Page last updated: 2024-09-03

gr 113808 and Muscle Contraction

gr 113808 has been researched along with Muscle Contraction in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (38.10)18.2507
2000's10 (47.62)29.6817
2010's3 (14.29)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ha, HS; Lee, JM; Nam, Y; Sohn, UD; Wang, Y1
Khin, PP; Sohn, UD; Zaw, TS1
Ariga, H; Ludwig, K; Mantyh, C; Pappas, TN; Takahashi, T; Taniguchi, H; Zheng, J1
Chai, W; Chan, KY; Danser, AH; de Maeyer, JH; de Vries, R; MaassenVanDenBrink, A; Saxena, PR; Schuurkes, JA; van den Bogeardt, AJ; Villalón, CM1
Fujii, H; Kadowaki, M; Kojima, Y; Nakagawa, T; Nakajima, Y; Shimatani, H; Takaki, M1
Anselmi, L; Balestra, B; Bassotti, G; De Giorgio, R; De Ponti, F; Di Nucci, A; Spelta, V; Tonini, M1
James, AN; Parkman, HP; Ryan, JP1
Chetty, N; Coupar, IM; Desmond, PV; Irving, HR; Liu, H; Pouton, CW; Tan, YY; Tochon-Danguy, N1
Bingham, S; Ellis, ES; Gaster, LM; Joiner, GF; King, FD; Sanger, GJ; Sutton, JM; Wardle, KA; Wyman, PA1
Balestra, B; Candura, SM; Lucchelli, A; Messori, E; Rizzi, CA; Tonini, M1
Bunce, KT; Gale, JD; Grossman, CJ; Humphrey, PP; Oxford, AW; Whitehead, JW1
Costall, B; Naylor, RJ; Tuladhar, BR1
Hosoki, K; Mine, Y; Nagai, R; Oku, S; Yoshida, N; Yoshikawa, T1
Läer, S; Müller, FU; Neumann, J; Remmers, F; Scholz, H; Stein, B1
Hosoki, K; Mine, Y; Yoshida, N; Yoshikawa, T1
Mizutani, Y; Suzuki, T; Takeda, M; Taniyama, K; Tsukamoto, K1
Akkermans, LM; Lefebvre, RA; Prins, NH; Schuurkes, JA2
Akkermans, LM; Lefebvre, RA; Prins, NH; Schuurkes, JA; van Der Grijn, A1
Fukushima, K; Isobe, Y; Ito, C; Kajita, S; Kawamura, R; Yasuda, S1
Bosmans, JP; Briejer, MR; Heylen, L; Jurzak, M; Leysen, JE; Prins, NH; Schuurkes, JA; Van Daele, P1

Other Studies

21 other study(ies) available for gr 113808 and Muscle Contraction

ArticleYear
The effect of Flos Lonicerae Japonicae extract on gastro-intestinal motility function.
    Journal of ethnopharmacology, 2016, Feb-17, Volume: 179

    Topics: Animals; Benzamides; Carbachol; Cats; Cells, Cultured; Domperidone; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; Esophageal Sphincter, Lower; Gastric Emptying; Gastrointestinal Motility; Gastrointestinal Transit; Herb-Drug Interactions; Indoles; Lonicera; Male; Morpholines; Muscle Contraction; Muscle, Smooth; Ondansetron; Plant Extracts; Rats; Sulfonamides

2016
Signal Transduction Underlying the Inhibitory Mechanism of Fluoxetine on Electrical Field Stimulation Response in Rat Ileal Smooth Muscle.
    Pharmacology, 2017, Volume: 99, Issue:5-6

    Topics: 4-Aminopyridine; Amides; Animals; Atropine; Azepines; Benzophenanthridines; Bicuculline; Calcimycin; Drug Interactions; Electric Stimulation; Estrenes; Fluoxetine; Glyburide; Ileum; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Ondansetron; Pyridines; Pyrrolidinones; Rats; Signal Transduction; Sulfonamides; Tetraethylammonium

2017
Endogenous ghrelin and 5-HT regulate interdigestive gastrointestinal contractions in conscious rats.
    American journal of physiology. Gastrointestinal and liver physiology, 2008, Volume: 295, Issue:2

    Topics: Animals; Duodenum; Gastrointestinal Motility; Ghrelin; Growth Hormone-Releasing Hormone; Indoles; Male; Muscle Contraction; Oligopeptides; Ondansetron; Postprandial Period; Rats; Rats, Sprague-Dawley; Serotonin; Sulfonamides; Vagotomy

