Page last updated: 2024-08-21

emetine and Malaria, Falciparum

emetine has been researched along with Malaria, Falciparum in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's5 (71.43)24.3611
2020's2 (28.57)2.80

Authors

AuthorsStudies
Breytenbach, WJ; de Kock, C; N'Da, DD; Pretorius, SI; Smith, PJ1
Chibale, K; Egan, TJ; Jurva, U; Masimirembwa, CM; Njoroge, M; Ongarora, DS; Strydom, N; Wicht, K; Wiesner, L; Wittlin, S1
Boesche, M; Crowther, GJ; Dasari, KS; Drewes, G; El Bakkouri, M; Fox, AM; Ghidelli-Disse, S; He, P; Hillesland, HK; Hui, R; Jones, JC; Keyloun, KR; Krahn, MM; Lafuente-Monasterio, MJ; Leonard, SE; Leroy, D; Maly, DJ; Mo, JS; Ojo, KK; Reid, MC; Rivas, KL; Van Voorhis, WC1
Combrinck, JM; de Villiers, KA; Egan, TJ; Hunter, R; L'abbate, FP; Müller, R; Openshaw, R1
Boone, M; Chibale, K; Combrinck, J; D'hooghe, M; Mangelinckx, S; Smith, PJ; Van de Walle, T; Van Puyvelde, J1
Abubaker, M; Bryce, RA; Burusco, KK; Fernández-Álvaro, E; Gutnov, A; Matthews, H; Nirmalan, N; Panwar, P; Wilkinson, J1
Deakin, J; Idris-Usman, M; Matthews, H; Nirmalan, NJ; Rajab, M1

Other Studies

7 other study(ies) available for emetine and Malaria, Falciparum

ArticleYear
Synthesis, characterization and antimalarial activity of quinoline-pyrimidine hybrids.
    Bioorganic & medicinal chemistry, 2013, Jan-01, Volume: 21, Issue:1

    Topics: Animals; Antimalarials; Cell Survival; CHO Cells; Cricetinae; Inhibitory Concentration 50; Malaria, Falciparum; Plasmodium falciparum; Pyrimidines; Quinolines

2013
Antimalarial benzoheterocyclic 4-aminoquinolines: Structure-activity relationship, in vivo evaluation, mechanistic and bioactivation studies.
    Bioorganic & medicinal chemistry, 2015, Sep-01, Volume: 23, Issue:17

    Topics: Aminoquinolines; Animals; Antimalarials; Benzene Derivatives; Humans; Malaria; Malaria, Falciparum; Mice; Mice, Inbred C57BL; Plasmodium berghei; Plasmodium falciparum; Structure-Activity Relationship

2015
Biochemical Screening of Five Protein Kinases from Plasmodium falciparum against 14,000 Cell-Active Compounds.
    PloS one, 2016, Volume: 11, Issue:3

    Topics: Antimalarials; Calcium; Cell Line, Tumor; Hep G2 Cells; Humans; Malaria, Falciparum; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase Kinases; Plasmodium falciparum; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Protozoan Proteins

2016
Hemozoin inhibiting 2-phenylbenzimidazoles active against malaria parasites.
    European journal of medicinal chemistry, 2018, Nov-05, Volume: 159

    Topics: Antimalarials; Benzimidazoles; Dose-Response Relationship, Drug; Hemeproteins; Malaria, Falciparum; Molecular Docking Simulation; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship

2018
Synthesis and biological evaluation of novel quinoline-piperidine scaffolds as antiplasmodium agents.
    European journal of medicinal chemistry, 2020, Jul-15, Volume: 198

    Topics: Antimalarials; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Molecular Structure; Parasitic Sensitivity Tests; Piperidines; Plasmodium falciparum; Quinolines; Structure-Activity Relationship

2020
Lead Optimization of Dehydroemetine for Repositioned Use in Malaria.
    Antimicrobial agents and chemotherapy, 2020, 03-24, Volume: 64, Issue:4

    Topics: Antimalarials; Atovaquone; Cell Line, Tumor; Drug Repositioning; Drug Resistance, Multiple; Drug Synergism; Emetine; Female; Hep G2 Cells; Humans; Malaria, Falciparum; Male; Membrane Potential, Mitochondrial; Plasmodium falciparum; Proguanil; Stereoisomerism

2020
Investigating antimalarial drug interactions of emetine dihydrochloride hydrate using CalcuSyn-based interactivity calculations.
    PloS one, 2017, Volume: 12, Issue:3

    Topics: Antimalarials; Artemisinins; Atovaquone; Chloroquine; Computational Biology; Drug Combinations; Drug Interactions; Drug Synergism; Drug Therapy, Combination; Emetine; Humans; Malaria, Falciparum; Plasmodium falciparum; Proguanil

2017