imatinib mesylate has been researched along with Acute Myelogenous Leukemia in 96 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 49 (51.04) | 29.6817 |
2010's | 34 (35.42) | 24.3611 |
2020's | 13 (13.54) | 2.80 |
Authors | Studies |
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Brunner, AM; Dal Cin, P; De Angelo, DJ; Dias-Santagata, D; Iafrate, AJ; Le, LP; Lennerz, JK; Luskin, MR; Marble, HD; Mueller, SB; Nardi, V; Stone, RM; Weinstock, MJ | 1 |
Abdel Hamid, M; Aref, S; Ayed, M; El-Sokkary, AMA; Fathy El-Metwaly, N | 1 |
Lv, K; Tong, W | 1 |
Chiriches, C; Guillen, N; Guy, C; Heesom, KJ; Khan, D; Ottmann, OG; Rokicki, M; Ruthardt, M; Wieske, M; Wilson, M | 1 |
Allan, JM; Blair, HJ; Dannoura, A; Dueñas, ME; Heidenreich, O; Heunis, T; Inns, J; Marín-Rubio, JL; Martin, MP; Peltier-Heap, RE; Saxty, B; Scott, J; Simpson, AJ; Trost, M; Watt, JE | 1 |
da Costa Guimarães, RF; da Silva Santos, N; de Carvalho Pires, MG; de Oliveira Mota, F; de Sousa, AVL; de Toledo, SRC; Delbuono, E; Gamba, FT; Gouveia, JT; Oliveira, ID; Rhein, BN | 1 |
Chada, K; D'Armiento, JM; Shiomi, T; Sonett, J; Unachukwu, U; Woode, D | 1 |
Chen, B; Guan, J; Ma, J | 1 |
Fei, J; Hu, H; Huang, G; Li, C; Liu, Y; Nie, H; Su, R; Wang, X; Wen, Z; Yang, J; Yin, Z; Zeng, X | 1 |
Bin, T; Chen, S; Chen, X; Cheng, J; Liao, Y; OUYang, J; Zou, W | 1 |
Ahmadi, A; Anower-E-Khuda, F; Bajaj, J; Blevins, A; Esko, JD; Ginsberg, MH; Hamilton, M; Ito, T; Karlseder, J; Koechlein, CS; Kritzik, M; Kwon, HY; Lytle, N; Park, PW; Reya, T; Spinler, K; Sun, H; Weeks, J; Zimdahl, B | 1 |
Adams, D; Advani, AS; Ali-Osman, F; Carew, JS; Cooper, B; Corrigan, D; Cotta, CV; Elson, P; Fensterl, J; Foster, B; Griffiths, EA; Jia, X; Kalaycio, M; Li, H; Maciejewski, JP; Park, J; Rao, AV; Rizzieri, DA; Rouphail, B; Rush, ML; Sekeres, MA; Sobecks, RM; Tripp, B; Tse, W; Wang, ES | 1 |
Cai, Y; Du, X; Fan, JC; Liu, HX; Wang, JX; You, WW | 1 |
Agarwal, K; Paulose, RM; Rani, PK; Tyagi, M | 1 |
Ankathil, R; Azlan, H; Baba, AA; Dzarr, AA | 1 |
Belyaeva, EA; Bernhardy, AJ; Bhatia, R; Bhatia, S; Bolton-Gillespie, E; Dasgupta, Y; Hanamshet, K; Johnson, N; Langer, S; Lee, J; Matlawska-Wasowska, K; Mazin, AV; Moore, M; Müschen, M; Nieborowska-Skorska, M; Siciliano, M; Skorski, T; Sullivan-Reed, K; Valent, P; Wasik, MA; Zhao, H | 1 |
Bombelli, S; Boultwood, J; Branford, S; Citterio, S; Crespiatico, I; D'Aliberti, D; Fontana, D; Gambacorti-Passerini, C; Khandelwal, P; Kim, DW; Magistroni, V; Massimino, L; Mauri, M; Mezzatesta, C; Morotti, A; Nava, M; Parker, W; Perego, R; Piazza, R; Pirola, A; Readelli, S; Rigolio, R; Saglio, G; Schreiber, A; Sharma, N; Viltadi, M; Wang, P; Yeung, D | 1 |
Guo, X; Zhang, X | 1 |
Battezzi, A; Bernardinetti, M; Bove, T; Parisella, L; Tomasino, S; Vetrugno, L | 1 |
Agrawal, S; Baruchel, A; Beverloo, BB; den Boer, ML; Dworzak, M; Kearns, PR; Lancaster, DL; Lehrnbecher, T; Manos, G; Mechinaud, F; Pieters, R; Reinhardt, D; Rizzari, C; Rosenberg, J; Strauss, L; van der Velden, VH; Zwaan, CM | 1 |
Arai, H; Handa, T; Iso, H; Mitani, K; Nagasawa, F; Nakamura, Y; Sasaki, K; Takahashi, W; Tokita, K; Tsurumi, S | 1 |
Druker, BJ | 2 |
Doki, N; Harada, H; Harada, Y; Inoue, D; Izawa, K; Kakihana, K; Katayama, Y; Kawabata, KC; Kitamura, T; Kitaura, J; Maehara, A; Matsui, T; Nakahara, F; Nishimura, K; Ohashi, K; Oki, T; Sada, A; Togami, K; Uchida, T; Yoshioka, K | 1 |
Garcia-Manero, G; Khoury, JD; Loghavi, S; Shah, S | 1 |
Fujii, S; Miura, I; Tanaka, H | 1 |
Goryainova, NV | 1 |
Mihaila, RG | 1 |
Ishikawa, T; Maruoka, H; Shimomura, Y | 1 |
Birgens, H; Brown, Pde N; Dalseg, AM; Dufva, IH; Hasselbalch, HC; Jensen, MK; Vangsted, A | 1 |
Abboud, C; Becker, M; Friedberg, J; Ifthikharuddin, J; Komrokji, RS; Liesveld, JL; Messina, P; Mulford, D; Oliva, J; Phillips, G; Walker, AR | 1 |
Becker, H; Berg, T; Binder, M; Dierks, C; Duque-Afonso, J; Hackanson, B; Lairmore, MD; Lübbert, M; Martens, U; Mertelsmann, R; Schäfer, HS; Schnitzler, M; Zeiser, R | 1 |
Berdel, WE; Choudhary, C; Evers, G; Hehn, S; Müller-Tidow, C; Ng, PR; Sargin, B; Serve, H; Tickenbrock, L | 1 |
Dvorak, P; Hruba, M; Subrt, I | 1 |
Chevallier, P; Dauriac, C; Garand, R; Harousseau, JL; Hunault-Berger, M; Larosa, F | 1 |
Cambazard, F; Chraïbi, R; Labeille, B; Perrot, JL | 1 |
Bendit, I; de Alencar Fischer Chamone, D; de Mello Conchon, MR; Dias, L; Dorlhiac-Llacer, PE; Ferreira, P; Kumeda, C; Lima, W | 1 |
Bacher, U; Bokemeyer, C; Bruemmendorf, TH; Dierlamm, J; Hochhaus, A; Schafhausen, P; Schnittger, S; Zander, AR | 1 |
Beelen, DW; Ditschkowski, M; Haferlach, C; Schulte, C; Trenschel, R | 1 |
Kondo, T; Kubo, Y; Matsuda, K; Matsuhashi, Y; Nakanishi, H; Sadahira, Y; Sano, F; Sugihara, T; Tasaka, T; Tohyama, K; Wada, H | 1 |
Hackanson, B; Lübbert, M; Rückert, A | 1 |
Adil, SN; Kumar, S; Masood, N | 1 |
Ozawa, K | 1 |
Ishizawa, J; Saya, H | 1 |
Jotterand, M; Muehlematter, D; Rausch, T; Spertini, O; Stalder, M; Védy, D | 1 |
Frankel, AE; Hogge, DE; Kim, HP | 1 |
