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cycloguanil and Plasmodium falciparum Malaria

cycloguanil has been researched along with Plasmodium falciparum Malaria in 38 studies

Research

Studies (38)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's15 (39.47)18.2507
2000's17 (44.74)29.6817
2010's6 (15.79)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bertaux, L; Bogreau, H; Bouchiba, H; Garnotel, E; Kraemer, P; Parzy, D; Pradines, B; Rogier, C; Savini, H; Simon, F1
Brun, R; Chitnumsub, P; Dartois, V; Diagana, TT; Goh, A; Kamchonwongpaisan, S; Keller, TH; Kiara, SM; Lakshminarayana, SB; Ma, NL; Maneeruttanarungroj, C; Nzila, A; Rottmann, M; Taweechai, S; Weaver, M; Wittlin, S; Wong, J; Yeung, BK; Yuthavong, Y; Zou, B1
Corral, MG; Leroux, J; Mylne, JS; Stubbs, KA1
Dinter, D; Domijan, AM; Gajski, G; Garaj-Vrhovac, V1
Diakite, I; Hartl, DL; Ogbunugafor, CB; Weinreich, DM; Wylie, CS1
Barata, L; Boutbibe, K; Clain, J; Franetich, JF; Houzé, P; Mazier, D; Zanghi, G1
Brown, KM; Costanzo, MS; Hartl, DL1
Delfino, RT; Figueroa-Villar, JD; Santos-Filho, OA1
Bouchaud, O; Durand, R; Godineau, N; Jezic, Z; Keundjian, A; Le Bras, J; Pradines, B; Ralaimazava, P1
Alifrangis, M; Jelinek, T; Salanti, A; Schwöbel, B1
Durand, R; Le Bras, J1
Ariey, F; Duchemin, JB; Harisoa, JL; Mauclere, P; Pietra, V; Rabarijaona, LP; Raharimalala, LA; Rakotomanana, F; Ranaivo, L; Randrianarivelojosia, M; Robert, V1
Ashley, E; Cho, D; Cho, T; Edstein, MD; Ginsberg, A; Looareesuwan, S; McGready, R; Nosten, F; Seaton, E; Stepniewska, K; White, NJ1
Rakotoson, JD; Randremanana, RV; Randriamanantena, A; Randrianarivelojosia, M; Randrianasolo, L; Ratsimbasoa, A1
Bienzle, U; Ehrhardt, S; Jelinek, T; Mockenhaupt, FP; Muehlen, M; Otchwemah, R; Schreiber, J1
Björkman, A; Gil, JP; Thapar, MM1
Peters, W; Robinson, BL; Stewart, LB1
Kioy, D; Konsil, J; Manyando, C; Miller, GB; Mulenga, M; Na-Bangchang, K; Ruengweerayut, R1
Aarons, L; Bojang, K; Edwards, G; Hughes, D; Manyando, C; Simpson, JA; Ward, S; Watkins, WA; Winstanley, P1
Chishimba, S; Mharakurwa, S; Mkulama, MA; Rouse, P; Sikalima, J; Thuma, PE1
Basco, LK; Eldin de Pécoulas, P; Le Bras, J; Mazabraud, A; Wilson, CM1
Ager, AL; Canfield, CJ; Jacobus, DP; Lewis, NJ; Milhous, WK; Rossan, RN; Sweeney, TR1
Basco, LK; Doury, JC; Le Bras, J; Ramiliarisoa, O; Ringwald, P1
Cowman, AF; Genton, B; Lorry, K; Reeder, JC; Rieckmann, KH; Wines, B1
Nguyen, DS; Nguyen, PD; Sköld, O; Swedberg, G; Zindrou, S1
Edstein, MD; Rieckmann, KH; Shanks, GD; Yeo, AE1
Basco, LK; Le Bras, J1
Doerig, C; Doury, JC; Fusai, T; Parzy, D; Pradines, B; Rico, A1
Mberu, EK; Nzila-Mounda, A; Plowe, CV; Sibley, CH; Watkins, WM; Winstanley, PA1
di Piazza, JP; Durand, R; Le Bras, J; Longuet, C; Parzy, D; Pradines, B1
Bergqvist, Y; Björkman, A; Ishizaki, T; Kalkoa, M; Kaneko, A; Kaneko, O; Kobayakawa, T; Takechi, M1
Bouchaud, O; di Piazza, JP; Durand, R; Godineau, N; Le Bras, J; Longuet, C; Marchou, B; Martet, G; Parzy, D; Pradines, B; Roué, R1
Fusai, T; Keundjian, A; Kombila, M; Lebeau, C; Mabika Mamfoumbi, M; Owono Medang, M; Parzy, D; Pradines, B; Rogier, C1
Howard, V; Mookherjee, S; Nzila-Mouanda, A; Sibley, CH; Watkins, W1
Clain, J; di Piazza, JP; Durand, R; le Bras, J; Longuet, C; Sécardin, Y1
Auparakkitanon, S; Chavalitshewinkoon-Petmitr, P; Pongvilairat, G; Wilairat, P1
Fusai, T; Mosnier, J; Parzy, D; Pradines, B; Rogier, C; Spiegel, A; Tall, A; Trape, JF1
Basco, LK; Ringwald, P1

