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ethylketocyclazocine and Muscle Contraction

ethylketocyclazocine has been researched along with Muscle Contraction in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-199020 (86.96)18.7374
1990's3 (13.04)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Corbett, AD; Gillan, MG; Kosterlitz, HW; McKnight, AT; Paterson, SJ; Robson, LE1
Huidobro-Toro, JP; Lee, NM; Loh, HH; Way, EL; Yoshimura, K3
Dickinson, SL; Slater, P1
Huidobro-Toro, JP; Lee, NM; Loh, HH; Way, EL; Zhu, YX1
Rezvani, A; Way, EL1
Fujino, M; Negishi, K; Oka, T; Sawa, A; Suda, M; Wakimasu, M1
Ishizuka, Y; Kajiwara, M; Matsumiya, T; Negishi, K; Oka, T; Watanabe, Y1
Bajusz, S; Berzétei, IP; Hársing, LG; Rónai, AZ; Vizi, ES1
Berzetei-Gurske, IP; Toll, L1
al-Shireida, MF; el-Sharkawy, TY; Pilcher, CW1
Jhamandas, K; Lapierre, C; Lemaire, S; Martinka, GP; Sabourin, L1
Friedmann, T; Furst, S; Kovacs, A; Wagner, T1
Cho, N; Hirobe, M; Koike, K; Konno, F; Okumura, K; Takayanagi, I1
Cho, N; Hirobe, M; Kobayashi, C; Konno, F; Morimoto, R; Takayanagi, I1
Hayes, A; Kelly, A1
Aoki, K; Ishii, K; Kajiwara, M; Matsumiya, T; Numata, H; Oka, T1
Larson, DL; Portoghese, PS; Ronsisvalle, G; Takemori, AE1
Seelhorst, A; Starke, K1
Hynes, MD; Leander, JD; Reel, JK; Zimmerman, DM1
Kadlec, O; Masek, K; Sebestová, L; Seferna, I1
Kadlec, O; Masek, K; Seferna, I1

Other Studies

23 other study(ies) available for ethylketocyclazocine and Muscle Contraction

ArticleYear
Radioligands for probing opioid receptors.
    Journal of receptor research, 1984, Volume: 4, Issue:1-6

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Binding Sites; Brain; Cyclazocine; Diprenorphine; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Naloxone; Pro-Opiomelanocortin; Protein Precursors; Pyrrolidines; Radioligand Assay; Rats; Receptors, Opioid; Vas Deferens

1984
Dynorphin interaction at the kappa-opiate site.
    European journal of pharmacology, 1981, Jun-19, Volume: 72, Issue:2-3

    Topics: Animals; Cyclazocine; Dynorphins; Electric Stimulation; Endorphins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Receptors, Opioid; Receptors, Opioid, kappa

1981
Opiate receptor antagonism by L-prolyl-L-leucyl-glycinamide, MIF-I.
    Peptides, 1980,Winter, Volume: 1, Issue:4

    Topics: Animals; Cyclazocine; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Female; Ileum; In Vitro Techniques; Male; Mice; Morphine; Motor Activity; MSH Release-Inhibiting Hormone; Muscle Contraction; Pain; Rats; Rats, Inbred Strains; Receptors, Opioid; Vas Deferens

1980
Kappa opioid properties of dynorphin and its peptide fragments on the guinea-pig Ileum.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 222, Issue:1

    Topics: Animals; Cyclazocine; Drug Interactions; Drug Tolerance; Dynorphins; Endorphins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Naloxone; Peptide Fragments; Receptors, Opioid; Receptors, Opioid, kappa

1982
Activation of K-opiate sites by dynorphin in the myenteric plexus.
    Advances in biochemical psychopharmacology, 1982, Volume: 33

    Topics: Animals; Cyclazocine; Drug Tolerance; Dynorphins; Electric Stimulation; Endorphins; Enkephalin, Leucine; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Narcotics; Receptors, Opioid; Receptors, Opioid, kappa

1982
Dynorphin inhibition of the neurotensin contractile activity on the myenteric plexus.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 228, Issue:2

    Topics: Animals; Atropine; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Dynorphins; Endorphins; Ethylketocyclazocine; Guinea Pigs; Ileum; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Naloxone; Nerve Tissue Proteins; Neurotensin; Peptide Fragments; Receptors, Opioid; Tetrodotoxin

1984
Dynorphin-(1-13) restores the potency of morphine on the tolerant guinea pig ileum.
    European journal of pharmacology, 1984, Jul-20, Volume: 102, Issue:3-4

    Topics: Animals; beta-Endorphin; Cyclazocine; Drug Interactions; Drug Tolerance; Dynorphins; Endorphins; Enkephalin, Leucine; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphine; Muscle Contraction; Muscle, Smooth; Naloxone; Peptide Fragments

1984
Evidence that dynorphin-(1-13) acts as an agonist on opioid kappa-receptors.
    European journal of pharmacology, 1982, Jan-22, Volume: 77, Issue:2-3

    Topics: Animals; Cyclazocine; Dynorphins; Electric Stimulation; Endorphins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Muscle Contraction; Muscle, Smooth; Naloxone; Peptide Fragments; Rabbits; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Vas Deferens

1982
The choice of opiate receptor subtype by neo-endorphins.
    European journal of pharmacology, 1982, Apr-23, Volume: 79, Issue:3-4

    Topics: Animals; Benzomorphans; beta-Endorphin; Cyclazocine; Drug Interactions; Endorphins; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Naloxone; Protein Precursors; Rabbits; Receptors, Opioid