Advani, AS; Bates, J; Copelan, EA; Cotta, CV; Egorin, MJ; Howard, M; Hsi, E; Jin, T; Kalaycio, M; Lim, K; Maciejewski, J; Noon, E; Price, C; Rush, ML; Salvado, A; Saunthararajah, Y; Sekeres, MA; Sobecks, R; Tiu, R; Tripp, B | 1 |
Czemerska, M; Grzybowska-Izydorczyk, O; Pluta, A; Robak, T; Szmigielska-Kapłon, A; Wierzbowska, A; Wolska, A | 1 |
Chen, Y; Li, D; Li, S; Peng, C | 1 |
Brandwein, JM; Chow, S; Gupta, V; Hedley, DW; Kamel-Reid, S; Minden, MD; Schimmer, AD; Schuh, AC; Xu, W; Yee, KW | 1 |
Angelopoulou, MK; Bartzi, V; Bitsani, A; Boutsikas, G; Dimou, M; Efthymiou, A; Georgiou, G; Kyrtsonis, MC; Panayiotidis, P; Pessach, I; Plata, E; Tofas, P; Vardounioti, I; Vassilakopoulos, TP | 1 |
Cho, JH; Hur, M; Kim, WS; Ko, YS; Lee, MH; Moon, HW; Yun, YM | 1 |
Fedorova, TV; Ilinskaya, ON; Kretova, OV; Makarov, AA; Mitkevich, VA; Petrushanko, IY; Prassolov, VS; Spirin, PV; Tchurikov, NA | 1 |
Allan, DS; Huang, H; Luo, Y; Sun, J; Tan, Y; Wang, Z | 1 |
Eisenberg, S | 1 |
Hamilton, MS; Hunter, H; Kerr, JP; Tucker, D; Wickham, C | 1 |
Huang, LS; Tong, JF; Xu, XH; Yang, J; Yu, T; Yuan, XG; Zhao, XY | 1 |
Kanzaki, S; Kure, A; Okuno, K; Sano, H; Tamoto, N; Ueyama, J | 1 |
Ding, YL; Ge, CH; Li, CY; Li, W; Lian, WX; Ning, HM; Xu, CW; Xu, WX; Yang, XM; Yang, Y; Yu, M; Zhan, YQ; Zhang, MJ | 1 |
Chan, M; Choong, A; Chu, S; Chuah, C; Goh, YT; Hwang, W; Koh, M; Lim, TJ; Linn, YC; Loh, Y; Ng, HJ; Niam, M; Suck, G; Yong, HX | 1 |
Aritaka, N; Ichikawa, K; Imai, H; Komatsu, N; Noguchi, M; Sekiguchi, Y; Sugimoto, KJ | 1 |
Bakhteeva, TD; Kalinkina, NV; Skliannaia, EV; Taradin, GG; Vatutin, NT | 1 |
Al-Riyami, AZ; Forrest, D; Hudoba, M; Young, S | 1 |
Boulton, C; Fabbro, D; Gilliland, DG; Griffin, JD; Kelly, LM; Manley, P; Meyer, T; Weisberg, E | 1 |
Breitenbuecher, F; Fischer, T; Gamm, H; Gschaidmeier, H; Hess, G; Huber, C; Kindler, T; Kirkpatrick, CJ; Marx, A | 1 |
Baker, LH; Bekele, BN; Benjamin, RS; Champlin, RE; Thall, PF; Wathen, JK | 1 |
Bishop, WR; Nakajima, A; Ohyashiki, K; Sumi, M; Tauchi, T | 1 |
Albitar, M; Cortes, J; Faderl, S; Garcia-Manero, G; Giles, F; Kantarjian, H; Letvak, L; O'Brien, S; Rios, MB; Salvado, A; Talpaz, M; Thomas, D | 1 |
Naoe, J | 1 |
Karp, JE; Lancet, JE | 1 |
Feng, R; Tan Tai, LF; Yi, ZS | 1 |
Cain, J; Grisolano, JL; O'Neal, J; Tomasson, MH | 1 |
Asaka, M; Ehira, N; Imamura, M; Kanamori, H; Kawamura, T; Masauzi, N; Miura, T; Obara, S; Tanaka, J; Tsutsumi, Y; Yamato, H | 1 |
Cortes, J; Faderl, S; Ferrajoli, A; Garcia-Manero, G; Giles, F; Hennessy, B; Kantarjian, H; O'brien, S; Ossa, G; Verstovsek, S | 1 |
Chen, B; Chen, GQ; Chen, J; Chen, SJ; Chen, Z; Jin, XL; Liang, WX; Liu, YW; Shen, ZX; Shi, JY; Wang, YY; Xiong, SM; Xu, F; Yang, G; Yin, T; You, JH; Zhou, GB | 1 |
Asou, N; Kawakita, T; Matsuno, N; Mitsuya, H; Nanri, T | 1 |
Bergholz, U; Besmer, P; Cammenga, J; Fiedler, W; Horn, S; Sommer, G; Stocking, C | 1 |
Chang, Y; Chen, SS; Fu, JY; Li, JL; Liu, YR; Ma, X; Qin, YZ; Ruan, GR; Wang, YZ | 1 |
Golovleva, I; Lazarevic, V; Nygren, I; Wahlin, A | 1 |
Kizaki, M | 1 |
Abruzzo, LV; Cortes, J; Garcia-Manero, G; Kantarjian, H; Kovitz, C | 1 |
Basic, I; Chandra, J; Giles, F; Golemovic, M; Kantarjian, H; Manshouri, T; Orsolic, N; Quintás-Cardama, A; Scappini, B; Verstovsek, S | 1 |
Horiike, S; Misawa, S; Taniwaki, M; Ueda, K; Zen, K | 1 |
Bainbridge, T; Corless, CL; Gatter, K; Granter, S; Harrell, P; Heinrich, MC; Lacouture, M; Le, C; White, C | 1 |
Arai, Y; Eguchi, M; Eguchi-Ishimae, M; Maki, K; Mitani, K; Nakamura, Y; Sasaki, K; Tadokoro, J; Tokita, K | 1 |
Baer, MR; Barcos, M; Coignet, LJ; Nganga, A; Pawarode, A; Sait, SN | 1 |
Borneo, J; Chan, RJ; Kapur, R; Munugalavadla, V; Sims, EC | 1 |
Colucci, F; Hamrouni, A; Hetuin, D; Jouy, N; Liu, J; Marchetti, P; Quesnel, B; Saudemont, A | 1 |
Cho, BS; Eom, KS; Kim, CC; Kim, HJ; Lee, JW; Lee, S; Min, WS | 1 |
Raaijmakers, MH | 1 |
Alberti, D; Arpinati, M; Baccarani, M; Candoni, A; Fanin, R; Lauria, F; Malagola, M; Martinelli, G; Messa, E; Paolini, S; Piccaluga, PP; Pirrotta, MT; Rancati, F; Rondoni, M; Russo, D; Saglio, G; Vinaccia, V; Visani, G | 1 |
Albitar, M; Bhalla, K; Cortes, J; Faraji, H; Giles, F; Gorre, M; Jilani, I; Kantarjian, H; O'Brien, S; Ottmann, O | 1 |
Kranz, S; Mohren, M; Neum, S; Schalk, E; Scheinpflug, K | 1 |
Baker, SD; Dahl, GV; Hu, S; Inaba, H; Minkin, P; Niu, H; Orwick, S; Rubnitz, J; Shimada, A | 1 |
Beran, M; Dong, L; Kantarjian, HM; Keating, MJ; Onida, F; Scappini, B; Verstovsek, S | 1 |
Draznin, J; Parisi, E; Porter, D; Schuster, SJ; Sollecito, TP; Stoopler, E | 1 |
22 review(s) available for imatinib mesylate and Acute Myelogenous Leukemia
Article | Year |
---|---|
De nove Philadelphia chromosome-positive myelodysplastic syndromes with complex karyotype and p230
Topics: Cell Transformation, Neoplastic; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; In Situ Hybridization, Fluorescence; Karyotype; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Myelodysplastic Syndromes; Philadelphia Chromosome | 2023 |
[Acute myeloid leukemia with FIP1L1-PDGFRA fusion gene treated with imatinib: a case report and literature review].
