Page last updated: 2024-09-02

fk 888 and Muscle Contraction

fk 888 has been researched along with Muscle Contraction in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's14 (82.35)18.2507
2000's3 (17.65)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bringas, A; Choppin, A; Dillon, MP; Groke, G; Stepan, G1
Calixto, JB; El Sayah, M1
Hamada, K; Hanioka, N; Imazumi, K; Maeda, Y; Manda, T; Matsuo, M; Mutoh, S; Yamamoto, T1
HÃ¥kanson, R; Strichartz, GR; Tung, SR; Wang, ZY1
Barthó, L; Maggi, CA; Patacchini, R; Wilhelm, M1
Giuliani, S; Maggi, CA; Zagorodnyuk, V1
Haga, N; Inatomi, N; Itoh, Z; Mizumoto, A; Shiba, Y; Yamamoto, O1
Fujii, T; Hagiwara, D; Ikari, N; Maeda, Y; Matsuo, M; Miyake, H; Murai, M1
Fujii, T; Hagiwara, D; Maeda, Y; Matsuo, M; Miyake, H; Murai, M; Yamaoka, M1
Calixto, JB; Campos, AH; Cechinel Filho, V; Dias, MA; Yunes, RA1
Caliendo, G; Calignano, A; Greco, G; Grieco, P; Mancuso, F; Novellino, E; Perissutti, E; Santagada, V1
Kojima, S; Shimo, Y1
Fujita, H; Kageyama, M; Kanai, A; Nakata, K; Shirasawa, E1
Fujita, H; Goto, W; Kageyama, M; Kanai, A; Nakata, K; Shirasawa, E1
Esteve, H; Hsieh, L; Knippenberg, R; Kudlacz, E; Logan, D; Maynard, G; Olsen, K; Shatzer, S1
Cirillo, R; Conte, B; Lopez, G; Maggi, CA; Manzini, S; Parlani, M1
Esposito, V; Griffiths, NM; Linard, C; Mathe, D; Wysocki, J1

Other Studies

17 other study(ies) available for fk 888 and Muscle Contraction

ArticleYear
Effect of YM-44781, YM-44778 and YM-49598, novel tachykinin antagonists, in a drug-induced bladder contraction model.
    Pharmacology, 2002, Volume: 65, Issue:2

    Topics: Animals; Binding, Competitive; CHO Cells; Cricetinae; Dipeptides; Female; Indoles; Muscle Contraction; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Spiro Compounds; Transfection; Urinary Bladder

2002
New evidence on the mechanisms underlying bradykinin-mediated contraction of the pig iris sphincter in vitro.
    Peptides, 2003, Volume: 24, Issue:7

    Topics: Animals; Benzamides; Bradykinin; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Calcium; Calcium Channels; Capsaicin; Carbazoles; Conotoxins; Dipeptides; Dose-Response Relationship, Drug; Egtazic Acid; In Vitro Techniques; Indoles; Iris; Maleimides; Muscle Contraction; Nicardipine; omega-Agatoxin IVA; Peptide Fragments; Piperidines; Protein Kinase Inhibitors; Protein Kinases; Pyrroles; Receptors, Calcitonin Gene-Related Peptide; Receptors, Drug; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Swine; Tachykinins

2003
Contribution of tachykinin receptor subtypes to micturition reflex in guinea pigs.
    European journal of pharmacology, 2003, Sep-23, Volume: 477, Issue:3

    Topics: Animals; Brain; Catheterization; CHO Cells; Cricetinae; Dipeptides; Dose-Response Relationship, Drug; Guinea Pigs; Humans; Indoles; Injections, Intravenous; Iodine Radioisotopes; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Piperidines; Radioligand Assay; Receptors, Neurokinin-1; Spinal Cord; Substance P; Succinimides; Tetrazoles; Tissue Extracts; Transfection; Urinary Bladder; Urination

2003
Investigation of the specificity of FK 888 as a tachykinin NK1 receptor antagonist.
    British journal of pharmacology, 1994, Volume: 111, Issue:4

    Topics: Action Potentials; Animals; Dipeptides; Female; Guinea Pigs; Histamine Release; In Vitro Techniques; Indoles; Iris; Male; Muscle Contraction; Neurokinin-1 Receptor Antagonists; Rabbits; Rana catesbeiana; Sciatic Nerve

1994
Tachykinin NK1 and NK2 receptors mediate atropine-resistant ileal circular muscle contractions evoked by capsaicin.
    European journal of pharmacology, 1994, Jul-01, Volume: 259, Issue:2

    Topics: Amino Acid Sequence; Animals; Atropine; Capsaicin; Dipeptides; Drug Resistance; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Oligopeptides; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Ruthenium Red; Substance P; Tetrodotoxin

1994
Specialization of tachykinin NK1 and NK2 receptors in producing fast and slow atropine-resistant neurotransmission to the circular muscle of the guinea-pig colon.
    Neuroscience, 1994, Volume: 63, Issue:4

    Topics: Action Potentials; Animals; Atropine; Autonomic Nervous System; Colon; Dipeptides; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neuromuscular Junction; Nifedipine; Oligopeptides; Physalaemin; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Synaptic Transmission

