dov-21947 has been researched along with Pain* in 1 studies
1 other study(ies) available for dov-21947 and Pain
Article | Year |
---|---|
Studies on the structure-activity relationship of bicifadine analogs as monoamine transporter inhibitors.
Compounds with various activities and selectivities were discovered through structure-activity relationship studies of bicifadine analogs as monoamine transporter inhibitors. The norepinephrine-selective 2-thienyl compound S-6j was efficacious in a rodent pain model. Topics: Animals; Bridged Bicyclo Compounds, Heterocyclic; Caco-2 Cells; Chemistry, Pharmaceutical; Drug Design; Humans; Inhibitory Concentration 50; Membrane Transport Proteins; Models, Chemical; Neurotransmitter Agents; Neurotransmitter Transport Proteins; Norepinephrine; Pain; Rats; Structure-Activity Relationship | 2008 |