Page last updated: 2024-09-03

deltorphin i, ala(2)- and Pain

deltorphin i, ala(2)- has been researched along with Pain in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (50.00)18.2507
2000's1 (25.00)29.6817
2010's1 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Balboni, G; Caliendo, G; Capasso, A; Guerrini, R; Lazarus, LH; Marastoni, M; Salvadori, S; Santagada, V; Sorrentino, L; Tomatis, R1
Fairbanks, CA; Kitto, KF; Messing, RO; Metcalf, MD; Schuster, DJ; Wilcox, GL1
Biondi, L; Filira, F; Giannini, E; Gobbo, M; Marastoni, M; Negri, L; Rocchi, R; Scolaro, B; Tomatisc, R1
Burks, TF; Carr, DB; Davis, P; Fang, L; Hruby, VJ; Knapp, RJ; Kramer, T; Lipkowski, AW; Misicka, A; Yamamura, HI1

Other Studies

4 other study(ies) available for deltorphin i, ala(2)- and Pain

ArticleYear
Synthesis and pharmacological activity of deltorphin and dermorphin-related glycopeptides.
    Journal of medicinal chemistry, 1997, Aug-29, Volume: 40, Issue:18

    Topics: Amino Acid Sequence; Analgesics, Opioid; Animals; Binding, Competitive; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Glycopeptides; Guinea Pigs; Ileum; In Vitro Techniques; Indicators and Reagents; Jejunum; Kinetics; Male; Mice; Muscle Contraction; Muscle, Smooth; Oligopeptides; Opioid Peptides; Pain; Rabbits; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Structure-Activity Relationship; Synaptosomes

1997
Ligand requirements for involvement of PKCε in synergistic analgesic interactions between spinal μ and δ opioid receptors.
    British journal of pharmacology, 2015, Volume: 172, Issue:2

    Topics: Analgesics, Opioid; Animals; Behavior, Animal; Drug Therapy, Combination; Female; Hot Temperature; Ligands; Male; Mice, Knockout; Morphine; Morpholines; Oligopeptides; Pain; Protein Kinase C-epsilon; Protein Multimerization; Receptors, Opioid, delta; Receptors, Opioid, mu; Spinal Cord

2015
Synthesis, conformation and biological activity of dermorphin and deltorphin I analogues containing N-alkylglycine in place of residues in position 1, 3, 5 and 6.
    Journal of peptide science : an official publication of the European Peptide Society, 2003, Volume: 9, Issue:10

    Topics: Analgesics, Opioid; Animals; CHO Cells; Cricetinae; Cricetulus; Guinea Pigs; Male; Mice; Muscle Contraction; Muscle, Smooth; N-substituted Glycines; Oligopeptides; Opioid Peptides; Pain; Protein Conformation; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu

2003
Topographical requirements for delta opioid ligands: presence of a carboxyl group in position 4 is not critical for deltorphin high delta receptor affinity and analgesic activity.
    Biochemical and biophysical research communications, 1991, Nov-14, Volume: 180, Issue:3

    Topics: Amino Acid Sequence; Analgesics; Animals; Binding, Competitive; Brain; Male; Models, Molecular; Molecular Sequence Data; Oligopeptides; Pain; Protein Conformation; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta

1991