Reviews

1 review(s) available for cycloguanil and Plasmodium falciparum Malaria

ArticleYear
The mechanisms of resistance to antimalarial drugs in Plasmodium falciparum.
    Fundamental & clinical pharmacology, 2003, Volume: 17, Issue:2

    Topics: Africa; Animals; Antimalarials; Antimetabolites; Chloroquine; Drug Resistance; Drug Resistance, Multiple; Humans; Malaria, Falciparum; Plasmodium falciparum; Proguanil; Pyrimethamine; Triazines

2003

Trials

2 trial(s) available for cycloguanil and Plasmodium falciparum Malaria

ArticleYear
Pregnancy and use of oral contraceptives reduces the biotransformation of proguanil to cycloguanil.
    European journal of clinical pharmacology, 2003, Volume: 59, Issue:7

    Topics: Antimalarials; Biotransformation; Case-Control Studies; Cohort Studies; Contraceptives, Oral, Hormonal; Female; Humans; Malaria, Falciparum; Pregnancy; Pregnancy Complications, Parasitic; Pregnancy Trimester, Third; Proguanil; Thailand; Triazines

2003
The pharmacokinetics and pharmacodynamics of atovaquone and proguanil for the treatment of uncomplicated falciparum malaria in third-trimester pregnant women.
    European journal of clinical pharmacology, 2005, Volume: 61, Issue:8

    Topics: Adolescent; Adult; Antimalarials; Atovaquone; Drug Combinations; Female; Humans; Malaria, Falciparum; Naphthoquinones; Pregnancy; Proguanil; Thailand; Triazines; Zambia

2005

Other Studies

35 other study(ies) available for cycloguanil and Plasmodium falciparum Malaria

ArticleYear
First case of emergence of atovaquone-proguanil resistance in Plasmodium falciparum during treatment in a traveler in Comoros.
    Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:6

    Topics: Animals; Antimalarials; Atovaquone; Comoros; Drug Resistance; France; Genotype; Humans; Malaria, Falciparum; Male; Parasitic Sensitivity Tests; Plasmodium falciparum; Proguanil; Travel; Treatment Failure

2008
Preclinical evaluation of the antifolate QN254, 5-chloro- N'6'-(2,5-dimethoxy-benzyl)-quinazoline-2,4,6-triamine, as an antimalarial drug candidate.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:6

    Topics: Administration, Oral; Animals; Antimalarials; Biological Availability; Drug Resistance; Female; Folic Acid Antagonists; Humans; In Vitro Techniques; Malaria; Malaria, Falciparum; Male; Mice; Models, Molecular; Mutation; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Pyrimethamine; Quinazolines; Rats; Rats, Wistar; Tetrahydrofolate Dehydrogenase

2010
Herbicidal properties of antimalarial drugs.
    Scientific reports, 2017, 03-31, Volume: 7

    Topics: Antimalarials; Arabidopsis; Herbicides; Humans; Malaria, Falciparum; Plasmodium falciparum; Proguanil; Pyrimethamine; Sulfadiazine; Sulfadoxine; Triazines

2017
Cytogenetic and oxidative status of human lymphocytes after exposure to clinically relevant concentrations of antimalarial drugs atovaquone and proguanil hydrochloride in vitro.
    Fundamental & clinical pharmacology, 2015, Volume: 29, Issue:6