Topics: Benzamides; Humans; Hypereosinophilic Syndrome; Imatinib Mesylate; Leukemia, Myeloid, Acute; mRNA Cleavage and Polyadenylation Factors; Oncogene Proteins, Fusion; Receptor, Platelet-Derived Growth Factor alpha | 2020 |
Pharmacogenetics and the treatment of chronic myeloid leukemia: how relevant clinically? An update.
Topics: Antineoplastic Agents; Drug Resistance, Neoplasm; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Pharmacogenetics; Polymorphism, Single Nucleotide; Protein Kinase Inhibitors | 2018 |
[Development of Ph negative acute myeloid leukemia in a patient with minor-BCR/ABL positive chronic myeloid leukemia achieving a partial cytogenetic response during tyrosine kinase inhibitor treatment].
Topics: Aged; Benzamides; Cytogenetic Analysis; Dasatinib; Fatal Outcome; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Male; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Remission Induction; Thiazoles | 2015 |
[THE CLINICAL SIGNIFICANCE OF GENETIC MUTATIONS IN ACUTE MYELOID LEUKEMIA].
Topics: Antineoplastic Agents; CCAAT-Enhancer-Binding Proteins; Core Binding Factor Alpha 2 Subunit; fms-Like Tyrosine Kinase 3; Gene Expression Regulation, Leukemic; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Mutation; Neoplasm Proteins; Nuclear Proteins; Nucleophosmin; Proto-Oncogene Proteins c-kit; Treatment Outcome; Tretinoin; WT1 Proteins | 2014 |
A minireview on NHE1 inhibitors. A rediscovered hope in oncohematology.
Topics: Amiloride; Antineoplastic Agents; Apoptosis; Cation Transport Proteins; Cell Line, Tumor; DNA Damage; Drug Interactions; fms-Like Tyrosine Kinase 3; Genes, abl; Guanidines; Heme Oxygenase-1; Humans; Hydrogen-Ion Concentration; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Mutation; Niacinamide; Osmolar Concentration; Patents as Topic; Phenylurea Compounds; Protein Kinase Inhibitors; Signal Transduction; Sodium-Hydrogen Exchanger 1; Sodium-Hydrogen Exchangers; Sorafenib; Sulfones; Tumor Hypoxia; Up-Regulation | 2015 |
[Novel medical treatment modalities in hematology].
Topics: Aminoglycosides; Anemia, Hemolytic; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antibodies, Monoclonal, Murine-Derived; Antineoplastic Agents; Benzamides; Benzoates; Boronic Acids; Bortezomib; Carbazoles; Carrier Proteins; Cyclophosphamide; Dasatinib; Furans; Gemtuzumab; Hematologic Diseases; Humans; Hydrazines; Imatinib Mesylate; Immunologic Factors; Indoles; Lenalidomide; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myeloid, Acute; Lymphoma; Multiple Myeloma; Myelodysplastic Syndromes; Piperazines; Purpura, Thrombocytopenic; Pyrazines; Pyrazoles; Pyrimidines; Receptors, Fc; Recombinant Fusion Proteins; Rituximab; Thalidomide; Thiazoles; Thrombopoietin; Vidarabine | 2008 |
Hyperleukocytotic secondary acute myeloid leukemia (AML) with sole monosomy 7 as sequela of Philadelphia-chromosome positive chronic myeloid leukemia (CML).
Topics: Aged; Anemia, Refractory, with Excess of Blasts; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Chromosome Deletion; Chromosomes, Human, Pair 7; Cytarabine; Disease Progression; Fatal Outcome; Humans; Imatinib Mesylate; Interferon-alpha; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Leukemia, Myeloid, Chronic, Atypical, BCR-ABL Negative; Leukocytosis; Male; Monosomy; Philadelphia Chromosome; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Selection, Genetic | 2009 |
Old disease, new targets. Part-II, haematological malignancies.
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Murine-Derived; Antineoplastic Agents; Benzamides; Drug Costs; Graft vs Host Disease; Hematologic Neoplasms; Humans; Imatinib Mesylate; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myeloid, Acute; Lymphoma, Non-Hodgkin; Piperazines; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Protein Kinase Inhibitors; Pyrimidines; Rituximab; Time Factors | 2009 |
[History, current status, and future prospects in clinical study of myeloid leukemia].
Topics: Antineoplastic Agents; Benzamides; Cytarabine; Drug Design; Drug Therapy, Combination; Gene Targeting; Granulocyte Colony-Stimulating Factor; Hematopoietic Stem Cell Transplantation; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Piperazines; Precision Medicine; Pyrimidines; Remission Induction; Risk; Tretinoin | 2009 |
[Current clinical trials using new targeted therapies for myeloid leukemia and the research trends].
Topics: Animals; Antineoplastic Agents; Benzamides; Chromosome Aberrations; Clinical Trials as Topic; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Leukemia, Promyelocytic, Acute; Neoplastic Stem Cells; Piperazines; Pyrimidines; Translational Research, Biomedical; Tretinoin | 2009 |
Novel and emerging drugs for acute myeloid leukemia: pharmacology and therapeutic activity.
Topics: Adenine Nucleotides; Animals; Arabinonucleosides; Azacitidine; Benzamides; Clofarabine; Cytarabine; Cytosine; Daunorubicin; Decitabine; Dioxolanes; Farnesyltranstransferase; Histone Deacetylase Inhibitors; Humans; Hydrazines; Imatinib Mesylate; Leukemia, Myeloid, Acute; Liposomes; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Sulfonamides; TOR Serine-Threonine Kinases; Valproic Acid; Vascular Endothelial Growth Factor Receptor-1 | 2011 |
Therapy-related acute leukemia with mixed phenotype and t(9;22)(q32;q11.2): a case report and review of the literature.
Topics: Adenocarcinoma; Antineoplastic Combined Chemotherapy Protocols; Back; Benzamides; Bone Marrow; Chromosomes, Human, Pair 22; Chromosomes, Human, Pair 9; Cytarabine; Endometrial Neoplasms; Female; Gene Rearrangement; Genes, abl; Humans; Idarubicin; Imatinib Mesylate; Immunophenotyping; Induction Chemotherapy; Karyotyping; Leukemia, Myeloid, Acute; Leukemic Infiltration; Middle Aged; Neoplasms, Second Primary; Piperazines; Pyrimidines; Remission Induction; Soft Tissue Neoplasms; Submandibular Gland Neoplasms; Translocation, Genetic | 2012 |
C-kit-positive acute myelogenous leukemia effectively treated with imatinib: a case report and review of the literature.
Topics: Aged, 80 and over; Antineoplastic Agents; Benzamides; Fatal Outcome; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines | 2012 |
[True polycythemia: current views of pathogenesis, diagnostics and treatment].