2008
Inotropic effects of prokinetic agents with 5-HT(4) receptor agonist actions on human isolated myocardial trabeculae.
    Life sciences, 2012, Apr-09, Volume: 90, Issue:13-14

    Topics: 5-Methoxytryptamine; Adolescent; Adult; Aged; Benzofurans; Calcium Channels; Child; Cisapride; Female; Gastrointestinal Agents; Heart Atria; Heart Ventricles; Humans; Indoles; Male; Middle Aged; Muscle Contraction; Myocardium; Pyridines; Quinuclidines; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin 5-HT4 Receptor Agonists; Serotonin Antagonists; Sulfonamides; Young Adult

2012
A 5-HT4 agonist mosapride enhances rectorectal and rectoanal reflexes in guinea pigs.
    American journal of physiology. Gastrointestinal and liver physiology, 2003, Volume: 285, Issue:2

    Topics: Anal Canal; Animals; Benzamides; Cisapride; Guinea Pigs; Indoles; Injections, Intravenous; Male; Morpholines; Muscle Contraction; Muscle Relaxation; Receptors, Serotonin; Rectum; Reflex; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Transducers, Pressure

2003
5-HT4 receptors contribute to the motor stimulating effect of levosulpiride in the guinea-pig gastrointestinal tract.
    Digestive and liver disease : official journal of the Italian Society of Gastroenterology and the Italian Association for the Study of the Liver, 2003, Volume: 35, Issue:4

    Topics: Animals; Colon; Dopamine Antagonists; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Pyloric Antrum; Receptors, Serotonin; Serotonin Antagonists; Sulfonamides; Sulpiride

2003
Effects of the selective serotonin reuptake inhibitor, fluoxetine, on regional gastric contractility.
    Neurogastroenterology and motility, 2005, Volume: 17, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Atropine; Drug Interactions; Fluoxetine; Gastric Fundus; Guinea Pigs; In Vitro Techniques; Indoles; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Phentolamine; Pylorus; Receptors, Neurotransmitter; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Stomach; Sulfonamides; Tetrodotoxin

2005
Comparison of 5-HT4 and 5-HT7 receptor expression and function in the circular muscle of the human colon.
    Life sciences, 2007, Mar-06, Volume: 80, Issue:13

    Topics: Aged; Aged, 80 and over; Animals; Colon; Dose-Response Relationship, Drug; Female; Gene Expression; Guinea Pigs; Humans; Ileum; Indoles; Male; Middle Aged; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Phenols; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; RNA, Messenger; Serotonin; Serotonin Antagonists; Sulfonamides

2007
N-[(1-butyl-4-piperidinyl)methyl]-3,4dihydro-2H-[1,3]oxazino[3,2- a]indole10-carboxamide hydrochloride: the first potent and selective 5-HT4 receptor antagonist amide with oral activity.
    Journal of medicinal chemistry, 1995, Nov-24, Volume: 38, Issue:24

    Topics: Administration, Oral; Animals; Dioxanes; Dogs; Guinea Pigs; Indoles; Muscle Contraction; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Structure-Activity Relationship; Sulfonamides

1995
5-Hydroxytryptamine receptors that facilitate excitatory neuromuscular transmission in the guinea-pig isolated detrusor muscle.
    British journal of pharmacology, 1995, Volume: 115, Issue:4

    Topics: Acetylcholine; Adenosine Triphosphate; Amphetamines; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Granisetron; Guinea Pigs; In Vitro Techniques; Indoles; Ketanserin; Male; Methiothepin; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Synaptic Transmission; Urinary Bladder

1995
GR113808: a novel, selective antagonist with high affinity at the 5-HT4 receptor.
    British journal of pharmacology, 1994, Volume: 111, Issue:1

    Topics: 5-Methoxytryptamine; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Colon; Dose-Response Relationship, Drug; Esophagus; Female; Guinea Pigs; Hemodynamics; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Rabbits; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sincalide; Sulfonamides

1994
5-HT3 and 5-HT4 receptor-mediated facilitation of the emptying phase of the peristaltic reflex in the marmoset isolated ileum.
    British journal of pharmacology, 1996, Volume: 117, Issue:8

    Topics: Acetylcholine; Analysis of Variance; Animals; Callithrix; Female; Indoles; Intestine, Small; Male; Muscle Contraction; Peristalsis; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides

