colforsin has been researched along with Muscle Contraction in 288 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 87 (30.21) | 18.7374 |
1990's | 112 (38.89) | 18.2507 |
2000's | 65 (22.57) | 29.6817 |
2010's | 21 (7.29) | 24.3611 |
2020's | 3 (1.04) | 2.80 |
Authors | Studies |
---|---|
Cho, HJ; Choi, JY; Engelhardt, JF; Joo, NS; Milla, CE; Shinbashi, M; Wine, JJ | 1 |
Hollywood, MA; Martin, SL; Morgan, LM; Mullins, ND; Sergeant, GP; Thornbury, KD | 1 |
Birulina, YG; Buyko, EE; Efremkina, EP; Gusakova, SV; Ivanov, VV; Kovalev, IV; Nosarev, AV; Smagliy, LV | 1 |
Cortese-Krott, MM; DeLalio, LJ; Diederich, L; Drake, JC; Isakson, BE; Jackson, EK; Keller, AS; Kelm, M; Panknin, C; Sherman, R; Yan, Z | 1 |
Baudenbacher, FJ; Brophy, CM; Cheung-Flynn, J; Hocking, KM; Komalavilas, P; Putumbaka, G; Venkatraman, S | 1 |
Inazumi, T; Iwasaki, R; Kawahara, A; Kawahara, O; Morimoto, K; Sugimoto, Y; Tsuchiya, S; Tsuge, K | 1 |
Chan, KY; Danser, AH; de Vries, R; Dirven, C; Garrelds, IM; Labruijere, S; MaassenVanDenBrink, A; Ramírez Rosas, MB; van den Bogaerdt, A; Villalón, CM | 1 |
Anoopkumar-Dukie, S; Grant, GD; Hempenstall, A; Johnson, PJ | 1 |
Cervantes, D; Fu, Q; Parikh, D; Xiang, YK; Xu, B | 1 |
Hill, MA; Lee, S; Li, M; Tanner, MA; Yang, Y | 1 |
Lorenz, K; Newe, M; Propping, S; Ravens, U; Wirth, MP | 1 |
Bouchelouche, P; Matras, C; Nordling, J; Sheykhzade, M; Svalø, J | 1 |
Gunst, SJ; Wu, Y | 1 |
Kanda, H; Kaneda, T; Saito, E; Shimizu, K; Urakawa, N | 1 |
Lim, KH; Loong, BJ; Mbaki, Y; Tan, JH; Ting, KN | 1 |
Bi, H; Cheng, L; Cui, Q; Fan, R; Feng, N; Guo, HT; Liu, JC; Ma, J; Pei, JM; Sun, X; Sun, XQ; Wang, YM; Yi, DH; Yin, W; Yin, Z; Yu, SQ; Zhang, QY; Zhang, SM | 1 |
Chen, S; Kaye, AD; Liu, L; Lu, SY; Mei, Q; Niu, X; Pei, J; Wei, J; Xing, B; Xiong, L; Zhu, M; Zhu, X | 1 |
Michel, MC; Sand, C | 1 |
Al-Chaer, ED; Chaloner, A; Greenwood-Van Meerveld, B; Rao, A | 1 |
HARA, Y; HARADA, Y; KANEDA, T; NEZU, Y; SHIMIZU, K; TAGAWA, M; URAKAWA, N; YOGO, T | 1 |
Hamada, C; Itoh, H; Jiang, B; Maruyama, J; Maruyama, K; Mitani, Y; Yokochi, A; Zhang, E | 1 |
Ehlert, FJ; Matsui, M; Ostrom, RS; Pak, KJ | 1 |
Britton, F; Dixon, R; Hwang, S; Sanders, K; Ward, S | 1 |
Coelho, LP; Cordeiro, RS; da Costa, JC; Martins, MA; Olsen, PC; Silva, PM | 1 |
Duarte, T; Godinho, RO; Menezes-Rodrigues, FS | 1 |
Kedia, GT; Kuczyk, MA; Merseburger, AS; Polat, H; Ückert, S | 1 |
Chappellaz, M; Grassie, ME; Kiss, E; MacDonald, JA; Sutherland, C; Ulke-Lemée, A; Walsh, MP | 1 |
Ballard, HJ; Cai, W; Lu, L; Tu, J | 1 |
Fujii, Y; Toyooka, H | 1 |
Advenier, C; Cortijo, J; Molimard, M; Morcillo, EJ; Moreau, J; Naline, E; Sarria, B; Therond, P; Zhang, Y | 1 |
Ckert, S; Frlich, Jr; Jonas, U; Machtens, S; Stief, CG; Tsikas, D | 1 |
Ehlert, FJ; Griffin, MT; Matsui, M; Shehnaz, D; Taketo, MM | 1 |
Fujii, Y; Toyooka, H; Uemura, A | 1 |
Amrani, Y; Chen, H; Panettieri, RA; Tliba, O; Van Besien, CR | 1 |
Brophy, CM; Joshi, L; Komalavilas, P; Panitch, A; Tessier, DJ | 1 |
Barnes, TA; Calo, G; Carra, G; Guerrini, R; Kitayama, M; Lambert, DG; McDonald, J; Rowbotham, DJ; Smith, G | 1 |
Boyd, JG; Gordon, T; Sulaiman, O | 1 |
