ici 118551 and Disease Models, Animal

ici 118551 has been researched along with Disease Models, Animal in 27 studies

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (18.52)18.2507
2000's11 (40.74)29.6817
2010's10 (37.04)24.3611
2020's1 (3.70)2.80

Authors

AuthorsStudies
Altenbach, RJ; Brioni, JD; Carr, TL; Chandran, P; Cowart, MD; Esbenshade, TA; Honore, P; Hsieh, GC; Lewis, LG; Liu, H; Manelli, AM; Marsh, KC; Milicic, I; Miller, TR; Strakhova, MI; Vortherms, TA; Wakefield, BD; Wetter, JM; Witte, DG1
Abrams, RPM; Bachani, M; Balasubramanian, A; Brimacombe, K; Dorjsuren, D; Eastman, RT; Hall, MD; Jadhav, A; Lee, MH; Li, W; Malik, N; Nath, A; Padmanabhan, R; Simeonov, A; Steiner, JP; Teramoto, T; Yasgar, A; Zakharov, AV1
Filipek, B; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pańczyk, K; Pękala, E; Rapacz, A; Słoczyńska, K; Waszkielewicz, AM; Żelaszczyk, D; Żesławska, E1
Kuda, Y; Kurata, Y; Shibamoto, T; Tanida, M; Yang, W; Zhang, T1
Azambuja, G; Jorge, CO; Krimon, S; Melo Aquino, B; Neves, JDS; Oliveira-Fusaro, MCG; Parada, CA; Santos, DFDSD; Schiavuzzo, JG1
Berthiaume, Y; Ferraro, P; Massé, C; Richard, C; Shabbir, W1
Branca, C; Caccamo, A; Hartman, LK; Oddo, S; Wisely, EV1
Agrawal, R; Giffard, RG; Han, RQ; Ouyang, YB; Patterson, AJ; Xu, L1
Barrot, M; Freund-Mercier, MJ; Hein, L; Petit-Demoulière, N; Tessier, LH; Waltisperger, E; Yalcin, I1
Barrot, M; Choucair-Jaafar, N; Freund-Mercier, MJ; Rodeau, JL; Waltisperger, E; Yalcin, I1
Lu, RC; Miao, D; Tan, L; Tian, Y; Wang, ND; Wang, XX; Yu, JT; Yu, NN1
Carbajal, AG; Dantzer, R; Eijkelkamp, N; Heijnen, CJ; Kavelaars, A; Kelley, KW; Schedlowski, M; Wang, H1
Bagnoli, P; Cupisti, E; Filippi, L; Fiorini, P; Martini, D; Mei, S; Monte, MD; Ristori, C1
Baiz, D; Cline, JM; D'Agostino, R; Danial, N; Datta, SR; Flores, A; Hassan, S; Karpova, Y; Kulik, G; Pullikuth, A; Register, T; Yancey, D1
Deng, J; Gamelli, R; Jones, SB; Muthu, K; Shankar, R1
Bennett, T; Gardiner, SM; Kemp, PA; March, JE1
Kishida, T; Kuroda, J; Murakami, M; Tanaka, S; Tsutsui, M; Yamagishi, R; Yoshida, T1
Laengle, UW; Markstein, R; Nogues, V; Provencher-Bollinger, A; Roman, D; Trendelenburg, AU1
Ammar-Aouchiche, Z; Bond, RA; Clement, C; Dickey, BF; Ehre, C; Frieske, JM; Ho, SB; Kesimer, M; Knoll, BJ; Nguyen, LP; Omoluabi, O; Parra, S; Tuvim, MJ1
Chupp, GL1
Acuna, G; Ai, X; Bers, DM; Desantiago, J; Islam, M; Pogwizd, SM; Ziolo, MT1
Chojnacka-Wójcik, E; Filip, M; Przegaliński, E; Tatarczyńska, E1
Collins, S; Daniel, KW; Gettys, TW; Ramkumar, V; Rohlfs, EM; Taylor, IL1
Sánchez, C1
Awender, NE; Lane, SM; Maender, KC; Maron, MB1
Gebhard, MM; Häcker, A; Martin, E; Schmidt, H; Schmidt, W1
McDonald, DM1