    Topics: Adult; Antimalarials; Atovaquone; Cell Survival; Cytogenetics; DNA Damage; Dose-Response Relationship, Drug; Drug Combinations; Glutathione; Humans; Lymphocytes; Malaria, Falciparum; Male; Malondialdehyde; Oxidative Stress; Plasmodium falciparum; Proguanil; Triazines

2015
Adaptive Landscape by Environment Interactions Dictate Evolutionary Dynamics in Models of Drug Resistance.
    PLoS computational biology, 2016, Volume: 12, Issue:1

    Topics: Antimalarials; Computational Biology; Drug Resistance; Evolution, Molecular; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Models, Biological; Mutation; Plasmodium falciparum; Proguanil; Pyrimethamine; Triazines

2016
In Vitro Analysis of the Interaction between Atovaquone and Proguanil against Liver Stage Malaria Parasites.
    Antimicrobial agents and chemotherapy, 2016, Volume: 60, Issue:7

    Topics: Antimalarials; Atovaquone; Drug Combinations; Hepatocytes; Humans; Inhibitory Concentration 50; Liver; Malaria, Falciparum; Plasmodium falciparum; Proguanil; Triazines

2016
Fitness trade-offs in the evolution of dihydrofolate reductase and drug resistance in Plasmodium falciparum.
    PloS one, 2011, Volume: 6, Issue:5

    Topics: Drug Resistance; Evolution, Molecular; Folic Acid Antagonists; Malaria, Falciparum; Plasmodium falciparum; Proguanil; Pyrimethamine; Tetrahydrofolate Dehydrogenase; Triazines

2011
Molecular modeling of wild-type and antifolate resistant mutant Plasmodium falciparum DHFR.
    Biophysical chemistry, 2002, Aug-02, Volume: 98, Issue:3

    Topics: Animals; Chickens; Drug Resistance; Folic Acid Antagonists; Humans; Liver; Malaria, Falciparum; Models, Chemical; Models, Genetic; Models, Molecular; Molecular Sequence Data; Plasmodium falciparum; Point Mutation; Proguanil; Pyrimethamine; Sequence Alignment; Tetrahydrofolate Dehydrogenase; Triazines

2002
Profile and evolution of the chemosusceptibility of falciparum malaria imported into France in 2000.
    Euro surveillance : bulletin Europeen sur les maladies transmissibles = European communicable disease bulletin, 2002, Volume: 7, Issue:7

    Topics: Adolescent; Adult; Aged; Animals; Antimalarials; Child; Child, Preschool; Chloroquine; Drug Resistance; Female; France; Humans; Infant; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Plasmodium falciparum; Proguanil; Quinine; Triazines

2002
Different mutation patterns of atovaquone resistance to Plasmodium falciparum in vitro and in vivo: rapid detection of codon 268 polymorphisms in the cytochrome b as potential in vivo resistance marker.
    Malaria journal, 2003, Mar-19, Volume: 2

    Topics: Animals; Antimalarials; Antiprotozoal Agents; Atovaquone; Codon; Drug Resistance; Electron Transport Complex III; Genetic Markers; Humans; Malaria, Falciparum; Mutation; Naphthoquinones; Plasmodium falciparum; Polymerase Chain Reaction; Polymorphism, Genetic; Polymorphism, Restriction Fragment Length; Proguanil; Triazines

2003
In vitro sensitivity of Plasmodium falciparum to amodiaquine compared with other major antimalarials in Madagascar.
    Parassitologia, 2002, Volume: 44, Issue:3-4

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Drug Resistance; Drug Resistance, Multiple; Humans; Inhibitory Concentration 50; Madagascar; Malaria, Falciparum; Mefloquine; Parasitemia; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinine; Triazines

2002
Susceptibility of Plasmodium falciparum to the drugs used to treat severe malaria (quinine) and to prevent malaria (mefloquine, cycloguanil) in Comoros Union and Madagascar.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 2004, Volume: 94, Issue:1

    Topics: Animals; Antimalarials; Comoros; Drug Resistance; Humans; In Vitro Techniques; Madagascar; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Proguanil; Quinine; Triazines

2004
Short communication: Prevalence of mutations associated with resistance to atovaquone and to the antifolate effect of proguanil in Plasmodium falciparum isolates from northern Ghana.
    Tropical medicine & international health : TM & IH, 2004, Volume: 9, Issue:3

