Page last updated: 2024-10-26

dilazep and Muscle Contraction

dilazep has been researched along with Muscle Contraction in 8 studies

Dilazep: Coronary vasodilator with some antiarrhythmic activity.
dilazep : A member of the class of diazepanes that is 1,4-diazepane substituted by 3-[(3,4,5-trimethoxybenzoyl)oxy]propyl groups at positions 1 and 4. It is a potent adenosine uptake inhibitor that exhibits antiplatelet, antianginal and vasodilator properties.

Muscle Contraction: A process leading to shortening and/or development of tension in muscle tissue. Muscle contraction occurs by a sliding filament mechanism whereby actin filaments slide inward among the myosin filaments.

Research Excerpts

ExcerptRelevanceReference
"Endogenous adenosine is an important modulator of intestinal neuro-effector activity, operating in the linear part of the dose-response curve."1.36Estimation of endogenous adenosine activity at adenosine receptors in guinea-pig ileum using a new pharmacological method. ( Glaumann, C; Grishina, VA; Gustafsson, LE; Nilsson, KF, 2010)

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19907 (87.50)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Nilsson, KF1
Grishina, VA1
Glaumann, C1
Gustafsson, LE2
Tonini, M1
Perucca, E1
Manzo, L1
Marcoli, M1
D'Angelo, L1
Saltarelli, P1
Onori, L1
Kobayashi, A1
Ogawa, K1
Yamazaki, N1
Gustafsson, L1
Fredholm, BB1
Hedqvist, P1
Fujita, S1
Ishida, Y1
Izumi, K1
Moritoki, H1
Ohara, M1
Takei, M1
Tamura, H1
Shirasawa, Y1
Hori, H1
Kondo, S1
Franco, R1
Hoyle, CH1
Centelles, JJ1
Burnstock, G1

Other Studies

8 other studies available for dilazep and Muscle Contraction

ArticleYear
Estimation of endogenous adenosine activity at adenosine receptors in guinea-pig ileum using a new pharmacological method.
    Acta physiologica (Oxford, England), 2010, Volume: 199, Issue:2

    Topics: 2-Chloroadenosine; Adenosine; Animals; Dilazep; Dose-Response Relationship, Drug; Guinea Pigs; Ileum

2010
Dilazep: an inhibitor of adenosine uptake with intrinsic calcium antagonistic properties.
    The Journal of pharmacy and pharmacology, 1983, Volume: 35, Issue:7

    Topics: Adenosine; Animals; Azepines; Calcium Channel Blockers; Dilazep; Female; Guinea Pigs; In Vitro Techn

1983
The effects of dilazep and SG 75 on cyclic nucleotides in the coronary artery.
    Japanese heart journal, 1980, Volume: 21, Issue:1

    Topics: Adenosine; Animals; Arteries; Azepines; Coronary Circulation; Coronary Vessels; Cyclic AMP; Cyclic G

1980
Theophylline interferes with the modulatory role of endogenous adenosine on cholinergic neurotransmission in guinea pig ileum.
    Acta physiologica Scandinavica, 1981, Volume: 111, Issue:3

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Animals; Cholin

1981
Potentiation by dilazep on the negative inotropic effect of adenosine on guinea-pig atria.
    British journal of pharmacology, 1980, Volume: 68, Issue:2

    Topics: Adenosine; Adenosine Deaminase; Animals; Azepines; Calcium; Dilazep; Drug Synergism; Female; Male; M

1980
[Effects of 1, 4-bis-(3-(3, 4, 5-trimethoxy benzoyl oxy)-propyl) perhydro-1, 4-diazepine (dilazep) on the isolated smooth muscles].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1975, Volume: 71, Issue:8

    Topics: Adenine Nucleotides; Adenosine; Animals; Aorta; Calcium; Dilazep; Dogs; Dose-Response Relationship,

1975
Mechanisms involved in the action of prostaglandins as modulators of neurotransmission.
    Annals of the New York Academy of Sciences, 1989, Volume: 559

    Topics: Acetylcholine; Adenosine; Animals; Blood Pressure; Dilazep; Electric Stimulation; Female; Heart Rate

1989
Degradation of adenosine by extracellular adenosine deaminase in the rat duodenum.
    General pharmacology, 1988, Volume: 19, Issue:5

    Topics: Adenosine; Adenosine Deaminase; Adenosine Deaminase Inhibitors; Animals; Coformycin; Dilazep; Duoden

1988