Brading, AF; Hashitani, H; Suzuki, H | 1 |
Agrawal, DK; Ariyarathna, K; Kelbe, PW | 1 |
Chan, SL; Dunn, WR; Garfield, B; Wang, M; Wilson, VG | 1 |
Chan, FL; Chan, YC; Chen, ZY; Huang, Y; Lau, CW; Yao, X | 1 |
Donini, A; Lange, AB | 1 |
Gillespie, JI | 1 |
Bespalova, ZhD; Khapchaev, AY; Krymsky, MA; Shirinsky, VP; Sidorova, MV; Vorotnikov, AV; Wang, CL | 1 |
Kaneda, T; Nakajyo, S; Shimizu, K; Urakawa, N | 1 |
Jin, Z; Meeks, MK; Rembold, CM; Ripley, ML | 1 |
Abe, DM; Ehlert, FJ; Griffin, MT; Manabe, T; Matsui, M; Taketo, MM; Vo, TH | 1 |
Benhamú, B; Caicoya, AG; Delgado, M; Fernández-Alfonso, MS; Fuentes, JA; Greciano, V; López-Rodríguez, ML; Manzanares, J; Pozo, MA | 1 |
Abete, P; Cacciatore, F; Calabrese, C; Corbi, G; Ferrara, N; Iaccarino, G; Leosco, D; Longobardi, G; Paolisso, G; Rengo, F; Scarpa, D; Trimarco, B | 1 |
Boterman, M; Elzinga, CR; Eppens, PB; Meurs, H; Wagemakers, D; Zaagsma, J | 1 |
Bubolz, AH; Li, H; Liu, Y; Wu, Q | 1 |
Batts, TW; Murphy, RA; Rembold, CM; Walker, JS | 1 |
Antunes, E; Baracat, JS; Claudino, MA; De Nucci, G; Priviero, FB; Teixeira, CE; Webb, RC | 1 |
Berg, KM; Evans, MC; Miner, AS; Porter, M; Ratz, PH; Ward, KR | 1 |
Honjo, H; Ito, S; Kamiya, K; Kodama, I; Kume, H; Oguma, T; Shimokata, K; Takeda, N | 1 |
Bai, Y; Sanderson, MJ | 1 |
Arreola, JL; Chávez, J; Flores-Soto, E; Montaño, LM; Segura, P; Vargas, MH | 1 |
Harada, M; Hirano, K; Hirano, M; Iwamoto, T; Kanaide, H; Karashima, E; Kita, S; Nishimura, J | 1 |
Ando, M; Mukuda, T; Sakihara, T; Watanabe, Y | 2 |
Minami, K; Ogata, J; Segawa, K | 1 |
Cornu, JN; Rouprêt, M | 1 |
Murthy, KS; Sriwai, W | 1 |
Alvarez, E; Cairrão, E; Morgado, M; Santos-Silva, AJ; Verde, I | 1 |
Araújo, PV; Clemente, CM; de Oliveira, RB; dos Santos, AA; Fernandes, GH; Magalhães, PJ; Palheta, RC; Ratts, ZM; Rola, FH | 1 |
Fatma, S; Grunstein, JS; Grunstein, MM; Hu, A; Nino, G | 1 |
Diamond, J; Vegesna, RV | 3 |
Göthert, M; Hentrich, F | 2 |
Bomzon, A; Finberg, JP; Hovevei-Sion, D; Youdim, MB | 1 |
Ajimal, GS; Gole, D; Haller, KA; Ram, JL; Williams, A | 1 |
Burka, JF | 2 |
Baer, HP; Muller, MJ | 1 |
Lindner, E; Metzger, H | 1 |
Gerthoffer, WT; Murphy, RA; Trevethick, MA | 1 |
Bylund, DB; Forte, LR; Jones, AW | 1 |
Forder, J; Kojima, I; Rasmussen, H; Scriabine, A | 1 |
Dhawan, BN; Dubey, MP; Nityanand, S; Srimal, RC | 1 |
Kendall, DA; Wilson, VG; Wright, IK | 1 |
Movahedi, H; Purdy, RE | 1 |
Bennett, JL; Blair, KL; Pax, RA | 1 |
Satoh, K; Taira, N; Yamagishi, T; Yanagisawa, T | 1 |
Dent, G; Magnussen, H; Nakashima, M; Rabe, KF; Schudt, C; Tenor, H | 1 |
Drescher, P; Eckert, RE; Madsen, PO | 1 |
Botella, A; Bueno, L; Delvaux, M; Fioramonti, J; Frexinos, J | 1 |
Eltze, M | 1 |
Linde, C; Quast, U | 1 |
Chowdhury, JU; Huang, SM; Pang, YW; Tomita, T; Tsugeno, M | 1 |
Rembold, CM; Stull, JT; Van Riper, DA; Weaver, BA | 1 |
Jino, H; Kurahashi, K; Nakata, Y; Shimizu, Y; Shirahase, H; Usui, H | 1 |
Latifpour, J; Nishimoto, T; Weiss, RM; Wheeler, MA; Yoshida, M | 1 |
McGrath, JC; Smith, GC | 1 |
Chess-Williams, R; Otter, DJ | 1 |
Giuliani, S; Maggi, CA; Santicioli, P | 1 |