    Topics: Animals; Antimalarials; Atovaquone; Child, Preschool; Cytochromes b; Drug Combinations; Drug Resistance; Drug Synergism; Drug Therapy, Combination; Female; Folic Acid Antagonists; Ghana; Humans; Infant; Malaria, Falciparum; Male; Mutation; Naphthoquinones; Plasmodium falciparum; Polymorphism, Restriction Fragment Length; Proguanil; Pyrimethamine; Sulfadoxine; Tetrahydrofolate Dehydrogenase; Triazines

2004
In vitro recrudescence of Plasmodium falciparum parasites suppressed to dormant state by atovaquone alone and in combination with proguanil.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 2005, Volume: 99, Issue:1

    Topics: Animals; Antimalarials; Atovaquone; Culture Media; Cytochrome b Group; Dose-Response Relationship, Drug; Drug Resistance; Drug Therapy, Combination; Humans; Malaria, Falciparum; Naphthoquinones; Parasitic Sensitivity Tests; Plasmodium falciparum; Proguanil; Recurrence; Triazines

2005
The chemotherapy of rodent malaria. LXII. Drug combinations to impede the selection of drug resistance, part 5: rates of development of resistance to some inhibitors of folate metabolism and to artesunate.
    Annals of tropical medicine and parasitology, 2004, Volume: 98, Issue:8

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Dapsone; Drug Resistance; Drug Therapy, Combination; Folic Acid Antagonists; Malaria, Falciparum; Male; Mice; Parasitemia; Plasmodium berghei; Plasmodium chabaudi; Plasmodium yoelii; Proguanil; Sesquiterpenes; Triazines

2004
Population pharmacokinetic and pharmacodynamic modelling of the antimalarial chemotherapy chlorproguanil/dapsone.
    British journal of clinical pharmacology, 2006, Volume: 61, Issue:3

    Topics: Adolescent; Adult; Animals; Antimalarials; Child; Child, Preschool; Dapsone; Humans; Infant; Malaria, Falciparum; Middle Aged; Plasmodium falciparum; Proguanil; Prospective Studies; Triazines

2006
Escalating Plasmodium falciparum antifolate drug resistance mutations in Macha, rural Zambia.
    Malaria journal, 2008, May-21, Volume: 7

    Topics: Animals; Antimalarials; Child; Child, Preschool; DNA, Protozoan; Drug Resistance; Folic Acid Antagonists; Humans; Malaria, Falciparum; Mutation, Missense; Peptide Synthases; Plasmodium falciparum; Point Mutation; Polymerase Chain Reaction; Polymorphism, Restriction Fragment Length; Proguanil; Protozoan Proteins; Pyrimethamine; Rural Population; Tetrahydrofolate Dehydrogenase; Triazines; Zambia

2008
Point mutations in the dihydrofolate reductase-thymidylate synthase gene and pyrimethamine and cycloguanil resistance in Plasmodium falciparum.
    Molecular and biochemical parasitology, 1995, Volume: 69, Issue:1

    Topics: Amino Acid Sequence; Animals; Base Sequence; Drug Resistance, Multiple; Humans; Malaria, Falciparum; Plasmodium falciparum; Point Mutation; Proguanil; Pyrimethamine; Tetrahydrofolate Dehydrogenase; Thymidylate Synthase; Triazines

1995
PS-15: a potent, orally active antimalarial from a new class of folic acid antagonists.
    The American journal of tropical medicine and hygiene, 1993, Volume: 49, Issue:1

    Topics: Administration, Oral; Animals; Antimalarials; Aotus trivirgatus; Atovaquone; Drug Synergism; Folic Acid Antagonists; Imides; Injections, Subcutaneous; Malaria, Falciparum; Mice; Naphthoquinones; Phenyl Ethers; Plasmodium falciparum; Proguanil; Sulfamethoxazole; Triazines

1993
In vitro activity of cycloguanil against African isolates of Plasmodium falciparum.
    Antimicrobial agents and chemotherapy, 1993, Volume: 37, Issue:4

    Topics: Animals; Erythrocytes; Humans; Liver; Malaria, Falciparum; Microbial Sensitivity Tests; Plasmodium falciparum; Proguanil; Triazines

