piperazines; Practice Guidelines as Topic; Prognosis; Protein Kinase Inhibitors; Pyrimidines; Risk Assessment; Trastuzumab; Treatment Outcome | 2006 |
[Targeted therapies of cancer: not lost in translation].
Topics: Antineoplastic Agents; Benzamides; Cell Transformation, Neoplastic; Gastrointestinal Stromal Tumors; Humans; Imatinib Mesylate; Mutation; Neoplasm Proteins; Neoplasms; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines | 2006 |
Mathematical models of targeted cancer therapy.
Topics: Antineoplastic Agents; Benzamides; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Models, Theoretical; Neoplasms; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Receptors, Growth Factor; Treatment Outcome | 2006 |
Protein kinases as drug targets in cancer.
Topics: Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Benzamides; Benzenesulfonates; Gefitinib; HSP90 Heat-Shock Proteins; Humans; Imatinib Mesylate; Neoplasms; Niacinamide; p38 Mitogen-Activated Protein Kinases; Phenylurea Compounds; Piperazines; Protein Kinase Inhibitors; Pyridines; Pyrimidines; Quinazolines; Signal Transduction; Sirolimus; Sorafenib; Trastuzumab | 2006 |
[Molecular targeted therapy].
Topics: Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antibodies, Monoclonal, Murine-Derived; Antineoplastic Agents; Benzamides; Cancer Vaccines; Cell Survival; Clinical Trials as Topic; Drug Delivery Systems; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Rituximab; Trastuzumab | 2006 |
Protein kinase inhibitors.
Topics: Animals; Benzamides; Cyclin-Dependent Kinases; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-kit; Pyrimidines; Receptors, Platelet-Derived Growth Factor | 2006 |
Why is cancer drug discovery so difficult?
Topics: Animals; Antineoplastic Agents; Benzamides; Drug Design; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Pyrimidines; Quantitative Trait Loci | 2007 |
[Current events about echography in 2006: position of the ultrasound functional imaging for the early evaluation of targeted therapeutics].
Topics: Antineoplastic Agents; Benzamides; Contrast Media; Gastrointestinal Stromal Tumors; Humans; Imatinib Mesylate; Kidney Neoplasms; Microcirculation; Neoplasms; Neovascularization, Pathologic; Phospholipids; Piperazines; Polysaccharides; Pyrimidines; Sulfur Hexafluoride; Treatment Outcome; Ultrasonography | 2006 |
Emerging safety issues with imatinib and other Abl tyrosine kinase inhibitors.
Topics: Benzamides; Clinical Trials as Topic; Follow-Up Studies; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-abl; Pyrimidines; Time Factors; United States; United States Food and Drug Administration | 2007 |
PDGF receptors as targets in tumor treatment.
Topics: Animals; Antineoplastic Agents; Benzamides; Clinical Trials, Phase III as Topic; Drug Delivery Systems; Extracellular Fluid; Fibroblasts; Humans; Imatinib Mesylate; Indoles; Mutation; Neoplasm Metastasis; Neoplasm Proteins; Neoplasms; Neovascularization, Pathologic; Piperazines; Platelet-Derived Growth Factor; Pressure; Protein Kinase Inhibitors; Pyrimidines; Pyrroles; Receptors, Platelet-Derived Growth Factor; Signal Transduction; Sunitinib; Translocation, Genetic | 2007 |
Targeted cancer therapy: promise and reality.
Topics: Angiogenesis Inhibitors; Animals; Antineoplastic Agents; Benzamides; Clinical Trials as Topic; Drug Delivery Systems; Drug Screening Assays, Antitumor; ErbB Receptors; Forecasting; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Mice; Mice, Transgenic; Neoplasm Proteins; Neoplasms; Neoplastic Stem Cells; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Signal Transduction | 2007 |
Risk assessment in haemotopoietic stem cell transplantation: disease and disease stage.
Topics: Acute Disease; Adult; Benzamides; Female; Hematopoietic Stem Cell Transplantation; Humans; Imatinib Mesylate; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid; Male; Multiple Myeloma; Myelodysplastic Syndromes; Neoplasm Staging; Neoplasms; Piperazines; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prognosis; Pyrimidines; Recurrence; Risk Assessment; Survival Analysis; Transplantation, Homologous | 2007 |
Spectrum of activity and mechanism of action of VEGF/PDGF inhibitors.
Topics: Angiogenesis Inhibitors; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Bevacizumab; Humans; Imatinib Mesylate; Immunologic Factors; Neoplasms; Neovascularization, Pathologic; Piperazines; Platelet-Derived Growth Factor; Pyrimidines; Receptors, Vascular Endothelial Growth Factor; Vascular Endothelial Growth Factor A | 2007 |
[Hypereosinophilic syndrome--recent developments in diagnosis and treatment].
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Glucocorticoids; Humans; Hypereosinophilic Syndrome; Hypersensitivity; Imatinib Mesylate; Immunosuppressive Agents; Interferon-alpha; Lung Diseases; Neoplasms; Parasitic Diseases; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Tumor Necrosis Factor-alpha; Vasculitis | 2007 |
Dissecting kinase signaling pathways.
Topics: Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Drug Delivery Systems; Humans; Imatinib Mesylate; Lapatinib; Neoplasms; Phosphoproteins; Phosphorylation; Piperazines; Protein Kinase Inhibitors; Protein Kinases; Proteomics; Pyrimidines; Quinazolines; Signal Transduction; Trastuzumab | 2007 |
New developments in multitargeted therapy for patients with solid tumours.
Topics: Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Benzenesulfonates; Clinical Trials as Topic; Dasatinib; Drug Delivery Systems; Humans; Imatinib Mesylate; Indoles; Neoplasms; Niacinamide; Phenylurea Compounds; Piperazines; Pyridines; Pyrimidines; Pyrroles; Sorafenib; Sunitinib; Thiazoles | 2008 |
Targeted therapies in solid tumours: results and promises.
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Bevacizumab; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Cetuximab; Clinical Trials as Topic; Colorectal Neoplasms; Female; Gastrointestinal Stromal Tumors; Humans; Imatinib Mesylate; Lung Neoplasms; Male; Neoplasms; Piperazines; Pyrimidines; Trastuzumab | 2007 |
Dendritic cells and innate defense against tumor cells.
Topics: Apoptosis; Benzamides; Biomarkers, Tumor; Cancer Vaccines; CpG Islands; Cytokines; Dendritic Cells; Fas Ligand Protein; Granulocyte-Macrophage Colony-Stimulating Factor; HMGB1 Protein; Humans; Imatinib Mesylate; Immunity, Innate; Interferon Type I; Interferon-gamma; Interferons; Interleukin-15; Killer Cells, Natural; Neoplasms; Oligodeoxyribonucleotides; Piperazines; Pyrimidines; Receptor Cross-Talk; T-Lymphocytes, Helper-Inducer; Uric Acid | 2008 |
[Imatinib and solid tumours].
Topics: Antineoplastic Agents; Benzamides; Dermatofibrosarcoma; Female; Fusion Proteins, bcr-abl; Gastrointestinal Stromal Tumors; Humans; Imatinib Mesylate; Male; Neoplasms; Neoplasms, Second Primary; Piperazines; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-abl; Proto-Oncogene Proteins c-kit; Pyrimidines; Receptors, Platelet-Derived Growth Factor; Skin Neoplasms | 2008 |
Application of PET/CT in the development of novel anticancer drugs.
Topics: Animals; Antineoplastic Agents; Benzamides; Humans; Imatinib Mesylate; Neoplasm Staging; Neoplasms; Piperazines; Positron-Emission Tomography; Pyrimidines; Tomography, X-Ray Computed | 2008 |
From single- to multi-target drugs in cancer therapy: when aspecificity becomes an advantage.
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Benzenesulfonates; Bevacizumab; Cetuximab; Clinical Trials as Topic; Enzyme Inhibitors; Erlotinib Hydrochloride; Gefitinib; Humans; Imatinib Mesylate; Indoles; Lapatinib; Neoplasms; Neovascularization, Pathologic; Niacinamide; Phenylurea Compounds; Piperazines; Piperidines; Protein-Tyrosine Kinases; Pyridines; Pyrimidines; Pyrroles; Quinazolines; Receptor Protein-Tyrosine Kinases; Sorafenib; Sunitinib; Trastuzumab | 2008 |
Acquired resistance to tyrosine kinase inhibitors during cancer therapy.
Topics: Antineoplastic Agents; Benzamides; Drug Resistance, Neoplasm; ErbB Receptors; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines | 2008 |
Commentary: Novel therapies for cancer: why dirty might be better.
Topics: Antineoplastic Agents; Benzamides; Drug Resistance, Neoplasm; ErbB Receptors; Erlotinib Hydrochloride; Fusion Proteins, bcr-abl; Gefitinib; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Microtubules; Neoplasms; Piperazines; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-kit; Pyrimidines; Quinazolines; Receptor Protein-Tyrosine Kinases; Receptors, Purinergic P2 | 2008 |
New agents in cancer clinical trials.
Topics: Antineoplastic Agents; Benzamides; Benzoquinones; Boronic Acids; Bortezomib; Clinical Trials as Topic; Dioxoles; Enzyme Inhibitors; Humans; Hydroxamic Acids; Imatinib Mesylate; Isoquinolines; Lactams, Macrocyclic; Neoplasms; Piperazines; Pyrazines; Pyrimidines; Rifabutin; Stilbenes; Tetrahydrofolates; Tetrahydroisoquinolines; Trabectedin; Vorinostat | 2000 |
Mechanisms of resistance to imatinib (STI571) and prospects for combination with conventional chemotherapeutic agents.
Topics: Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Drug Resistance, Neoplasm; Gene Amplification; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines | 2001 |
Targeting protein kinases for tumor therapy.
Topics: Antineoplastic Agents; Benzamides; Cell Division; Cell Survival; Clinical Trials as Topic; Enzyme Inhibitors; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Pyrimidines; Receptor Protein-Tyrosine Kinases | 2001 |
Tyrosine kinase inhibitors: a clinical perspective.
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Enzyme Inhibitors; ErbB Receptors; Humans; Imatinib Mesylate; Molecular Structure; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines; Trastuzumab | 2002 |
[Selective tyrosine kinase inhibitor imatinib (STI571) in haematological and oncological disease].
Topics: Adult; Antineoplastic Agents; Benzamides; Carcinoma, Small Cell; Clinical Trials, Phase I as Topic; Clinical Trials, Phase II as Topic; Cytogenetics; Drug Resistance, Neoplasm; Drug Therapy, Combination; Enzyme Inhibitors; Female; Fusion Proteins, bcr-abl; Gastrointestinal Neoplasms; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myelomonocytic, Chronic; Lung Neoplasms; Male; Mastocytosis; Multicenter Studies as Topic; Mutation; Neoplasms; Piperazines; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Primary Myelofibrosis; Protein-Tyrosine Kinases; Pyrimidines; Remission Induction; Time Factors | 2002 |
Inhibition of KIT tyrosine kinase activity: a novel molecular approach to the treatment of KIT-positive malignancies.
Topics: Angiogenesis Inhibitors; Benzamides; Enzyme Inhibitors; Humans; Imatinib Mesylate; Indoles; Mutation; Neoplasms; Oxindoles; Piperazines; Propionates; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-kit; Pyrimidines; Pyrroles | 2002 |
Interaction of tyrosine kinase inhibitors with the human multidrug transporter proteins, MDR1 and MRP1.
Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzamides; Enzyme Inhibitors; Humans; Imatinib Mesylate; In Vitro Techniques; Multidrug Resistance-Associated Proteins; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines; Recombinant Proteins; Tumor Cells, Cultured | 2002 |
13 trial(s) available for imatinib mesylate and Benign Neoplasms
Article | Year |
---|---|
Topics: A549 Cells; Acetylmuramyl-Alanyl-Isoglutamine; Acinetobacter baumannii; Acute Lung Injury; Adaptor Proteins, Signal Transducing; Adenine; Adenocarcinoma; Adipogenesis; Administration, Cutaneous; Administration, Ophthalmic; Adolescent; Adsorption; Adult; Aeromonas hydrophila; Aerosols; Aged; Aged, 80 and over; Aging; Agriculture; Air Pollutants; Air Pollution; Airway Remodeling; Alanine Transaminase; Albuminuria; Aldehyde Dehydrogenase 1 Family; Algorithms; AlkB Homolog 2, Alpha-Ketoglutarate-Dependent Dioxygenase; Alzheimer Disease; Amino Acid Sequence; Ammonia; Ammonium Compounds; Anaerobiosis; Anesthetics, Dissociative; Anesthetics, Inhalation; Animals; Anti-Bacterial Agents; Anti-HIV Agents; Anti-Infective Agents; Anti-Inflammatory Agents; Antibiotics, Antineoplastic; Antibodies, Antineutrophil Cytoplasmic; Antibodies, Monoclonal, Humanized; Antifungal Agents; Antigens, Bacterial; Antigens, CD; Antigens, Differentiation, Myelomonocytic; Antimetabolites, Antineoplastic; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Antioxidants; Antitubercular Agents; Antiviral Agents; Apolipoproteins E; Apoptosis; Arabidopsis; Arabidopsis Proteins; Arsenic; Arthritis, Rheumatoid; Asthma; Atherosclerosis; ATP-Dependent Proteases; Attitude of Health Personnel; Australia; Austria; Autophagy; Axitinib; Bacteria; Bacterial Outer Membrane Proteins; Bacterial Proteins; Bacterial Toxins; Bacterial Typing Techniques; Bariatric Surgery; Base Composition; Bayes Theorem; Benzoxazoles; Benzylamines; beta Catenin; Betacoronavirus; Betula; Binding Sites; Biological Availability; Biological Oxygen Demand Analysis; Biomarkers; Biomarkers, Tumor; Biopsy; Bioreactors; Biosensing Techniques; Birth Weight; Blindness; Blood Chemical Analysis; Blood Gas Analysis; Blood Glucose; Blood Pressure; Blood Pressure Monitoring, Ambulatory; Blood-Brain Barrier; Blotting, Western; Body Mass Index; Body Weight; Bone and Bones; Bone Density; Bone Resorption; Borates; Brain; Brain Infarction; Brain Injuries, Traumatic; Brain Neoplasms; Breakfast; Breast Milk Expression; Breast Neoplasms; Bronchi; Bronchoalveolar Lavage Fluid; Buffaloes; Cadherins; Calcification, Physiologic; Calcium Compounds; Calcium, Dietary; Cannula; Caprolactam; Carbon; Carbon Dioxide; Carboplatin; Carcinogenesis; Carcinoma, Ductal; Carcinoma, Ehrlich Tumor; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Pancreatic Ductal; Carcinoma, Renal Cell; Cardiovascular Diseases; Carps; Carrageenan; Case-Control Studies; Catalysis; Catalytic Domain; Cattle; CD8-Positive T-Lymphocytes; Cell Adhesion; Cell Cycle Proteins; Cell Death; Cell Differentiation; Cell Line; Cell Line, Tumor; Cell Movement; Cell Nucleus; Cell Phone Use; Cell Proliferation; Cell Survival; Cell Transformation, Neoplastic; Cell Transformation, Viral; Cells, Cultured; Cellulose; Chemical Phenomena; Chemoradiotherapy; Child; Child Development; Child, Preschool; China; Chitosan; Chlorocebus aethiops; Cholecalciferol; Chromatography, Liquid; Circadian Clocks; Circadian Rhythm; Circular Dichroism; Cisplatin; Citric Acid; Clinical Competence; Clinical Laboratory Techniques; Clinical Trials, Phase I as Topic; Clinical Trials, Phase II as Topic; Clostridioides difficile; Clostridium Infections; Coculture Techniques; Cohort Studies; Cold Temperature; Colitis; Collagen Type I; Collagen Type I, alpha 1 Chain; Collagen Type XI; Color; Connective Tissue Diseases; Copper; Coronary Angiography; Coronavirus 3C Proteases; Coronavirus Infections; Cost of Illness; Counselors; COVID-19; COVID-19 Testing; Creatine Kinase; Creatinine; Cross-Over Studies; Cross-Sectional Studies; Cryoelectron Microscopy; Cryosurgery; Crystallography, X-Ray; Cues; Cultural Competency; Cultural Diversity; Curriculum; Cyclic AMP Response Element-Binding Protein; Cyclin-Dependent Kinase Inhibitor p21; Cycloparaffins; Cysteine Endopeptidases; Cytokines; Cytoplasm; Cytoprotection; Databases, Factual; Denitrification; Deoxycytidine; Diabetes Complications; Diabetes Mellitus; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Diagnosis, Differential; Diatoms; Diet; Diet, High-Fat; Dietary Exposure; Diffusion Magnetic Resonance Imaging; Diketopiperazines; Dipeptidyl Peptidase 4; Dipeptidyl-Peptidase IV Inhibitors; Disease Models, Animal; Disease Progression; Disease-Free Survival; DNA; DNA Damage; DNA Glycosylases; DNA Repair; DNA-Binding Proteins; DNA, Bacterial; DNA, Viral; Docetaxel; Dose Fractionation, Radiation; Dose-Response Relationship, Drug; Down-Regulation; Doxorubicin; Drosophila; Drosophila melanogaster; Drug Carriers; Drug Delivery Systems; Drug Liberation; Drug Repositioning; Drug Resistance, Bacterial; Drug Resistance, Multiple, Bacterial; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Drug Synergism; Drug Therapy, Combination; Edema; Edible Grain; Education, Graduate; Education, Medical, Graduate; Education, Pharmacy; Ehlers-Danlos Syndrome; Electron Transport Complex III; Electron Transport Complex IV; Electronic Nicotine Delivery Systems; Emergency Service, Hospital; Empathy; Emulsions; Endothelial Cells; Endurance Training; Energy Intake; Enterovirus A, Human; Environment; Environmental Monitoring; Enzyme Assays; Enzyme Inhibitors; Epithelial Cells; Epithelial-Mesenchymal Transition; Epoxide Hydrolases; Epoxy Compounds; Erythrocyte Count; Erythrocytes; Escherichia coli; Escherichia coli Infections; Escherichia coli Proteins; Esophageal Neoplasms; Esophageal Squamous Cell Carcinoma; Esophagectomy; Estrogens; Etanercept; Ethiopia; Ethnicity; Ethylenes; Exanthema; Exercise; Exercise Test; Exercise Tolerance; Extracellular Matrix; Extracorporeal Membrane Oxygenation; Eye Infections, Fungal; False Negative Reactions; Fatty Acids; Fecal Microbiota Transplantation; Feces; Female; Femur Neck; Fermentation; Ferritins; Fetal Development; Fibroblast Growth Factor-23; Fibroblast Growth Factors; Fibroblasts; Fibroins; Fish Proteins; Flavanones; Flavonoids; Focus Groups; Follow-Up Studies; Food Handling; Food Supply; Food, Formulated; Forced Expiratory Volume; Forests; Fractures, Bone; Fruit and Vegetable Juices; Fusobacteria; G1 Phase Cell Cycle Checkpoints; G2 Phase Cell Cycle Checkpoints; Gamma Rays; Gastrectomy; Gastrointestinal Microbiome; Gastrointestinal Stromal Tumors; Gefitinib; Gels; Gemcitabine; Gene Amplification; Gene Expression; Gene Expression Regulation; Gene Expression Regulation, Bacterial; Gene Expression Regulation, Neoplastic; Gene Expression Regulation, Plant; Gene Knockdown Techniques; Gene-Environment Interaction; Genotype; Germany; Glioma; Glomerular Filtration Rate; Glucagon; Glucocorticoids; Glycemic Control; Glycerol; Glycogen Synthase Kinase 3 beta; Glycolipids; Glycolysis; Goblet Cells; Gram-Negative Bacterial Infections; Granulocyte Colony-Stimulating Factor; Graphite; Greenhouse Effect; Guanidines; Haemophilus influenzae; HCT116 Cells; Health Knowledge, Attitudes, Practice; Health Personnel; Health Services Accessibility; Health Services Needs and Demand; Health Status Disparities; Healthy Volunteers; Heart Failure; Heart Rate; Heart Transplantation; Heart-Assist Devices; HEK293 Cells; Heme; Heme Oxygenase-1; Hemolysis; Hemorrhage; Hepatitis B; Hepatitis B e Antigens; Hepatitis B Surface Antigens; Hepatitis B virus; Hepatitis B, Chronic; Hepatocytes; Hexoses; High-Throughput Nucleotide Sequencing; Hippo Signaling Pathway; Histamine; Histamine Agonists; Histidine; Histone Deacetylase 2; HIV Infections; HIV Reverse Transcriptase; HIV-1; Homebound Persons; Homeodomain Proteins; Homosexuality, Male; Hospice and Palliative Care Nursing; HSP70 Heat-Shock Proteins; Humans; Hyaluronan Receptors; Hydrogen; Hydrogen Peroxide; Hydrogen-Ion Concentration; Hydrolysis; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypoglycemia; Hypoglycemic Agents; Hypoxia; Idiopathic Interstitial Pneumonias; Imaging, Three-Dimensional; Imatinib Mesylate; Immunotherapy; Implementation Science; Incidence; INDEL Mutation; Induced Pluripotent Stem Cells; Industrial Waste; Infant; Infant, Newborn; Inflammation; Inflammation Mediators; Infliximab; Infusions, Intravenous; Inhibitory Concentration 50; Injections; Insecticides; Insulin-Like Growth Factor Binding Protein 5; Insulin-Secreting Cells; Interleukin-1; Interleukin-17; Interleukin-8; Internship and Residency; Intestines; Intracellular Signaling Peptides and Proteins; Ion Transport; Iridaceae; Iridoid Glucosides; Islets of Langerhans Transplantation; Isodon; Isoflurane; Isotopes; Italy; Joint Instability; Ketamine; Kidney; Kidney Failure, Chronic; Kidney Function Tests; Kidney Neoplasms; Kinetics; Klebsiella pneumoniae; Knee Joint; Kruppel-Like Factor 4; Kruppel-Like Transcription Factors; Lactate Dehydrogenase 5; Laparoscopy; Laser Therapy; Lasers, Semiconductor; Lasers, Solid-State; Laurates; Lead; Leukocyte L1 Antigen Complex; Leukocytes, Mononuclear; Light; Lipid Peroxidation; Lipopolysaccharides; Liposomes; Liver; Liver Cirrhosis; Liver Neoplasms; Liver Transplantation; Locomotion; Longitudinal Studies; Lopinavir; Lower Urinary Tract Symptoms; Lubricants; Lung; Lung Diseases, Interstitial; Lung Neoplasms; Lymphocyte Activation; Lymphocytes, Tumor-Infiltrating; Lymphoma, Mantle-Cell; Lysosomes; Macrophages; Male; Manganese Compounds; MAP Kinase Kinase 4; Mass Screening; Maternal Health; Medicine, Chinese Traditional; Melanoma, Experimental; Memantine; Membrane Glycoproteins; Membrane Proteins; Mesenchymal Stem Cell Transplantation; Metal Nanoparticles; Metalloendopeptidases; Metalloporphyrins; Methadone; Methane; Methicillin-Resistant Staphylococcus aureus; Mexico; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Inbred ICR; Mice, Knockout; Mice, Nude; Mice, SCID; Mice, Transgenic; Microarray Analysis; Microbial Sensitivity Tests; Microbiota; Micronutrients; MicroRNAs; Microscopy, Confocal; Microsomes, Liver; Middle Aged; Milk; Milk, Human; Minority Groups; Mitochondria; Mitochondrial Membranes; Mitochondrial Proteins; Models, Animal; Models, Molecular; Molecular Conformation; Molecular Docking Simulation; Molecular Dynamics Simulation; Molecular Epidemiology; Molecular Structure; Molecular Weight; Multilocus Sequence Typing; Multimodal Imaging; Muscle Strength; Muscle, Skeletal; Muscular Diseases; Mutation; Mycobacterium tuberculosis; Myocardial Stunning; Myristates; NAD(P)H Dehydrogenase (Quinone); Nanocomposites; Nanogels; Nanoparticles; Nanotechnology; Naphthalenes; Nasal Cavity; National Health Programs; Necrosis; Needs Assessment; Neoadjuvant Therapy; Neonicotinoids; Neoplasm Invasiveness; Neoplasm Metastasis; Neoplasm Proteins; Neoplasm Recurrence, Local; Neoplasm Staging; Neoplasm Transplantation; Neoplasms; Neoplastic Stem Cells; Netherlands; Neuroblastoma; Neuroprotective Agents; Neutrophils; NF-kappa B; NFATC Transcription Factors; Nicotiana; Nicotine; Nitrates; Nitrification; Nitrites; Nitro Compounds; Nitrogen; Nitrogen Dioxide; North Carolina; Nuclear Magnetic Resonance, Biomolecular; Nuclear Proteins; Nucleic Acid Hybridization; Nucleosomes; Nutrients; Obesity; Obesity, Morbid; Oceans and Seas; Oncogene Protein v-akt; Oncogenes; Oocytes; Open Reading