Topics: Age Factors; Algorithms; Antineoplastic Agents; Aspirin; Benzamides; Combined Modality Therapy; Hematocrit; Hemodilution; Humans; Hydroxyurea; Imatinib Mesylate; Janus Kinase 2; Leukemia, Myeloid, Acute; Mutation; Piperazines; Platelet Aggregation Inhibitors; Polycythemia Vera; Prevalence; Primary Myelofibrosis; Pyrimidines; Randomized Controlled Trials as Topic; Risk Assessment; Thrombosis; Treatment Outcome | 2012 |
[Pathophysiology and treatment of acute myeloid leukemia].
Topics: Animals; Antineoplastic Agents; Benzamides; fms-Like Tyrosine Kinase 3; Genetic Therapy; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Piperazines; Proto-Oncogene Proteins; Pyrimidines; Receptor Protein-Tyrosine Kinases; Tretinoin | 2003 |
Farnesyl transferase inhibitors in myeloid malignancies.
Topics: Alkyl and Aryl Transferases; Antineoplastic Agents; Benzamides; Benzodiazepines; Clinical Trials as Topic; Enzyme Inhibitors; Farnesyltranstransferase; Hematologic Neoplasms; Humans; Imatinib Mesylate; Imidazoles; Leukemia, Myeloid, Acute; Models, Biological; Myeloproliferative Disorders; Piperazines; Pyrimidines; Quinolones; ras Proteins; Signal Transduction | 2003 |
Management of patients with systemic mastocytosis: review of M. D. Anderson Cancer Center experience.
Topics: Adult; Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Cladribine; Combined Modality Therapy; Cytarabine; Female; Humans; Idarubicin; Imatinib Mesylate; Interferon-alpha; Leukemia, Myeloid, Acute; Male; Mastocytosis, Systemic; Middle Aged; Myelodysplastic Syndromes; Piperazines; Prospective Studies; Pyrimidines; Stem Cell Transplantation; Treatment Outcome | 2004 |
New therapeutic approach for myeloid leukemia: induction of apoptosis via modulation of reactive oxygen species production by natural compounds.
Topics: Animals; Antineoplastic Agents, Phytogenic; Apoptosis; Benzamides; Hemorrhage; Humans; Imatinib Mesylate; Infections; Leukemia, Myeloid, Acute; Piperazines; Pyrimidines; Reactive Oxygen Species | 2006 |
Myelodysplastic syndromes and acute leukemia developing after imatinib mesylate therapy for chronic myeloid leukemia.
Topics: Antineoplastic Agents; Benzamides; Chromosome Aberrations; Female; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Leukemia, Myeloid, Chronic, Atypical, BCR-ABL Negative; Male; Middle Aged; Myelodysplastic Syndromes; Piperazines; Pyrimidines; Risk Factors | 2006 |
ATP-binding-cassette transporters in hematopoietic stem cells and their utility as therapeutical targets in acute and chronic myeloid leukemia.
Topics: Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Benzamides; Cell Differentiation; Drug Resistance, Neoplasm; Gene Expression Regulation, Leukemic; Hematopoietic Stem Cells; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Mice; Models, Biological; Phenotype; Piperazines; Protein Binding; Pyrimidines | 2007 |
Acute myelogenous leukemia: advances and limitations of treatment.
Topics: Adult; Aminoglycosides; Anthracyclines; Anti-Bacterial Agents; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antigens, CD; Antigens, Differentiation, Myelomonocytic; Antimetabolites, Antineoplastic; Antineoplastic Agents; Benzamides; Case-Control Studies; Cytarabine; Fatal Outcome; Gemtuzumab; Gingiva; Hematopoietic Stem Cell Transplantation; Humans; Imatinib Mesylate; Immunosuppressive Agents; Immunotoxins; Leukemia, Myeloid, Acute; Leukemic Infiltration; Male; Piperazines; Pyrimidines; Remission Induction; Sialic Acid Binding Ig-like Lectin 3 | 2002 |
9 trial(s) available for imatinib mesylate and Acute Myelogenous Leukemia
Article | Year |
---|---|
A Phase II Trial of Imatinib Mesylate as Maintenance Therapy for Patients With Newly Diagnosed C-kit-positive Acute Myeloid Leukemia.
Topics: Adult; Aged; Aged, 80 and over; Female; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Maintenance Chemotherapy; Male; Middle Aged; Neoplasm Recurrence, Local; Progression-Free Survival; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-kit; Young Adult | 2021 |
Dasatinib in children and adolescents with relapsed or refractory leukemia: results of the CA180-018 phase I dose-escalation study of the Innovative Therapies for Children with Cancer Consortium.
Topics: Adolescent; Antineoplastic Agents; Benzamides; Child; Child, Preschool; Dasatinib; Diarrhea; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Headache; Humans; Imatinib Mesylate; Infant; Kaplan-Meier Estimate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Male; Nausea; Piperazines; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Sample Size; Therapies, Investigational; Thiazoles; Treatment Outcome; Vomiting; Young Adult | 2013 |
Hes1 upregulation contributes to the development of FIP1L1-PDGRA-positive leukemia in blast crisis.
Topics: Amino Acid Substitution; Animals; Antineoplastic Agents; Basic Helix-Loop-Helix Transcription Factors; Benzamides; Blast Crisis; Female; Gene Expression Regulation, Leukemic; Homeodomain Proteins; Humans; Imatinib Mesylate; Interleukin-3; Leukemia, Myeloid, Acute; Male; Mice; Mice, Inbred BALB C; mRNA Cleavage and Polyadenylation Factors; Mutation, Missense; Neoplasms, Experimental; Oncogene Proteins, Fusion; Piperazines; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Pyrimidines; Receptor, Platelet-Derived Growth Factor alpha; Transcription Factor HES-1 | 2014 |
Phase I study of cladribine, cytarabine (Ara-C), granulocyte colony stimulating factor (G-CSF) (CLAG Regimen) and simultaneous escalating doses of imatinib mesylate (Gleevec) in relapsed/refractory AML.
Topics: Adult; Aged; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Blast Crisis; Bone Marrow; Cladribine; Cytarabine; Disease-Free Survival; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Granulocyte Colony-Stimulating Factor; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Middle Aged; Piperazines; Pyrimidines; Recurrence; Time Factors | 2008 |
A phase II trial of high-dose imatinib mesylate for relapsed or refractory c-kit positive and Bcr-Abl negative acute myeloid leukaemia: the AFR-15 trial.
Topics: Adult; Aged; Antineoplastic Agents; Benzamides; Disease-Free Survival; Female; Genes, abl; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Middle Aged; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines; Survival Rate; Time Factors | 2009 |
A Phase 1 study of imatinib mesylate in combination with cytarabine and daunorubicin for c-kit positive relapsed acute myeloid leukemia.
Topics: Adult; Aged; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Cytarabine; Daunorubicin; Female; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Maximum Tolerated Dose; Middle Aged; Phosphorylation; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines; Recurrence; STAT5 Transcription Factor | 2010 |
A phase I/II study of imatinib plus reinduction therapy for c-kit-positive relapsed/refractory acute myeloid leukemia: inhibition of Akt activation correlates with complete response.
Topics: Adult; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Female; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Middle Aged; Phosphorylation; Piperazines; Prognosis; Proto-Oncogene Proteins c-akt; Proto-Oncogene Proteins c-kit; Pyrimidines; Remission Induction; Salvage Therapy; Treatment Outcome | 2011 |
A phase I/II clinical trial of autologous cytokine-induced killer cells as adjuvant immunotherapy for acute and chronic myeloid leukemia in clinical remission.