Other Studies

27 other study(ies) available for ici 118551 and Disease Models, Animal

ArticleYear
cis-4-(Piperazin-1-yl)-5,6,7a,8,9,10,11,11a-octahydrobenzofuro[2,3-h]quinazolin-2-amine (A-987306), a new histamine H4R antagonist that blocks pain responses against carrageenan-induced hyperalgesia.
    Journal of medicinal chemistry, 2008, Nov-27, Volume: 51, Issue:22

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzofurans; Carrageenan; Disease Models, Animal; Drug Design; Drug Evaluation, Preclinical; Humans; Hyperalgesia; Ligands; Mice; Molecular Structure; Pain; Peritonitis; Quinazolines; Rats; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Stereoisomerism; Structure-Activity Relationship

2008
Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors.
    Proceedings of the National Academy of Sciences of the United States of America, 2020, 12-08, Volume: 117, Issue:49

    Topics: Animals; Antiviral Agents; Artificial Intelligence; Chlorocebus aethiops; Disease Models, Animal; Drug Evaluation, Preclinical; High-Throughput Screening Assays; Immunocompetence; Inhibitory Concentration 50; Methacycline; Mice, Inbred C57BL; Protease Inhibitors; Quantitative Structure-Activity Relationship; Small Molecule Libraries; Vero Cells; Zika Virus; Zika Virus Infection

2020
Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH
    Bioorganic & medicinal chemistry, 2017, 01-15, Volume: 25, Issue:2

    Topics: Amino Alcohols; Animals; Anticonvulsants; Crystallography, X-Ray; Disease Models, Animal; Dose-Response Relationship, Drug; Electroshock; Mice; Models, Molecular; Molecular Structure; Rats; Seizures; Structure-Activity Relationship

2017
Blockade of β2-adrenoceptor, rather than β1-adrenoceptor, deteriorates cardiac anaphylaxis in isolated blood-perfused rat hearts.
    Cardiology journal, 2017, Volume: 24, Issue:4

    Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Anaphylaxis; Animals; Atenolol; Coronary Vasospasm; Coronary Vessels; Disease Models, Animal; Isolated Heart Preparation; Male; Myocardial Contraction; Ovalbumin; Propanolamines; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Time Factors; Vasoconstriction; Ventricular Dysfunction, Left; Ventricular Function, Left; Ventricular Pressure

2017
Muscle pain induced by static contraction in rats is modulated by peripheral inflammatory mechanisms.
    Neuroscience, 2017, 09-01, Volume: 358

    Topics: Analysis of Variance; Animals; Anti-Arrhythmia Agents; Anti-Inflammatory Agents; Atenolol; Bradykinin; Bradykinin B1 Receptor Antagonists; Creatine Kinase; Dexamethasone; Disease Models, Animal; Electric Stimulation; Hyperalgesia; L-Lactate Dehydrogenase; Locomotion; Male; Muscle Contraction; Myalgia; Neutrophils; Propanolamines; Prostaglandins; Rats; Rats, Wistar

2017
Alveolar liquid clearance in lung injury: Evaluation of the impairment of the β
    Respiratory physiology & neurobiology, 2019, Volume: 259

    Topics: Aminophylline; Animals; Blood Pressure; Bronchodilator Agents; Cyclic AMP; Disease Models, Animal; Dogs; Dose-Response Relationship, Drug; Epithelial Sodium Channels; Female; Heart Rate; Imidazoles; Iodine Radioisotopes; Iodocyanopindolol; Lung Injury; Male; Propanolamines; Protein Binding; Pulmonary Alveoli; Pulmonary Edema; Receptors, Adrenergic, beta-2; Reperfusion Injury; RNA, Messenger

2019
Administration of a selective β2 adrenergic receptor antagonist exacerbates neuropathology and cognitive deficits in a mouse model of Alzheimer's disease.
    Neurobiology of aging, 2014, Volume: 35, Issue:12

