Page last updated: 2024-09-05

etravirine and HIV

etravirine has been researched along with HIV in 27 studies

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's10 (37.04)29.6817
2010's15 (55.56)24.3611
2020's2 (7.41)2.80

Authors

AuthorsStudies
De Clercq, E; Du, D; Liu, H; Liu, X; Pannecouque, C; Rai, D; Tian, Y; Wang, L; Zhan, P1
Elgaher, WA; Hartmann, RW; Haupenthal, J; Mély, Y; Pires, M; Real, E; Saladini, F; Sharma, KK1
Chen, FE; Gu, SX; Liu, GY; Meng, G; Pannecouque, C; Tang, JF; Wu, FS; Xiao, T; Xu, ZQ; Zhu, YY1
De Clercq, E; Gao, P; Liu, X; Pannecouque, C; Song, S; Sun, L; Wang, Z; Zhan, P; Zhang, J1
Challenger, E; Clotet, B; Curran, A; Khoo, S; Miranda, C; Moltó, J; Ribera, E; Santos, JR; Valle, M1
Kichula, E; Lynch, DR; Schadt, K1
Borghetti, A; D'Avino, A; De Luca, A; Del Puente, F; Di Biagio, A; Irene Bonelli, S; Riccardi, N; Taramasso, L; Zazzi, M1
DeMasi, R; Kakuda, TN; Mohammed, P; van Delft, Y1
Bell, CS; Contreras, GA; Del Bianco, GP; Heresi, GP; Kleinosky, MT; Murphy, JR; Pérez, N1
Aldieri, C; Bonora, S; Calcagno, A; Carbone, A; Castagna, A; D'Avolio, A; Di Perri, G; Ghisetti, V; Marinaro, L; Nozza, S; Trentalange, A1
Bañón, S; Casado, JL; Moreno, A; Moreno, S; Rodriguez, MA1
Belkhir, L; Capron, A; De Laveleye, M; Delongie, KA; Elens, L; Haufroid, V; Vandercam, B; Vincent, A; Yombi, J; Zech, F1
Cartledge, JD; Lascar, M1
Couzigou, C; Escaut, L; Morand-Joubert, L; Roque-Afonso, AM; Seang, S; Vittecoq, D1
García Deltoro, M1
Sanne, I; Stevens, WS; Venter, F; Wallis, CL1
Antinori, A; Ceccherini-Silberstein, F; Cozzi-Lepri, A; Monforte, Ad; Mussini, C; Palamara, G; Perno, CF; Santoro, MM; Spagnuolo, V; Zaccarelli, M1
Arribas, JR1
Castagna, A; De Wit, S; Florence, E; Hill, A; Marks, S; Ribera, E; van Delft, Y; Vanaken, H1
Aleixo, AW; Arruda, MB; de M Brindeiro, R; Greco, DB; Martins, AN; Pires, AF; Tanuri, A1
Durant, J; Duvivier, C; Fätkenheuer, G; Hill, A; Marks, S; Rey, D; Rieger, A; Schmidt, W; van Delft, Y1
Dilanchian, P; Jayaweera, D1
Nelson, MR; Waters, L1
Alcorn, K1
Geretti, AM1
Stephenson, J1

Reviews

6 review(s) available for etravirine and HIV

ArticleYear
New protease inhibitors and non-nucleoside reverse transcriptase inhibitors.
    Journal of HIV therapy, 2008, Volume: 13, Issue:2

    Topics: Clinical Trials as Topic; Darunavir; Drug Resistance, Viral; Drug Therapy, Combination; HIV; HIV Infections; HIV Protease Inhibitors; Humans; Nitriles; Pyridazines; Pyridines; Pyrimidines; Pyrones; Sulfonamides; Treatment Outcome

2008
[Resistance to darunavir].
    Enfermedades infecciosas y microbiologia clinica, 2008, Volume: 26 Suppl 10

    Topics: Adult; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Darunavir; Dose-Response Relationship, Drug; Drug Resistance, Viral; Female; HIV; HIV Infections; HIV Protease; HIV Protease Inhibitors; Humans; Lopinavir; Male; Multicenter Studies as Topic; Mutagenesis, Site-Directed; Mutation, Missense; Nitriles; Phenotype; Point Mutation; Pyridazines; Pyrimidines; Pyrimidinones; Randomized Controlled Trials as Topic; Sulfonamides