Frames; Osteoclasts; Osteogenesis; Osteoporosis; Osteoporosis, Postmenopausal; Outpatients; Ovarian Neoplasms; Ovariectomy; Overweight; Oxazines; Oxidants; Oxidation-Reduction; Oxidative Stress; Oxides; Oxidoreductases; Oxygen; Oxygen Inhalation Therapy; Oxygenators, Membrane; Ozone; Paclitaxel; Paenibacillus; Pain Measurement; Palliative Care; Pancreatic Neoplasms; Pandemics; Parasympathetic Nervous System; Particulate Matter; Pasteurization; Patient Preference; Patient Satisfaction; Pediatric Obesity; Permeability; Peroxiredoxins; Peroxynitrous Acid; Pharmaceutical Services; Pharmacists; Pharmacy; Phaseolus; Phenotype; Phoeniceae; Phosphates; Phosphatidylinositol 3-Kinases; Phospholipid Transfer Proteins; Phospholipids; Phosphorus; Phosphorylation; Photoperiod; Photosynthesis; Phylogeny; Physical Endurance; Physicians; Pilot Projects; Piperidines; Pituitary Adenylate Cyclase-Activating Polypeptide; Plant Extracts; Plant Leaves; Plant Proteins; Plant Roots; Plaque, Atherosclerotic; Pneumonia; Pneumonia, Viral; Point-of-Care Testing; Polyethylene Glycols; Polymers; Polysorbates; Pore Forming Cytotoxic Proteins; Positron Emission Tomography Computed Tomography; Positron-Emission Tomography; Postprandial Period; Poverty; Pre-Exposure Prophylaxis; Prediabetic State; Predictive Value of Tests; Pregnancy; Pregnancy Trimester, First; Pregnancy, High-Risk; Prenatal Exposure Delayed Effects; Pressure; Prevalence; Primary Graft Dysfunction; Primary Health Care; Professional Role; Professionalism; Prognosis; Progression-Free Survival; Prolactin; Promoter Regions, Genetic; Proof of Concept Study; Proportional Hazards Models; Propylene Glycol; Prospective Studies; Prostate; Protein Binding; Protein Biosynthesis; Protein Isoforms; Protein Kinase Inhibitors; Protein Phosphatase 2; Protein Processing, Post-Translational; Protein Serine-Threonine Kinases; Protein Structure, Tertiary; Protein Transport; Proteoglycans; Proteome; Proto-Oncogene Proteins c-akt; Proto-Oncogene Proteins c-myc; Proto-Oncogene Proteins c-ret; Proto-Oncogene Proteins p21(ras); Proton Pumps; Protons; Protoporphyrins; Pseudomonas aeruginosa; Pseudomonas fluorescens; Pulmonary Artery; Pulmonary Disease, Chronic Obstructive; Pulmonary Gas Exchange; Pulmonary Veins; Pyrazoles; Pyridines; Pyrimidines; Qualitative Research; Quinoxalines; Rabbits; Random Allocation; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Histamine H3; Receptors, Immunologic; Receptors, Transferrin; Recombinant Proteins; Recurrence; Reference Values; Referral and Consultation; Regional Blood Flow; Registries; Regulon; Renal Insufficiency, Chronic; Reperfusion Injury; Repressor Proteins; Reproducibility of Results; Republic of Korea; Research Design; Resistance Training; Respiration, Artificial; Respiratory Distress Syndrome; Respiratory Insufficiency; Resuscitation; Retinal Dehydrogenase; Retreatment; Retrospective Studies; Reverse Transcriptase Inhibitors; Rhinitis, Allergic; Ribosomal Proteins; Ribosomes; Risk Assessment; Risk Factors; Ritonavir; Rivers; RNA Interference; RNA-Seq; RNA, Messenger; RNA, Ribosomal, 16S; RNA, Small Interfering; Rosuvastatin Calcium; Rural Population; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Salivary Ducts; Salivary Gland Neoplasms; San Francisco; SARS-CoV-2; Satiation; Satiety Response; Schools; Schools, Pharmacy; Seasons; Seawater; Selection, Genetic; Sequence Analysis, DNA; Serine-Threonine Kinase 3; Sewage; Sheep; Sheep, Domestic; Shock, Hemorrhagic; Signal Transduction; Silver; Silymarin; Single Photon Emission Computed Tomography Computed Tomography; Sirolimus; Sirtuin 1; Skin; Skin Neoplasms; Skin Physiological Phenomena; Sleep Initiation and Maintenance Disorders; Social Class; Social Participation; Social Support; Soil; Soil Microbiology; Solutions; Somatomedins; Soot; Specimen Handling; Spectrophotometry, Ultraviolet; Spectroscopy, Fourier Transform Infrared; Spectrum Analysis; Spinal Fractures; Spirometry; Staphylococcus aureus; STAT1 Transcription Factor; STAT3 Transcription Factor; Streptomyces coelicolor; Stress, Psychological; Stroke; Stroke Volume; Structure-Activity Relationship; Students, Medical; Students, Pharmacy; Substance Abuse Treatment Centers; Sulfur Dioxide; Surface Properties; Surface-Active Agents; Surveys and Questionnaires; Survival Analysis; Survival Rate; Survivin; Sweden; Swine; Swine, Miniature; Sympathetic Nervous System; T-Lymphocytes, Regulatory; Talaromyces; Tandem Mass Spectrometry; tau Proteins; Telemedicine; Telomerase; Telomere; Telomere Homeostasis; Temperature; Terminally Ill; Th1 Cells; Thiamethoxam; Thiazoles; Thiophenes; Thioredoxin Reductase 1; Thrombosis; Thulium; Thyroid Cancer, Papillary; Thyroid Carcinoma, Anaplastic; Thyroid Neoplasms; Time Factors; Titanium; Tomography, Emission-Computed, Single-Photon; Tomography, X-Ray Computed; TOR Serine-Threonine Kinases; Transcription Factor AP-1; Transcription Factors; Transcription, Genetic; Transcriptional Activation; Transcriptome; Transforming Growth Factor beta1; Transistors, Electronic; Translational Research, Biomedical; Transplantation Tolerance; Transplantation, Homologous; Transportation; Treatment Outcome; Tretinoin; Tuberculosis, Multidrug-Resistant; Tuberculosis, Pulmonary; Tubulin Modulators; Tumor Microenvironment; Tumor Necrosis Factor Inhibitors; Tumor Necrosis Factor-alpha; Twins; Ultrasonic Therapy; Ultrasonography; Ultraviolet Rays; United States; Up-Regulation; Uranium; Urethra; Urinary Bladder; Urodynamics; Uromodulin; Uveitis; Vasoconstrictor Agents; Ventricular Function, Left; Vero Cells; Vesicular Transport Proteins; Viral Nonstructural Proteins; Visual Acuity; Vital Capacity; Vitamin D; Vitamin D Deficiency; Vitamin K 2; Vitamins; Volatilization; Voriconazole; Waiting Lists; Waste Disposal, Fluid; Wastewater; Water Pollutants, Chemical; Whole Genome Sequencing; Wine; Wnt Signaling Pathway; Wound Healing; Wounds and Injuries; WW Domains; X-linked Nuclear Protein; X-Ray Diffraction; Xanthines; Xenograft Model Antitumor Assays; YAP-Signaling Proteins; Yogurt; Young Adult; Zebrafish; Zebrafish Proteins; Ziziphus | 2016 |
Phase I clinical trial of combination imatinib and ipilimumab in patients with advanced malignancies.
Topics: Adult; Aged; Antineoplastic Combined Chemotherapy Protocols; Female; Humans; Imatinib Mesylate; Ipilimumab; Male; Middle Aged; Neoplasms; Young Adult | 2017 |
A dose-escalating phase I of imatinib mesylate with fixed dose of metronomic cyclophosphamide in targeted solid tumours.
Topics: Administration, Metronomic; Adult; Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Chordoma; Cyclophosphamide; Disease-Free Survival; Dose-Response Relationship, Drug; Feasibility Studies; Female; Gastrointestinal Neoplasms; Humans; Imatinib Mesylate; Male; Maximum Tolerated Dose; Melanoma; Middle Aged; Molecular Targeted Therapy; Neoplasms; Piperazines; Pyrimidines; Skin Neoplasms | 2013 |
A phase I dose-escalation study of imatinib mesylate (Gleevec/STI571) plus capecitabine (Xeloda) in advanced solid tumors.
Topics: Adult; Aged; Antineoplastic Combined Chemotherapy Protocols; Becaplermin; Benzamides; Capecitabine; Cohort Studies; Deoxycytidine; Drug Administration Schedule; Female; Fluorouracil; Humans; Imatinib Mesylate; Male; Middle Aged; Neoplasms; Neovascularization, Physiologic; Piperazines; Platelet-Derived Growth Factor; Proto-Oncogene Proteins c-sis; Pyrimidines; Skin | 2010 |
Phase I study of gemcitabine, docetaxel and imatinib in refractory and relapsed solid tumors.
Topics: Adult; Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Deoxycytidine; Diffusion Magnetic Resonance Imaging; Docetaxel; Drug Administration Schedule; Drug Interactions; Drug Resistance, Neoplasm; Female; Gemcitabine; Humans; Imatinib Mesylate; Male; Maximum Tolerated Dose; Michigan; Middle Aged; Neoplasm Recurrence, Local; Neoplasms; New Jersey; Perfusion Imaging; Piperazines; Pyrimidines; Taxoids; Time Factors; Treatment Outcome | 2012 |
Cyclophosphamide induces differentiation of Th17 cells in cancer patients.
Topics: Adult; Aged; Animals; Antineoplastic Agents, Alkylating; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Cell Differentiation; Cyclophosphamide; Female; Humans; Imatinib Mesylate; Interleukin-2; Lymphocyte Subsets; Male; Melanoma, Experimental; Mice; Mice, Inbred C57BL; Middle Aged; Neoplasms; Piperazines; Pyrimidines; T-Lymphocytes, Regulatory; Th17 Cells | 2011 |
A phase I trial to determine the safety of imatinib in combination with vatalanib in patients with advanced malignancies.
Topics: Administration, Oral; Adult; Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Biopsy; Drug Administration Schedule; Female; Humans; Imatinib Mesylate; Male; Maximum Tolerated Dose; Middle Aged; Neoplasms; Phthalazines; Piperazines; Protein Kinase Inhibitors; Pyridines; Pyrimidines; Risk Assessment; Tennessee; Time Factors; Treatment Outcome; Young Adult | 2011 |
A Phase I clinical trial of the combination of imatinib and paclitaxel in patients with advanced or metastatic solid tumors refractory to standard therapy.
Topics: Adult; Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Chemotherapy, Adjuvant; Cohort Studies; Disease Progression; Drug Administration Schedule; Drug Resistance, Neoplasm; Female; Humans; Imatinib Mesylate; Male; Maximum Tolerated Dose; Middle Aged; Neoplasms; Neutropenia; Paclitaxel; Piperazines; Pyrimidines; Radiotherapy, Adjuvant; Severity of Illness Index; Treatment Outcome | 2012 |
A phase II study of imatinib mesylate in children with refractory or relapsed solid tumors: a Children's Oncology Group study.
Topics: Adolescent; Adult; Antineoplastic Agents; Benzamides; Bone Neoplasms; Carcinoma, Small Cell; Child; Child, Preschool; Female; Gastrointestinal Stromal Tumors; Humans; Imatinib Mesylate; Male; Neoplasm Recurrence, Local; Neoplasms; Neuroblastoma; Osteosarcoma; Piperazines; Pyrimidines; Sarcoma, Ewing; Sarcoma, Synovial | 2008 |
Phase I and pharmacokinetic study of imatinib mesylate (Gleevec) and gemcitabine in patients with refractory solid tumors.
Topics: Adult; Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Cohort Studies; Deoxycytidine; Drug Resistance, Neoplasm; Female; Gemcitabine; Humans; Imatinib Mesylate; Male; Maximum Tolerated Dose; Middle Aged; Neoplasms; Piperazines; Pyrimidines; Treatment Outcome | 2007 |
Phase I and pharmacokinetic study of imatinib mesylate in patients with advanced malignancies and varying degrees of liver dysfunction: a study by the National Cancer Institute Organ Dysfunction Working Group.
Topics: Administration, Oral; Adult; Aged; Aged, 80 and over; Antineoplastic Agents; Benzamides; Bilirubin; Female; Gastrointestinal Diseases; Humans; Imatinib Mesylate; Liver Diseases; Liver Function Tests; Male; Middle Aged; Neoplasms; Piperazines; Pyrimidines | 2008 |
Phase I and pharmacokinetic study of imatinib mesylate in patients with advanced malignancies and varying degrees of renal dysfunction: a study by the National Cancer Institute Organ Dysfunction Working Group.
Topics: Administration, Oral; Adolescent; Adult; Aged; Antineoplastic Agents; Area Under Curve; Benzamides; Biological Availability; Creatinine; Female; Half-Life; Humans; Hypophosphatemia; Imatinib Mesylate; Kidney Diseases; Kidney Function Tests; Male; Middle Aged; Neoplasms; Piperazines; Pyrimidines | 2008 |
Phase II, open-label study evaluating the activity of imatinib in treating life-threatening malignancies known to be associated with imatinib-sensitive tyrosine kinases.
