ici 118551 has been researched along with Disease Models, Animal in 27 studies
Timeframe | Studies, this research(%) | All Research% |
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pre-1990 | 0 (0.00) | 18.7374 |
1990's | 5 (18.52) | 18.2507 |
2000's | 11 (40.74) | 29.6817 |
2010's | 10 (37.04) | 24.3611 |
2020's | 1 (3.70) | 2.80 |
Authors | Studies |
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Altenbach, RJ; Brioni, JD; Carr, TL; Chandran, P; Cowart, MD; Esbenshade, TA; Honore, P; Hsieh, GC; Lewis, LG; Liu, H; Manelli, AM; Marsh, KC; Milicic, I; Miller, TR; Strakhova, MI; Vortherms, TA; Wakefield, BD; Wetter, JM; Witte, DG | 1 |
Abrams, RPM; Bachani, M; Balasubramanian, A; Brimacombe, K; Dorjsuren, D; Eastman, RT; Hall, MD; Jadhav, A; Lee, MH; Li, W; Malik, N; Nath, A; Padmanabhan, R; Simeonov, A; Steiner, JP; Teramoto, T; Yasgar, A; Zakharov, AV | 1 |
Filipek, B; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pańczyk, K; Pękala, E; Rapacz, A; Słoczyńska, K; Waszkielewicz, AM; Żelaszczyk, D; Żesławska, E | 1 |
Kuda, Y; Kurata, Y; Shibamoto, T; Tanida, M; Yang, W; Zhang, T | 1 |
Azambuja, G; Jorge, CO; Krimon, S; Melo Aquino, B; Neves, JDS; Oliveira-Fusaro, MCG; Parada, CA; Santos, DFDSD; Schiavuzzo, JG | 1 |
Berthiaume, Y; Ferraro, P; Massé, C; Richard, C; Shabbir, W | 1 |
Branca, C; Caccamo, A; Hartman, LK; Oddo, S; Wisely, EV | 1 |
Agrawal, R; Giffard, RG; Han, RQ; Ouyang, YB; Patterson, AJ; Xu, L | 1 |
Barrot, M; Freund-Mercier, MJ; Hein, L; Petit-Demoulière, N; Tessier, LH; Waltisperger, E; Yalcin, I | 1 |
Barrot, M; Choucair-Jaafar, N; Freund-Mercier, MJ; Rodeau, JL; Waltisperger, E; Yalcin, I | 1 |
Lu, RC; Miao, D; Tan, L; Tian, Y; Wang, ND; Wang, XX; Yu, JT; Yu, NN | 1 |
Carbajal, AG; Dantzer, R; Eijkelkamp, N; Heijnen, CJ; Kavelaars, A; Kelley, KW; Schedlowski, M; Wang, H | 1 |
Bagnoli, P; Cupisti, E; Filippi, L; Fiorini, P; Martini, D; Mei, S; Monte, MD; Ristori, C | 1 |
Baiz, D; Cline, JM; D'Agostino, R; Danial, N; Datta, SR; Flores, A; Hassan, S; Karpova, Y; Kulik, G; Pullikuth, A; Register, T; Yancey, D | 1 |
Deng, J; Gamelli, R; Jones, SB; Muthu, K; Shankar, R | 1 |
Bennett, T; Gardiner, SM; Kemp, PA; March, JE | 1 |
Kishida, T; Kuroda, J; Murakami, M; Tanaka, S; Tsutsui, M; Yamagishi, R; Yoshida, T | 1 |
Laengle, UW; Markstein, R; Nogues, V; Provencher-Bollinger, A; Roman, D; Trendelenburg, AU | 1 |
Ammar-Aouchiche, Z; Bond, RA; Clement, C; Dickey, BF; Ehre, C; Frieske, JM; Ho, SB; Kesimer, M; Knoll, BJ; Nguyen, LP; Omoluabi, O; Parra, S; Tuvim, MJ | 1 |
Chupp, GL | 1 |
Acuna, G; Ai, X; Bers, DM; Desantiago, J; Islam, M; Pogwizd, SM; Ziolo, MT | 1 |
Chojnacka-Wójcik, E; Filip, M; Przegaliński, E; Tatarczyńska, E | 1 |
Collins, S; Daniel, KW; Gettys, TW; Ramkumar, V; Rohlfs, EM; Taylor, IL | 1 |
Sánchez, C | 1 |
Awender, NE; Lane, SM; Maender, KC; Maron, MB | 1 |
Gebhard, MM; Häcker, A; Martin, E; Schmidt, H; Schmidt, W | 1 |
McDonald, DM | 1 |
27 other study(ies) available for ici 118551 and Disease Models, Animal
Article | Year |
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cis-4-(Piperazin-1-yl)-5,6,7a,8,9,10,11,11a-octahydrobenzofuro[2,3-h]quinazolin-2-amine (A-987306), a new histamine H4R antagonist that blocks pain responses against carrageenan-induced hyperalgesia.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzofurans; Carrageenan; Disease Models, Animal; Drug Design; Drug Evaluation, Preclinical; Humans; Hyperalgesia; Ligands; Mice; Molecular Structure; Pain; Peritonitis; Quinazolines; Rats; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Stereoisomerism; Structure-Activity Relationship | 2008 |
Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors.