Topics: Adult; Benzamides; CD3 Complex; CD56 Antigen; Cytokine-Induced Killer Cells; Female; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Immunotherapy; Immunotherapy, Adoptive; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Male; Middle Aged; Neoplasm Recurrence, Local; Peripheral Blood Stem Cell Transplantation; Piperazines; Pyrimidines | 2012 |
Imatinib mesylate in the treatment of newly diagnosed or refractory/resistant c-KIT positive acute myeloid leukemia. Results of an Italian Multicentric Phase II Study.
Topics: Adolescent; Adult; Antineoplastic Agents; Benzamides; Disease-Free Survival; Drug Resistance, Neoplasm; Female; Humans; Imatinib Mesylate; Italy; Leukemia, Myeloid, Acute; Male; Middle Aged; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines; Survival Rate | 2007 |
65 other study(ies) available for imatinib mesylate and Acute Myelogenous Leukemia
Article | Year |
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t(4;12)(q12;p13) ETV6-rearranged AML without eosinophilia does not involve PDGFRA: relevance for imatinib insensitivity.
Topics: Eosinophilia; Humans; Imatinib Mesylate; In Situ Hybridization, Fluorescence; Leukemia, Myeloid, Acute; Receptor Protein-Tyrosine Kinases; Retrospective Studies | 2022 |
CD34+/CD38- Stem Cell Burden Could Predict Chronic Myeloid Leukemia Patients' Outcome.
Topics: Adolescent; ADP-ribosyl Cyclase 1; Adult; Aged; Aged, 80 and over; Antigens, CD34; Antineoplastic Agents; Biomarkers, Tumor; Cell Transformation, Neoplastic; Drug Resistance, Neoplasm; Female; Flow Cytometry; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Male; Middle Aged; Neoplastic Stem Cells; Protein Kinase Inhibitors; Treatment Outcome; Young Adult | 2021 |
Waking up CML leukemia stem cells for the kill.
Topics: Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Stem Cells | 2022 |
Activation of signaling pathways in models of t(6;9)-acute myeloid leukemia.
Topics: Chromosomal Proteins, Non-Histone; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Oncogene Proteins; Oncogene Proteins, Fusion; Poly-ADP-Ribose Binding Proteins; Signal Transduction; Translocation, Genetic | 2022 |
A Matrix-Assisted Laser Desorption/Ionization Time-of-Flight Assay Identifies Nilotinib as an Inhibitor of Inflammation in Acute Myeloid Leukemia.
Topics: Cytokines; Drug Resistance, Neoplasm; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Inflammation; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Protein Kinase Inhibitors; Proteome; Pyrimidines; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization | 2022 |
NUP214::ABL1: A Ph-like fusion found in a pediatric acute myeloid leukemia patient with normal karyotype.
Topics: Child; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Karyotype; Leukemia, Myeloid, Acute; Nuclear Pore Complex Proteins; Oncogene Proteins, Fusion; Protein-Tyrosine Kinases | 2023 |
Tyrosine Kinase Inhibitors Diminish Renal Neoplasms in a Tuberous Sclerosis Model Via Induction of Apoptosis.
Topics: Angiomyolipoma; Animals; Apoptosis; Imatinib Mesylate; Kidney Neoplasms; Leukemia, Myeloid, Acute; Mice; Mice, Inbred C57BL; TOR Serine-Threonine Kinases; Tuberous Sclerosis; Tumor Suppressor Proteins; Tyrosine Kinase Inhibitors | 2023 |
System analysis of Huang-Lian-Jie-Du-Tang and their key active ingredients for overcoming CML resistance by suppression of leukemia stem cells.
Topics: Animals; Berberine; Drug Resistance, Neoplasm; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Mice; Myeloid Cell Leukemia Sequence 1 Protein; Protein Kinase Inhibitors; Stem Cells | 2023 |
Secondary chronic myeloid leukemia following acute myeloid leukemia treated with autologous hematopoietic stem cell transplantation: a case report.
Topics: Adult; Antineoplastic Combined Chemotherapy Protocols; Combined Modality Therapy; Cytarabine; Etoposide; Hematopoietic Stem Cell Transplantation; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Male; Mitoxantrone; Pyrimidines; Remission Induction; Transplantation, Autologous | 2020 |
A stem cell reporter based platform to identify and target drug resistant stem cells in myeloid leukemia.
Topics: Animals; Antineoplastic Agents; Blast Crisis; Chemoradiotherapy; Disease Models, Animal; Drug Resistance, Neoplasm; Gene Knock-In Techniques; Gene Knockout Techniques; Genes, Reporter; Green Fluorescent Proteins; High-Throughput Screening Assays; Humans; Imatinib Mesylate; Integrin beta Chains; Leukemia, Myeloid, Acute; Mice, Transgenic; Neoplastic Stem Cells; RNA-Binding Proteins; RNA-Seq; Signal Transduction; Syndecan-1 | 2020 |
Retinal haemorrhages: a clue to the underlying leukaemia.
Topics: Adult; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Fluorescein Angiography; Fovea Centralis; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Referral and Consultation; Retinal Hemorrhage; Tomography, Optical Coherence; Vision, Low; Visual Fields | 2017 |
Simultaneous Targeting of PARP1 and RAD52 Triggers Dual Synthetic Lethality in BRCA-Deficient Tumor Cells.
Topics: Animals; BRCA1 Protein; BRCA2 Protein; DNA Repair; Female; Fusion Proteins, bcr-abl; Homologous Recombination; Humans; Imatinib Mesylate; Kaplan-Meier Estimate; Leukemia, Myeloid, Acute; Male; Mice; Mice, Inbred NOD; Mice, Knockout; Phthalazines; Piperazines; Poly (ADP-Ribose) Polymerase-1; Rad52 DNA Repair and Recombination Protein; Synthetic Lethal Mutations; Tumor Suppressor p53-Binding Protein 1 | 2018 |
Topics: Blast Crisis; Cell Differentiation; Disease Progression; Drug Resistance, Neoplasm; Exome Sequencing; Female; HEK293 Cells; Humans; Imatinib Mesylate; K562 Cells; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Male; Mutation; Protein Kinase Inhibitors; Sequence Analysis, DNA; Ubiquitin-Conjugating Enzymes | 2019 |
Coexistence of BCR/ABL1 p190 transcript and CEBPA double mutations in de novo acute myeloid leukemia.
Topics: Antineoplastic Combined Chemotherapy Protocols; CCAAT-Enhancer-Binding Proteins; Cytarabine; Fusion Proteins, bcr-abl; Humans; Idarubicin; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Middle Aged; Mutation; Prognosis; Remission Induction | 2019 |
Cardiac tamponade and graft versus host disease: one more reason to remember.
Topics: Biomarkers; Cardiac Tamponade; Echocardiography; Graft vs Host Disease; Heart Function Tests; Hematopoietic Stem Cell Transplantation; Hemodynamics; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Middle Aged; Pericardiocentesis; Treatment Outcome | 2018 |
[Detection of BCR-ABL1 chimeric gene-positive neutrophils in a patient with mixed phenotype acute leukemia].
Topics: Adult; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Dasatinib; Diagnosis, Differential; Female; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Male; Middle Aged; Neutrophils; Phenotype; Piperazines; Pyrimidines; Thiazoles | 2013 |
Janet Rowley (1925-2013).
Topics: Benzamides; Genetics, Medical; History, 20th Century; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Leukemia, Promyelocytic, Acute; Neoplasms; Piperazines; Pyrimidines; Translocation, Genetic; United States | 2014 |
Discovery of imatinib-responsive FIP1L1-PDGFRA mutation during refractory acute myeloid leukemia transformation of chronic myelomonocytic leukemia.