Topics: Antineoplastic Agents; Benzamides; Hematologic Neoplasms; Humans; Imatinib Mesylate; Kaplan-Meier Estimate; Mutation; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-kit; Pyrimidines; Receptor, Platelet-Derived Growth Factor alpha; Receptor, Platelet-Derived Growth Factor beta | 2008 |
160 other study(ies) available for imatinib mesylate and Benign Neoplasms
Article | Year |
---|---|
Synthesis and apoptosis inducing ability of new anilino substituted pyrimidine sulfonamides as potential anticancer agents.
Topics: Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Cyclin D1; Down-Regulation; G1 Phase; Humans; Neoplasms; NF-kappa B; Pyrimidines; Sulfonamides | 2011 |
Design, synthesis and anti-cancer activity of pyrrole-imidazole polyamides through target-downregulation of c-kit gene expression.
Topics: A549 Cells; Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Down-Regulation; Drug Design; Humans; Imidazoles; Neoplasms; Nylons; Promoter Regions, Genetic; Proto-Oncogene Proteins c-kit; Pyrroles | 2020 |
[Successful treatment with imatinib for a patient with myeloid neoplasms with eosinophilia and abnormalities of PDGFRB due to t (5;14)(q33;q22)].
Topics: Eosinophilia; Humans; Imatinib Mesylate; Male; Middle Aged; Myeloproliferative Disorders; Neoplasms; Receptor, Platelet-Derived Growth Factor beta | 2021 |
New Imatinib Derivatives with Antiproliferative Activity against A549 and K562 Cancer Cells.
Topics: A549 Cells; Antineoplastic Agents; Apoptosis; Cell Proliferation; Cell Survival; Cells, Cultured; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Humans; Imatinib Mesylate; K562 Cells; Neoplasms; Protein Kinase Inhibitors | 2022 |
Tyrosine kinase inhibitors and direct oral anticoagulants: In vitro evaluation of drug-drug interaction mediated by P-glycoprotein.
Topics: Administration, Oral; Anticoagulants; ATP Binding Cassette Transporter, Subfamily B, Member 1; Axitinib; Crizotinib; Dabigatran; Drug Interactions; Humans; Imatinib Mesylate; Neoplasms; Protein Kinase Inhibitors; Pyrazoles; Pyridones; Rivaroxaban | 2022 |
Pharmacological PDGFRβ inhibitors imatinib and sunitinib cause human brain pericyte death in vitro.
Topics: Brain; Humans; Imatinib Mesylate; Neoplasms; Pericytes; Protein Kinase Inhibitors; Receptor, Platelet-Derived Growth Factor beta; Sunitinib | 2022 |
Automated gathering of real-world data from online patient forums can complement pharmacovigilance for rare cancers.
Topics: Drug-Related Side Effects and Adverse Reactions; Humans; Imatinib Mesylate; Neoplasms; Pharmacovigilance; Quality of Life | 2022 |
Imatinib responsive erythrocytosis in a patient with FIP1L1::PDGFRA rearranged myeloid neoplasm with hypereosinophilia - Another manifestation of a stem cell neoplasm.
Topics: Humans; Hypereosinophilic Syndrome; Imatinib Mesylate; Myeloproliferative Disorders; Neoplasms; Oncogene Proteins, Fusion; Polycythemia; Stem Cells | 2022 |
Pseudo-Gaucher cells in a myeloid neoplasm with PDGFRB rearrangement: imitating the imitator.
Topics: Gene Rearrangement; Humans; Imatinib Mesylate; Myeloproliferative Disorders; Neoplasms; Receptor, Platelet-Derived Growth Factor beta | 2022 |
A challenging diagnosis of myeloid/lymphoid neoplasm with eosinophilia and FIP1L1::PDGFRA rearrangement.
Topics: Eosinophilia; Humans; Imatinib Mesylate; mRNA Cleavage and Polyadenylation Factors; Myeloproliferative Disorders; Neoplasms; Oncogene Proteins, Fusion; Receptor, Platelet-Derived Growth Factor alpha | 2023 |
False-Negative Testing for FIP1L1::PDGFRA by Fluorescence in situ Hybridization Is a Frequent Cause of Diagnostic Delay.
Topics: Benzamides; Delayed Diagnosis; Humans; Imatinib Mesylate; In Situ Hybridization, Fluorescence; Myeloproliferative Disorders; Neoplasms; Oncogene Proteins, Fusion; Piperazines; Pyrimidines | 2023 |
Screening and Analysis of Possible Drugs Binding to PDGFRα: A Molecular Modeling Study.
Topics: Humans; Imatinib Mesylate; Models, Molecular; Molecular Docking Simulation; Neoplasms; Quantitative Structure-Activity Relationship; Receptor, Platelet-Derived Growth Factor alpha | 2023 |
A cryptic imatinib-sensitive G3BP1-PDGFRB rearrangement in a myeloid neoplasm with eosinophilia.
Topics: DNA Helicases; Eosinophilia; Humans; Imatinib Mesylate; Male; Neoplasms; Poly-ADP-Ribose Binding Proteins; Receptor, Platelet-Derived Growth Factor beta; RNA Helicases; RNA Recognition Motif Proteins; Young Adult | 2020 |
Progressive multifocal leukoencephalopathy responsive to withdrawal of imatinib in a patient with FIP1L1-PDGFRA positive myeloid neoplasm.
Topics: Humans; Hypereosinophilic Syndrome; Imatinib Mesylate; Leukoencephalopathy, Progressive Multifocal; mRNA Cleavage and Polyadenylation Factors; Myeloproliferative Disorders; Neoplasms; Oncogene Proteins, Fusion; Receptor, Platelet-Derived Growth Factor alpha | 2020 |
Myeloid neoplasm with the abnormality of PDGFRB gene secondary interstitial pneumonia: A case report.
Topics: Aged; Humans; Imatinib Mesylate; Lung Diseases, Interstitial; Male; Myeloproliferative Disorders; Neoplasms; Receptor, Platelet-Derived Growth Factor beta | 2020 |
Mathematical Oncology Comes to the Clinic: A Data-Driven Treatment for Financial Toxicity?
Topics: Humans; Imatinib Mesylate; Medical Oncology; Neoplasms | 2020 |
Cumulative mechanism of several major imatinib-resistant mutations in Abl kinase.
Topics: Adenosine Triphosphate; Amino Acid Sequence; Antineoplastic Agents; Drug Resistance, Neoplasm; Humans; Imatinib Mesylate; Neoplasms; Oncogene Proteins v-abl | 2020 |
Identification of benzimidazole containing 4
Topics: Adenosine Triphosphate; Allosteric Site; Benzimidazoles; Computer Simulation; Drug Design; Drug Screening Assays, Antitumor; Humans; Imatinib Mesylate; Molecular Docking Simulation; Molecular Structure; Neoplasms; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Structure-Activity Relationship | 2021 |
Benzylidene thiazolidinediones: Synthesis, in vitro investigations of antiproliferative mechanisms and in vivo efficacy determination in combination with Imatinib.
Topics: Animals; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Benzylidene Compounds; Cell Line, Tumor; Cell Proliferation; Female; G1 Phase Cell Cycle Checkpoints; Humans; Imatinib Mesylate; Male; Mice, Nude; Molecular Structure; Neoplasms; Structure-Activity Relationship; Thiazolidinediones; Xenograft Model Antitumor Assays | 2020 |
A Cryptic BCR-PDGFRB Fusion Resulting in a Chronic Myeloid Neoplasm With Monocytosis and Eosinophilia: A Novel Finding With Treatment Implications.
Topics: Eosinophilia; Humans; Imatinib Mesylate; Myeloproliferative Disorders; Neoplasms; Oncogene Proteins, Fusion; Receptor, Platelet-Derived Growth Factor beta; Translocation, Genetic | 2020 |
Osteonecrosis of the jaw associated with imatinib therapy in myeloproliferative neoplasm: a rare case report.
Topics: Bisphosphonate-Associated Osteonecrosis of the Jaw; Bone Density Conservation Agents; Diphosphonates; Humans; Imatinib Mesylate; Neoplasms; Osteonecrosis | 2021 |
Optimizing the dose in cancer patients treated with imatinib, sunitinib and pazopanib.
Topics: Adolescent; Adult; Aged; Aged, 80 and over; Antineoplastic Agents; Child; Chromatography, High Pressure Liquid; Drug Monitoring; Feasibility Studies; Female; Humans; Imatinib Mesylate; Indazoles; Indoles; Male; Middle Aged; Neoplasms; Protein Kinase Inhibitors; Pyrimidines; Pyrroles; Retrospective Studies; Sulfonamides; Sunitinib; Tandem Mass Spectrometry; Treatment Outcome; Young Adult | 2017 |
Mesoporous nano-bioglass designed for the release of imatinib and in vitro inhibitory effects on cancer cells.
Topics: Biocompatible Materials; Ceramics; Glass; Humans; Imatinib Mesylate; Neoplasms; Porosity; X-Ray Diffraction | 2017 |
QnAs with Tony Hunter and James Allison.
Topics: Antineoplastic Agents; Humans; Imatinib Mesylate; Neoplasms | 2017 |
Effect of Adherence on Pharmacokinetic/Pharmacodynamic Relationships of Oral Targeted Anticancer Drugs.
Topics: Administration, Oral; Antineoplastic Agents; Bayes Theorem; Dose-Response Relationship, Drug; Drug Monitoring; Humans; Imatinib Mesylate; Medication Adherence; Models, Biological; Molecular Targeted Therapy; Neoplasms | 2018 |
Amplification of F-Actin Disassembly and Cellular Repulsion by Growth Factor Signaling.
Topics: Actins; Animals; Axon Guidance; Biocatalysis; Biomechanical Phenomena; Cell Adhesion Molecules; Cell Proliferation; Drosophila melanogaster; Humans; Imatinib Mesylate; Intercellular Signaling Peptides and Proteins; Mice, Nude; Mixed Function Oxygenases; Models, Biological; Neoplasms; Nerve Tissue Proteins; Oxidation-Reduction; Phosphorylation; Protein Binding; Protein Domains; Proto-Oncogene Proteins c-abl; Semaphorins; Signal Transduction | 2017 |
[Therapeutic drug monitoring - 4th edition of the congress of pharmacology of anticancer drugs].
Topics: Antineoplastic Agents; Bayes Theorem; Bevacizumab; Colorectal Neoplasms; Drug Monitoring; Erlotinib Hydrochloride; Humans; Imatinib Mesylate; Liver; Neoplasms; Phenylurea Compounds; Pyridines | 2017 |
Kinase Inhibitors: The Reality Behind the Success.
Topics: Animals; Carcinogenesis; Humans; Imatinib Mesylate; Medical Oncology; Neoplasms; Protein Kinase Inhibitors | 2017 |
Precision Medicine: Where have we reached and where are we headed?
Topics: Antineoplastic Agents; Evidence-Based Medicine; Forecasting; Humans; Imatinib Mesylate; Neoplasms; Precision Medicine; Rituximab; Trastuzumab | 2017 |
Pleural and pericardial effusions in patient on tyrosine kinase inhibitor.
Topics: Aged; Female; Humans; Imatinib Mesylate; Neoplasms; Pericardial Effusion; Pleural Effusion; Protein Kinase Inhibitors; Protein-Tyrosine Kinases | 2018 |
Regulatory T cell-targeted hybrid nanoparticles combined with immuno-checkpoint blockage for cancer immunotherapy.
Topics: Animals; Antineoplastic Agents; Apoptosis; CD8-Positive T-Lymphocytes; Cell Line, Tumor; Cell Survival; CTLA-4 Antigen; Humans; Imatinib Mesylate; Immunosuppression Therapy; Immunotherapy; Mice, Inbred C57BL; Nanoparticles; Neoplasms; Peptides; Phosphorylation; STAT3 Transcription Factor; STAT5 Transcription Factor; T-Lymphocytes, Cytotoxic; T-Lymphocytes, Regulatory; Tumor Microenvironment | 2018 |
Design, synthesis and 3D QSAR based pharmacophore study of novel imatinib analogs as antitumor-apoptotic agents.
Topics: A549 Cells; Antineoplastic Agents; Apoptosis; Caspase 3; Cell Cycle Checkpoints; Cell Line, Tumor; Drug Design; Drug Screening Assays, Antitumor; Humans; Imatinib Mesylate; Models, Molecular; Neoplasms; Quantitative Structure-Activity Relationship | 2018 |
Out-of-Pocket Spending Not Associated with Oral Oncolytic Survival Benefit.
