Page last updated: 2024-10-28

fasudil and Lupus Erythematosus, Systemic

fasudil has been researched along with Lupus Erythematosus, Systemic in 2 studies

fasudil: intracellular calcium antagonist; structure in first source
fasudil : An isoquinoline substituted by a (1,4-diazepan-1-yl)sulfonyl group at position 5. It is a Rho-kinase inhibitor and its hydrochloride hydrate form is approved for the treatment of cerebral vasospasm and cerebral ischemia.

Lupus Erythematosus, Systemic: A chronic, relapsing, inflammatory, and often febrile multisystemic disorder of connective tissue, characterized principally by involvement of the skin, joints, kidneys, and serosal membranes. It is of unknown etiology, but is thought to represent a failure of the regulatory mechanisms of the autoimmune system. The disease is marked by a wide range of system dysfunctions, an elevated erythrocyte sedimentation rate, and the formation of LE cells in the blood or bone marrow.

Research Excerpts

ExcerptRelevanceReference
"Fasudil treatment significantly improved survival and decreased proteinuria, particularly when treatment was started at 18 weeks."1.38Administration of fasudil, a ROCK inhibitor, attenuates disease in lupus-prone NZB/W F1 female mice. ( Bhagat, G; Biswas, PS; Gupta, S; Pernis, AB; Song, L; Stirzaker, RA, 2012)

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Pernis, AB2
Ricker, E1
Weng, CH1
Rozo, C1
Yi, W1
Stirzaker, RA1
Biswas, PS1
Gupta, S1
Song, L1
Bhagat, G1

Reviews

1 review available for fasudil and Lupus Erythematosus, Systemic

ArticleYear
Rho Kinases in Autoimmune Diseases.
    Annual review of medicine, 2016, Volume: 67

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amides; Animals; Arthritis, Rheumatoid; Autoimmune Di

2016

Other Studies

1 other study available for fasudil and Lupus Erythematosus, Systemic

ArticleYear
Administration of fasudil, a ROCK inhibitor, attenuates disease in lupus-prone NZB/W F1 female mice.
    Lupus, 2012, Volume: 21, Issue:6

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Administration, Oral; Animals; Antigen-Antibody Compl

2012