Topics: Benzamides; Eosinophilia; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Leukemia, Myelomonocytic, Chronic; Male; Middle Aged; mRNA Cleavage and Polyadenylation Factors; Mutation; Oncogene Proteins, Fusion; Piperazines; Pyrimidines; Receptor, Platelet-Derived Growth Factor alpha; Treatment Outcome | 2014 |
Marked response to imatinib mesylate in a patient with platelet-derived growth factor receptor beta-associated acute myeloid leukemia.
Topics: Aged; Antineoplastic Agents; Chromosomes, Human, Pair 5; Cyclic GMP-Dependent Protein Kinase Type II; Cytogenetic Analysis; Fatal Outcome; Gene Fusion; Gene Rearrangement; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Receptor, Platelet-Derived Growth Factor beta; Remission Induction; Signal Transduction; Translocation, Genetic; Treatment Outcome | 2017 |
XXIII International Association for Comparative Research on Leukemia and Related Diseases Symposium: from molecular pathogenesis to targeted therapy in leukemia and solid tumors.
Topics: Adolescent; Adult; Age Factors; Aged; Animals; Benzamides; Humans; Imatinib Mesylate; Leukemia; Leukemia, Myeloid, Acute; Medical Oncology; Mice; Middle Aged; Myelodysplastic Syndromes; Neoplasms; Piperazines; Protein-Tyrosine Kinases; Pyrimidines; Transcription Factors | 2008 |
Activation of Wnt signaling in cKit-ITD mediated transformation and imatinib sensitivity in acute myeloid leukemia.
Topics: Animals; Antineoplastic Agents; Benzamides; beta Catenin; Cell Line; Cell Transformation, Neoplastic; fms-Like Tyrosine Kinase 3; Gene Expression Regulation, Leukemic; Glycogen Synthase Kinase 3; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Mice; Phosphorylation; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines; Signal Transduction; Tandem Repeat Sequences; Transfection; Wnt Proteins | 2008 |
Development of acute myeloid leukemia associated with Ph-negative clone with inv(3)(q21q26) during imatinib therapy for chronic myeloid leukemia.
Topics: Adult; Antineoplastic Agents; Benzamides; Chromosome Banding; Chromosome Inversion; Chromosomes, Human, Pair 3; Female; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Piperazines; Pyrimidines | 2009 |
[Porphyria cutanea tarda in a patient presenting hepatitis C treated with imatinib].
Topics: Benzamides; Hepatitis C; Humans; Imatinib Mesylate; Interferon-alpha; Leukemia, Myeloid, Acute; Male; Middle Aged; Piperazines; Porphyria Cutanea Tarda; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines | 2008 |
Emergence of abnormal clone with monsomy 7 in Philadelphia negative cells of CML patients treated with tyrosine kinase inhibitors.
Topics: Benzamides; Chromosomes, Human, Pair 7; Clone Cells; Dasatinib; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Male; Middle Aged; Monosomy; Myelodysplastic Syndromes; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Thiazoles; Young Adult | 2009 |
Development of AML with t(8;21)(q22;q22) and RUNX1-RUNX1T1 fusion following Philadelphia-negative clonal evolution during treatment of CML with Imatinib.
Topics: Antineoplastic Agents; Benzamides; Chromosomes, Human, Pair 21; Chromosomes, Human, Pair 8; Core Binding Factor Alpha 2 Subunit; Female; Humans; Imatinib Mesylate; Karyotyping; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Leukemia, Myeloid, Chronic, Atypical, BCR-ABL Negative; Middle Aged; Oncogene Proteins, Fusion; Piperazines; Pyrimidines; RUNX1 Translocation Partner 1 Protein; Translocation, Genetic | 2009 |
Occurrence of AML in cells of donor origin after treatment of CML in relapse with imatinib and donor stem cell boost 16 years after the original allogeneic BMT.
Topics: Aged; Antineoplastic Agents; Benzamides; Bone Marrow Transplantation; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Male; Piperazines; Pyrimidines | 2009 |
Philadelphia chromosome-positive acute myeloid leukemia (Ph + AML) treated with imatinib mesylate (IM): a report with IM plasma concentration and bcr-abl transcripts.
Topics: Aged; Antineoplastic Agents; Benzamides; Chromatography, High Pressure Liquid; Genes, abl; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Leukemia, Myeloid, Chronic, Atypical, BCR-ABL Negative; Male; Mass Spectrometry; Piperazines; Polymerase Chain Reaction; Pyrimidines | 2009 |
Acute myeloid leukemia with myeloid sarcoma and eosinophilia: prolonged remission and molecular response to imatinib.
Topics: Antineoplastic Agents; Benzamides; Eosinophilia; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Middle Aged; Piperazines; Pyrimidines; Remission Induction; Sarcoma, Myeloid | 2010 |
A diphtheria toxin interleukin-3 fusion protein synergizes with tyrosine kinase inhibitors in killing leukemic progenitors from BCR/ABL positive acute leukemia.
Topics: Adult; Aged; Benzamides; Blotting, Western; Cell Cycle; Cell Proliferation; Cells, Cultured; Dasatinib; Diphtheria Toxin; Drug Synergism; Female; Flow Cytometry; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Interleukin-3; Interleukin-3 Receptor alpha Subunit; Leukemia, Myeloid, Acute; Male; Middle Aged; Neoplastic Stem Cells; Piperazines; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Protein-Tyrosine Kinases; Pyrimidines; Recombinant Fusion Proteins; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiazoles | 2010 |
Role of Pten in leukemia stem cells.
Topics: Animals; Benzamides; Dasatinib; Drug Resistance, Neoplasm; Genes, Tumor Suppressor; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Mice; Neoplastic Stem Cells; Piperazines; PTEN Phosphohydrolase; Pyrimidines; Signal Transduction; Thiazoles | 2010 |
Development of acute myeloid leukemia with NPM1 mutation, in Ph-negative clone, during treatment of CML with imatinib.
Topics: Antineoplastic Agents; Benzamides; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Male; Middle Aged; Mutation; Nuclear Proteins; Nucleophosmin; Philadelphia Chromosome; Piperazines; Pyrimidines | 2012 |
Sensitivity of acute myeloid leukemia Kasumi-1 cells to binase toxic action depends on the expression of KIT and АML1-ETO oncogenes.
Topics: Animals; Apoptosis; Bacillus; Benzamides; Cell Line, Tumor; Cell Proliferation; Cell Survival; Core Binding Factor Alpha 2 Subunit; Drug Screening Assays, Antitumor; Endoribonucleases; Gene Expression Regulation, Leukemic; Gene Knockdown Techniques; Humans; Imatinib Mesylate; Inhibitory Concentration 50; Lentivirus; Leukemia, Myeloid, Acute; Mice; Oncogene Proteins, Fusion; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines; RNA, Small Interfering; RUNX1 Translocation Partner 1 Protein; Time Factors | 2011 |
Prolonged survival with imatinib mesylate combined with chemotherapy and allogeneic stem cell transplantation in de novo Ph+ acute myeloid leukemia.
Topics: Antineoplastic Agents; Benzamides; Combined Modality Therapy; Daunorubicin; Disease-Free Survival; Female; Fusion Proteins, bcr-abl; Hematopoietic Stem Cell Transplantation; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Middle Aged; Philadelphia Chromosome; Piperazines; Pyrimidines; Transplantation, Homologous; Young Adult | 2012 |
The case of the harmful herbs.
