Page last updated: 2024-09-02

fr 139317 and Muscle Contraction

fr 139317 has been researched along with Muscle Contraction in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's15 (88.24)18.2507
2000's2 (11.76)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Halaka, NN; Lodge, NJ1
Cheng, XM; Cody, WL; Davis, LS; DePue, PL; Doherty, AM; Flynn, MA; He, JX; LaDouceur, DM; Reynolds, EE; Welch, KM1
Clayton, RA; McGrath, JC; Nally, JE; Thomson, NC; Wakelam, MJ1
Fujii, E; Irie, K; Muraki, T; Uchida, Y1
Adner, M; Edvinsson, L; Erlinge, D; Salford, LG; Wahlestedt, C; Yee, F1
Adner, M; Edvinsson, L; Jansen, I1
Aghai, Z; Bax, WA; Saxena, PR; van Tricht, CL; Wassenaar, C1
Lüscher, TF; Tschudi, MR1
Battistini, B; Fournier, A; Vane, JR; Warner, TD1
Abboa-Offei, B; McMullen, D; Moreland, S; Seymour, A1
Adner, M; Cardell, LO; Edvinsson, L; Ottosson, A; Sjöberg, T1
Bakken, IJ; Edvinsson, L; Elsås, T; Sjaavaag, I; Vincent, MB; White, LR1
Kamikawa, Y; Uchida, K; Yuzuki, R1
Henry, PJ; King, SH1
Bellissant, E; Durand-Castel, X; Goineau, S; Guillo, P; Pape, D1
MacLean, MR; Mullaney, I; Vaughan, DM1
Huang, SC1

Other Studies

17 other study(ies) available for fr 139317 and Muscle Contraction

ArticleYear
Endothelin receptor subtype(s) in rabbit jugular vein smooth muscle.
    Journal of cardiovascular pharmacology, 1993, Volume: 22 Suppl 8

    Topics: Animals; Azepines; Endothelin Receptor Antagonists; Endothelins; In Vitro Techniques; Indoles; Jugular Veins; Male; Muscle Contraction; Muscle, Smooth, Vascular; Peptides, Cyclic; Rabbits; Receptors, Endothelin; Viper Venoms

1993
In vitro and in vivo studies with a series of hexapeptide endothelin antagonists.
    Journal of cardiovascular pharmacology, 1993, Volume: 22 Suppl 8

    Topics: Amino Acid Sequence; Animals; Arachidonic Acid; Azepines; Endothelin Receptor Antagonists; Endothelins; Ganglionic Blockers; Hemodynamics; In Vitro Techniques; Indoles; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth, Vascular; Oligopeptides; Rabbits; Rats; Receptors, Endothelin; Structure-Activity Relationship; Vasoconstriction

1993
Angiotensin II enhances responses to endothelin-1 in bovine bronchial smooth muscle.
    Pulmonary pharmacology, 1994, Volume: 7, Issue:6

    Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Azepines; Biphenyl Compounds; Bronchi; Cattle; Drug Synergism; Endothelins; Imidazoles; In Vitro Techniques; Indoles; Losartan; Muscle Contraction; Muscle, Smooth; Receptors, Angiotensin; Receptors, Endothelin; Tetrazoles

1994
Developmental changes in response to endothelins and receptor subtypes of isolated rat duodenum.
    European journal of pharmacology, 1995, Feb-24, Volume: 275, Issue:1

    Topics: Aging; Animals; Animals, Newborn; Azepines; Duodenum; Endothelin Receptor Antagonists; Endothelins; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Peptide Fragments; Rats; Rats, Wistar; Receptors, Endothelin

1995
Human endothelin ETA receptor antisense oligodeoxynucleotides inhibit endothelin-1 evoked vasoconstriction.
    European journal of pharmacology, 1994, Aug-22, Volume: 261, Issue:3

    Topics: Azepines; Base Sequence; Endothelin Receptor Antagonists; Endothelins; Humans; In Vitro Techniques; Indoles; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth, Vascular; Oligonucleotides, Antisense; Receptors, Endothelin; RNA, Messenger; Vasoconstriction

1994
Endothelin-A receptors mediate contraction in human cerebral, meningeal and temporal arteries.
    Journal of the autonomic nervous system, 1994, Volume: 49 Suppl

    Topics: Azepines; Cerebral Arteries; Endothelin Receptor Antagonists; Endothelins; Humans; In Vitro Techniques; Indoles; Meningeal Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Temporal Arteries; Vasoconstriction

1994
Different endothelin receptors involved in endothelin-1- and sarafotoxin S6B-induced contractions of the human isolated coronary artery.
    British journal of pharmacology, 1994, Volume: 113, Issue:4

    Topics: Adolescent; Adult; Azepines; Child; Child, Preschool; Coronary Vessels; Endothelin Receptor Antagonists; Endothelin-1; Endothelins; Endothelium, Vascular; Female; Glycopeptides; Humans; In Vitro Techniques; Indoles; Infant; Male; Middle Aged; Muscle Contraction; Muscle, Smooth, Vascular; Peptides, Cyclic; Protease Inhibitors; Protein Precursors; Receptors, Endothelin; Vasoconstrictor Agents; Viper Venoms

1994
Characterization of contractile endothelin and angiotensin receptors in human resistance arteries: evidence for two endothelin and one angiotensin receptor.
    Biochemical and biophysical research communications, 1994, Oct-28, Volume: 204, Issue:2