1996
Comparison of effect of mosapride citrate and existing 5-HT4 receptor agonists on gastrointestinal motility in vivo and in vitro.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 283, Issue:3

    Topics: Animals; Benzamides; Carbachol; Dogs; Female; Gastrointestinal Motility; Guinea Pigs; In Vitro Techniques; Indoles; Male; Morpholines; Muscle Contraction; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin Receptor Agonists; Sulfonamides

1997
Receptor mechanisms involved in the 5-HT-induced inotropic action in the rat isolated atrium.
    British journal of pharmacology, 1998, Volume: 123, Issue:6

    Topics: Animals; Atrial Function; Blotting, Southern; Cyclic AMP; Heart Atria; In Vitro Techniques; Indoles; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Polymerase Chain Reaction; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; RNA, Messenger; Serotonin; Serotonin Antagonists; Sulfonamides

1998
Affinity of mosapride citrate, a new gastroprokinetic agent, for 5-HT4 receptors in guinea pig ileum.
    Japanese journal of pharmacology, 1998, Volume: 77, Issue:1

    Topics: Animals; Benzamides; Binding, Competitive; Dopamine Antagonists; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Male; Morpholines; Muscle Contraction; Radioligand Assay; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Sulfonamides; Tritium

1998
Identification of SK-951, a novel benzofuran derivative, as an agonist to 5-HT4 receptors.
    Japanese journal of pharmacology, 1999, Volume: 79, Issue:2

    Topics: Acetylcholine; Animals; Benzofurans; Bridged Bicyclo Compounds, Heterocyclic; Carbachol; Cisapride; Electric Stimulation; Esophagus; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Muscarinic; Serotonin Receptor Agonists; Sulfonamides

1999
5-HT(4) receptors on cholinergic nerves involved in contractility of canine and human large intestine longitudinal muscle.
    British journal of pharmacology, 2000, Volume: 131, Issue:5

    Topics: Animals; Dogs; Electric Stimulation; Female; Humans; In Vitro Techniques; Indoles; Intestine, Large; Male; Muscle Contraction; Muscle, Smooth; Nitroarginine; Parasympathetic Nervous System; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Sulfonamides; Tetrodotoxin

2000
5-HT(4) receptors mediating enhancement of contractility in canine stomach; an in vitro and in vivo study.
    British journal of pharmacology, 2001, Volume: 132, Issue:8

    Topics: Animals; Benzofurans; Dogs; Electric Stimulation; Female; In Vitro Techniques; Indoles; Manometry; Muscle Contraction; Muscle, Smooth; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stomach; Sulfonamides

2001
Pharmacological characterization of a novel 5-HT4 receptor agonist, TS-951, in vitro.
    Pharmacology, 2001, Volume: 63, Issue:1

    Topics: Animals; Brain; Colon; Corpus Striatum; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Male; Mice; Mice, Inbred ICR; Molecular Structure; Muscle Contraction; Muscle, Smooth; Quinolines; Radioligand Assay; Receptors, Neurotransmitter; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides

2001
The in vitro pharmacological profile of prucalopride, a novel enterokinetic compound.
    European journal of pharmacology, 2001, Jun-29, Volume: 423, Issue:1

    Topics: Acetylcholine; Animals; Benzofurans; Binding, Competitive; Carbachol; Cell Line; CHO Cells; Colon; Cricetinae; Dioxanes; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; Esophagus; Female; Gallbladder; Gastrointestinal Agents; Granisetron; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Indoles; Indomethacin; Male; Motilin; Muscle Contraction; Piperidines; Rabbits; Rats; Rats, Wistar; Receptors, Cholecystokinin; Receptors, Dopamine D2; Receptors, Dopamine D4; Receptors, Gastrointestinal Hormone; Receptors, Neuropeptide; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sincalide; Stomach; Sulfonamides; Vasodilator Agents

2001
Characterization of the receptors involved in the 5-HT-induced excitation of canine antral longitudinal muscle.
    British journal of pharmacology, 2001, Volume: 134, Issue:6

    Topics: Animals; Atropine; Dogs; Electric Stimulation; Female; Gastrointestinal Motility; Granisetron; In Vitro Techniques; Indoles; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Nitroarginine; Pyloric Antrum; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sulfonamides; Tetrodotoxin; Tryptamines

2001