Topics: Adult; Antineoplastic Agents; Dasatinib; Disease-Free Survival; Drug Prescriptions; Female; Health Expenditures; Humans; Imatinib Mesylate; Lenalidomide; Male; Middle Aged; Neoplasms; Prescription Fees; Retrospective Studies; Survival Analysis; Thalidomide; United States; Young Adult | 2018 |
A pharmacovigilance system for treatment access and medical donation programs: The Max Foundation experience.
Topics: Antineoplastic Agents; Developing Countries; Drug Industry; Health Services Accessibility; Humans; Imatinib Mesylate; Neoplasms; Pharmacovigilance; Program Evaluation | 2018 |
Embracing the complexity in cancer therapy.
Topics: Animals; Antibodies, Blocking; Antibodies, Monoclonal; Antineoplastic Combined Chemotherapy Protocols; CTLA-4 Antigen; Humans; Imatinib Mesylate; Immunotherapy; Neoplasms; Nobel Prize; Physiology; Programmed Cell Death 1 Receptor | 2018 |
Tyrosine Kinase Inhibitor Imatinib Mesylate Alters DMBA-Induced Early Onco/Suppressor Gene Expression with Tissue-Specificity in Mice.
Topics: Animals; Anthracenes; Anticarcinogenic Agents; Gene Expression Regulation, Neoplastic; Humans; Imatinib Mesylate; Mice; Neoplasms; Organ Specificity; Piperidines; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-myc; Proto-Oncogene Proteins p21(ras); Tumor Suppressor Protein p53 | 2019 |
The Time Has Come!
Topics: Humans; Imatinib Mesylate; Neoplasms | 2019 |
"Variant-specific discrepancy when quantitating BCR-ABL1 e13a2 and e14a2 transcripts using the Europe Against Cancer qPCR assay." Is dPCR the key?
Topics: Europe; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Neoplasms; Real-Time Polymerase Chain Reaction | 2019 |
Factors Influencing Imatinib-Induced Hepatotoxicity.
Topics: Adult; Aged; Antineoplastic Agents; Biomarkers, Tumor; Chemical and Drug Induced Liver Injury; Female; Humans; Imatinib Mesylate; Male; Middle Aged; Neoplasms; Odds Ratio; Prognosis; Protein Kinase Inhibitors; Risk Assessment; Risk Factors; Treatment Outcome | 2020 |
Evolutionary variation and adaptation in a conserved protein kinase allosteric network: implications for inhibitor design.
Topics: Allosteric Regulation; Allosteric Site; Archaea; Bacteria; Benzamides; Biocatalysis; Drug Design; Eukaryotic Cells; Evolution, Molecular; Genetic Variation; Humans; Hydrogen Bonding; Hydrophobic and Hydrophilic Interactions; Imatinib Mesylate; Models, Molecular; Neoplasms; Phosphorylation; Piperazines; Protein Kinase Inhibitors; Protein Kinases; Protein Structure, Secondary; Protein Structure, Tertiary; Proto-Oncogene Proteins c-pim-1; Pyrimidines | 2013 |
India's patent case victory rattles Big Pharma.
Topics: Antineoplastic Agents; Benzamides; Drug Industry; Drugs, Generic; Humans; Imatinib Mesylate; India; Legislation, Drug; Neoplasms; Patents as Topic; Piperazines; Pyrimidines | 2013 |
Computational analysis of the binding specificity of Gleevec to Abl, c-Kit, Lck, and c-Src tyrosine kinases.
Topics: Antineoplastic Agents; Benzamides; Binding Sites; CSK Tyrosine-Protein Kinase; Humans; Imatinib Mesylate; Lymphocyte Specific Protein Tyrosine Kinase p56(lck); Molecular Dynamics Simulation; Neoplasms; Piperazines; Protein Binding; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-abl; Proto-Oncogene Proteins c-kit; Pyrimidines; src-Family Kinases; Thermodynamics | 2013 |
Plasma concentrations of tyrosine kinase inhibitors imatinib, erlotinib, and sunitinib in routine clinical outpatient cancer care.
Topics: Aged; Antineoplastic Agents; Benzamides; Body Weight; Chromatography, High Pressure Liquid; Cytochrome P-450 CYP3A Inhibitors; Dose-Response Relationship, Drug; Drug Monitoring; Erlotinib Hydrochloride; Female; Gastric Acid; Half-Life; Histamine H2 Antagonists; Humans; Imatinib Mesylate; Indoles; Male; Middle Aged; Neoplasms; Outpatients; Piperazines; Protein Kinase Inhibitors; Proton Pump Inhibitors; Pyrimidines; Pyrroles; Quinazolines; Sunitinib; Tandem Mass Spectrometry | 2014 |
Janet Rowley (1925-2013).
Topics: Benzamides; Genetics, Medical; History, 20th Century; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Leukemia, Promyelocytic, Acute; Neoplasms; Piperazines; Pyrimidines; Translocation, Genetic; United States | 2014 |
Therapy: This time it's personal.
Topics: Adult; Aged; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Biological Evolution; Biopsy; Disease Progression; DNA Mutational Analysis; DNA, Neoplasm; Drug Delivery Systems; Drug Resistance, Neoplasm; Genes, Tumor Suppressor; Genetics, Medical; Genomics; Humans; Imatinib Mesylate; Immunotherapy; Indoles; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Middle Aged; Nanoparticles; Neoplasms; Pharmacogenetics; Piperazines; Precision Medicine; Proto-Oncogene Proteins B-raf; Pyrimidines; RNA Interference; RNA, Small Interfering; Sulfonamides; Time Factors; Transcriptome; Vemurafenib | 2014 |
Biology: Three known unknowns.
Topics: Antineoplastic Combined Chemotherapy Protocols; Benzamides; Biological Evolution; Drug Resistance, Neoplasm; Genes, Tumor Suppressor; Humans; Imatinib Mesylate; Immunity; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasm Metastasis; Neoplasms; Piperazines; Pyrimidines; Tumor Microenvironment | 2014 |
This time it's personal.
Topics: Antineoplastic Agents; Benzamides; Humans; Imatinib Mesylate; Mutation; Neoplasms; Piperazines; Precision Medicine; Pyrimidines; Transcriptome | 2014 |
Inhibition of c-Abl kinase activity renders cancer cells highly sensitive to mitoxantrone.
Topics: Antineoplastic Agents; Apoptosis; Benzamides; Caspase 3; Caspase 7; Cell Line, Tumor; DNA Damage; Down-Regulation; Drug Resistance, Neoplasm; Fibroblasts; Gene Expression Regulation, Neoplastic; Humans; Imatinib Mesylate; Mitoxantrone; Neoplasms; Oncogene Proteins, Viral; Piperazines; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-abl; Pyrimidines; RNA Interference; S Phase Cell Cycle Checkpoints; Topoisomerase II Inhibitors; Tumor Suppressor Protein p53 | 2014 |
Energetic dissection of Gleevec's selectivity toward human tyrosine kinases.
Topics: Antineoplastic Agents; Benzamides; Cell Line; Humans; Imatinib Mesylate; Kinetics; Neoplasms; Piperazines; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-abl; Pyrimidines; src-Family Kinases; Thermodynamics | 2014 |
Concurrent effects of ABCB1 C3435T, ABCG2 C421A, and XRCC1 Arg194Trp genetic polymorphisms with risk of cancer, clinical output, and response to treatment with imatinib mesylate in patients with chronic myeloid leukemia.
Topics: Adult; ATP Binding Cassette Transporter, Subfamily B; Case-Control Studies; Cytogenetics; DNA-Binding Proteins; Female; Gene Expression Regulation, Leukemic; Genotype; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Male; Middle Aged; Neoplasms; Polymorphism, Restriction Fragment Length; Prevalence; Treatment Outcome; X-ray Repair Cross Complementing Protein 1 | 2016 |
Sos1 Regulates Macrophage Podosome Assembly and Macrophage Invasive Capacity.
Topics: Animals; Cell Movement; Chlorocebus aethiops; COS Cells; Humans; Imatinib Mesylate; Macrophages; Mice; Neoplasm Invasiveness; Neoplasms; Phosphorylation; Podosomes; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-abl; rac GTP-Binding Proteins; SOS1 Protein; src-Family Kinases | 2015 |
Reversing cancer stemness.
Topics: Epithelial-Mesenchymal Transition; Humans; Imatinib Mesylate; Neoplasm Metastasis; Neoplasms; Neoplastic Stem Cells; Receptor, Platelet-Derived Growth Factor alpha | 2015 |
Target prices for mass production of tyrosine kinase inhibitors for global cancer treatment.
Topics: Antineoplastic Agents; Commerce; Drug Industry; Erlotinib Hydrochloride; Global Health; Humans; Imatinib Mesylate; Lapatinib; Neoplasms; Niacinamide; Phenylurea Compounds; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Quinazolines; Sorafenib | 2016 |
Nanoporous capsules of block co-polymers of [(MeO-PEG-NH)-b-(L-GluA)]-PCL for the controlled release of anticancer drugs for therapeutic applications.
Topics: Antineoplastic Agents; Capsules; Cell Survival; Delayed-Action Preparations; Doxorubicin; Glucose Transporter Type 1; HEK293 Cells; Humans; Imatinib Mesylate; K562 Cells; Nanopores; Neoplasms; Particle Size; Polyesters; Polymers | 2016 |
Pathological fracture due to lytic lesion caused by a myeloid neoplasm with FIP1L1-PDGFRA.
Topics: Adult; Eosinophilia; Femur Neck; Fractures, Bone; Humans; Imatinib Mesylate; Male; mRNA Cleavage and Polyadenylation Factors; Myeloproliferative Disorders; Neoplasms; Oncogene Proteins, Fusion; Receptor, Platelet-Derived Growth Factor alpha | 2016 |
Theory and practice of clinical pharmacodynamics in oncology drug development.
Topics: Antineoplastic Agents; Biomarkers, Tumor; Biopsy; Chemistry Techniques, Analytical; Drug Design; Drug Discovery; Humans; Imatinib Mesylate; Molecular Targeted Therapy; Neoplasms; Reproducibility of Results; Specimen Handling | 2016 |
Disease progression in some cancers may be due to low blood levels of targeted therapies.
Topics: Administration, Oral; Antineoplastic Agents; Benzamides; Biological Availability; Dasatinib; Disease Progression; Drug Administration Schedule; Drug Interactions; Drug Resistance, Neoplasm; Gastrointestinal Stromal Tumors; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Patient Compliance; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Thiazoles | 2008 |
XXIII International Association for Comparative Research on Leukemia and Related Diseases Symposium: from molecular pathogenesis to targeted therapy in leukemia and solid tumors.
Topics: Adolescent; Adult; Age Factors; Aged; Animals; Benzamides; Humans; Imatinib Mesylate; Leukemia; Leukemia, Myeloid, Acute; Medical Oncology; Mice; Middle Aged; Myelodysplastic Syndromes; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines; Transcription Factors | 2008 |
[Pharmazie in unserer Zeit 5/2008].
Topics: Antineoplastic Agents; Benzamides; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Tyrosine 3-Monooxygenase | 2008 |
Inhibition of imatinib transport by uremic toxins during renal failure.
Topics: Animals; Antineoplastic Agents; Area Under Curve; Benzamides; Biological Availability; Biological Transport; Humans; Imatinib Mesylate; Kidney Failure, Chronic; Liver Failure; Neoplasms; Organic Anion Transporters; Paclitaxel; Piperazines; Pyrimidines; Xenopus laevis | 2008 |
[Cardiac toxicity and edema].
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Edema, Cardiac; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Prodrugs; Pyrimidines; Risk Factors; Trastuzumab | 2008 |
[Practical approach to hypereosinophilia].
Topics: Benzamides; Eosinophils; Food Hypersensitivity; Glucocorticoids; Hematologic Diseases; Humans; Hypereosinophilic Syndrome; Imatinib Mesylate; Leukocyte Count; Mutation; Neoplasms; Parasitic Diseases; Piperazines; Prednisone; Protein-Tyrosine Kinases; Pulmonary Eosinophilia; Pyrimidines | 2008 |
Comparison of the effects of the kinase inhibitors imatinib, sorafenib, and transforming growth factor-beta receptor inhibitor on extravasation of nanoparticles from neovasculature.
Topics: Animals; Benzamides; Benzenesulfonates; Cell Line, Tumor; Extravasation of Diagnostic and Therapeutic Materials; Humans; Imatinib Mesylate; Mice; Mice, Inbred BALB C; Nanoparticles; Neoplasms; Niacinamide; Phenylurea Compounds; Piperazines; Protein Kinase Inhibitors; Pyrazoles; Pyridines; Pyrimidines; Pyrroles; Receptors, Transforming Growth Factor beta; Signal Transduction; Sorafenib; Vascular Endothelial Growth Factor A | 2009 |
Catastrophic tumour lysis syndrome following single dose of imatinib.