Topics: Benzamides; Drug Interactions; Herbal Medicine; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Piperazines; Pyrimidines | 2012 |
Lytic bone disease as the presenting feature of Philadelphia-positive monosomy 7 myelodysplasia progressing to acute myeloid leukaemia.
Topics: Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Bone Diseases; Chromosome Deletion; Chromosomes, Human, Pair 19; Chromosomes, Human, Pair 7; Chromosomes, Human, Pair 9; Cytarabine; Humans; Idarubicin; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Middle Aged; Myelodysplastic Syndromes; Pain; Philadelphia Chromosome; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Radiography; Vidarabine | 2012 |
Chronic myeloid leukemia arising from acute myeloid leukemia: response to imatinib mesylate with favorable outcome.
Topics: Adult; Antineoplastic Agents; Benzamides; Bone Marrow; Humans; Imatinib Mesylate; Karyotyping; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Male; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Treatment Outcome | 2013 |
[Treatment with a tyrosine-kinase inhibitor of for c-KIT mutation and AML1-ETO double positive refractory acute myeloid leukemia].
Topics: Adolescent; Benzamides; Core Binding Factor Alpha 2 Subunit; Dasatinib; Fatal Outcome; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Mutation; Palliative Care; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-kit; Pyrimidines; RUNX1 Translocation Partner 1 Protein; Thiazoles; Transcription Factors | 2012 |
Erythroid differentiation-associated gene interacts with NPM1 (nucleophosmin/B23) and increases its protein stability, resisting cell apoptosis.
Topics: Apoptosis; Benzamides; Cycloheximide; Down-Regulation; Gene Knockdown Techniques; HEK293 Cells; Humans; Imatinib Mesylate; Immunoprecipitation; K562 Cells; Leukemia, Myeloid, Acute; Nuclear Proteins; Nucleophosmin; Piperazines; Pyrimidines; Tetradecanoylphorbol Acetate | 2012 |
Sorafenib is effective for imatinib-resistant FIP1L1/PDGFRA T674I mutation-positive acute myeloid leukemia with eosinophilia.
Topics: Antineoplastic Agents; Benzamides; Drug Resistance, Neoplasm; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; mRNA Cleavage and Polyadenylation Factors; Mutation; Niacinamide; Phenylurea Compounds; Piperazines; Pyrimidines; Receptor, Platelet-Derived Growth Factor alpha; Sorafenib; Treatment Outcome | 2013 |
Inhibition of mutant FLT3 receptors in leukemia cells by the small molecule tyrosine kinase inhibitor PKC412.
Topics: Animals; Antineoplastic Agents; Apoptosis; Benzamides; Bone Marrow Cells; Bone Marrow Transplantation; Cell Cycle; Cell Division; Cell Transformation, Neoplastic; Drug Resistance, Neoplasm; Enzyme Inhibitors; Flow Cytometry; fms-Like Tyrosine Kinase 3; Humans; Imatinib Mesylate; Immunoblotting; Interleukin-3; Leukemia, Myeloid, Acute; Male; Mice; Mice, Inbred BALB C; Mice, Nude; Mutation; Phosphorylation; Piperazines; Protein Kinase C; Proto-Oncogene Proteins; Pyrimidines; Receptor Protein-Tyrosine Kinases; Staurosporine; Transfection; Tumor Cells, Cultured | 2002 |
Sustained complete hematologic remission after administration of the tyrosine kinase inhibitor imatinib mesylate in a patient with refractory, secondary AML.
Topics: Anemia, Refractory; Anemia, Refractory, with Excess of Blasts; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Bone Marrow; Cytarabine; Daunorubicin; Disease Progression; Drug Resistance, Neoplasm; Enzyme Inhibitors; Exons; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Middle Aged; Neoplasm Proteins; Neoplastic Stem Cells; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines; Receptors, Platelet-Derived Growth Factor; Recurrence; Remission Induction; Salvage Therapy | 2003 |
Hierarchical Bayesian approaches to phase II trials in diseases with multiple subtypes.
Topics: Antineoplastic Agents; Bayes Theorem; Benzamides; Bone Marrow Transplantation; Busulfan; Clinical Trials, Phase II as Topic; Disease Progression; Humans; Imatinib Mesylate; Immunosuppressive Agents; Leukemia, Myeloid, Acute; Myelodysplastic Syndromes; Piperazines; Pyrimidines; Research Design; Sarcoma; Treatment Outcome; Vidarabine | 2003 |
Efficacy of SCH66336, a farnesyl transferase inhibitor, in conjunction with imatinib against BCR-ABL-positive cells.
Topics: Alkyl and Aryl Transferases; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Benzamides; Cell Division; Colony-Forming Units Assay; Cytarabine; Daunorubicin; Drug Resistance, Neoplasm; Enzyme Inhibitors; Etoposide; Farnesyltranstransferase; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Interleukin-3; Leukemia, Myeloid, Acute; Piperazines; Piperidines; Protein-Tyrosine Kinases; Pyridines; Pyrimidines; Transfection; Treatment Outcome; Tumor Cells, Cultured | 2003 |
Overcoming resistance to imatinib by combining targeted agents.
Topics: Alkyl and Aryl Transferases; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Benzamides; Cell Division; Drug Resistance, Neoplasm; Enzyme Inhibitors; Farnesyltranstransferase; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Piperazines; Piperidines; Pyridines; Pyrimidines | 2003 |
Results of imatinib mesylate therapy in patients with refractory or recurrent acute myeloid leukemia, high-risk myelodysplastic syndrome, and myeloproliferative disorders.
Topics: Adult; Aged; Aged, 80 and over; Antineoplastic Agents; Benzamides; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Leukemia, Myelomonocytic, Chronic; Middle Aged; Myelodysplastic Syndromes; Myeloproliferative Disorders; Piperazines; Polycythemia Vera; Primary Myelofibrosis; Pyrimidines; Recurrence | 2003 |
[In vitro effect of STI571 on expression of c-kit in bone marrow cells from patients with acute non-lymphocytic leukemia].
Topics: Adolescent; Adult; Aged; Antineoplastic Agents; Benzamides; Bone Marrow Cells; Female; Gene Expression Regulation, Neoplastic; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Middle Aged; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger | 2003 |
An activated receptor tyrosine kinase, TEL/PDGFbetaR, cooperates with AML1/ETO to induce acute myeloid leukemia in mice.
Topics: 3T3 Cells; Acetylation; Animals; Benzamides; Blotting, Southern; Bone Marrow Transplantation; Core Binding Factor Alpha 2 Subunit; DNA; Flow Cytometry; Histone Deacetylases; Histones; Humans; Hydroxamic Acids; Imatinib Mesylate; Leukemia, Myeloid, Acute; Mice; Mice, Inbred BALB C; Mice, Transgenic; Models, Genetic; Mutation; Oncogene Proteins, Fusion; Phenotype; Piperazines; Plasmids; Protein Binding; Protein Structure, Tertiary; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-kit; Pyrimidines; Retroviridae; RUNX1 Translocation Partner 1 Protein; Time Factors; Transcription Factors; Vorinostat | 2003 |
Monitoring of plasma imatinib concentration for the effective treatment of CML patients.
Topics: Adult; Aged; Antineoplastic Agents; Benzamides; Body Height; Body Weight; Dose-Response Relationship, Drug; Gastrointestinal Stromal Tumors; Humans; Imatinib Mesylate; Japan; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Middle Aged; Piperazines; Pyrimidines; Treatment Outcome | 2004 |
AML1-ETO and C-KIT mutation/overexpression in t(8;21) leukemia: implication in stepwise leukemogenesis and response to Gleevec.