2008
Drugs in traditional drug classes (nucleoside reverse transcriptase inhibitor/nonnucleoside reverse transcriptase inhibitor/protease inhibitors) with activity against drug-resistant virus (tipranavir, darunavir, etravirine).
    Current opinion in HIV and AIDS, 2009, Volume: 4, Issue:6

    Topics: Anti-HIV Agents; Darunavir; Drug Resistance, Viral; HIV; HIV Infections; HIV Protease Inhibitors; Humans; Nitriles; Pyridazines; Pyridines; Pyrimidines; Pyrones; Ritonavir; Sulfonamides

2009
New therapeutic landscape of NNRTIs for treatment of HIV: a look at recent data.
    Expert opinion on pharmacotherapy, 2012, Volume: 13, Issue:18

    Topics: Antiretroviral Therapy, Highly Active; Clinical Trials as Topic; Drug Resistance, Viral; HIV; HIV Infections; Humans; Nitriles; Pyridazines; Pyrimidines; Reverse Transcriptase Inhibitors; Rilpivirine

2012
New drugs.
    HIV medicine, 2005, Volume: 6, Issue:4

    Topics: Anti-HIV Agents; Benzophenones; Cytidine Triphosphate; Darunavir; Deoxycytidine; Emtricitabine; HIV; HIV Fusion Inhibitors; HIV Reverse Transcriptase; Humans; Imidazoles; Nitriles; Protease Inhibitors; Pyridazines; Pyridines; Pyrimidines; Pyrones; Reverse Transcriptase Inhibitors; Sulfonamides; Sulfur Compounds; Zalcitabine

2005
Resistance testing methodologies and mechanisms of resistance.
    Journal of HIV therapy, 2007, Volume: 12, Issue:4

    Topics: Adenine; Anti-HIV Agents; CCR5 Receptor Antagonists; Drug Resistance, Viral; HIV; Humans; Lopinavir; Nitriles; Organophosphonates; Pyridazines; Pyrimidines; Pyrimidinones; Tenofovir

2007

Trials

4 trial(s) available for etravirine and HIV

ArticleYear
Pharmacokinetics of darunavir/cobicistat and etravirine alone and co-administered in HIV-infected patients.
    The Journal of antimicrobial chemotherapy, 2018, 03-01, Volume: 73, Issue:3

    Topics: Adult; Anti-HIV Agents; Cobicistat; Cohort Studies; Darunavir; Drug Therapy, Combination; Female; HIV; HIV Infections; HIV Protease Inhibitors; Humans; Male; Middle Aged; Nitriles; Pyridazines; Pyrimidines; RNA, Viral; Young Adult

2018
Pharmacokinetic interaction between etravirine or darunavir/ritonavir and artemether/lumefantrine in healthy volunteers: a two-panel, two-way, two-period, randomized trial.
    HIV medicine, 2013, Volume: 14, Issue:7

    Topics: Adult; Anti-HIV Agents; Antimalarials; Artemether; Artemisinins; Cross-Over Studies; Darunavir; Drug Interactions; Ethanolamines; Fluorenes; Healthy Volunteers; HIV; HIV Infections; Humans; Lumefantrine; Malaria; Middle Aged; Nitriles; Pyridazines; Pyrimidines; Ritonavir; Sulfonamides

2013
HIV RNA suppression rates after 24 weeks of treatment with etravirine, darunavir/ritonavir and raltegravir in the etravirine early access programme.
    International journal of STD & AIDS, 2010, Volume: 21, Issue:3

    Topics: Antiretroviral Therapy, Highly Active; CD4 Lymphocyte Count; Cohort Studies; Darunavir; Drug Administration Schedule; Female; HIV; HIV Infections; Humans; Immunosuppression Therapy; Male; Middle Aged; Nitriles; Pyridazines; Pyrimidines; Pyrrolidinones; Raltegravir Potassium; Reverse Transcriptase Inhibitors; Ritonavir; RNA, Viral; Sulfonamides; Treatment Outcome

2010
Lipid profiles for etravirine versus efavirenz in treatment-naive patients in the randomized, double-blind SENSE trial.
    The Journal of antimicrobial chemotherapy, 2012, Volume: 67, Issue:3

    Topics: Adolescent; Adult; Aged; Alkynes; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Benzoxazines; Cyclopropanes; Double-Blind Method; Female; HIV; HIV Infections; Humans; Lipids; Male; Middle Aged; Nitriles; Placebos; Pyridazines; Pyrimidines; Viral Load; Young Adult