Daniel, EE; Eng, R; Hipworth, S; Lu, S; McGrogan, I; Preocanin, D; Sormaz, L | 1 |
Ganten, D; Kreutz, R; Pfitzer, G; Satoh, S; Wilm, C | 1 |
Kurosawa, S; Owyang, C; Takahashi, T | 1 |
Bennett, JL; Day, TA; Pax, RA | 1 |
Conte Camerino, D; De Luca, A; Pierno, S; Tricarico, D | 1 |
Kamata, K; Kasuya, Y; Suenaga, H | 1 |
Begonha, R; Guimarães, S; Mota, A | 1 |
Botella, A; Bueno, L; Delvaux, M; Frexinos, J; Jeanneton, O | 1 |
Ichikawa, K; Ito, M; Itoh, H; Konishi, T; Nakano, T; Okubo, S; Shimomura, A | 1 |
Abe, A; Karaki, H | 4 |
Ito, S; Itoh, T; Suzuki, S | 1 |
Buxton, IL; Gerthoffer, WT; Keef, KD; Sanders, KM; Smith, TK; Ward, SM; Zhang, L | 1 |
Black, C; Curry, C; Emala, C; Hirshman, CA; Levine, MA | 1 |
Hori, M; Karaki, H; Mitsui, M; Ozaki, H; Tajimi, M | 1 |
Barnett, NL; Luttmann, W; Osborne, NN | 1 |
Ehlert, FJ; Thomas, EA | 2 |
Blankesteijn, WM; Raat, NJ; Thien, T; Willems, PH | 1 |
Forssmann, WG; Jonas, U; Kuczyk, M; Schulz-Knappe, P; Stief, CG; Truss, MC; Uckert, S | 1 |
Elzinga, CR; Hoiting, BH; Kuipers, R; Meurs, H; Schuiling, M; Zaagsma, J | 1 |
Delpy, E; le Monnier de Gouville, AC | 1 |
Edwards, SC; Hinsch, GW; Spaziani, EP | 1 |
Coste, H; Delpy, E; Gouville, AC | 1 |
Pfaffendorf, M; van Zwieten, PA; Winkler Prins, EA; Zwaveling, J | 1 |
Fredberg, JJ; Heyder, J; Hubmayr, RD; Moller, W; Panettieri, RA; Planus, E; Shore, SA; Wang, N | 1 |
Jino, H; Kurahashi, K; Nakata, Y; Shimizu, Y; Temma, S; Usui, H | 1 |
Huang, Y; Kwok, KH | 1 |
Satake, N; Shibata, S | 1 |
Collado, MC; Fuentes, T; Hernández, J; Martinez, E | 1 |
Drescher, P; Knes, JM; Madsen, PO; Rauch, D; Sparwasser, C | 1 |
Buus, C; Mulvany, MJ; Nilsson, H; Prieto, D | 1 |
Briscoe, JA; Leggett, RE; Longhurst, PA; Rosenberg, DJ | 1 |
Goldstein, I; Huang, YH; Moreland, RB; Traish, AM | 1 |
Ekblad, E; Sundler, F | 1 |
Hsieh, CM; Li, L; Shen, Y; Xi, M; Yang, LZ | 1 |
Kline, LW; Pang, PK | 1 |
Beall, A; Brophy, CM; Dickinson, M; Lamb, S; Ware, DJ | 1 |
Ehlert, FJ; Sawyer, GW | 1 |
Beall, A; Brophy, C; Epstein, A; Jerius, H; Woodrum, D | 1 |
Honjo, H; Kodama, I; Satake, K; Shibata, S; Takagi, K; Toyama, J | 1 |
Blackwell, K; Bodmer, JE; Moy, AB; Shasby, DM; Shasby, S | 1 |
Dickenson, JM; Hill, SJ | 1 |
Brooman, JE; Holden-Dye, L; Trim, N; Walker, RJ | 1 |
Fujimoto, N; Hanawa, T; Kimura, T | 1 |
Coutts, AA; Pertwee, RG | 1 |
Kendall, DA; Roberts, RE; Tomlinson, AE; Wilson, VG | 1 |
Fujimoto, S; Hiramoto, A; Inoue, Y; Itoh, T; Nagai, K; Ohashi, M; Shiokawa, H | 1 |
Christensen, G; Holt, E; Lunde, PK; Sejersted, OM; Semb, SO; Tønnessen, T; Wasserstrom, JA | 1 |
Gong, GX; Scholz, PM; Tse, J; Weiss, HR; Yan, L | 1 |
Tanaka, S; Tsuchida, H | 1 |
Mitchelson, F; Shen, A | 1 |
Bueno, L; Delvaux, M; Frexinos, J; Rekik, M | 1 |
Parkington, HC; Raymond, GL; Tonta, MA; Wendt, IR | 1 |
Kim, CJ; Sim, SS | 1 |
Bali, JP; Bataille, D; Geneviève, R; Jarrousse, C; Le Nguyen, D; Magous, R; Martinez, J; Mochizuki, T; Rodier, G | 1 |
Beall, A; Brophy, CM; Epstein, A; Woodrum, D | 1 |
Ehlert, F; Sawyer, G | 1 |
Makhlouf, GM; Murthy, KS | 1 |
Kendall, DA; Roberts, RE; Wilson, VG | 1 |
Crocker, P; Gibson, TM; Pertwee, RG; Razdan, RK; Ross, RA; Saha, B; Stevenson, LA | 1 |