Topics: Adolescent; Adult; Antineoplastic Agents; Apoptosis; Benzamides; Child; Child, Preschool; Chromosomes, Human, Pair 21; Chromosomes, Human, Pair 8; Core Binding Factor Alpha 2 Subunit; Female; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Middle Aged; Mutation; Oncogene Proteins, Fusion; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines; RUNX1 Translocation Partner 1 Protein; Transcription Factors; Translocation, Genetic | 2005 |
Imatinib mesylate for refractory acute myeloblastic leukemia harboring inv(16) and a C-KIT exon 8 mutation.
Topics: Benzamides; Chromosome Aberrations; Chromosomes, Human, Pair 16; Exons; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Middle Aged; Mutation; Neoplasm, Residual; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines; Recurrence; Remission Induction | 2005 |
Extracellular KIT receptor mutants, commonly found in core binding factor AML, are constitutively active and respond to imatinib mesylate.
Topics: Animals; Antineoplastic Agents; Apoptosis; Benzamides; Core Binding Factors; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Mice; Mutagenesis, Site-Directed; Mutation; Piperazines; Pyrimidines; Stem Cell Factor | 2005 |
Abnormal expression of the programmed cell death 5 gene in acute and chronic myeloid leukemia.
Topics: Adult; Apoptosis Regulatory Proteins; Benzamides; Bone Marrow Cells; Female; Fusion Proteins, bcr-abl; Gene Expression Regulation, Leukemic; Humans; Imatinib Mesylate; K562 Cells; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Male; Neoplasm Proteins; Piperazines; Protein Kinase Inhibitors; Pyrimidines | 2006 |
Induction chemotherapy and post-remission imatinib therapy for de Novo BCR-ABL-positive AML.
Topics: Aged; Antineoplastic Agents; Benzamides; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Male; Piperazines; Pyrimidines; Remission Induction | 2006 |
Adaphostin has significant and selective activity against chronic and acute myeloid leukemia cells.
Topics: Adamantane; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Benzamides; Blotting, Western; Cell Proliferation; Cells, Cultured; Drug Resistance, Neoplasm; Drug Synergism; Flow Cytometry; Humans; Hydroquinones; Imatinib Mesylate; Inhibitory Concentration 50; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Leukemia, Myeloid, Chronic, Atypical, BCR-ABL Negative; Phosphorylation; Piperazines; Pyrimidines; Tyrosine | 2006 |
Complete cytogenetic and molecular response to treatment with imatinib mesylate for philadelphia chromosome positive acute myeloid leukemia with multilineage dysplasia.
Topics: Antineoplastic Agents; Benzamides; Cytogenetic Analysis; Female; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Middle Aged; Piperazines; Prognosis; Protein-Tyrosine Kinases; Pyrimidines; Treatment Outcome | 2006 |
Allele-specific polymerase chain reaction for the imatinib-resistant KIT D816V and D816F mutations in mastocytosis and acute myelogenous leukemia.
Topics: Adult; Aged; Alleles; Animals; Benzamides; Cell Line; Female; Genes, ras; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Mastocytosis; Mice; Middle Aged; Mutation; Piperazines; Polymerase Chain Reaction; Protein Kinase Inhibitors; Pyrimidines; Receptor Protein-Tyrosine Kinases; Sensitivity and Specificity | 2006 |
Chronic idiopathic myelofibrosis expressing a novel type of TEL-PDGFRB chimaera responded to imatinib mesylate therapy.
Topics: Adult; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Chromosomes, Human, Pair 12; Chromosomes, Human, Pair 5; Chronic Disease; Fatal Outcome; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Male; Oncogene Proteins, Fusion; Piperazines; Primary Myelofibrosis; Pyrimidines; Transcription, Genetic; Translocation, Genetic | 2007 |
Acute myeloid leukemia developing during imatinib mesylate therapy for chronic myeloid leukemia in the absence of new cytogenetic abnormalities.
Topics: Adult; Antineoplastic Agents; Base Sequence; Benzamides; DNA Primers; DNA, Complementary; Female; Humans; Imatinib Mesylate; In Situ Hybridization, Fluorescence; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Piperazines; Pyrimidines | 2007 |
Genetic and pharmacologic evidence implicating the p85 alpha, but not p85 beta, regulatory subunit of PI3K and Rac2 GTPase in regulating oncogenic KIT-induced transformation in acute myeloid leukemia and systemic mastocytosis.
Topics: Amino Acid Substitution; Animals; Antibiotics, Antineoplastic; Benzamides; Cell Proliferation; Cell Transformation, Neoplastic; Cytokines; Drug Resistance, Neoplasm; Enzyme Inhibitors; Hematopoietic Stem Cells; Imatinib Mesylate; Leukemia, Myeloid, Acute; Mastocytosis, Systemic; Mice; Mice, Knockout; Mutation, Missense; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Piperazines; Protein Subunits; Proto-Oncogene Proteins c-kit; Pyrimidines; rac GTP-Binding Proteins; RAC2 GTP-Binding Protein; Sirolimus | 2007 |
Dormant tumor cells develop cross-resistance to apoptosis induced by CTLs or imatinib mesylate via methylation of suppressor of cytokine signaling 1.
Topics: Animals; Apoptosis; Benzamides; DNA Methylation; Gene Expression Regulation, Leukemic; Gene Silencing; Imatinib Mesylate; Janus Kinases; Leukemia, Myeloid, Acute; Mice; Mice, Inbred C3H; Piperazines; Promoter Regions, Genetic; Pyrimidines; STAT Transcription Factors; Suppressor of Cytokine Signaling 1 Protein; Suppressor of Cytokine Signaling Proteins; T-Lymphocytes, Cytotoxic; Transfection | 2007 |
Successful interim therapy with imatinib prior to allogeneic stem cell transplantation in Philadelphia chromosome-positive acute myeloid leukemia.
Topics: Adolescent; Adult; Benzamides; Chromosomes, Human; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Male; Piperazines; Pyrimidines; Stem Cell Transplantation; Transplantation, Homologous; Treatment Outcome | 2007 |
An immunological method for the detection of BCR-ABL fusion protein and monitoring its activation.
Topics: Antineoplastic Agents; Benzamides; Flow Cytometry; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Immunoassay; Immunoprecipitation; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Phosphorylation; Piperazines; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prognosis; Protein-Tyrosine Kinases; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sensitivity and Specificity | 2008 |
Long-term remission in a patient with BCR/ABL-positive acute myeloid leukaemia on maintenance therapy with imatinib.
Topics: Benzamides; Female; Humans; Imatinib Mesylate; Leukemia, Myeloid, Acute; Middle Aged; Philadelphia Chromosome; Piperazines; Pyrimidines; Remission Induction | 2009 |
Comparison of antitumor effects of multitargeted tyrosine kinase inhibitors in acute myelogenous leukemia.
Topics: Antineoplastic Agents; Apoptosis; Benzamides; Benzenesulfonates; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Imatinib Mesylate; Indoles; Leukemia, Myeloid, Acute; Niacinamide; Phenylurea Compounds; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyridines; Pyrimidines; Pyrroles; Sorafenib; Sunitinib | 2008 |
Effects of signal transduction inhibitor 571 in acute myelogenous leukemia cells.
Topics: Benzamides; Cell Division; Cytarabine; Granulocyte-Macrophage Colony-Stimulating Factor; Humans; Imatinib Mesylate; Interleukin-3; Kinetics; Leukemia, Myeloid, Acute; Leukocyte Count; Phosphorylation; Piperazines; Proto-Oncogene Proteins c-kit; Pyrimidines; Recurrence; Signal Transduction; Stem Cell Factor | 2001 |