    Topics: Adrenergic beta-2 Receptor Antagonists; Alzheimer Disease; Amyloid beta-Peptides; Animals; Cerebral Cortex; Cognition; Disease Models, Animal; Disease Progression; Female; Hippocampus; Male; Mice, Transgenic; Phosphorylation; Propanolamines; Receptors, Adrenergic, beta-2; tau Proteins

2014
Postischemic brain injury is attenuated in mice lacking the beta2-adrenergic receptor.
    Anesthesia and analgesia, 2009, Volume: 108, Issue:1

    Topics: Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Disease Models, Animal; HSP72 Heat-Shock Proteins; Infarction, Middle Cerebral Artery; Ischemic Attack, Transient; Male; Mice; Mice, Knockout; Motor Activity; Neuroprotective Agents; Propanolamines; Receptors, Adrenergic, beta-2; Up-Regulation

2009
Chronic treatment with agonists of beta(2)-adrenergic receptors in neuropathic pain.
    Experimental neurology, 2010, Volume: 221, Issue:1

    Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Functional Laterality; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Naltrexone; Narcotic Antagonists; Pain Measurement; Pain Threshold; Propanolamines; Receptors, Adrenergic, beta-2; Sciatica; Time Factors

2010
Beta2-adrenoceptor agonists alleviate neuropathic allodynia in mice after chronic treatment.
    British journal of pharmacology, 2009, Volume: 158, Issue:7

    Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Disease Models, Animal; Drug Administration Schedule; Male; Mice; Mice, Inbred C57BL; Neuralgia; Pain Measurement; Propanolamines; Propranolol

2009
Blocking beta2-adrenergic receptor attenuates acute stress-induced amyloid beta peptides production.
    Brain research, 2010, Mar-04, Volume: 1317

    Topics: Acute Disease; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alzheimer Disease; Amyloid beta-Peptides; Animals; Clenbuterol; Disease Models, Animal; Hippocampus; Male; Mice; Mice, Inbred C57BL; Peptide Fragments; Propanolamines; Proto-Oncogene Proteins c-fos; Random Allocation; Receptors, Adrenergic, beta-2; Restraint, Physical; RNA, Messenger; Stress, Psychological

2010
GRK2 in sensory neurons regulates epinephrine-induced signalling and duration of mechanical hyperalgesia.
    Pain, 2011, Volume: 152, Issue:7

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Disease Models, Animal; Enzyme Inhibitors; Epinephrine; Female; G-Protein-Coupled Receptor Kinase 2; Ganglia, Spinal; Gene Expression Regulation; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neuroglia; Pain Measurement; Pain Threshold; Phentolamine; Propanolamines; Sensory Receptor Cells; Signal Transduction

2011
Antiangiogenic effects of β2 -adrenergic receptor blockade in a mouse model of oxygen-induced retinopathy.
    Journal of neurochemistry, 2011, Volume: 119, Issue:6

    Topics: Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Angiogenesis Inhibitors; Animals; Animals, Newborn; Atenolol; Cyclic AMP-Dependent Protein Kinases; Disease Models, Animal; Dose-Response Relationship, Drug; Electroretinography; Enzyme-Linked Immunosorbent Assay; Female; Gene Expression Regulation, Developmental; Humans; Infant, Newborn; Insulin-Like Growth Factor I; Male; Mice; Mice, Inbred C57BL; Organ Culture Techniques; Oxygen; Platelet Endothelial Cell Adhesion Molecule-1; Propanolamines; Receptors, Adrenergic, beta-2; Retinal Neovascularization; Retinopathy of Prematurity; RNA, Messenger; RNA, Small Interfering; Statistics, Nonparametric; Transfection; Vascular Endothelial Growth Factor A

2011
Behavioral stress accelerates prostate cancer development in mice.
    The Journal of clinical investigation, 2013, Volume: 123, Issue:2