Topics: Animals; Antiviral Agents; Artificial Intelligence; Chlorocebus aethiops; Disease Models, Animal; Drug Evaluation, Preclinical; High-Throughput Screening Assays; Immunocompetence; Inhibitory Concentration 50; Methacycline; Mice, Inbred C57BL; Protease Inhibitors; Quantitative Structure-Activity Relationship; Small Molecule Libraries; Vero Cells; Zika Virus; Zika Virus Infection | 2020 |
Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH
Topics: Amino Alcohols; Animals; Anticonvulsants; Crystallography, X-Ray; Disease Models, Animal; Dose-Response Relationship, Drug; Electroshock; Mice; Models, Molecular; Molecular Structure; Rats; Seizures; Structure-Activity Relationship | 2017 |
Blockade of β2-adrenoceptor, rather than β1-adrenoceptor, deteriorates cardiac anaphylaxis in isolated blood-perfused rat hearts.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Anaphylaxis; Animals; Atenolol; Coronary Vasospasm; Coronary Vessels; Disease Models, Animal; Isolated Heart Preparation; Male; Myocardial Contraction; Ovalbumin; Propanolamines; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Time Factors; Vasoconstriction; Ventricular Dysfunction, Left; Ventricular Function, Left; Ventricular Pressure | 2017 |
Muscle pain induced by static contraction in rats is modulated by peripheral inflammatory mechanisms.
Topics: Analysis of Variance; Animals; Anti-Arrhythmia Agents; Anti-Inflammatory Agents; Atenolol; Bradykinin; Bradykinin B1 Receptor Antagonists; Creatine Kinase; Dexamethasone; Disease Models, Animal; Electric Stimulation; Hyperalgesia; L-Lactate Dehydrogenase; Locomotion; Male; Muscle Contraction; Myalgia; Neutrophils; Propanolamines; Prostaglandins; Rats; Rats, Wistar | 2017 |
Alveolar liquid clearance in lung injury: Evaluation of the impairment of the β
Topics: Aminophylline; Animals; Blood Pressure; Bronchodilator Agents; Cyclic AMP; Disease Models, Animal; Dogs; Dose-Response Relationship, Drug; Epithelial Sodium Channels; Female; Heart Rate; Imidazoles; Iodine Radioisotopes; Iodocyanopindolol; Lung Injury; Male; Propanolamines; Protein Binding; Pulmonary Alveoli; Pulmonary Edema; Receptors, Adrenergic, beta-2; Reperfusion Injury; RNA, Messenger | 2019 |
Administration of a selective β2 adrenergic receptor antagonist exacerbates neuropathology and cognitive deficits in a mouse model of Alzheimer's disease.
Topics: Adrenergic beta-2 Receptor Antagonists; Alzheimer Disease; Amyloid beta-Peptides; Animals; Cerebral Cortex; Cognition; Disease Models, Animal; Disease Progression; Female; Hippocampus; Male; Mice, Transgenic; Phosphorylation; Propanolamines; Receptors, Adrenergic, beta-2; tau Proteins | 2014 |
Postischemic brain injury is attenuated in mice lacking the beta2-adrenergic receptor.
Topics: Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Disease Models, Animal; HSP72 Heat-Shock Proteins; Infarction, Middle Cerebral Artery; Ischemic Attack, Transient; Male; Mice; Mice, Knockout; Motor Activity; Neuroprotective Agents; Propanolamines; Receptors, Adrenergic, beta-2; Up-Regulation | 2009 |
Chronic treatment with agonists of beta(2)-adrenergic receptors in neuropathic pain.
Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Functional Laterality; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Naltrexone; Narcotic Antagonists; Pain Measurement; Pain Threshold; Propanolamines; Receptors, Adrenergic, beta-2; Sciatica; Time Factors | 2010 |
Beta2-adrenoceptor agonists alleviate neuropathic allodynia in mice after chronic treatment.
Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Disease Models, Animal; Drug Administration Schedule; Male; Mice; Mice, Inbred C57BL; Neuralgia; Pain Measurement; Propanolamines; Propranolol | 2009 |
Blocking beta2-adrenergic receptor attenuates acute stress-induced amyloid beta peptides production.