Kitazawa, T; Maezono, Y; Taneike, T | 1 |
Fox, LE; Lloyd, PE | 1 |
Banner, WK; Gibson, TM; Martin, BR; Pertwee, RG; Razdan, RK; Ross, RA; Saha, B; Stevenson, LA | 1 |
Sekiguchi, F; Shimamura, K; Sunano, S; Yamamoto, K | 1 |
Elliott, RA; Hudman, D; Norman, RI | 1 |
Goldstein, I; Huang, YH; Kim, NN; Moreland, RB; Traish, A | 1 |
Furuya, K; Kato, K; Ozaki, T; Tsutsui, I; Yamagishi, S | 1 |
Matsuda, N; Sellke, FW | 1 |
Ahmad, M; Andersson, KE; Aszòdi, A; Fässler, R; Pandita, RK; Persson, K; Pfeifer, A | 1 |
Frith, D; Gibson, A | 1 |
Kidokoro, Y; Suzuki, K; Yoshihara, M | 1 |
Choi, JC; Hahn, SJ; Jo, YH; Kim, MS; Kim, YC; Min, DS; Rhie, DJ; Shim, HS; Sim, SS; Yoon, SH | 1 |
Fujii, Y; Hoshi, T; Toyooka, H | 1 |
Hashimoto, K; Igarashi, T; Imai, T; Mitani, A; Nakazawa, T; Noguchi, K; Otsuka, K; Saitoh, M; Shigenobu, K; Someya, S; Tanaka, H; Tanaka, Y; Yamaki, F | 1 |
Brixius, K; Fässler, R; Fleischmann, B; Herr, C; Hescheler, J; Lasek, K; Noegel, AA; Sasse, P; Schröder, R; Schwinger, RH; Smyth, N; Ullrich, S; Yun, F | 1 |
Ito, S; Ito, Y; Kume, H; Yamaki, K | 1 |
Bessard, G; Bréant, D; Caron, F; Corompt, E; Devillier, P | 1 |
Kalodimos, PJ; Ventura, S | 1 |
Craig, EC; Haynes-Johnson, D; Kraft, P; Liu, X; Qiu, Y | 1 |
Krymsky, MA; Kudryashov, DS; Lukas, TJ; Shirinsky, VP; Vorotnikov, AV; Watterson, DM | 1 |
Frölich, JC; Heuer, O; Jonas, U; Machtens, SA; Stief, CG; Tsikas, D; Uckert, S | 1 |
Chen, CF; Chiou, WF | 1 |
Ito, Y; Kume, H; Mizutani, H; Takagi, K; Yamaki, K | 1 |
Botella, A; Bueno, L; Delvaux, M; Frexinos, J | 1 |
Bradley, ME; Buxton, IL; Keef, KD; Zhang, L | 1 |
Abdel-Latif, AA; Akhtar, RA; Tachado, SD; Zhou, CJ | 1 |
Beck-Sickinger, AG; Gaida, W; Grouzmann, E; Hoffmann, E; Jung, G; van Meir, EG; Waeber, B | 1 |
Feniuk, W; Humphrey, PP; McCormick, JD; Sumner, MJ | 1 |
Yamakage, M | 1 |
Ahn, HY; Chang, KC; Kang, SE; Karaki, H | 1 |
Kubota, K; Matsuoka, Y; Nagahamaya, K; Shirane, M; Sunagane, N; Tsunematsu, R; Uruno, T; Wada, K | 1 |
Cheng, JT; Tsai, LH | 1 |
Adler, M; Filbert, MG; Moore, DH | 1 |
Aikawa, T; Itabashi, S; Morikawa, M; Sasaki, H; Sekizawa, K; Takishima, T | 1 |
Alibhai, KN; Huizinga, JD; Richardson, D | 1 |
Mouzou, A; Poindessault, JP; Raymond, G | 1 |
Duty, S; Weston, AH | 1 |
Boswell, CA; Joris, I; Majno, G; Ostrom, KA | 1 |
Bast, A; Van der Vliet, A | 1 |
Roberts, JM; Russell, JA | 1 |
Den Hertog, A; Manolopoulos, VG; Nelemans, A; Pipili-Synetos, E | 1 |
Morley, GP; Neild, TO | 1 |
Fujimoto, S; Matsuda, T | 1 |
De Mey, JG; Dijkstra, EH; Vrijdag, MJ | 1 |
De Mey, JG; Heesen, BJ | 1 |
Kohno, S; Matsubayashi, H; Tsuru, H | 1 |
Berkenboom, G; Fang, ZY; Fontaine, J; Goldman, M; Unger, P | 2 |
Huizinga, JD; Pintin-Quezada, J; Tomlinson, J | 1 |
Arnold, R; Casiano, F; Childers, SR; Pacheco, M; Ward, SJ | 1 |
Lloyd, PE; Lotshaw, DP | 1 |
Grider, JR | 1 |
Hori, M; Ishihara, H; Karaki, H; Kasai, H; Ozaki, H; Sato, K | 1 |
Blackshear, PJ; Lobaugh, LA | 1 |
Gustafsson, LE; Hedqvist, P; Ohlén, A; Wiklund, CU; Wiklund, NP | 1 |
Stuart-Smith, K; Vanhoutte, PM | 1 |
King, AD; Milavec-Krizman, M; Müller-Schweinitzer, E | 1 |
