Page last updated: 2024-08-21

emetine and Malaria

emetine has been researched along with Malaria in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19907 (43.75)18.7374
1990's0 (0.00)18.2507
2000's1 (6.25)29.6817
2010's8 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Adrián, F; Anderson, P; Brinker, A; Caldwell, JS; Chatterjee, A; Gray, NS; Henson, K; Janes, J; Kato, N; Kuhen, K; Matzen, JT; McNamara, C; Nagle, A; Nam, TG; Plouffe, D; Schultz, PG; Trager, R; Winzeler, EA; Yan, SF; Zhou, Y1
Chibale, K; Egan, TJ; Hunter, R; Joshi, MC; Martin, RE; Smith, PJ; Summers, RL; Zishiri, VK1
Barnes, SW; Bonamy, GM; Bopp, SE; Borboa, R; Bright, AT; Chatterjee, A; Che, J; Cohen, S; Dharia, NV; Diagana, TT; Fidock, DA; Froissard, P; Gagaring, K; Gettayacamin, M; Glynne, RJ; Gordon, P; Groessl, T; Kato, N; Kuhen, KL; Lee, MC; Mazier, D; McNamara, CW; Meister, S; Nagle, A; Nam, TG; Plouffe, DM; Richmond, W; Roland, J; Rottmann, M; Sattabongkot, J; Schultz, PG; Tuntland, T; Walker, JR; Winzeler, EA; Wu, T; Zhou, B; Zhou, Y1
Fortuin, EE; Joubert, J; Malan, SF; Smith, PJ; Taylor, D1
Chibale, K; Egan, TJ; Jurva, U; Masimirembwa, CM; Njoroge, M; Ongarora, DS; Strydom, N; Wicht, K; Wiesner, L; Wittlin, S1
Hoppe, HC; Isaacs, M; Khanye, SD; Svogie, AL; Veale, CG1
Barnard, L; Birkholtz, LM; Botha, M; Brunschwig, C; Burrows, JN; Chibale, K; Churchyard, A; Coetzer, TL; Denti, P; Egan, TJ; Laing, L; Lauterbach, S; Machado, M; Ndubi, F; Njogu, PM; Njoroge, M; Nondaba, S; Okombo, J; Prudêncio, M; Reader, J; Singh, K; Wiesner, L; Wilkinson, C; Wittlin, S; Yeates, C1
Chibale, K; Egan, TJ; Hunter, R; Joshi, MC; Ndove, J; Nsumiwa, S; Okombo, J; Taylor, D; Wiesner, L1
Baartzes, N; Chibale, K; Seldon, R; Smith, GS; Stringer, T; Taylor, D; Warner, DF; Wittlin, S1
DURIEUX, C; TANGUY, F; TRENOUS, J1
TELLA, A1
Degrémont, A1
Fernex, M1
James, RF1
Esposito, R1
Brossi, A1

Other Studies

16 other study(ies) available for emetine and Malaria

ArticleYear
In silico activity profiling reveals the mechanism of action of antimalarials discovered in a high-throughput screen.
    Proceedings of the National Academy of Sciences of the United States of America, 2008, Jul-01, Volume: 105, Issue:26

    Topics: Animals; Antimalarials; Cluster Analysis; Computational Biology; Drug Evaluation, Preclinical; Drug Resistance; Folic Acid Antagonists; Malaria; Models, Molecular; Parasites; Plasmodium falciparum; Reproducibility of Results; Structure-Activity Relationship; Tetrahydrofolate Dehydrogenase

2008
Quinoline antimalarials containing a dibemethin group are active against chloroquinone-resistant Plasmodium falciparum and inhibit chloroquine transport via the P. falciparum chloroquine-resistance transporter (PfCRT).
    Journal of medicinal chemistry, 2011, Oct-13, Volume: 54, Issue:19

    Topics: Animals; Antimalarials; Biological Transport; Cell Survival; Chloroquine; CHO Cells; Cricetinae; Cricetulus; Crystallography, X-Ray; Female; Malaria; Membrane Transport Proteins; Mice; Molecular Structure; Oocytes; Parasitemia; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Protozoan Proteins; Structure-Activity Relationship; Xenopus laevis

2011
Imaging of Plasmodium liver stages to drive next-generation antimalarial drug discovery.
    Science (New York, N.Y.), 2011, Dec-09, Volume: 334, Issue:6061

    Topics: Animals; Antimalarials; Cell Line, Tumor; Drug Discovery; Drug Evaluation, Preclinical; Drug Resistance; Erythrocytes; Humans; Imidazoles; Liver; Malaria; Mice; Mice, Inbred BALB C; Molecular Structure; Piperazines; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Plasmodium yoelii; Polymorphism, Single Nucleotide; Protozoan Proteins; Random Allocation; Small Molecule Libraries; Sporozoites

2011
Pentacycloundecylamines and conjugates thereof as chemosensitizers and reversed chloroquine agents.
    Bioorganic & medicinal chemistry letters, 2014, Dec-01, Volume: 24, Issue:23