Topics: Antineoplastic Agents; Benzamides; Humans; Imatinib Mesylate; Male; Middle Aged; Neoplasms; Piperazines; Pyrimidines; Tumor Lysis Syndrome | 2009 |
Targeting homologous recombination using imatinib results in enhanced tumor cell chemosensitivity and radiosensitivity.
Topics: Animals; Benzamides; Cell Line, Tumor; Humans; Imatinib Mesylate; Male; Mice; Mice, Inbred BALB C; Mice, Nude; Mitosis; Neoplasms; Piperazines; Pyrimidines; Rad51 Recombinase; Radiation Tolerance; Recombination, Genetic; Xenograft Model Antitumor Assays | 2009 |
Target-driven exploratory study of imatinib mesylate in children with solid malignancies by the Innovative Therapies for Children with Cancer (ITCC) European Consortium.
Topics: Adolescent; Antineoplastic Agents; Benzamides; Child; Child, Preschool; Drug Administration Schedule; Exons; Female; Humans; Imatinib Mesylate; Male; Neoplasms; Piperazines; Positron-Emission Tomography; Proto-Oncogene Proteins c-kit; Pyrimidines; Receptor, Platelet-Derived Growth Factor beta; Treatment Outcome; Young Adult | 2009 |
A Bayesian case study in oncology Phase I combination dose-finding using logistic regression with covariates.
Topics: Antineoplastic Combined Chemotherapy Protocols; Bayes Theorem; Benzamides; Clinical Trials, Phase I as Topic; Cohort Studies; Dose-Response Relationship, Drug; Drug Administration Schedule; Humans; Imatinib Mesylate; Logistic Models; Maximum Tolerated Dose; Multivariate Analysis; Neoplasms; Piperazines; Probability; Pyrimidines | 2009 |
Promises and pitfalls of oral cancer chemotherapy.
Topics: Administration, Oral; Antineoplastic Agents; Benzamides; Drug Monitoring; Imatinib Mesylate; Medication Adherence; Neoplasms; Patient Education as Topic; Physician-Patient Relations; Piperazines; Pyrimidines | 2009 |
The therapeutic benefits of heme oxygenase (HO-1) inhibition in the management of systemic malignancies besides hepatocellular carcinomas.
Topics: Antineoplastic Agents; Benzamides; Carcinoma, Hepatocellular; Enzyme Inhibitors; Heme Oxygenase-1; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Liver Neoplasms; Nasopharyngeal Neoplasms; Neoplasms; Piperazines; Protoporphyrins; Pyrimidines; Sarcoma, Kaposi | 2009 |
Quality of reporting of serious adverse drug events to an institutional review board: a case study with the novel cancer agent, imatinib mesylate.
Topics: Adverse Drug Reaction Reporting Systems; Antineoplastic Agents; Benzamides; Clinical Trials as Topic; Drug Utilization Review; Fractures, Bone; Heart Failure; Humans; Imatinib Mesylate; Infections; Neoplasms; Piperazines; Product Surveillance, Postmarketing; Professional Staff Committees; Pulmonary Edema; Pyrimidines; Time Factors | 2009 |
Therapeutic Drug Monitoring of the new targeted anticancer agents imatinib, nilotinib, dasatinib, sunitinib, sorafenib and lapatinib by LC tandem mass spectrometry.
Topics: Antineoplastic Agents; Benzamides; Benzenesulfonates; Chromatography, Liquid; Dasatinib; Drug Monitoring; Humans; Imatinib Mesylate; Indoles; Lapatinib; Neoplasms; Niacinamide; Phenylurea Compounds; Piperazines; Pyridines; Pyrimidines; Pyrroles; Quinazolines; Sorafenib; Sunitinib; Tandem Mass Spectrometry; Thiazoles | 2009 |
Perspectives on the development of imatinib and the future of cancer research.
Topics: Awards and Prizes; Benzamides; Clinical Trials as Topic; History, 20th Century; History, 21st Century; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Research; United States | 2009 |
Attacking cancer at its foundation.
Topics: Academic Medical Centers; Awards and Prizes; Benzamides; Clinical Trials as Topic; Drug Design; Drug Discovery; Drug Industry; History, 20th Century; History, 21st Century; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein Kinase Inhibitors; Pyrimidines; United States | 2009 |
Shifting paradigms: the seeds of oncogene addiction.
Topics: Awards and Prizes; Benzamides; Clinical Trials as Topic; DNA, Complementary; Drug Resistance; History, 20th Century; History, 21st Century; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Mutation; Neoplasms; Oncogenes; Piperazines; Protein Kinase Inhibitors; Protein Structure, Tertiary; Pyrimidines; Sequence Analysis, DNA; United States | 2009 |
Imatinib and nilotinib reverse multidrug resistance in cancer cells by inhibiting the efflux activity of the MRP7 (ABCC10).
Topics: Antineoplastic Agents; Benzamides; Cell Line; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Gene Expression Regulation, Neoplastic; Humans; Imatinib Mesylate; Models, Chemical; Multidrug Resistance-Associated Proteins; Neoplasms; Paclitaxel; Piperazines; Pyrimidines; Tetrazolium Salts; Thiazoles | 2009 |
Anticipating drug resistance in the MAP kinase pathway.
Topics: Adenosine Triphosphate; Animals; Antineoplastic Agents; Benzamides; Catalytic Domain; Drug Design; Drug Resistance, Neoplasm; Enzyme Activation; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; MAP Kinase Signaling System; Neoplasms; Phosphatidylinositol 3-Kinases; Piperazines; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Pyrimidines | 2010 |
Tyrosine kinase inhibitor-induced macrocytosis.
Topics: Anemia, Macrocytic; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Benzenesulfonates; Erlotinib Hydrochloride; Humans; Imatinib Mesylate; Indoles; Neoplasm Staging; Neoplasms; Niacinamide; Phenylurea Compounds; Piperazines; Prognosis; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-kit; Pyridines; Pyrimidines; Pyrroles; Quinazolines; Retrospective Studies; Sorafenib; Sunitinib; Survival Rate | 2009 |
Inhibitors of the Abl kinase directed at either the ATP- or myristate-binding site.
Topics: Adenosine Triphosphate; Allosteric Regulation; Benzamides; Crystallography, X-Ray; Drug Resistance, Neoplasm; Humans; Imatinib Mesylate; Mutation, Missense; Myristic Acid; Neoplasms; Nuclear Magnetic Resonance, Biomolecular; Piperazines; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-abl; Pyrimidines | 2010 |
Molecular dynamics simulations show that conformational selection governs the binding preferences of imatinib for several tyrosine kinases.
Topics: Animals; Benzamides; Chickens; Computer Simulation; Humans; Imatinib Mesylate; Models, Molecular; Neoplasms; Piperazines; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Secondary; Protein-Tyrosine Kinases; Pyrimidines | 2010 |
Counterpoint: Data first.
Topics: Antineoplastic Agents; Benzamides; Drug Discovery; Fusion Proteins, bcr-abl; Genome, Human; Genomics; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Piperazines; Precision Medicine; Pyrimidines | 2010 |
Imatinib (Gleevec) as a paradigm of targeted cancer therapies.
Topics: Antineoplastic Agents; Benzamides; Biomedical Research; History, 19th Century; History, 20th Century; History, 21st Century; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Piperazines; Pyrimidines | 2010 |
Preclinical evaluation of nilotinib efficacy in an imatinib-resistant KIT-driven tumor model.
Topics: Amino Acid Substitution; Animals; Antineoplastic Agents; Benzamides; Cell Line, Tumor; Disease Models, Animal; Drug Evaluation, Preclinical; Drug Resistance, Neoplasm; Humans; Imatinib Mesylate; Mice; Mice, Inbred DBA; Neoplasm Transplantation; Neoplasms; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines; Transplantation, Isogeneic; Treatment Outcome | 2010 |
Effect of the tyrosine kinase inhibitors (sunitinib, sorafenib, dasatinib, and imatinib) on blood glucose levels in diabetic and nondiabetic patients in general clinical practice.
Topics: Aged; Antineoplastic Agents; Benzamides; Benzenesulfonates; Blood Glucose; Dasatinib; Diabetes Mellitus; Female; Humans; Hypoglycemia; Hypoglycemic Agents; Imatinib Mesylate; Indoles; Linear Models; Male; Middle Aged; Neoplasms; Niacinamide; Pennsylvania; Phenylurea Compounds; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyridines; Pyrimidines; Pyrroles; Retrospective Studies; Risk Assessment; Risk Factors; Sorafenib; Sunitinib; Thiazoles; Time Factors; Treatment Outcome | 2011 |
Targeting targeted therapies.
Topics: Antibodies, Monoclonal; Antigens, Neoplasm; Benzamides; Cancer Vaccines; Clinical Trials as Topic; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines | 2010 |
Who is in charge of assessing therapeutic drug monitoring? The case of imatinib.
Topics: Antineoplastic Agents; Benzamides; Drug Industry; Drug Monitoring; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein Kinase Inhibitors; Pyrimidines | 2011 |
16-Hydroxycleroda-3,13-dien-15,16-olide deregulates PI3K and Aurora B activities that involve in cancer cell apoptosis.
Topics: Antineoplastic Agents; Apoptosis; Aurora Kinase B; Aurora Kinases; Benzamides; Cell Cycle; Cell Line, Tumor; Cell Survival; Diterpenes; DNA Damage; Drug Resistance, Neoplasm; Gene Expression Regulation, Neoplastic; Gene Silencing; Humans; Imatinib Mesylate; Neoplasms; Phosphoinositide-3 Kinase Inhibitors; Piperazines; Protein Serine-Threonine Kinases; Pyrimidines; Signal Transduction | 2011 |
NPB001-05 inhibits Bcr-Abl kinase leading to apoptosis of imatinib-resistant cells.
Topics: Apoptosis; Benzamides; Cell Cycle; Cell Line, Tumor; Drug Resistance, Neoplasm; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Mutation; Neoplasms; Phosphorylation; Piperazines; Plant Extracts; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines | 2011 |
From genome to drugs: where do we stand?
Topics: Antineoplastic Agents; Benzamides; Drug Approval; Drug Design; Drug Industry; Drug Resistance, Neoplasm; Genome, Human; Genomics; Humans; Imatinib Mesylate; Indoles; Molecular Targeted Therapy; Mutation; Neoplasm Proteins; Neoplasms; Orphan Drug Production; Piperazines; Protein Kinase Inhibitors; Proto-Oncogene Proteins B-raf; Pyrimidines; Rare Diseases; Sulfonamides; United States; United States Food and Drug Administration; Vemurafenib | 2011 |
ASCO 2011: broadening the horizons of cancer research.
Topics: Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Cell Proliferation; Disease Models, Animal; Global Health; Humans; Imatinib Mesylate; Medical Oncology; Mice; Neoplasms; Neoplastic Stem Cells; Piperazines; Pyrimidines; Receptor, ErbB-2; Research; Societies, Medical; Trastuzumab; United States; United States Food and Drug Administration | 2011 |
[Therapeutic adherence to oral cancer therapy and interdisciplinary management].
Topics: Adenocarcinoma; Administration, Oral; Aged; Algorithms; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Capecitabine; Cecal Neoplasms; Deoxycytidine; Female; Fluorouracil; Gastrointestinal Stromal Tumors; Humans; Imatinib Mesylate; Interdisciplinary Communication; Male; Medication Adherence; Neoplasms; Outpatients; Patient-Centered Care; Pharmacists; Physician's Role; Pilot Projects; Piperazines; Prospective Studies; Pyrimidines; Switzerland; Time Factors; Treatment Outcome | 2011 |
miRNAs in the spotlight: Understanding cancer gene dependency.
Topics: Animals; Antineoplastic Agents; Benzamides; Drug Delivery Systems; Gene Expression Regulation, Neoplastic; Genes, Neoplasm; Humans; Imatinib Mesylate; Mice; MicroRNAs; Mutation; Neoplasms; Piperazines; Pyrimidines | 2011 |
Use and costs of oral anticancer agents in the Netherlands in the period 2000-2008.
Topics: Administration, Oral; Antineoplastic Agents; Benzamides; Capecitabine; Deoxycytidine; Fluorouracil; Humans; Imatinib Mesylate; Neoplasms; Netherlands; Pharmacies; Piperazines; Protein-Tyrosine Kinases; Pyrimidines | 2012 |
Serum creatine kinase increase in patients treated with tyrosine kinase inhibitors for solid tumors.
Topics: Adult; Aged; Aged, 80 and over; Benzamides; Creatine Kinase; Female; Gastrointestinal Stromal Tumors; Humans; Imatinib Mesylate; Male; Middle Aged; Neoplasms; Piperazines; Prospective Studies; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines | 2012 |
Lab reports and cat scans: can veterinary oncology guide our way to new treatments for human cancers?