Karaki, H; Kwon, SC; Ozaki, H; Tajimi, M | 1 |
Chapman, RW; Gulbenkian, A; Kreutner, W; Tozzi, S | 1 |
Forder, J; Rasmussen, H; Scriabine, A | 1 |
Park, S; Rasmussen, H | 2 |
Lange, AB; Orchard, I | 1 |
Kondo, S; Miyagawa, I; Morita, T; Weiss, RM; Wheeler, MA | 1 |
Hoffman, BB; Lee, CH; Tsujimoto, G | 1 |
Cline, WH; Nickols, GA | 1 |
Carlsen, RC; Gourley, IM; Klein, HW; Matthews, CC | 1 |
Dorsett, JA; Yau, WM; Youther, ML | 1 |
Ahn, HY; Karaki, H; Urakawa, N | 1 |
Iida, H; Page, E | 1 |
Goy, MF; Kravitz, EA | 1 |
Asano, M; Masuzawa, K; Matsuda, T | 1 |
Auguet, M; Braquet, P; Clostre, F; Delaflotte, S; Pirotzky, E | 1 |
Kelly, E; Koenig, SM; Leff, AR; Mitchell, RW; Popovich, KJ; White, SR | 1 |
Fujimoto, M; Mihara, S; Shigeri, Y | 1 |
Danthuluri, NR; Deth, RC | 1 |
Moummi, C; Rattan, S | 2 |
Owen, DA; Wood, LM | 1 |
Kamata, K; Kasuya, Y; Miyata, N | 1 |
Bandyopadhyay, S; Gunst, SJ | 1 |
Nishimura, J; van Breemen, C | 1 |
DeFeo, TT; Morgan, KG | 1 |
Dale, MM; Obianime, AW | 1 |
Baskin, EP; Vlasuk, GP; Winquist, RJ | 1 |
Giesa, FR; Grimes, D; Heaslip, RJ; Rimele, TJ | 1 |
Orth, DN; Watanabe, T | 1 |
Linz, W; Schölkens, BA; Wiemer, G | 1 |
Gunst, SJ; Stropp, JQ | 1 |
Sasaguri, T; Stanley, AF; Watson, SP | 1 |
Hagiwara, M; Hidaka, H; Ishikawa, T; Itoh, H; Onoda, K; Tanaka, T | 1 |
Brown, JK; Madison, JM | 1 |
Carlsen, RC; Gourley, I; Klein, HW | 1 |
Baba, K; Honda, Y; Ito, H; Ito, M; Tomita, T | 2 |
Goldie, RG; Paterson, JW; Spina, D | 1 |
Ito, Y; Kuriyama, H; Miledi, R; Parker, I | 1 |
Auguet, M; Braquet, P; Clostre, F; Hellegouarch, A | 1 |
Bowman, WC; Lam, FY; Rodger, IW; Shahid, M | 1 |
Gustafsson, LE; Hedqvist, P; Lundin, J; Wiklund, NP | 1 |
Rubin, LL | 1 |
Edvinsson, L; Fredholm, BB; Jansen, I | 1 |
Pappano, AJ; Smith, CJ | 1 |
McMahon, EG; Paul, RJ | 1 |
Goldie, RG; Papadimitriou, JM; Paterson, JW; Rigby, PJ; Self, HM; Spina, D | 1 |
Satake, T; Suzuki, K; Takagi, K; Tsukawaki, M | 1 |
Honda, K; Satake, T; Takagi, K; Tomita, T | 1 |
Morita, T; Weiss, RM; Wheeler, MA | 1 |
Hwang, KS; Van Breemen, C | 1 |
Dohkita, S; Kondo, S; Morita, T; Tsuchida, S | 1 |
Itoh, H; Lederis, K | 1 |
Satake, T; Suzuki, K; Suzuki, R; Takagi, K; Tsukawaki, M | 1 |
Boyle, JP; Cortijo, J; Curtis-Prior, PB; Davies, JM; Foster, RW; Hofer, P; Small, RC | 1 |
Lodge, NJ; Nouailhetas, VL; Twort, CH; Van Breemen, C | 1 |
Kelley, G; Rasmussen, H; Takuwa, N; Takuwa, Y | 1 |
Huang, M; Lederis, K; Rorstad, OP; Suzuki, Y | 1 |
Rasmussen, H; Takuwa, N; Takuwa, Y | 1 |
Denborough, MA; Sim, AT; White, MD | 1 |
Bradley, RJ; Edge, MT | 1 |
Flaim, SF; Gleason, MM | 1 |
Prostran, M; Varagić, VM | 1 |
Cho, YH; Housman, A; Weiss, RM; Wheeler, MA | 1 |
Armour, CL; Hogg, JC; Paré, PD; Schellenberg, RR; Taylor, SM | 1 |
Burke, JA; Potter, DE; Temple, JR | 1 |
Waldeck, B; Widmark, E | 1 |
Addison, B; Babich, M; Piascik, MT | 1 |
Dale, MM; Obianime, W | 1 |
Cawthorpe, DR; Colmers, WF; Drummond, GI; Lukowiak, K; Rosenberg, J | 1 |
2 review(s) available for colforsin and Muscle Contraction
Article | Year |
---|---|
[Effects of colforsin daropate hydrochloride on myocardium, smooth muscle and renal function].