1993
Point mutations in the dihydrofolate reductase and dihydropteroate synthetase genes and in vitro susceptibility to pyrimethamine and cycloguanil of Plasmodium falciparum isolates from Papua New Guinea.
    The American journal of tropical medicine and hygiene, 1996, Volume: 55, Issue:2

    Topics: Animals; Antimalarials; Base Sequence; Dihydropteroate Synthase; DNA Primers; Drug Resistance; Folic Acid Antagonists; Humans; Malaria, Falciparum; Molecular Sequence Data; Plasmodium falciparum; Point Mutation; Polymerase Chain Reaction; Proguanil; Pyrimethamine; Sequence Analysis, DNA; Tetrahydrofolate Dehydrogenase; Triazines

1996
Plasmodium falciparum: mutation pattern in the dihydrofolate reductase-thymidylate synthase genes of Vietnamese isolates, a novel mutation, and coexistence of two clones in a Thai patient.
    Experimental parasitology, 1996, Volume: 84, Issue:1

    Topics: Animals; Antimalarials; Base Sequence; DNA, Protozoan; Drug Resistance; Folic Acid Antagonists; Humans; Malaria, Falciparum; Molecular Sequence Data; Plasmodium falciparum; Point Mutation; Proguanil; Pyrimethamine; Tetrahydrofolate Dehydrogenase; Thailand; Thymidylate Synthase; Triazines; Vietnam

1996
Ex vivo antimalarial activity of proguanil combined with dapsone against cycloguanil-resistant Plasmodium falciparum isolates.
    Acta tropica, 1997, Sep-10, Volume: 66, Issue:3

    Topics: Animals; Antimalarials; Dapsone; Drug Resistance; Drug Therapy, Combination; Humans; Malaria, Falciparum; Plasmodium falciparum; Proguanil; Triazines

1997
In vitro sensitivity of Plasmodium falciparum to anti-folinic agents (trimethoprim, pyrimethamine, cycloguanil): a study of 29 African strains.
    Bulletin de la Societe de pathologie exotique (1990), 1997, Volume: 90, Issue:2

    Topics: Animals; Antimalarials; Confidence Intervals; Drug Resistance; Folic Acid Antagonists; Humans; Lethal Dose 50; Malaria, Falciparum; Nonlinear Dynamics; Plasmodium falciparum; Proguanil; Pyrimethamine; Tetrahydrofolate Dehydrogenase; Triazines; Trimethoprim

1997
Proguanil resistance in Plasmodium falciparum African isolates: assessment by mutation-specific polymerase chain reaction and in vitro susceptibility testing.
    The American journal of tropical medicine and hygiene, 1997, Volume: 57, Issue:6

    Topics: Africa; Amino Acid Substitution; Animals; Asparagine; Codon; DNA, Protozoan; Drug Resistance, Microbial; Humans; Malaria, Falciparum; Microbial Sensitivity Tests; Plasmodium falciparum; Point Mutation; Polymerase Chain Reaction; Proguanil; Sequence Analysis, DNA; Serine; Tetrahydrofolate Dehydrogenase; Triazines

1997
Kenyan Plasmodium falciparum field isolates: correlation between pyrimethamine and chlorcycloguanil activity in vitro and point mutations in the dihydrofolate reductase domain.
    Antimicrobial agents and chemotherapy, 1998, Volume: 42, Issue:1

    Topics: Animals; Antimalarials; Humans; Kenya; Malaria, Falciparum; Plasmodium falciparum; Point Mutation; Proguanil; Protozoan Proteins; Pyrimethamine; Sensitivity and Specificity; Tetrahydrofolate Dehydrogenase; Triazines

1998
[Considering disparities in resistance of Plasmodium falciparum in Africa in chemoprevention decisions].
    Presse medicale (Paris, France : 1983), 1998, Sep-26, Volume: 27, Issue:28

    Topics: Africa; Animals; Antimalarials; Chloroquine; Cross-Cultural Comparison; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Folic Acid Antagonists; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Proguanil; Seasons; Travel; Triazines

1998
Intrinsic efficacy of proguanil against falciparum and vivax malaria independent of the metabolite cycloguanil.
    The Journal of infectious diseases, 1999, Volume: 179, Issue:4