    Topics: Amines; Antimalarials; Chloroquine; Humans; Malaria; Molecular Structure

2014
Antimalarial benzoheterocyclic 4-aminoquinolines: Structure-activity relationship, in vivo evaluation, mechanistic and bioactivation studies.
    Bioorganic & medicinal chemistry, 2015, Sep-01, Volume: 23, Issue:17

    Topics: Aminoquinolines; Animals; Antimalarials; Benzene Derivatives; Humans; Malaria; Malaria, Falciparum; Mice; Mice, Inbred C57BL; Plasmodium berghei; Plasmodium falciparum; Structure-Activity Relationship

2015
Indolyl-3-ethanone-α-thioethers: A promising new class of non-toxic antimalarial agents.
    European journal of medicinal chemistry, 2016, May-23, Volume: 114

    Topics: Antimalarials; Dose-Response Relationship, Drug; HeLa Cells; Humans; Indoles; Malaria; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship; Sulfides

2016
Antimalarial Pyrido[1,2-a]benzimidazoles: Lead Optimization, Parasite Life Cycle Stage Profile, Mechanistic Evaluation, Killing Kinetics, and in Vivo Oral Efficacy in a Mouse Model.
    Journal of medicinal chemistry, 2017, 02-23, Volume: 60, Issue:4

    Topics: Animals; Antimalarials; Benzimidazoles; Life Cycle Stages; Malaria; Male; Mice; Plasmodium berghei; Structure-Activity Relationship

2017
4-Aminoquinoline Antimalarials Containing a Benzylmethylpyridylmethylamine Group Are Active against Drug Resistant Plasmodium falciparum and Exhibit Oral Activity in Mice.
    Journal of medicinal chemistry, 2017, 12-28, Volume: 60, Issue:24

    Topics: Administration, Oral; Aminopyridines; Aminoquinolines; Animals; Antimalarials; Cell Membrane Permeability; Chloroquine; CHO Cells; Cricetulus; Drug Evaluation, Preclinical; Drug Resistance, Microbial; ERG1 Potassium Channel; Hemeproteins; Humans; Malaria; Male; Mice, Inbred BALB C; Plasmodium berghei; Plasmodium falciparum; Solubility; Structure-Activity Relationship

2017
Bioisosteric ferrocenyl aminoquinoline-benzimidazole hybrids: Antimicrobial evaluation and mechanistic insights.
    European journal of medicinal chemistry, 2019, Oct-15, Volume: 180

    Topics: Animals; Anti-Bacterial Agents; Antimalarials; Benzimidazoles; Disease Models, Animal; Dose-Response Relationship, Drug; Ferrous Compounds; Malaria; Mice; Molecular Structure; Mycobacterium tuberculosis; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolines; Structure-Activity Relationship

2019
Research on the therapeutic properties of conessine, preliminary trials in the treatment of malaria and intestinal amebiasis; will emin be ruled by the conessine?
    Medecine tropicale : revue du Corps de sante colonial, 1948, Jan-01, Volume: 8, Issue:1

    Topics: Alkaloids; Amebiasis; Dysentery, Amebic; Emetine; Humans; Malaria

1948
CHEMOTHERAPY OF TROPICAL DISEASES.
    Current medicine and drugs, 1964, Volume: 4, Issue:10

    Topics: Amebiasis; Amebicides; Anti-Bacterial Agents; Antimalarials; Antimony; Arsenicals; Chagas Disease; Chloroquine; Dysentery, Amebic; Emetine; Humans; Iodoquinol; Leishmaniasis; Leishmaniasis, Mucocutaneous; Leishmaniasis, Visceral; Malaria; Suramin; Trypanosomiasis; Trypanosomiasis, African; United States

1964
[Biological diagnosis of malaria and amebiasis].
    Schweizerische medizinische Wochenschrift, 1977, May-07, Volume: 107, Issue:18

    Topics: Acetamides; Amebiasis; Chloroquine; Emetine; Entamoeba histolytica; Feces; Humans; Malaria; Methods; Nitroimidazoles; Primaquine; Quinine; Serologic Tests

1977
[Prevention and therapy of malaria and amebiasis].
    Schweizerische medizinische Wochenschrift, 1977, May-07, Volume: 107, Issue:18

    Topics: Acetamides; Amebiasis; Chloroquine; Drug Combinations; Drug Resistance, Microbial; Emetine; Humans; Malaria; Nitroimidazoles; Protective Devices; Pyrimethamine; Sulfadoxine; Tetracycline

1977
Malaria treated with emetine or metronidazole.
    Lancet (London, England), 1985, Aug-31, Volume: 2, Issue:8453

    Topics: Emetine; Humans; Malaria; Metronidazole; Plasmodium falciparum; Plasmodium vivax

1985
Emetine and metronidazole as antimalarial drugs.
    Lancet (London, England), 1985, Oct-05, Volume: 2, Issue:8458

    Topics: Emetine; Humans; Malaria; Metronidazole

1985
Some recent results on the chemotherapy of amebiasis, coccidiosis, and malaria.
    Pure and applied chemistry. Chimie pure et appliquee, 1969, Volume: 19, Issue:1

    Topics: Amebiasis; Animals; Animals, Domestic; Anti-Bacterial Agents; Coccidiosis; Emetine; Malaria; Pyrimethamine; Quinine; Sulfadimethoxine

1969