Topics: Adenylyl Cyclases; Animals; Cell Proliferation; Colforsin; Cyclic AMP; Glomerular Filtration Rate; Glomerulonephritis, Membranoproliferative; Heart Failure; Humans; Mesangial Cells; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Contraction; Receptors, Adrenergic, beta-1; Renal Circulation; Signal Transduction | 2007 |
Functional role of M2 muscarinic receptors in the guinea pig ileum.
Topics: Animals; Colforsin; Cyclic AMP; Guinea Pigs; Heart; Histamine; Ileum; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Pertussis Toxin; Piperidines; Rats; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Signal Transduction; Submandibular Gland; Virulence Factors, Bordetella | 1995 |
286 other study(ies) available for colforsin and Muscle Contraction
Article | Year |
---|---|
Combined agonists act synergistically to increase mucociliary clearance in a cystic fibrosis airway model.
Topics: Animals; Carbachol; Colforsin; Cystic Fibrosis; Disease Models, Animal; Drug Synergism; Drug Therapy, Combination; Ferrets; Isoproterenol; Mucociliary Clearance; Muscle Contraction; Muscle, Smooth; Swine | 2021 |
Modulation of carbachol-induced Ca
Topics: Animals; Calcium; Carbachol; Colforsin; Dinoprostone; Mice; Muscle Contraction; Muscle, Smooth; Myocytes, Smooth Muscle | 2022 |
Regulation of Vascular Smooth Muscle Contractions in the Model of Metabolic Syndrome.
Topics: Acetylcholine; Animals; Aorta; Body Weight; Calcium; Carbohydrates; Colforsin; Disease Models, Animal; Endothelium, Vascular; Glucose; Hemodynamics; Lipids; Male; Metabolic Syndrome; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Nitroprusside; Phenylephrine; Potassium Channels; Rats; Rats, Wistar; Stress, Mechanical; Triglycerides; Vasoconstriction | 2020 |
Possible roles for ATP release from RBCs exclude the cAMP-mediated Panx1 pathway.
Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Adenosine Triphosphate; Adenylyl Cyclases; Adult; Animals; Colforsin; Connexins; Cyclic AMP; Energy Metabolism; Erythrocytes; Exercise Tolerance; Female; Genotype; Gluconates; Hemolysis; Humans; Male; Mice, Inbred C57BL; Mice, Knockout; Muscle Contraction; Muscle, Skeletal; Nerve Tissue Proteins; Phenotype; Second Messenger Systems; Time Factors; Young Adult | 2017 |
Role of cyclic nucleotide-dependent actin cytoskeletal dynamics:Ca(2+)](i) and force suppression in forskolin-pretreated porcine coronary arteries.
Topics: Actin Cytoskeleton; Actin Depolymerizing Factors; Actins; Animals; Biomechanical Phenomena; Calcium; Cell Adhesion Molecules; Colforsin; Coronary Vessels; Histamine; HSP20 Heat-Shock Proteins; Intracellular Space; Microfilament Proteins; Muscle Contraction; Myosin Light Chains; Nucleotides, Cyclic; Paxillin; Phosphoproteins; Phosphorylation; Sus scrofa | 2013 |
Molecular and pharmacological characterization of zebrafish 'contractile' and 'inhibitory' prostanoid receptors.
Topics: Animals; Calcium; Chlorocebus aethiops; Cloning, Molecular; Colforsin; COS Cells; Gene Expression Profiling; Gene Expression Regulation; Humans; Mice; Muscle Contraction; Pertussis Toxin; Phylogeny; Receptors, G-Protein-Coupled; Receptors, Prostaglandin; Receptors, Prostaglandin E, EP3 Subtype; Receptors, Thromboxane; Signal Transduction; Tissue Distribution; Zebrafish; Zebrafish Proteins | 2013 |
Cranioselectivity of sumatriptan revisited: pronounced contractions to sumatriptan in small human isolated coronary artery.
Topics: Adolescent; Adult; Aged; Biphenyl Compounds; Child; Colforsin; Coronary Vessels; Cyclic AMP; Dose-Response Relationship, Drug; Female; Humans; Male; Meningeal Arteries; Middle Aged; Muscle Contraction; Piperazines; Piperidones; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Spiro Compounds; Sumatriptan; Tissue Culture Techniques; Vasoconstrictor Agents; Vasodilator Agents; Young Adult | 2014 |
Pyocyanin inhibits both nitric oxide-dependent and -independent relaxation in porcine coronary arteries.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Colforsin; Coronary Vessels; Cyclic AMP; Cyclic GMP; Diethylamines; Dinoprost; Female; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Nitric Oxide; Pseudomonas aeruginosa; Pyocyanine; Swine; Vasodilation | 2015 |
Insulin induces IRS2-dependent and GRK2-mediated β2AR internalization to attenuate βAR signaling in cardiomyocytes.
Topics: Animals; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Fluorescence Resonance Energy Transfer; G-Protein-Coupled Receptor Kinase 2; Insulin; Insulin Receptor Substrate Proteins; Mice; Mice, Knockout; Muscle Contraction; Myocytes, Cardiac; Phosphorylation; Protein Transport; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Signal Transduction | 2015 |
Heterogeneity in Kv7 channel function in the cerebral and coronary circulation.