    Topics: Adolescent; Antimalarials; Aryl Hydrocarbon Hydroxylases; Child; Child, Preschool; Cytochrome P-450 CYP2C19; Cytochrome P-450 Enzyme System; Genotype; Humans; Infant; Malaria, Falciparum; Malaria, Vivax; Mixed Function Oxygenases; Proguanil; Tetrahydrofolate Dehydrogenase; Triazines

1999
[Resistance to chloroquine and cycloguanil of Plasmodium falciparum in patients arriving in France after travel in Africa without chemoprophylaxis].
    Bulletin de la Societe de pathologie exotique (1990), 1998, Volume: 91, Issue:5 Pt 1-2

    Topics: Africa; Animals; Antimalarials; Chloroquine; Codon; Drug Resistance, Multiple; Folic Acid Antagonists; France; Humans; Malaria, Falciparum; Plasmodium falciparum; Proguanil; Seasons; Tetrahydrofolate Dehydrogenase; Travel; Triazines

1998
[In vitro sensitivity of Plasmodium falciparum isolates from Gabon to chloroquine and cycloguanil].
    Bulletin de la Societe de pathologie exotique (1990), 1999, Volume: 92, Issue:2

    Topics: Adolescent; Animals; Antimalarials; Child; Child, Preschool; Chloroquine; Drug Resistance; Gabon; Humans; Infant; Malaria, Falciparum; Plasmodium falciparum; Proguanil; Triazines

1999
Identification and analysis of dihydrofolate reductase alleles from Plasmodium falciparum present at low frequency in polyclonal patient samples.
    The American journal of tropical medicine and hygiene, 1999, Volume: 61, Issue:1

    Topics: Alleles; Animals; Antimalarials; DNA Primers; DNA Restriction Enzymes; DNA, Protozoan; Humans; Inhibitory Concentration 50; Kenya; Malaria, Falciparum; Plasmodium falciparum; Polymerase Chain Reaction; Proguanil; Pyrimethamine; Saccharomyces cerevisiae; Tetrahydrofolate Dehydrogenase; Triazines

1999
Increased incidence of cycloguanil resistance in malaria cases entering France from Africa, determined as point mutations in the parasites' dihydrofolate-reductase genes.
    Annals of tropical medicine and parasitology, 1999, Volume: 93, Issue:1

    Topics: Africa; Animals; Antimalarials; Drug Resistance; Folic Acid Antagonists; France; Genes, Protozoan; Humans; Malaria, Falciparum; Plasmodium falciparum; Point Mutation; Polymerase Chain Reaction; Polymorphism, Restriction Fragment Length; Proguanil; Tetrahydrofolate Dehydrogenase; Triazines

1999
Gametocytocidal activity of pyronaridine and DNA topoisomerase II inhibitors against multidrug-resistant Plasmodium falciparum in vitro.
    Parasitology international, 2000, Volume: 48, Issue:4

    Topics: Amsacrine; Animals; Antimalarials; Chloroquine; Drug Resistance, Multiple; Enzyme Inhibitors; Etoposide; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Mefloquine; Naphthyridines; Norfloxacin; Nucleic Acid Synthesis Inhibitors; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Thailand; Topoisomerase II Inhibitors; Triazines

2000
Antibiotics for prophylaxis of Plasmodium falciparum infections: in vitro activity of doxycycline against Senegalese isolates.
    The American journal of tropical medicine and hygiene, 2000, Volume: 62, Issue:1

    Topics: Amodiaquine; Animals; Anti-Bacterial Agents; Antibiotic Prophylaxis; Antimalarials; Artemether; Artemisinins; Chloroquine; Doxycycline; Drug Resistance; Erythrocytes; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinine; Scintillation Counting; Senegal; Sesquiterpenes; Statistics, Nonparametric; Triazines

2000
Molecular epidemiology of malaria in Yaounde, Cameroon. VI. Sequence variations in the Plasmodium falciparum dihydrofolate reductase-thymidylate synthase gene and in vitro resistance to pyrimethamine and cycloguanil.
    The American journal of tropical medicine and hygiene, 2000, Volume: 62, Issue:2

    Topics: Animals; Antimalarials; Cameroon; DNA Primers; DNA, Protozoan; Drug Resistance; Folic Acid Antagonists; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Plasmodium falciparum; Point Mutation; Polymerase Chain Reaction; Proguanil; Pyrimethamine; Sequence Analysis, DNA; Tetrahydrofolate Dehydrogenase; Triazines

2000
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