    Topics: Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Angiotensin-Converting Enzyme Inhibitors; Azepines; Benzazepines; Bosentan; Endothelin Receptor Antagonists; Endothelins; Humans; In Vitro Techniques; Indoles; Mammary Arteries; Muscle Contraction; Plasmids; Receptors, Angiotensin; Receptors, Endothelin; Sulfonamides; Tetrazoles; Valine; Valsartan; Vasoconstrictor Agents; Viper Venoms

1994
Characterization of ETB receptors mediating contractions induced by endothelin-1 or IRL 1620 in guinea-pig isolated airways: effects of BQ-123, FR139317 or PD 145065.
    British journal of pharmacology, 1994, Volume: 111, Issue:4

    Topics: Animals; Azepines; Dose-Response Relationship, Drug; Endothelin Receptor Antagonists; Endothelins; Guinea Pigs; In Vitro Techniques; Indoles; Male; Muscle Contraction; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Receptors, Endothelin; Respiratory Physiological Phenomena; Respiratory System

1994
Evidence for a differential location of vasoconstrictor endothelin receptors in the vasculature.
    British journal of pharmacology, 1994, Volume: 112, Issue:2

    Topics: Animals; Azepines; Blood Pressure; Blood Vessels; Dogs; Endothelin Receptor Antagonists; Female; In Vitro Techniques; Indoles; Isometric Contraction; Macaca fascicularis; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Peptides, Cyclic; Rabbits; Rats; Rats, Sprague-Dawley; Receptors, Endothelin; Species Specificity; Swine; Vasoconstrictor Agents; Viper Venoms

1994
Contractile endothelin-B (ETB) receptors in human small bronchi.
    The European respiratory journal, 1996, Volume: 9, Issue:2

    Topics: Acetylcholine; Azepines; Bronchi; Bronchoconstriction; Dose-Response Relationship, Drug; Endothelin Receptor Antagonists; Endothelins; Histamine; Humans; In Vitro Techniques; Indoles; Lung Neoplasms; Muscle Contraction; Muscle, Smooth; Oligopeptides; Peptide Fragments; Receptor, Endothelin B; Receptors, Endothelin

1996
Vasoactivity mediated by endothelin ETA and ETB receptors in isolated porcine ophthalmic artery.
    Acta physiologica Scandinavica, 1996, Volume: 157, Issue:2

    Topics: Animals; Azepines; Bosentan; Dinoprost; Endothelin Receptor Antagonists; Endothelin-1; Endothelin-3; In Vitro Techniques; Indoles; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Ophthalmic Artery; Receptors, Endothelin; Sulfonamides; Swine; Vasoconstrictor Agents; Viper Venoms

1996
Pharmacological characterization of endothelin-induced contraction in the guinea-pig oesophageal muscularis mucosae.
    British journal of pharmacology, 1998, Volume: 125, Issue:4

    Topics: Animals; Azepines; Calcium Channels; Endothelin Receptor Antagonists; Endothelin-1; Endothelin-2; Endothelin-3; Endothelins; Esophagus; Guinea Pigs; Humans; Imidazoles; Indoles; Male; Muscle Contraction; Muscle, Smooth; Peptides, Cyclic; Receptors, Endothelin; Viper Venoms

1998
Typical endothelin ETA receptors mediate atypical endothelin-1-induced contractions in sheep isolated tracheal smooth muscle.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:3

    Topics: Animals; Azepines; Binding, Competitive; Endothelin Receptor Antagonists; Endothelin-1; In Vitro Techniques; Indoles; Kinetics; Muscle Contraction; Muscle, Smooth; Peptides, Cyclic; Radioligand Assay; Receptor, Endothelin A; Receptors, Endothelin; Sheep; Trachea; Vasoconstrictor Agents; Viper Venoms

1999
Endothelin, but not angiotensin II, contributes to the hypoxic contractile response of large isolated pulmonary arteries in the rat.
    Fundamental & clinical pharmacology, 1999, Volume: 13, Issue:4

    Topics: Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Angiotensin-Converting Enzyme Inhibitors; Animals; Azepines; Bosentan; Calcium; Calcium Channel Blockers; Endothelin Receptor Antagonists; Endothelins; Endothelium, Vascular; Extracellular Space; Glycopeptides; Hypoxia; In Vitro Techniques; Indoles; Lisinopril; Losartan; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nicardipine; Pulmonary Artery; Rats; Rats, Wistar; Sulfonamides

1999
Regional modulation of cyclic nucleotides by endothelin-1 in rat pulmonary arteries: direct activation of G(i)2-protein in the main pulmonary artery.
    British journal of pharmacology, 2000, Volume: 129, Issue:5

    Topics: Adenosine Diphosphate Ribose; Animals; Azepines; Cell Membrane; Cholera Toxin; Cyclic AMP; Cyclic GMP; Endothelin Receptor Antagonists; Endothelin-1; Endothelium, Vascular; GTP-Binding Protein alpha Subunits, Gi-Go; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth, Vascular; Oligopeptides; Piperidines; Pulmonary Artery; Rats; Rats, Wistar; Receptor, Endothelin A; Receptor, Endothelin B; Signal Transduction

2000
Two classes of endothelin receptors mediating contraction in esophageal muscularis mucosae.
    Regulatory peptides, 2002, May-30, Volume: 105, Issue:3

    Topics: Animals; Atropine; Autoradiography; Azepines; Binding, Competitive; Carbachol; Cell Membrane; Cells, Cultured; Endothelin Receptor Antagonists; Endothelins; Esophagus; Guinea Pigs; In Vitro Techniques; Indoles; Male; Mucous Membrane; Muscle Contraction; Oligopeptides; Piperidines; Protein Binding; Receptors, Endothelin; Tetrodotoxin; Viper Venoms

2002