    Topics: Adrenergic beta-Antagonists; Animals; Apoptosis; bcl-Associated Death Protein; Cell Line, Tumor; Disease Models, Animal; Epinephrine; Humans; Hypothalamo-Hypophyseal System; Male; Mice; Mice, Inbred BALB C; Mice, Nude; Pituitary-Adrenal System; Propanolamines; Prostatic Neoplasms; Proto-Oncogene Proteins c-myc; PTEN Phosphohydrolase; Receptors, Adrenergic, beta-2; Signal Transduction; Stress, Psychological; Transplantation, Heterologous

2013
Adrenergic modulation of cytokine release in bone marrow progenitor-derived macrophage following polymicrobial sepsis.
    Journal of neuroimmunology, 2005, Volume: 158, Issue:1-2

    Topics: Adrenergic beta-Antagonists; Animals; Antibodies; Atenolol; Bone Marrow; Cell Differentiation; Cytokines; Disease Models, Animal; Drug Interactions; Endotoxins; Enzyme-Linked Immunosorbent Assay; Epinephrine; Interleukin-10; Laparotomy; Lipopolysaccharides; Macrophage Activation; Macrophages; Male; Mice; Myeloid Progenitor Cells; Propanolamines; Random Allocation; Sepsis

2005
Involvement of CB1-receptors and beta-adrenoceptors in the regional hemodynamic responses to lipopolysaccharide infusion in conscious rats.
    American journal of physiology. Heart and circulatory physiology, 2005, Volume: 288, Issue:5

    Topics: Adrenergic beta-Antagonists; Animals; Blood Pressure; Consciousness; Disease Models, Animal; Drug Interactions; Endotoxemia; Lipopolysaccharides; Male; Piperidines; Propanolamines; Propranolol; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Adrenergic, beta; Sympathetic Nervous System; Tachycardia; Vasodilation

2005
Tissue- and dose-dependent alteration of stress-inducible proteins by beta2-adrenoceptor agonist, salbutamol, in rats.
    The Journal of toxicological sciences, 2005, Volume: 30, Issue:4

    Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Albuterol; Animals; Cytokines; Disease Models, Animal; Dose-Response Relationship, Drug; Heart; Heat-Shock Proteins; Heme Oxygenase (Decyclizing); Inflammation; Lipopolysaccharides; Liver; Lung; Male; Myocardium; Nitric Oxide Synthase Type II; Propanolamines; Rats; Rats, Sprague-Dawley; RNA, Messenger

2005
GLC756 decreases TNF-alpha via an alpha2 and beta2 adrenoceptor related mechanism.
    Experimental eye research, 2006, Volume: 83, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Disease Models, Animal; Lipopolysaccharides; Medetomidine; Propanolamines; Quinolines; Rats; Rats, Inbred Lew; Receptors, Adrenergic; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta-2; Receptors, Dopamine D1; Receptors, Dopamine D2; Serotonin 5-HT1 Receptor Antagonists; Serotonin Receptor Agonists; Tumor Necrosis Factor-alpha; Uveitis

2006
Chronic exposure to beta-blockers attenuates inflammation and mucin content in a murine asthma model.
    American journal of respiratory cell and molecular biology, 2008, Volume: 38, Issue:3

    Topics: Administration, Oral; Adrenergic beta-Antagonists; Animals; Asthma; Disease Models, Animal; Female; Inflammation; Infusion Pumps; Injections, Intraperitoneal; Ligands; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mucins; Nadolol; Ovalbumin; Propanolamines; Specific Pathogen-Free Organisms

2008
Say what, beta-blockers for asthma?
    American journal of respiratory cell and molecular biology, 2008, Volume: 38, Issue:3

    Topics: Administration, Oral; Adrenergic beta-Antagonists; Animals; Asthma; Bronchoalveolar Lavage Fluid; Cytokines; Disease Models, Animal; Infusion Pumps; Injections, Intraperitoneal; Mice; Mucins; Nadolol; Ovalbumin; Propanolamines; Reproducibility of Results

2008
Arrhythmogenic effects of beta2-adrenergic stimulation in the failing heart are attributable to enhanced sarcoplasmic reticulum Ca load.
    Circulation research, 2008, Jun-06, Volume: 102, Issue:11