Topics: Animals; Antineoplastic Agents; Benzamides; Breast Neoplasms; Cats; Disease Models, Animal; Dogs; Female; Humans; Imatinib Mesylate; Indoles; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Mast-Cell Sarcoma; Neoplasms; Piperazines; Piperidines; Protein Kinase Inhibitors; Pyridines; Pyrimidines; Pyrroles; Thiazoles; Transcriptome | 2012 |
Assessment of tracer 99mTc(V)-DMSA uptake as a measure of tumor cell proliferation in vitro.
Topics: Benzamides; Biomarkers; Cell Line, Tumor; Cell Proliferation; Fluorodeoxyglucose F18; Gene Expression Regulation, Neoplastic; Humans; Imatinib Mesylate; MCF-7 Cells; Neoplasms; Piperazines; Pyrimidines; Radiopharmaceuticals; S Phase; Technetium Tc 99m Dimercaptosuccinic Acid | 2013 |
Changes and challenges--the world post-Gleevec (Glivec).
Topics: Animals; Antineoplastic Agents; Benzamides; Drug Delivery Systems; Enzyme Inhibitors; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Pyrimidines | 2002 |
[Targeted treatment of cancers with imatinib mesylate (STI571, Gleevec): results of Asco 2002].
Topics: Antineoplastic Agents; Benzamides; Dermatofibrosarcoma; Florida; Gastrointestinal Neoplasms; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-kit; Pyrimidines; Sarcoma; Skin Neoplasms | 2002 |
Cancer drugs. Smart weapons prove tough to design.
Topics: Advisory Committees; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Carcinoma, Non-Small-Cell Lung; Clinical Trials as Topic; Drug Approval; Drug Industry; Epidermal Growth Factor; Erlotinib Hydrochloride; Gefitinib; Humans; Imatinib Mesylate; Lung Neoplasms; Neoplasms; Patient Selection; Piperazines; Pyrimidines; Quinazolines; United States; United States Food and Drug Administration | 2002 |
Synthetic lethality: killing cancer with cancer.
Topics: Animals; Antineoplastic Agents; Benzamides; Benzoquinones; Cell Cycle Proteins; DNA-Binding Proteins; E2F Transcription Factors; Gefitinib; Genes, Tumor Suppressor; HSP90 Heat-Shock Proteins; Humans; Imatinib Mesylate; Indoles; Lactams, Macrocyclic; Mutation; Neoplasms; Phosphoric Monoester Hydrolases; Piperazines; PTEN Phosphohydrolase; Pyrimidines; Pyrroles; Quinazolines; Rifabutin; Signal Transduction; Sirolimus; Transcription Factors; Tumor Suppressor Proteins | 2002 |
[The new mechanisms and reversal of drug resistance].
Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Benzamides; Drug Resistance, Neoplasm; Humans; Imatinib Mesylate; Neoplasms; Oligonucleotide Array Sequence Analysis; Pharmacogenetics; Piperazines; Pyrimidines | 2003 |
A new era in cancer therapeutics?
Topics: Antineoplastic Agents; Benzamides; Enzyme Inhibitors; Humans; Imatinib Mesylate; Neoplasms; Pharmacogenetics; Piperazines; Pyrimidines | 2003 |
The hypereosinophilic syndrome and the biology of cancer.
Topics: Benzamides; Chromosome Deletion; Enzyme Inhibitors; Eosinophilia; Eosinophils; Humans; Hypereosinophilic Syndrome; Imatinib Mesylate; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines; T-Lymphocytes; Translocation, Genetic | 2003 |
Drug maker's vow to donate cancer medicine falls short.
Topics: Antineoplastic Agents; Benzamides; Developing Countries; Drug Industry; Humans; Imatinib Mesylate; India; Internationality; Neoplasms; Piperazines; Pyrimidines; United States | 2003 |
Combinations of targeted therapies take aim at multiple pathways.
Topics: Animals; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Boronic Acids; Bortezomib; Clinical Trials as Topic; Gefitinib; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Pyrazines; Pyrimidines; Quinazolines; Research Design | 2003 |
Targeted therapy in cancer and transgenic animal model.
Topics: Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Breast Neoplasms; Chemoprevention; Disease Models, Animal; Genes, erbB-2; Humans; Imatinib Mesylate; Mice; Mice, Transgenic; Neoplasms; Piperazines; Pyrimidines; Signal Transduction; Trastuzumab | 2003 |
[New reversing agents that target membrane transporters].
Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Benzamides; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Imatinib Mesylate; Membrane Glycoproteins; Membrane Transport Proteins; Neoplasms; Piperazines; Pyrimidines | 2004 |
Advances in molecular targets and cancer therapeutics.
Topics: Antineoplastic Agents; Benzamides; Drug Delivery Systems; Drug Design; Genomics; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Proteomics; Pyrimidines; Technology, Pharmaceutical | 2004 |
Tyrosine kinase inhibitor STI-571: the new wonder drug of cancer therapy.
Topics: Antineoplastic Agents; Benzamides; Cell Transformation, Neoplastic; Chemoprevention; Colorectal Neoplasms; Drug Design; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines | 2004 |
Development and validation of a simple liquid chromatographic method with ultraviolet detection for the determination of imatinib in biological samples.
Topics: Administration, Oral; Antineoplastic Agents; Benzamides; Calibration; Chromatography, High Pressure Liquid; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Pyrimidines; Sensitivity and Specificity; Spectrophotometry, Ultraviolet | 2004 |
A widening prospect: Imatinib and novel applications of targeted therapy.
Topics: Antineoplastic Agents; Benzamides; Enzyme Inhibitors; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines; Receptors, Platelet-Derived Growth Factor; Signal Transduction | 2004 |
Protein kinase C theta is highly expressed in gastrointestinal stromal tumors but not in other mesenchymal neoplasias.
Topics: Benzamides; Blotting, Western; Gastrointestinal Neoplasms; Gene Expression Regulation; Humans; Imatinib Mesylate; Immunohistochemistry; Isoenzymes; Mesoderm; Neoplasms; Oligonucleotide Array Sequence Analysis; Piperazines; Protein Isoforms; Protein Kinase C; Protein Kinase C-theta; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-kit; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; Sarcoma; Stromal Cells; T-Lymphocytes; Transcription, Genetic | 2004 |
Imatinib: paradigm or anomaly?
Topics: Antineoplastic Agents; Benzamides; Clinical Trials as Topic; Drug Design; Early Diagnosis; Gefitinib; Humans; Imatinib Mesylate; Mutation; Neoplasms; Piperazines; Pyrimidines; Quinazolines; Receptors, Growth Factor; Signal Transduction | 2004 |
Other malignant neoplasms in patients with gastrointestinal stromal tumors (GIST).
Topics: Adult; Antineoplastic Agents; Benzamides; Female; Gastrointestinal Neoplasms; Humans; Imatinib Mesylate; Male; Middle Aged; Neoplasms; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines | 2004 |
Gold standard or wrong standard?
Topics: Antineoplastic Agents; Benzamides; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Pyrimidines; Randomized Controlled Trials as Topic; Survival Rate; Treatment Outcome | 2004 |
Imatinib mesylate (STI-571) enhances antigen-presenting cell function and overcomes tumor-induced CD4+ T-cell tolerance.
Topics: Amino Acid Sequence; Animals; Antigen-Presenting Cells; Antineoplastic Agents; Benzamides; Bone Marrow Cells; CD4-Positive T-Lymphocytes; Dendritic Cells; Imatinib Mesylate; Immune Tolerance; Lymphoma; Macrophages; Mice; Mice, Inbred BALB C; Molecular Sequence Data; Neoplasms; Ovalbumin; Peptide Fragments; Piperazines; Pyrimidines | 2005 |
[Target-oriented tumor therapy -- proof of the principle].
Topics: Antibodies, Monoclonal; Antineoplastic Agents; Benzamides; Drug Delivery Systems; Gastrointestinal Neoplasms; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Piperazines; Pyrimidines | 2004 |
Prevalence of KIT expression in human tumors.
Topics: Antineoplastic Agents; Benzamides; Gastrointestinal Stromal Tumors; Gene Expression Profiling; Humans; Imatinib Mesylate; Immunohistochemistry; Neoplasms; Oligonucleotide Array Sequence Analysis; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines | 2004 |
New drugs in cancer therapy, National Tumor Institute, Naples, 17-18 June 2004.
Topics: Angiogenesis Inhibitors; Antineoplastic Agents; Benzamides; Clinical Trials as Topic; Drug Resistance, Neoplasm; Drugs, Investigational; Genes, erbB; Imatinib Mesylate; Neoplasms; Piperazines; Pyrimidines; Signal Transduction | 2005 |
[Targeted drugs in radiation therapy].
Topics: Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Cetuximab; Clinical Trials, Phase I as Topic; Clinical Trials, Phase III as Topic; Combined Modality Therapy; ErbB Receptors; Gefitinib; Humans; Imatinib Mesylate; Mice; Mice, Nude; Mutation; Neoplasms; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Quinazolines; Radiation-Sensitizing Agents; Randomized Controlled Trials as Topic; Trastuzumab; Tumor Cells, Cultured | 2004 |
A functional approach to questions about life, death, and phosphorylation.
Topics: Antineoplastic Agents; Apoptosis; Benzamides; Cell Survival; Drug Synergism; HeLa Cells; Humans; Imatinib Mesylate; Neoplasms; Phosphoprotein Phosphatases; Phosphorylation; Piperazines; Protein Kinase Inhibitors; Protein Kinases; Pyrimidines; RNA Interference; RNA, Small Interfering | 2005 |
Chronic imatinib mesylate exposure leads to reduced intracellular drug accumulation by induction of the ABCG2 (BCRP) and ABCB1 (MDR1) drug transport pumps.
Topics: Administration, Oral; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Benzamides; Biological Transport; Chlorocebus aethiops; Constitutive Androstane Receptor; COS Cells; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Gene Expression; Humans; Imatinib Mesylate; Membrane Transport Proteins; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Neoplasms; Piperazines; Pregnane X Receptor; Protein-Tyrosine Kinases; Pyrimidines; Receptors, Cytoplasmic and Nuclear; Receptors, Steroid; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Transcription Factors; Transcriptional Activation; Tumor Cells, Cultured | 2005 |
Phosphorylations of DEAD box p68 RNA helicase are associated with cancer development and cell proliferation.
Topics: Antineoplastic Agents; Antineoplastic Agents, Phytogenic; Benzamides; Blotting, Western; Caco-2 Cells; Cell Line, Tumor; Cell Proliferation; Etoposide; HeLa Cells; Humans; Imatinib Mesylate; K562 Cells; Neoplasms; Paclitaxel; Phosphorus Radioisotopes; Phosphorylation; Piperazines; Precipitin Tests; Pyrimidines; RNA Helicases; RNA Interference; Stilbenes; Tumor Necrosis Factor-alpha | 2005 |
Imatinib: the narrow line between immune tolerance and activation.
Topics: Adjuvants, Immunologic; Antineoplastic Agents; Benzamides; Humans; Imatinib Mesylate; Immune Tolerance; Immunosuppressive Agents; Neoplasms; Piperazines; Pyrimidines | 2005 |
FMS receptor for M-CSF (CSF-1) is sensitive to the kinase inhibitor imatinib and mutation of Asp-802 to Val confers resistance.
Topics: Animals; Antineoplastic Agents; Aspartic Acid; Benzamides; Disease Progression; Dose-Response Relationship, Drug; Down-Regulation; Drug Resistance, Neoplasm; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Inflammation; Inhibitory Concentration 50; Macrophage Colony-Stimulating Factor; Mice; Mutation; Neoplasms; Oncogene Protein v-cbl; Phosphorylation; Piperazines; Protein Structure, Tertiary; Proto-Oncogene Proteins c-crk; Proto-Oncogene Proteins c-kit; Pyrimidines; Rats; Receptor Protein-Tyrosine Kinases; Receptor, Macrophage Colony-Stimulating Factor; Signal Transduction; Time Factors; Valine | 2006 |
Drug discovery: playing dirty.
Topics: Animals; Benzamides; Cardiovascular Diseases; Clinical Trials as Topic; Clozapine; Depression; Drug Approval; Drug Design; Drug Evaluation, Preclinical; Drug Industry; Gefitinib; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Pyrimidines; Quinazolines; Sensitivity and Specificity; Substrate Specificity; Therapeutics; United States; United States Food and Drug Administration | 2005 |
Active (p)CrkL is overexpressed in human malignancies: potential role as a surrogate parameter for therapeutic tyrosine kinase inhibition.
Topics: Adaptor Proteins, Signal Transducing; Benzamides; Biomarkers, Tumor; Blotting, Western; Cell Line, Tumor; Enzyme Activation; Female; Humans; Imatinib Mesylate; Immunohistochemistry; Male; Neoplasms; Nuclear Proteins; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Up-Regulation | 2006 |
[Current status and prospect of neoplasm targeted therapy].