Topics: Animals; Basilar Artery; Carbamates; Cerebrovascular Circulation; Circle of Willis; Colforsin; Coronary Circulation; Indoles; KCNQ Potassium Channels; KCNQ1 Potassium Channel; Male; Mice; Mice, Knockout; Muscle Contraction; Muscle, Smooth, Vascular; Organ Specificity; Phenylenediamines; Potassium Channel Blockers; Pyridines; Vasoconstriction; Vasodilation; Vasodilator Agents | 2015 |
β-Adrenoceptor-Mediated Relaxation of Carbachol-Pre-Contracted Mouse Detrusor.
Topics: Aminophenols; Animals; Carbachol; Cholinergic Agonists; Colforsin; Homozygote; Imidazoles; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Mucous Membrane; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-2; Sulfonamides; Urinary Bladder | 2015 |
Functional and molecular evidence for Kv7 channel subtypes in human detrusor from patients with and without bladder outflow obstruction.
Topics: Aged; Colforsin; Female; Gene Expression Regulation; Humans; Isoproterenol; KCNQ Potassium Channels; Male; Middle Aged; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Receptors, Adrenergic, beta; Urinary Bladder; Urinary Bladder Neck Obstruction | 2015 |
Vasodilator-stimulated phosphoprotein (VASP) regulates actin polymerization and contraction in airway smooth muscle by a vinculin-dependent mechanism.
Topics: Acetylcholine; Actins; Animals; Biocatalysis; Cell Adhesion Molecules; Cell Membrane; Chickens; Colforsin; Dogs; Epinephrine; Humans; Microfilament Proteins; Muscle Contraction; Muscle, Smooth; Phosphoproteins; Phosphorylation; Profilins; Protein Multimerization; Protein Structure, Quaternary; Protein Transport; Trachea; Tyrosine; Vinculin | 2015 |
Effects of papaverine on carbachol- and high K+ -induced contraction in the bovine abomasum.
Topics: Abomasum; Adjuvants, Immunologic; Animals; Carbachol; Cattle; Cholinergic Agonists; Colforsin; Muscle Contraction; Muscle, Smooth; Nitric Oxide Donors; Nitroprusside; Papaverine; Phosphodiesterase Inhibitors; Potassium | 2015 |
Contractile function of smooth muscle retained after overnight storage.
Topics: Animals; Carbachol; Colforsin; Endothelium, Vascular; Isoproterenol; Male; Models, Animal; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Phenylephrine; Rats; Rats, Sprague-Dawley; Time Factors; Tissue Preservation | 2015 |
Modulation of {beta}-adrenoceptor signaling in the hearts of 4-wk simulated weightlessness rats.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Anesthesia; Animals; Body Weight; Colforsin; Cyclic AMP; Electric Stimulation; Heart; Hindlimb Suspension; Isoproterenol; Male; Muscle Contraction; Myocardial Contraction; Myocytes, Cardiac; Organ Size; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Signal Transduction; Weightlessness Simulation | 2008 |
Inhibition of cardiomyocyte contractile/relaxation by MN9202 and mechanisms involved.
Topics: Animals; Calcium; Cell Shape; Colforsin; Dihydropyridines; Methylene Blue; Muscle Contraction; Muscle Relaxation; Myocytes, Cardiac; Nitrobenzenes; Rats; Tetraethylammonium | 2008 |
Effect of pre-contraction on β-adrenoceptor-mediated relaxation of rat urinary bladder.
Topics: Adrenergic beta-Agonists; Animals; Bradykinin; Carbachol; Colforsin; Dose-Response Relationship, Drug; Humans; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Potassium Chloride; Rats; Rats, Wistar; Serotonin; Urinary Bladder; Urinary Bladder, Overactive | 2009 |
Importance of neural mechanisms in colonic mucosal and muscular dysfunction in adult rats following neonatal colonic irritation.
Topics: Animals; Animals, Newborn; Carbachol; Chlorides; Cholinergic Agonists; Colforsin; Colon; Colonic Diseases; Electric Stimulation; Feces; In Vitro Techniques; Intestinal Mucosa; Male; Muscle Contraction; Muscle, Smooth; Permeability; Peroxidase; Potassium; Random Allocation; Rats; Rats, Sprague-Dawley | 2010 |
Effects of various selective phosphodiesterase inhibitors on relaxation and cyclic nucleotide contents in porcine iris sphincter.
Topics: Animals; Carbachol; Colforsin; Female; Iris; Male; Muscle Contraction; Nitroprusside; Phosphodiesterase Inhibitors; Swine; Tissue Culture Techniques | 2009 |
Colforsin-induced vasodilation in chronic hypoxic pulmonary hypertension in rats.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Chronic Disease; Colforsin; Dinoprost; Drug Synergism; Fluorescent Dyes; Fura-2; Hypertension, Pulmonary; Hypertrophy, Right Ventricular; Hypoxia; In Vitro Techniques; Isometric Contraction; Male; Muscle Contraction; Potassium Chloride; Pulmonary Artery; Rats; Rats, Wistar; Vasodilation; Vasodilator Agents | 2010 |
Impaired M3 and enhanced M2 muscarinic receptor contractile function in a streptozotocin model of mouse diabetic urinary bladder.