Topics: Acute Disease; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alzheimer Disease; Amyloid beta-Peptides; Animals; Clenbuterol; Disease Models, Animal; Hippocampus; Male; Mice; Mice, Inbred C57BL; Peptide Fragments; Propanolamines; Proto-Oncogene Proteins c-fos; Random Allocation; Receptors, Adrenergic, beta-2; Restraint, Physical; RNA, Messenger; Stress, Psychological | 2010 |
GRK2 in sensory neurons regulates epinephrine-induced signalling and duration of mechanical hyperalgesia.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Disease Models, Animal; Enzyme Inhibitors; Epinephrine; Female; G-Protein-Coupled Receptor Kinase 2; Ganglia, Spinal; Gene Expression Regulation; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neuroglia; Pain Measurement; Pain Threshold; Phentolamine; Propanolamines; Sensory Receptor Cells; Signal Transduction | 2011 |
Antiangiogenic effects of β2 -adrenergic receptor blockade in a mouse model of oxygen-induced retinopathy.
Topics: Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Angiogenesis Inhibitors; Animals; Animals, Newborn; Atenolol; Cyclic AMP-Dependent Protein Kinases; Disease Models, Animal; Dose-Response Relationship, Drug; Electroretinography; Enzyme-Linked Immunosorbent Assay; Female; Gene Expression Regulation, Developmental; Humans; Infant, Newborn; Insulin-Like Growth Factor I; Male; Mice; Mice, Inbred C57BL; Organ Culture Techniques; Oxygen; Platelet Endothelial Cell Adhesion Molecule-1; Propanolamines; Receptors, Adrenergic, beta-2; Retinal Neovascularization; Retinopathy of Prematurity; RNA, Messenger; RNA, Small Interfering; Statistics, Nonparametric; Transfection; Vascular Endothelial Growth Factor A | 2011 |
Behavioral stress accelerates prostate cancer development in mice.
Topics: Adrenergic beta-Antagonists; Animals; Apoptosis; bcl-Associated Death Protein; Cell Line, Tumor; Disease Models, Animal; Epinephrine; Humans; Hypothalamo-Hypophyseal System; Male; Mice; Mice, Inbred BALB C; Mice, Nude; Pituitary-Adrenal System; Propanolamines; Prostatic Neoplasms; Proto-Oncogene Proteins c-myc; PTEN Phosphohydrolase; Receptors, Adrenergic, beta-2; Signal Transduction; Stress, Psychological; Transplantation, Heterologous | 2013 |
Adrenergic modulation of cytokine release in bone marrow progenitor-derived macrophage following polymicrobial sepsis.
Topics: Adrenergic beta-Antagonists; Animals; Antibodies; Atenolol; Bone Marrow; Cell Differentiation; Cytokines; Disease Models, Animal; Drug Interactions; Endotoxins; Enzyme-Linked Immunosorbent Assay; Epinephrine; Interleukin-10; Laparotomy; Lipopolysaccharides; Macrophage Activation; Macrophages; Male; Mice; Myeloid Progenitor Cells; Propanolamines; Random Allocation; Sepsis | 2005 |
Involvement of CB1-receptors and beta-adrenoceptors in the regional hemodynamic responses to lipopolysaccharide infusion in conscious rats.
Topics: Adrenergic beta-Antagonists; Animals; Blood Pressure; Consciousness; Disease Models, Animal; Drug Interactions; Endotoxemia; Lipopolysaccharides; Male; Piperidines; Propanolamines; Propranolol; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Adrenergic, beta; Sympathetic Nervous System; Tachycardia; Vasodilation | 2005 |
Tissue- and dose-dependent alteration of stress-inducible proteins by beta2-adrenoceptor agonist, salbutamol, in rats.
Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Albuterol; Animals; Cytokines; Disease Models, Animal; Dose-Response Relationship, Drug; Heart; Heat-Shock Proteins; Heme Oxygenase (Decyclizing); Inflammation; Lipopolysaccharides; Liver; Lung; Male; Myocardium; Nitric Oxide Synthase Type II; Propanolamines; Rats; Rats, Sprague-Dawley; RNA, Messenger | 2005 |
GLC756 decreases TNF-alpha via an alpha2 and beta2 adrenoceptor related mechanism.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Disease Models, Animal; Lipopolysaccharides; Medetomidine; Propanolamines; Quinolines; Rats; Rats, Inbred Lew; Receptors, Adrenergic; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta-2; Receptors, Dopamine D1; Receptors, Dopamine D2; Serotonin 5-HT1 Receptor Antagonists; Serotonin Receptor Agonists; Tumor Necrosis Factor-alpha; Uveitis | 2006 |
Chronic exposure to beta-blockers attenuates inflammation and mucin content in a murine asthma model.
