Page last updated: 2024-09-04

fidarestat and Diabetes Mellitus

fidarestat has been researched along with Diabetes Mellitus in 3 studies

*Diabetes Mellitus: A heterogeneous group of disorders characterized by HYPERGLYCEMIA and GLUCOSE INTOLERANCE. [MeSH]

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Demopoulos, VJ; Nicolaou, I1
El-Kabbani, O; Podjarny, A1
Aoki, T; Makino, M; Mizuno, K; Sassa, H; Sobajima, H; Suzuki, T; Taniko, K1

Reviews

1 review(s) available for fidarestat and Diabetes Mellitus

ArticleYear
Selectivity determinants of the aldose and aldehyde reductase inhibitor-binding sites.
    Cellular and molecular life sciences : CMLS, 2007, Volume: 64, Issue:15

    Topics: Aldehyde Reductase; Amino Acid Substitution; Animals; Catalytic Domain; Diabetes Mellitus; Enzyme Inhibitors; Glucose; Humans; Imidazolidines; In Vitro Techniques; Models, Molecular; Mutagenesis, Site-Directed; Protein Conformation; Recombinant Proteins

2007

Other Studies

2 other study(ies) available for fidarestat and Diabetes Mellitus

ArticleYear
Substituted pyrrol-1-ylacetic acids that combine aldose reductase enzyme inhibitory activity and ability to prevent the nonenzymatic irreversible modification of proteins from monosaccharides.
    Journal of medicinal chemistry, 2003, Jan-30, Volume: 46, Issue:3

    Topics: Acetates; Aldehyde Reductase; Animals; Diabetes Mellitus; Enzyme Inhibitors; Female; Fructose; Male; Monosaccharides; Oxidation-Reduction; Proteins; Pyrroles; Rats; Rats, Inbred F344; Serum Albumin; Structure-Activity Relationship

2003
Pharmacological properties of fidarestat, a potent aldose reductase inhibitor, clarified by using sorbitol in human and rat erythrocytes.
    Pharmacology, 2001, Volume: 62, Issue:4

    Topics: Age Factors; Aldehyde Reductase; Animals; Blood Glucose; Body Weight; Diabetes Mellitus; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Enzyme Inhibitors; Erythrocytes; Fasting; Female; Glycated Hemoglobin; Humans; Imidazoles; Imidazolidines; Male; Rats; Rats, Sprague-Dawley; Rhodanine; Sciatic Nerve; Sex Factors; Sorbitol; Thiazolidines

2001