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ethylketocyclazocine and Ache

ethylketocyclazocine has been researched along with Ache in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-199021 (84.00)18.7374
1990's3 (12.00)18.2507
2000's1 (4.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Domino, EF; Gwynn, GJ1
Dickinson, SL; Slater, P1
Tung, AS; Yaksh, TL1
Sewell, RD; Spencer, PS; Upton, N1
Kamerling, SG; Martin, WR; Wettstein, JG; Wu, KM2
Han, JS; Xie, GX1
Bakthavachalam, V; Bidlack, JM; Cohen, DJ; Gao, P; Mello, NK; Negus, SS; Neumeyer, JL; Zong, R1
Gent, JP; Goodchild, CS; Serrao, JM1
Abbott, FV2
Edwards, M; Gent, JP; Goodchild, CS; Serrao, JM1
Dequick, DJ; Kamerling, SG; Tobin, T; Weckman, TJ1
Inoki, R; Kudo, T; Ohkubo, T; Shibata, M; Takahashi, H1
Russell, NJ; Schaible, HG; Schmidt, RF1
Dickenson, AH; Knox, RJ1
Candeletti, S; Cavicchini, E; Ferri, S; Romualdi, P; Spampinato, S; Speroni, E1
Kitchen, I; McDowell, J1
Kameyama, T; Matsuno, K; Nabeshima, T1
Hayes, AG; Skingle, M; Tyers, MB1
Barr, GA; Erickson, KL; Paredes, W; Zukin, RS1
Abbott, FV; Franklin, KB; Libman, RB1
Barr, GA; Giordano, J2
Belknap, JK; Danielson, PW; Laursen, SE; Noordewier, B1

Other Studies

25 other study(ies) available for ethylketocyclazocine and Ache

ArticleYear
Genotype-dependent behavioral sensitivity to mu vs. kappa opiate agonists. II. Antinociceptive tolerance and physical dependence.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 231, Issue:2

    Topics: Analgesics; Animals; Cyclazocine; Drug Tolerance; Ethylketocyclazocine; Genotype; Humans; Male; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Morphine; Opioid-Related Disorders; Pain; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Species Specificity

1984
Opiate receptor antagonism by L-prolyl-L-leucyl-glycinamide, MIF-I.
    Peptides, 1980,Winter, Volume: 1, Issue:4

    Topics: Animals; Cyclazocine; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Female; Ileum; In Vitro Techniques; Male; Mice; Morphine; Motor Activity; MSH Release-Inhibiting Hormone; Muscle Contraction; Pain; Rats; Rats, Inbred Strains; Receptors, Opioid; Vas Deferens

1980
In vivo evidence for multiple opiate receptors mediating analgesia in the rat spinal cord.
    Brain research, 1982, Sep-09, Volume: 247, Issue:1

    Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Injections, Spinal; Male; Naloxone; Pain; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Spinal Cord

1982
Analgesic actions of mu- and kappa-opiate agonists in rats.
    Archives internationales de pharmacodynamie et de therapie, 1983, Volume: 262, Issue:2

    Topics: Analgesics, Opioid; Animals; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Hot Temperature; Male; Nociceptors; Pain; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1983
Medullary kappa hyperalgesic mechanisms II. The effects of ethylketazocine administered into the fourth cerebral ventricle of the conscious dog.
    Life sciences, 1983, Oct-31, Volume: 33, Issue:18

    Topics: Analgesics, Opioid; Animals; Cerebral Ventricles; Cyclazocine; Dogs; Ethylketocyclazocine; Female; Injections; Medulla Oblongata; Pain; Receptors, Opioid; Reflex

1983
Possible medullary kappa hyperalgesic mechanism. I. A new potential role for endogenous opioid peptides in pain perception.
    Life sciences, 1983, Oct-31, Volume: 33, Issue:18

    Topics: Animals; Cyclazocine; Dogs; Dynorphins; Endorphins; Ethylketocyclazocine; Medulla Oblongata; Naloxone; Pain; Receptors, Opioid; Reflex

1983
[Dynorphin: analgesic effect via kappa receptors in spinal cord of the spinal cords of rats].
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1984, Volume: 5, Issue:4

    Topics: Analgesics; Animals; Cyclazocine; Dynorphins; Ethylketocyclazocine; Female; Morphine; Naloxone; Pain; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Sensory Thresholds; Spinal Cord

1984
Synthesis and opioid receptor affinity of morphinan and benzomorphan derivatives: mixed kappa agonists and mu agonists/antagonists as potential pharmacotherapeutics for cocaine dependence.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Acetic Acid; Animals; Benzomorphans; Brain; Dose-Response Relationship, Drug; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Morphinans; Morphine; Narcotic Antagonists; Pain; Pain Measurement; Reaction Time; Receptors, Opioid, kappa; Receptors, Opioid, mu

2000
Reversal by naloxone of spinal antinociceptive effects of fentanyl, ketocyclazocine and midazolam.
    European journal of anaesthesiology, 1991, Volume: 8, Issue:5

    Topics: Analgesia, Epidural; Animals; Catheters, Indwelling; Dose-Response Relationship, Drug; Drug Tolerance; Electric Stimulation; Ethylketocyclazocine; Fentanyl; Flumazenil; Injections, Spinal; Lumbar Vertebrae; Male; Midazolam; Naloxone; Nociceptors; Pain; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Opioid; Sensory Thresholds

1991
beta-Funaltrexamine antagonizes the analgesic effects of mu and kappa agonists in the formalin test.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 37, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Dose-Response Relationship, Drug; Ethylketocyclazocine; Formaldehyde; Male; Morphine; Naltrexone; Narcotic Antagonists; Pain; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Urination

1990
On the mechanism by which midazolam causes spinally mediated analgesia.
    Anesthesiology, 1990, Volume: 73, Issue:2