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Arrhythmias, Cardiac; Calcium; Cells, Cultured; Disease Models, Animal; Ethanolamines; Female; Heart Failure; Heart Ventricles; Humans; Male; Myocytes, Cardiac; Patch-Clamp Techniques; Phosphorylation; Propanolamines; Rabbits; Receptors, Adrenergic, beta-2; Sarcoplasmic Reticulum

2008
The role of 5-hydroxytryptamine1A (5-HT1A) receptors in the anticonflict activity of beta-adrenoceptor antagonists.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 47, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Anxiety; Betaxolol; Conflict, Psychological; Disease Models, Animal; Drug Interactions; Male; p-Chloroamphetamine; Pindolol; Piperazines; Prazosin; Propanolamines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists

1994
Impaired expression and functional activity of the beta 3- and beta 1-adrenergic receptors in adipose tissue of congenitally obese (C57BL/6J ob/ob) mice.
    Molecular endocrinology (Baltimore, Md.), 1994, Volume: 8, Issue:4

    Topics: Adenylyl Cyclases; Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Base Sequence; Cells, Cultured; Cyclic AMP; Diabetes Mellitus, Type 2; Disease Models, Animal; Dose-Response Relationship, Drug; Enzyme Activation; Epinephrine; Gene Expression Regulation; Hyperglycemia; Imidazoles; Lipolysis; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Molecular Sequence Data; Obesity; Propanolamines; Propranolol; Receptors, Adrenergic, beta; RNA Splicing; RNA, Messenger

1994
Serotonergic mechanisms involved in the exploratory behaviour of mice in a fully automated two-compartment black and white text box.
    Pharmacology & toxicology, 1995, Volume: 77, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Anti-Anxiety Agents; Anxiety Disorders; Buspirone; Chlordiazepoxide; Darkness; Diazepam; Disease Models, Animal; Exploratory Behavior; Fenfluramine; Light; Male; Mice; Penbutolol; Propanolamines; Pyrimidines; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Receptor Agonists

1995
Adrenal epinephrine increases alveolar liquid clearance in a canine model of neurogenic pulmonary edema.
    American journal of respiratory and critical care medicine, 1998, Volume: 158, Issue:3

    Topics: Adrenal Glands; Adrenalectomy; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amiloride; Animals; Blood; Blood Pressure; Brain Diseases; Central Nervous System Agents; Cisterna Magna; Disease Models, Animal; Diuretics; Dogs; Epinephrine; Extravascular Lung Water; Female; Hypertension, Pulmonary; Injections; Male; Propanolamines; Proteins; Pulmonary Alveoli; Pulmonary Artery; Pulmonary Edema; Sodium Channel Blockers; Veratrine

1998
Dopexamine attenuates endotoxin-induced microcirculatory changes in rat mesentery: role of beta2 adrenoceptors.
    Critical care medicine, 1998, Volume: 26, Issue:10

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bacteremia; Capillary Permeability; Disease Models, Animal; Dopamine; Drug Evaluation, Preclinical; Escherichia coli Infections; Leukocytes; Male; Mesentery; Microcirculation; Propanolamines; Random Allocation; Rats; Rats, Wistar; Receptors, Adrenergic, beta-2; Vasodilator Agents

1998
Angiogenesis and remodeling of airway vasculature in chronic inflammation.
    American journal of respiratory and critical care medicine, 2001, Nov-15, Volume: 164, Issue:10 Pt 2

    Topics: Adrenergic beta-Antagonists; Adult; Albuterol; Angiopoietin-1; Animals; Asthma; Bronchitis; Bronchodilator Agents; Capillary Permeability; Chronic Disease; Disease Models, Animal; Endothelial Growth Factors; Endothelium; Humans; Inflammation; Lung; Lymphokines; Membrane Glycoproteins; Mice; Mice, Inbred C57BL; Microcirculation; Nebulizers and Vaporizers; Neovascularization, Pathologic; Pneumonia, Mycoplasma; Propanolamines; Rats; Rats, Wistar; Research; Respiratory Mucosa; Salmeterol Xinafoate; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors

2001