1982
[Met5]enkephalin-Arg-Phe ACTS on vascular opiate receptors.
    European journal of pharmacology, 1982, Apr-23, Volume: 79, Issue:3-4

    Topics: Animals; Cyclazocine; Electric Stimulation; Endorphins; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Rabbits; Receptors, Opioid

1982
The mu-opioid activity of kappa-opioid receptor agonist compounds in the guinea pig ileum.
    European journal of pharmacology, 1992, Mar-03, Volume: 212, Issue:2-3

    Topics: Animals; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nalorphine; Naltrexone; Phenazocine; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1992
Vascular effects of some opioid receptor agonists.
    Canadian journal of physiology and pharmacology, 1991, Volume: 69, Issue:6

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzomorphans; Calcium Channel Blockers; Dinoprost; Endothelium, Vascular; Ethylketocyclazocine; In Vitro Techniques; Male; Morphine; Muscle Contraction; Muscle, Smooth, Vascular; Narcotic Antagonists; Norepinephrine; Potassium; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Vasodilation

1991
Dynorphin A-(1-13)-Tyr14-Leu15-Phe16-Asn17-Gly18-Pro19 : a potent and selective kappa opioid peptide.
    European journal of pharmacology, 1991, Apr-17, Volume: 196, Issue:2

    Topics: Amino Acid Sequence; Animals; Dynorphins; Ethylketocyclazocine; Guinea Pigs; Kinetics; Male; Mice; Molecular Sequence Data; Muscle Contraction; Nociceptors; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1991
Comparison of the opioid activity of CAM and kappa agonists.
    NIDA research monograph, 1986, Volume: 75

    Topics: Animals; Cyclazocine; Diuresis; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Morphinans; Muscle Contraction; Narcotic Antagonists; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1986
Intrinsic activity and effects of guanyl-5'-yl imidodiphosphate, Gpp(NH)p and sodium ion on the affinity of dynorphin 1-13, nalorphine and nalorphine-7,8-oxide to kappa-opioid receptor.
    General pharmacology, 1985, Volume: 16, Issue:6

    Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Dynorphins; Ethylketocyclazocine; Guanosine Triphosphate; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle, Smooth; Nalorphine; Naloxone; Peptide Fragments; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Sodium; Synaptosomes; Vas Deferens

1985
Pharmacological effects of nalorphine and nalorphine-7,8-oxide (nalorphine-epoxide): interaction of the intrinsic activity, affinity and pharmacological responses.
    Archives internationales de pharmacodynamie et de therapie, 1986, Volume: 282, Issue:2

    Topics: Analgesics; Animals; Brain; Cyclazocine; Dihydromorphine; Dynorphins; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Nalorphine; Peptide Fragments; Rabbits; Rats; Rats, Inbred Strains; Reaction Time; Receptors, Opioid

1986
Profile of activity of kappa receptor agonists in the rabbit vas deferens.
    European journal of pharmacology, 1985, Apr-16, Volume: 110, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Butorphanol; Cyclazocine; Ethylketocyclazocine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nalorphine; Naloxone; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Vas Deferens

1985
Agonist and antagonist actions of buprenorphine on three types of opioid receptor in isolated preparations.
    Japanese journal of pharmacology, 1986, Volume: 40, Issue:1

    Topics: Animals; Benzomorphans; Buprenorphine; Cyclazocine; Electric Stimulation; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Morphinans; Morphine; Muscle Contraction; Muscle, Smooth; Naloxone; Rabbits; Rats; Rats, Inbred Strains; Receptors, Opioid; Species Specificity; Time Factors; Vas Deferens

1986
Synthesis and opioid antagonist potencies of naltrexamine bivalent ligands with conformationally restricted spacers.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:9

    Topics: Animals; Biological Assay; Chemical Phenomena; Chemistry; Cyclazocine; Endorphins; Ethylketocyclazocine; Guinea Pigs; Ileum; Molecular Conformation; Morphine; Muscle Contraction; Naltrexone; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Structure-Activity Relationship

1986
Prejunctional opioid receptors in the pulmonary artery of the rabbit.
    Archives internationales de pharmacodynamie et de therapie, 1986, Volume: 281, Issue:2

    Topics: Animals; Cyclazocine; Electric Stimulation; Ethylketocyclazocine; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Naloxone; Narcotics; Norepinephrine; Pulmonary Artery; Rabbits; Receptors, Opioid; Tetrodotoxin

1986
Use of beta-funaltrexamine to determine mu opioid receptor involvement in the analgesic activity of various opioid ligands.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Animals; Biological Assay; Buprenorphine; Butorphanol; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Etorphine; Fentanyl; Methadone; Mice; Morphine; Muscle Contraction; Nalbuphine; Nalorphine; Naltrexone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, mu

1987
The topography and dynamics of cholinergic transmission in the myenteric plexus-smooth muscle preparation of the guinea-pig ileum; the effect of ketocyclazocine, a kappa opiate ligand.
    Physiologia Bohemoslovaca, 1987, Volume: 36, Issue:1

    Topics: Acetylcholine; Animals; Cyclazocine; Electric Stimulation; Electromyography; Ethylketocyclazocine; Guinea Pigs; Ileum; Ligands; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Narcotics; Parasympathetic Nervous System; Synaptic Transmission

1987
The topography of cholinergic transmission in the mechanism of drug action at muscarinic synapses of the guinea-pig ileum.
    European journal of pharmacology, 1987, Apr-14, Volume: 136, Issue:2

    Topics: Action Potentials; Animals; Axons; Cholinergic Fibers; Cyclazocine; Electric Stimulation; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Synaptic Transmission

1987