Topics: Administration, Oral; Adrenergic beta-Antagonists; Animals; Asthma; Disease Models, Animal; Female; Inflammation; Infusion Pumps; Injections, Intraperitoneal; Ligands; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mucins; Nadolol; Ovalbumin; Propanolamines; Specific Pathogen-Free Organisms | 2008 |
Say what, beta-blockers for asthma?
Topics: Administration, Oral; Adrenergic beta-Antagonists; Animals; Asthma; Bronchoalveolar Lavage Fluid; Cytokines; Disease Models, Animal; Infusion Pumps; Injections, Intraperitoneal; Mice; Mucins; Nadolol; Ovalbumin; Propanolamines; Reproducibility of Results | 2008 |
Arrhythmogenic effects of beta2-adrenergic stimulation in the failing heart are attributable to enhanced sarcoplasmic reticulum Ca load.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Arrhythmias, Cardiac; Calcium; Cells, Cultured; Disease Models, Animal; Ethanolamines; Female; Heart Failure; Heart Ventricles; Humans; Male; Myocytes, Cardiac; Patch-Clamp Techniques; Phosphorylation; Propanolamines; Rabbits; Receptors, Adrenergic, beta-2; Sarcoplasmic Reticulum | 2008 |
The role of 5-hydroxytryptamine1A (5-HT1A) receptors in the anticonflict activity of beta-adrenoceptor antagonists.
Topics: Adrenergic beta-Antagonists; Animals; Anxiety; Betaxolol; Conflict, Psychological; Disease Models, Animal; Drug Interactions; Male; p-Chloroamphetamine; Pindolol; Piperazines; Prazosin; Propanolamines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists | 1994 |
Impaired expression and functional activity of the beta 3- and beta 1-adrenergic receptors in adipose tissue of congenitally obese (C57BL/6J ob/ob) mice.
Topics: Adenylyl Cyclases; Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Base Sequence; Cells, Cultured; Cyclic AMP; Diabetes Mellitus, Type 2; Disease Models, Animal; Dose-Response Relationship, Drug; Enzyme Activation; Epinephrine; Gene Expression Regulation; Hyperglycemia; Imidazoles; Lipolysis; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Molecular Sequence Data; Obesity; Propanolamines; Propranolol; Receptors, Adrenergic, beta; RNA Splicing; RNA, Messenger | 1994 |
Serotonergic mechanisms involved in the exploratory behaviour of mice in a fully automated two-compartment black and white text box.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Anti-Anxiety Agents; Anxiety Disorders; Buspirone; Chlordiazepoxide; Darkness; Diazepam; Disease Models, Animal; Exploratory Behavior; Fenfluramine; Light; Male; Mice; Penbutolol; Propanolamines; Pyrimidines; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Receptor Agonists | 1995 |
Adrenal epinephrine increases alveolar liquid clearance in a canine model of neurogenic pulmonary edema.
Topics: Adrenal Glands; Adrenalectomy; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amiloride; Animals; Blood; Blood Pressure; Brain Diseases; Central Nervous System Agents; Cisterna Magna; Disease Models, Animal; Diuretics; Dogs; Epinephrine; Extravascular Lung Water; Female; Hypertension, Pulmonary; Injections; Male; Propanolamines; Proteins; Pulmonary Alveoli; Pulmonary Artery; Pulmonary Edema; Sodium Channel Blockers; Veratrine | 1998 |
Dopexamine attenuates endotoxin-induced microcirculatory changes in rat mesentery: role of beta2 adrenoceptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bacteremia; Capillary Permeability; Disease Models, Animal; Dopamine; Drug Evaluation, Preclinical; Escherichia coli Infections; Leukocytes; Male; Mesentery; Microcirculation; Propanolamines; Random Allocation; Rats; Rats, Wistar; Receptors, Adrenergic, beta-2; Vasodilator Agents | 1998 |
Angiogenesis and remodeling of airway vasculature in chronic inflammation.
Topics: Adrenergic beta-Antagonists; Adult; Albuterol; Angiopoietin-1; Animals; Asthma; Bronchitis; Bronchodilator Agents; Capillary Permeability; Chronic Disease; Disease Models, Animal; Endothelial Growth Factors; Endothelium; Humans; Inflammation; Lung; Lymphokines; Membrane Glycoproteins; Mice; Mice, Inbred C57BL; Microcirculation; Nebulizers and Vaporizers; Neovascularization, Pathologic; Pneumonia, Mycoplasma; Propanolamines; Rats; Rats, Wistar; Research; Respiratory Mucosa; Salmeterol Xinafoate; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors | 2001 |