1994
Stimulatory mechanism of EM523-induced contractions in postprandial stomach of conscious dogs.
    Gastroenterology, 1995, Volume: 109, Issue:5

    Topics: Animals; Anti-Bacterial Agents; Atropine; Dipeptides; Dogs; Dopamine; Eating; Erythromycin; Hexamethonium; Indoles; Motilin; Muscle Contraction; Naloxone; Ondansetron; Serotonin Antagonists; Stomach; Substance P

1995
Effects of an NK1 receptor antagonist, FK888, on constriction and plasma extravasation induced in guinea pig airway by neurokinins and capsaicin.
    European journal of pharmacology, 1993, May-12, Volume: 236, Issue:1

    Topics: Animals; Capillary Permeability; Capsaicin; Dipeptides; Guinea Pigs; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Trachea

1993
The pharmacological properties of FK888, a novel dipeptide NK1 antagonist.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Animals; Bronchoconstriction; Capsaicin; Cell Membrane; Dipeptides; Edema; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Indoles; Kinetics; Lung; Muscle Contraction; Muscle, Smooth; Neurokinin A; Receptors, Neurokinin-1; Substance P

1993
Analysis of the mechanisms underlying the contractile response induced by the hydroalcoholic extract of Phyllanthus urinaria in the guinea-pig urinary bladder in-vitro.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:10

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Benzamides; Dipeptides; Ethanol; Female; Guinea Pigs; In Vitro Techniques; Indoles; Ion Channels; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Neurokinin A; Piperidines; Plant Extracts; Plants, Medicinal; Receptors, Tachykinin; Substance P; Urinary Bladder

1995
Modification of the potent peptide FK888 with unusual aminoacids: effects on activity on neurokinin receptors.
    Farmaco (Societa chimica italiana : 1989), 1996, Volume: 51, Issue:3

    Topics: Amino Acid Sequence; Amino Acids; Animals; Chromatography, High Pressure Liquid; Colon; Dipeptides; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth, Vascular; Neurokinin-1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Spectrometry, Mass, Fast Atom Bombardment

1996
Investigation into the 5-hydroxytryptamine-induced atropine-resistant neurogenic contraction of guinea-pig proximal colon.
    British journal of pharmacology, 1996, Volume: 117, Issue:8

    Topics: 5-Methoxytryptamine; Animals; Atropine; Colon; Dipeptides; Dose-Response Relationship, Drug; Guinea Pigs; Indoles; Male; Methiothepin; Muscarinic Antagonists; Muscle Contraction; Ondansetron; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1996
Effects of the immunosuppressant cyclosporin A on neurotransmitter release from peripheral non-adrenergic, non-cholinergic nerves.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:3

    Topics: Animals; Atropine; Calcium Channel Blockers; Capsaicin; Cyclosporine; Dipeptides; Immunosuppressive Agents; Indoles; Iris; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Nerve Fibers; Neurokinin-1 Receptor Antagonists; Rabbits; Sodium Channel Blockers; Substance P

1997
FK506-binding proteins regulate smooth muscle contractility by altering neurotransmitter release.
    European journal of pharmacology, 1997, Aug-27, Volume: 333, Issue:2-3

    Topics: Animals; Calcium Channel Blockers; Capsaicin; Dipeptides; Dose-Response Relationship, Drug; Immunosuppressive Agents; Indoles; Iris; Male; Muscle Contraction; Muscle, Smooth; Polyenes; Rabbits; Receptors, Tachykinin; Sirolimus; Synaptic Transmission; Tachykinins; Tacrolimus

1997
A role for histamine and substance P in immediate allergic responses in guinea pig airways: characterization of MDL 108,207DA, a dual H1/NK-1 receptor antagonist.
    International archives of allergy and immunology, 1998, Volume: 115, Issue:2

    Topics: Animals; Benzimidazoles; Bronchi; Capillary Permeability; CHO Cells; Cricetinae; Dipeptides; Drug Combinations; Guinea Pigs; Histamine; Histamine H1 Antagonists; Indoles; Inositol Phosphates; Muscle Contraction; Neurokinin-1 Receptor Antagonists; Ovalbumin; Pyrilamine; Pyrrolidines; Radioligand Assay; Receptors, Histamine H1; Receptors, Neurokinin-1; Respiratory Hypersensitivity; Skin Tests; Substance P; Trachea; Tumor Cells, Cultured

1998
Inflammatory and motor responses by tachykinins in the guinea-pig oesophageal sphincter.
    Journal of autonomic pharmacology, 1998, Volume: 18, Issue:5

    Topics: Animals; Dipeptides; Diphenhydramine; Dose-Response Relationship, Drug; Esophagogastric Junction; Evans Blue; Extravasation of Diagnostic and Therapeutic Materials; Guinea Pigs; Indoles; Inflammation; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Peptides, Cyclic; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P

1998
A substance P receptor antagonist (FK 888) modifies gut alterations induced by ionizing radiation.
    International journal of radiation biology, 1998, Volume: 74, Issue:5

    Topics: Animals; Dipeptides; Ileum; Indoles; Intestinal Mucosa; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Rats; Rats, Wistar; Substance P

1998