    Topics: Analgesia, Epidural; Animals; Bicuculline; Cyclazocine; Dose-Response Relationship, Drug; Electric Stimulation; Ethylketocyclazocine; Fentanyl; Flumazenil; Male; Midazolam; Pain; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sensory Thresholds

1990
Dose-related effects of ethylketazocine on nociception, behaviour and autonomic responses in the horse.
    The Journal of pharmacy and pharmacology, 1986, Volume: 38, Issue:1

    Topics: Analgesics, Opioid; Animals; Autonomic Nervous System; Behavior, Animal; Body Temperature; Cyclazocine; Ethylketocyclazocine; Female; Horses; Male; Motor Activity; Pain; Pupil; Reaction Time

1986
[Peripheral analgesic actions of opioid peptides and morphine analogues].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1986, Volume: 88, Issue:2

    Topics: Analgesics, Opioid; Animals; Cyclazocine; Dynorphins; Enkephalin, Methionine; Ethylketocyclazocine; Levallorphan; Lidocaine; Male; Mice; Morphine; Naloxone; Pain; Peptide Fragments

1986
Opiates inhibit the discharges of fine afferent units from inflamed knee joint of the cat.
    Neuroscience letters, 1987, Apr-23, Volume: 76, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Arthritis; Cats; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ethylketocyclazocine; Morphine; Naloxone; Nociceptors; Pain; Peripheral Nerves; Pyrrolidines

1987
Effects of selective and non-selective kappa-opioid receptor agonists on cutaneous C-fibre-evoked responses of rat dorsal horn neurones.
    Brain research, 1987, Jul-07, Volume: 415, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Action Potentials; Animals; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Electric Stimulation; Ethylketocyclazocine; Injections, Spinal; Male; Naloxone; Nerve Fibers; Pain; Peptide Fragments; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Skin; Spinal Cord; Time Factors

1987
Investigations on dynorphin structurally-related opioid peptides. I. Impact on nociceptive transmission. II. Regulation of pituitary content.
    Annali dell'Istituto superiore di sanita, 1988, Volume: 24, Issue:3

    Topics: Animals; Benzomorphans; Cyclazocine; Dynorphins; Estradiol; Ethylketocyclazocine; Female; Hypothalamo-Hypophyseal System; Male; Ovary; Pain; Pain Measurement; Rats; Rats, Inbred Strains; Structure-Activity Relationship

1988
Peripheral and central antinociceptive actions of ethylketocyclazocine in the formalin test.
    European journal of pharmacology, 1988, Jul-26, Volume: 152, Issue:1-2

    Topics: Analgesics; Analgesics, Opioid; Animals; Behavior, Animal; Cyclazocine; Ethylketocyclazocine; Formaldehyde; Injections, Intraventricular; Male; Naloxone; Pain; Rats

1988
Impairment of ketocyclazocine antinociception in rats by perinatal lead exposure.
    Toxicology letters, 1985, Volume: 26, Issue:2-3

    Topics: Animals; Animals, Newborn; Animals, Suckling; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Female; Lead; Lead Poisoning; Pain; Pregnancy; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Sensory Thresholds

1985
Involvement of different opioid receptor subtypes in electric shock-induced analgesia and motor suppression in the rat.
    European journal of pharmacology, 1985, Aug-15, Volume: 114, Issue:2

    Topics: Animals; Cyclazocine; Electroshock; Enkephalin, Methionine; Ethylketocyclazocine; Male; Motor Activity; Naloxone; Pain; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Time Factors

1985
Reversal by beta-funaltrexamine of the antinociceptive effect of opioid agonists in the rat.
    British journal of pharmacology, 1986, Volume: 88, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Buprenorphine; Cyclazocine; Ethylketocyclazocine; Fentanyl; Male; Naltrexone; Pain; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1986
Kappa opioid receptor-mediated analgesia in the developing rat.
    Brain research, 1986, Volume: 394, Issue:2

    Topics: Age Factors; Animals; Brain; Cyclazocine; Drug Tolerance; Ethylketocyclazocine; Hot Temperature; Morphine; Pain; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1986
A dose-ratio comparison of mu and kappa agonists in formalin and thermal pain.
    Life sciences, 1986, Nov-24, Volume: 39, Issue:21

    Topics: Analgesia; Animals; Benzomorphans; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Fentanyl; Formaldehyde; Hot Temperature; Male; Naloxone; Pain; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sufentanil

1986
Morphine- and ketocyclazocine-induced analgesia in the developing rat: differences due to type of noxious stimulus and body topography.
    Brain research, 1987, Volume: 429, Issue:2

    Topics: Age Factors; Analgesics; Animals; Animals, Suckling; Central Nervous System; Cyclazocine; Ethylketocyclazocine; Morphine; Naloxone; Pain; Pain Measurement; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1987
Effects of neonatal spinal cord serotonin depletion on opiate-induced analgesia in tests of thermal and mechanical pain.
    Brain research, 1988, Jun-01, Volume: 469, Issue:1-2

    Topics: 5,7-Dihydroxytryptamine; Analgesia; Animals; Animals, Newborn; Cyclazocine; Desipramine; Dihydroxytryptamines; Ethylketocyclazocine; Hot Temperature; Morphine; Pain; Physical Stimulation; Rats; Serotonin; Spinal Cord

1988
Selective breeding for levorphanol-induced antinociception on the hot-plate assay: commonalities in mechanism of action with morphine, pentazocine, ethylketocyclazocine, U-50488H and clonidine in mice.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Animals; Clonidine; Cyclazocine; Ethylketocyclazocine; Female; Levorphanol; Male; Mice; Morphine; Narcotics; Pain; Pentazocine; Pyrrolidines

1987