2012

Other Studies

17 other study(ies) available for etravirine and HIV

ArticleYear
Fused heterocyclic compounds bearing bridgehead nitrogen as potent HIV-1 NNRTIs. Part 1: design, synthesis and biological evaluation of novel 5,7-disubstituted pyrazolo[1,5-a]pyrimidine derivatives.
    Bioorganic & medicinal chemistry, 2014, Apr-01, Volume: 22, Issue:7

    Topics: Anti-HIV Agents; Dose-Response Relationship, Drug; Drug Design; Heterocyclic Compounds; HIV; HIV Reverse Transcriptase; Microbial Sensitivity Tests; Models, Molecular; Molecular Structure; Nitrogen; Pyrazoles; Pyrimidines; Reverse Transcriptase Inhibitors; Structure-Activity Relationship

2014
Discovery and Structure-Based Optimization of 2-Ureidothiophene-3-carboxylic Acids as Dual Bacterial RNA Polymerase and Viral Reverse Transcriptase Inhibitors.
    Journal of medicinal chemistry, 2016, Aug-11, Volume: 59, Issue:15

    Topics: Anti-Bacterial Agents; Anti-HIV Agents; Carboxylic Acids; DNA-Directed RNA Polymerases; Dose-Response Relationship, Drug; Drug Discovery; Enzyme Inhibitors; Escherichia coli; HEK293 Cells; HeLa Cells; HIV; Humans; Microbial Sensitivity Tests; Molecular Structure; RNA-Directed DNA Polymerase; Structure-Activity Relationship; Thiophenes

2016
Indazolyl-substituted piperidin-4-yl-aminopyrimidines as HIV-1 NNRTIs: Design, synthesis and biological activities.
    European journal of medicinal chemistry, 2020, Jan-15, Volume: 186

    Topics: Anti-HIV Agents; Dose-Response Relationship, Drug; Drug Design; HIV; HIV Reverse Transcriptase; Humans; Indazoles; Microbial Sensitivity Tests; Molecular Structure; Piperidines; Pyrimidines; Reverse Transcriptase Inhibitors; Structure-Activity Relationship

2020
Design, synthesis and anti-HIV evaluation of novel 5-substituted diarylpyrimidine derivatives as potent HIV-1 NNRTIs.
    Bioorganic & medicinal chemistry, 2021, 06-15, Volume: 40

    Topics: Anti-HIV Agents; Cell Line, Tumor; Dose-Response Relationship, Drug; Drug Design; HIV; HIV Reverse Transcriptase; Humans; Microbial Sensitivity Tests; Models, Molecular; Molecular Structure; Pyrimidines; Reverse Transcriptase Inhibitors; Structure-Activity Relationship

2021
Etravirine in Friedreich's ataxia: Lessons from HIV?
    Movement disorders : official journal of the Movement Disorder Society, 2019, Volume: 34, Issue:3

    Topics: Drug Repositioning; Friedreich Ataxia; HIV; Humans; Nitriles; Pyridazines; Pyrimidines

2019
Is it time to re-think the use of etravirine in patients with available genotypic resistance test?
    Infectious diseases (London, England), 2019, Volume: 51, Issue:6

    Topics: HIV; HIV Infections; Humans; Nitriles; Pyridazines; Pyrimidines; Sweden

2019
Prevalence and risk factors associated with resistance-associated mutations to etravirine in a cohort of perinatally HIV-infected children.
    The Journal of antimicrobial chemotherapy, 2013, Volume: 68, Issue:10

    Topics: Anti-HIV Agents; Child; Child, Preschool; Cohort Studies; Drug Resistance, Viral; Female; HIV; HIV Infections; Humans; Male; Mutation, Missense; Nitriles; Prevalence; Pyridazines; Pyrimidines; Retrospective Studies; Risk Factors

2013
Etravirine plasma exposure is associated with virological efficacy in treatment-experienced HIV-positive patients.
    Antiviral research, 2014, Volume: 108

    Topics: Adult; CD4 Lymphocyte Count; Female; HIV; HIV Infections; Humans; Male; Middle Aged; Nitriles; Plasma; Pyridazines; Pyrimidines; Retrospective Studies; Reverse Transcriptase Inhibitors; RNA, Viral; Treatment Outcome; Viral Load

2014
Efficacy and pharmacokinetics of the combination of etravirine plus raltegravir as novel dual antiretroviral maintenance regimen in HIV-infected patients.
    Antiviral research, 2015, Volume: 113

