dov-21947 and Pain

dov-21947 has been researched along with Pain* in 1 studies

Other Studies

1 other study(ies) available for dov-21947 and Pain

ArticleYear
Studies on the structure-activity relationship of bicifadine analogs as monoamine transporter inhibitors.
    Bioorganic & medicinal chemistry letters, 2008, Jul-01, Volume: 18, Issue:13

    Compounds with various activities and selectivities were discovered through structure-activity relationship studies of bicifadine analogs as monoamine transporter inhibitors. The norepinephrine-selective 2-thienyl compound S-6j was efficacious in a rodent pain model.

    Topics: Animals; Bridged Bicyclo Compounds, Heterocyclic; Caco-2 Cells; Chemistry, Pharmaceutical; Drug Design; Humans; Inhibitory Concentration 50; Membrane Transport Proteins; Models, Chemical; Neurotransmitter Agents; Neurotransmitter Transport Proteins; Norepinephrine; Pain; Rats; Structure-Activity Relationship

2008