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Cetuximab; Drug Delivery Systems; Drug Design; Erlotinib Hydrochloride; Gefitinib; Humans; Imatinib Mesylate; Immunologic Factors; Neoplasms; Palliative Care; Piperazines; Pyrimidines; Quinazolines; Signal Transduction | 2005 |
Selective kinase inhibition with daily imatinib intensifies toxicity of chemotherapy in patients with solid tumours.
Topics: Adult; Aged; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Cohort Studies; Deoxycytidine; Doxorubicin; Female; Gemcitabine; Humans; Imatinib Mesylate; Male; Maximum Tolerated Dose; Middle Aged; Neoplasms; Piperazines; Protein Kinase Inhibitors; Pyrimidines | 2006 |
Imatinib (Gleevec, Glivec) tumour tissue analysis by measurement of sediment and by liquid chromatography tandem mass spectrometry.
Topics: Animals; Antineoplastic Agents; Benzamides; Calibration; Chromatography, High Pressure Liquid; Erythrocytes; Humans; Imatinib Mesylate; Mass Spectrometry; Molecular Structure; Neoplasms; Piperazines; Pyrimidines | 2006 |
TGFbeta in cancer and other disease - AACR special conference in cancer research.
Topics: Animals; Antibodies, Monoclonal; Benzamides; Humans; Imatinib Mesylate; Neoplasms; Oligonucleotides, Antisense; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Transforming Growth Factor beta; Transforming Growth Factor beta2 | 2006 |
[The diagnostic and predictive role of kit (CD117)].
Topics: Antineoplastic Agents; Benzamides; Female; Gastrointestinal Stromal Tumors; Genetic Markers; Humans; Imatinib Mesylate; Immunohistochemistry; Male; Mutation; Neoplasms; Piperazines; Predictive Value of Tests; Prognosis; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-kit; Pyrimidines; Sensitivity and Specificity; Signal Transduction | 2006 |
Imatinib mesylate--uncovering a fast track to adaptive immunity.
Topics: Adoptive Transfer; Animals; Benzamides; Cytotoxicity, Immunologic; Dendritic Cells; Imatinib Mesylate; Interferon-gamma; Interferons; Killer Cells, Natural; Mice; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines | 2006 |
Targeting tyrosine kinases in cancer: the second wave.
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Drug Resistance, Neoplasm; ErbB Receptors; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Mutation; Neoplasms; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-kit; Pyrimidines; Receptor, ErbB-2; Receptors, Platelet-Derived Growth Factor; Trastuzumab | 2006 |
Ongoing challenges of a global international patient assistance program.
Topics: Administration, Oral; Antineoplastic Agents; Benzamides; Developing Countries; Gastrointestinal Stromal Tumors; Global Health; Health Services Accessibility; Humans; Imatinib Mesylate; International Cooperation; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Piperazines; Program Development; Program Evaluation; Public Health; Pyrimidines; Thailand | 2006 |
Targeted cancer therapeutics: the heartbreak of success.
Topics: Antibodies, Monoclonal; Antineoplastic Agents; Benzamides; Drug Delivery Systems; Enzyme Inhibitors; Heart Failure; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Models, Biological; Neoplasms; Piperazines; Pyrimidines; src-Family Kinases; Ventricular Dysfunction, Left | 2006 |
Antivascular therapy of cancer metastasis.
Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Bone Neoplasms; Disease Progression; Growth Substances; Humans; Imatinib Mesylate; Male; Mice; Mice, Nude; Neoplasm Metastasis; Neoplasms; Paclitaxel; Piperazines; Platelet-Derived Growth Factor; Prostatic Neoplasms; Pyrimidines; Receptors, Growth Factor; Receptors, Platelet-Derived Growth Factor | 2006 |
Evaluation of the function of human invariant NKT cells from cancer patients using alpha-galactosylceramide-loaded murine dendritic cells.
Topics: Animals; Benzamides; Cell Differentiation; Cells, Cultured; Coculture Techniques; Dendritic Cells; Galactosylceramides; Humans; Imatinib Mesylate; Interferon-gamma; Interleukin-12; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lymphocyte Activation; Mice; Monocytes; Neoplasms; Piperazines; Pyrimidines; T-Lymphocytes, Regulatory | 2006 |
Pharmacy benefit spending on oral chemotherapy drugs.
Topics: Administration, Oral; Ambulatory Care; Antineoplastic Agents; Benzamides; Benzenesulfonates; Capecitabine; Dasatinib; Deoxycytidine; Drug Costs; Employer Health Costs; Erlotinib Hydrochloride; Fluorouracil; Gefitinib; Health Benefit Plans, Employee; Humans; Imatinib Mesylate; Indoles; Insurance, Pharmaceutical Services; Lenalidomide; Neoplasms; Niacinamide; Phenylurea Compounds; Piperazines; Prescription Fees; Pyridines; Pyrimidines; Pyrroles; Quinazolines; Sorafenib; Sunitinib; Thalidomide; Thiazoles; United States | 2006 |
In vitro and in vivo activity of SKI-606, a novel Src-Abl inhibitor, against imatinib-resistant Bcr-Abl+ neoplastic cells.
Topics: Aniline Compounds; Animals; Benzamides; Cell Line; Cell Line, Tumor; Cell Proliferation; Dasatinib; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Fusion Proteins, bcr-abl; Genotype; Humans; Imatinib Mesylate; K562 Cells; Mice; Mice, Nude; Models, Molecular; Mutation; Neoplasms; Nitriles; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Quinolines; src-Family Kinases; Survival Analysis; Thiazoles; U937 Cells; Xenograft Model Antitumor Assays | 2006 |
EORTC-NCI-AACR - 18th Symposium - Molecular Targets and Cancer Therapeutics. Pediatric drugs, biomarkers and new therapies.
Topics: Angiogenesis Inhibitors; Antibodies, Monoclonal; Antineoplastic Agents; Benzamides; Biomarkers, Tumor; Child; Drug Design; Humans; Imatinib Mesylate; Neoplasm Metastasis; Neoplasms; Piperazines; Pyrimidines | 2007 |
In reply to 'Cardiotoxicity of the cancer therapeutic agent imatinib mesylate'.
Topics: Antineoplastic Agents; Benzamides; Heart Failure; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Piperazines; Pyrimidines | 2007 |
In reply to 'Cardiotoxicity of the cancer therapeutic agent imatinib mesylate'.
Topics: Antineoplastic Agents; Benzamides; Heart Failure; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Piperazines; Pyrimidines | 2007 |
In reply to 'Cardiotoxicity of the cancer therapeutic agent imatinib mesylate'.
Topics: Antineoplastic Agents; Benzamides; Heart Failure; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Piperazines; Pyrimidines | 2007 |
In reply to 'Cardiotoxicity of the cancer therapeutic agent imatinib mesylate'.
Topics: Antineoplastic Agents; Benzamides; Heart Failure; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Piperazines; Pyrimidines | 2007 |
New insights into oncogene addiction found.
Topics: Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Apoptosis; Benzamides; Cyclin D1; Erlotinib Hydrochloride; Gefitinib; Gene Expression Regulation, Neoplastic; Gene Silencing; Genes, bcl-1; Humans; Imatinib Mesylate; Mutation; Neoplasms; Oncogenes; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Quinazolines; Signal Transduction; Trastuzumab | 2007 |
Imaging the modulation of adenoviral kinetics and biodistribution for cancer gene therapy.
Topics: Adenoviridae; Animals; Antineoplastic Agents; Benzamides; Cell Line, Tumor; Clodronic Acid; Genetic Therapy; Genetic Vectors; Humans; Imatinib Mesylate; Immunohistochemistry; Kinetics; Liver; Luciferases; Luminescent Measurements; Male; Mice; Mice, SCID; Microscopy, Fluorescence; Neoplasms; Phosphorylation; Piperazines; Pyrimidines; Receptor, Platelet-Derived Growth Factor beta; Recombinant Fusion Proteins; Reverse Transcriptase Polymerase Chain Reaction; Time Factors; Tissue Distribution | 2007 |
Cancer therapy: new drugs are emerging based on molecular targeting but still many challenges.
Topics: Antineoplastic Agents; Benzamides; Humans; Imatinib Mesylate; Neoplasms; Oncogenes; Piperazines; Pyrimidines; TNF-Related Apoptosis-Inducing Ligand | 2007 |
Unexplored pharmacokinetic opportunities with microdosing in oncology.
Topics: Antineoplastic Agents; Benzamides; Dose-Response Relationship, Drug; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Pyrimidines | 2007 |
Progressive thoughts about progressive disease.
Topics: Antineoplastic Agents; Benzamides; Clone Cells; Disease Progression; Drug Resistance, Neoplasm; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Pyrimidines | 2007 |
In vitro biotransformation of imatinib by the tumor expressed CYP1A1 and CYP1B1.
Topics: Antineoplastic Agents; Aryl Hydrocarbon Hydroxylases; Benzamides; Biotransformation; Cytochrome P-450 CYP1A1; Cytochrome P-450 CYP1B1; Humans; Imatinib Mesylate; Kinetics; Mass Spectrometry; Neoplasms; Piperazines; Proto-Oncogene Proteins c-abl; Pyrimidines | 2008 |
Distinct angiogenic mediators are required for basic fibroblast growth factor- and vascular endothelial growth factor-induced angiogenesis: the role of cytoplasmic tyrosine kinase c-Abl in tumor angiogenesis.
Topics: Angiogenesis Inducing Agents; Animals; Benzamides; Cell Line; Cell Proliferation; Cytoplasm; Cytoskeleton; Endothelial Cells; Enzyme Activation; Fibroblast Growth Factor 2; Humans; Imatinib Mesylate; Mice; Mice, SCID; Models, Biological; Mutant Proteins; Neoplasms; Neovascularization, Pathologic; Piperazines; Proto-Oncogene Proteins c-abl; Pyrimidines; Signal Transduction; Vascular Endothelial Growth Factor A | 2008 |
Telomerase inhibition combined with other chemotherapeutic reagents to enhance anti-cancer effect.
Topics: Animals; Antineoplastic Agents; Benzamides; Drug Synergism; Humans; Imatinib Mesylate; K562 Cells; Neoplasms; Oxazoles; Piperazines; Pyrimidines; Telomerase | 2007 |
In vitro cytotoxic effects of a tyrosine kinase inhibitor STI571 in combination with commonly used antileukemic agents.
Topics: Antineoplastic Agents; Apoptosis; Benzamides; Cytarabine; Dose-Response Relationship, Drug; Drug Interactions; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Drug Synergism; Enzyme Inhibitors; Fusion Proteins, bcr-abl; Harringtonines; Homoharringtonine; Humans; Hydroxyurea; Imatinib Mesylate; Interferon-alpha; Leukemia; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Methotrexate; Microbial Sensitivity Tests; Neoplasm Proteins; Neoplasms; Piperazines; Pyrimidines; Tumor Cells, Cultured; Vincristine | 2001 |
New hope for cancer.
Topics: Animals; Antineoplastic Agents; Benzamides; Drug Design; Drug Industry; Enzyme Inhibitors; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines; United States | 2001 |
Researchers optimistic about sea change in cancer treatment.
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzamides; Cetuximab; Clinical Trials as Topic; Enzyme Inhibitors; Gastrointestinal Neoplasms; Humans; Imatinib Mesylate; Medical Oncology; Neoplasms; Piperazines; Pyrimidines; Receptor Protein-Tyrosine Kinases | 2001 |
STI571 revolution: can the newer targeted drugs measure up?
Topics: Antineoplastic Agents; Benzamides; Biomarkers, Tumor; Drug Industry; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Mutation; Neoplasms; Piperazines; Pyrimidines | 2001 |
Cancer treatment. New drugs, new hope.
Topics: Angiogenesis Inhibitors; Antibodies, Monoclonal; Antineoplastic Agents; Benzamides; Enzyme Inhibitors; Gastrointestinal Neoplasms; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines; Sarcoma | 2001 |
92nd Annual Meeting of the American Association for Cancer Research. 24-28 March, 2001, New Orleans, Louisiana, USA.
Topics: Animals; Benzamides; Carrier Proteins; Clinical Trials as Topic; Dimethylallyltranstransferase; Enzyme Inhibitors; Humans; Imatinib Mesylate; Intracellular Signaling Peptides and Proteins; Neoplasms; Piperazines; Pyrimidines; Societies, Medical; United States | 2001 |
The advent of targeted therapeutics and implications for pathologists.
Topics: Antineoplastic Agents; Benzamides; Drug Design; Humans; Imatinib Mesylate; Neoplasms; Pathology; Piperazines; Protein-Tyrosine Kinases; Pyrimidines | 2002 |
On the offensive.
Topics: Antineoplastic Agents; Benzamides; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Pyrimidines; Research | 2002 |