    Topics: Adult; Aged; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Female; Follow-Up Studies; HIV; HIV Infections; Humans; Male; Middle Aged; Nitriles; Prospective Studies; Pyridazines; Pyrimidines; Pyrrolidinones; Raltegravir Potassium; Viral Load

2015
Quantification of darunavir and etravirine in human peripheral blood mononuclear cells using high performance liquid chromatography tandem mass spectrometry (LC-MS/MS), clinical application in a cohort of 110 HIV-1 infected patients and evidence of a pote
    Clinical biochemistry, 2016, Volume: 49, Issue:7-8

    Topics: Biomarkers; Chromatography, High Pressure Liquid; Cohort Studies; Darunavir; Drug Interactions; Drug Monitoring; Female; Follow-Up Studies; HIV; HIV Infections; HIV Protease Inhibitors; Humans; Leukocytes, Mononuclear; Limit of Detection; Male; Middle Aged; Nitriles; Prognosis; Pyridazines; Pyrimidines; Reverse Transcriptase Inhibitors; Tandem Mass Spectrometry

2016
Efficacy of etravirine for treatment of acute HIV meningoencephalitis.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2009, Mar-15, Volume: 48, Issue:6

    Topics: Adult; Anti-HIV Agents; Cerebrospinal Fluid; Female; Hepatitis C; HIV; HIV Infections; Humans; Meningoencephalitis; Nitriles; Pyridazines; Pyrimidines; Treatment Outcome

2009
Will etravirine work in patients failing nonnucleoside reverse transcriptase inhibitor-based treatment in southern Africa?
    Journal of acquired immune deficiency syndromes (1999), 2009, Volume: 52, Issue:5

    Topics: Africa, Southern; Drug Resistance, Viral; HIV; HIV Infections; Humans; Mutation; Nitriles; Pyridazines; Pyrimidines; Reverse Transcriptase Inhibitors; Treatment Failure

2009
Is there any potential for first-line etravirine use? Analysis from a large data set of antiretroviral therapy-naive HIV-infected patients undergoing resistance test.
    Journal of acquired immune deficiency syndromes (1999), 2010, Volume: 53, Issue:1

    Topics: Adolescent; Adult; Aged; Clinical Trials as Topic; Drug Resistance, Viral; Female; HIV; HIV Infections; Humans; Male; Middle Aged; Mutation; Nitriles; Pyridazines; Pyrimidines; Young Adult

2010
Prevalence of etravirine-associated mutations in clinical samples with genotypic resistance to nevirapine and efavirenz in Brazilian clinics.
    Journal of acquired immune deficiency syndromes (1999), 2011, Volume: 57 Suppl 3

    Topics: Alkynes; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Benzoxazines; Brazil; Cyclopropanes; Drug Resistance, Viral; HIV; HIV Infections; Humans; Mutation, Missense; Nevirapine; Nitriles; Prevalence; Pyridazines; Pyrimidines

2011
TMC 125 possibly effective against NNRTI-resistant HIV.
    IAPAC monthly, 2004, Volume: 10, Issue:1

    Topics: Drug Resistance, Viral; HIV; HIV Infections; Humans; Mutation; Nitriles; Pyridazines; Pyrimidines; Reverse Transcriptase Inhibitors; Virus Replication

2004
TMC125 study highlights failing NNRTI regimen task.
    IAPAC monthly, 2006, Volume: 12, Issue:11

    Topics: Clinical Trials, Phase II as Topic; Drug Resistance, Viral; HIV; Humans; Mutation; Nitriles; Pyridazines; Pyrimidines; Randomized Controlled Trials as Topic; Reverse Transcriptase Inhibitors; Viral Load

2006
Researchers explore new anti-HIV agents.
    JAMA, 2002, Apr-03, Volume: 287, Issue:13

    Topics: Anti-HIV Agents; CCR5 Receptor Antagonists; Clinical Trials as Topic; Cyclic N-Oxides; Drugs, Investigational; Enfuvirtide; Furans; HIV; HIV Envelope Protein gp120; HIV Envelope Protein gp41; HIV Infections; HIV Integrase Inhibitors; Humans; Nitriles; Oximes; Peptide Fragments; Piperazines; Piperidines; Pyridazines; Pyridines; Pyrimidines; Reverse Transcriptase Inhibitors; Triazoles

2002
chemdatabank.com