Topics: Animals; Colforsin; Diabetes Mellitus, Experimental; Disease Models, Animal; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscarinic Agonists; Muscle Contraction; Oxotremorine; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Streptozocin; Time Factors; Urinary Bladder | 2010 |
Inhibitory effect of caffeine on pacemaker activity in the oviduct is mediated by cAMP-regulated conductances.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; ATP-Binding Cassette Transporters; Biological Clocks; Caffeine; Colforsin; Cyclic AMP; Drug Interactions; Female; Glyburide; KATP Channels; Membrane Potentials; Mice; Mice, Inbred BALB C; Muscle Contraction; Muscle, Smooth; Oviducts; Phosphodiesterase Inhibitors; Pinacidil; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Sulfonylurea Receptors | 2011 |
Two for one: cyclic AMP mediates the anti-inflammatory and anti-spasmodic properties of the non-anesthetic lidocaine analog JMF2-1.
Topics: Adenylyl Cyclases; Animals; Anti-Inflammatory Agents; Apoptosis; Asthma; Carbachol; Caspase 8; Cell Proliferation; Cell Survival; Colforsin; Cyclic AMP; Epithelium; Guinea Pigs; Inflammation; Lidocaine; Lymph Nodes; Male; Mice; Mice, Inbred BALB C; Muscle Contraction; Myocytes, Smooth Muscle; NG-Nitroarginine Methyl Ester; Nitric Oxide; Parasympatholytics; Rats; Rats, Wistar; Respiratory System; T-Lymphocytes; Trachea | 2012 |
Contribution of the extracellular cAMP-adenosine pathway to dual coupling of β2-adrenoceptors to Gs and Gi proteins in mouse skeletal muscle.
Topics: Adenosine; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Animals; Clenbuterol; Colforsin; Cyclic AMP; Diaphragm; Electric Stimulation; Feedback, Physiological; Fenoterol; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Male; Mice; Muscle Contraction; Receptors, Adrenergic, beta-2; Rolipram; Signal Transduction | 2012 |
Evaluating the significance of cyclic adenosine monophosphate-mediated signaling in human prostate: a functional and biochemical study.
Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Aged; Benzamides; Colforsin; Cyclic AMP; Humans; In Vitro Techniques; Inhibitory Concentration 50; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Papaverine; Phosphodiesterase 4 Inhibitors; Phosphodiesterase 5 Inhibitors; Phosphodiesterase Inhibitors; Piperazines; Prostate; Purines; Pyridines; Rolipram; Signal Transduction; Sildenafil Citrate; Sulfones | 2012 |
Cross-talk between Rho-associated kinase and cyclic nucleotide-dependent kinase signaling pathways in the regulation of smooth muscle myosin light chain phosphatase.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Amino Acid Substitution; Animals; Colforsin; Cyclic AMP; Male; Muscle Contraction; Mutation, Missense; Myocytes, Smooth Muscle; Phosphorylation; Protein Phosphatase 1; Rats; Rats, Sprague-Dawley; rho-Associated Kinases; rhoA GTP-Binding Protein; Second Messenger Systems; Smooth Muscle Myosins; Vasoconstrictor Agents | 2012 |
cAMP/protein kinase A activates cystic fibrosis transmembrane conductance regulator for ATP release from rat skeletal muscle during low pH or contractions.
Topics: 1-Methyl-3-isobutylxanthine; Adenosine Triphosphate; Animals; Benzoates; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cystic Fibrosis Transmembrane Conductance Regulator; Glyburide; Hydrogen-Ion Concentration; Lactic Acid; Male; Muscle Contraction; Muscle, Skeletal; Myoblasts; Rats; Rats, Sprague-Dawley; Signal Transduction; Sodium-Calcium Exchanger; Sodium-Hydrogen Exchangers; Thiazolidines | 2012 |
High-dose colforsin daropate increases diaphragmatic contractility in dogs.
Topics: Animals; Cardiac Output; Colforsin; Diaphragm; Dogs; Hemodynamics; Muscle Contraction | 2002 |
Muscarinic M2 receptors in acetylcholine-isoproterenol functional antagonism in human isolated bronchus.
Topics: Acetylcholine; Bronchi; Colforsin; Cyclic AMP; Humans; In Vitro Techniques; Isoproterenol; Lung Neoplasms; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Piperidines; Receptor, Muscarinic M2; Receptors, Muscarinic | 2002 |
Effects of various nitric oxide-donating drugs on adrenergic tension of human seminal vesicles in vitro.
Topics: Adrenergic alpha-Agonists; Aged; Colforsin; Cyclic GMP; Ejaculation; Erectile Dysfunction; Humans; In Vitro Techniques; Isometric Contraction; Male; Middle Aged; Molsidomine; Muscle Contraction; Muscle, Smooth; Nitric Oxide Donors; Nitroprusside; Norepinephrine; S-Nitroso-N-Acetylpenicillamine; S-Nitrosoglutathione; Seminal Vesicles; Sexual Dysfunction, Physiological; Signal Transduction | 2003 |
Increased relaxant action of forskolin and isoproterenol against muscarinic agonist-induced contractions in smooth muscle from M2 receptor knockout mice.
Topics: Adrenergic beta-Agonists; Animals; Colforsin; Drug Combinations; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscle Contraction; Muscle Relaxants, Central; Muscle, Smooth; Receptor, Muscarinic M2; Receptors, Muscarinic | 2003 |
The effect of inhaled colforsin daropate on contractility of fatigued diaphragm in dogs.
Topics: Administration, Inhalation; Animals; Blood Pressure; Colforsin; Diaphragm; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; Electrophysiology; Heart Rate; Hemodynamics; Muscle Contraction; Muscle Fatigue; Muscle, Skeletal | 2003 |
TNF-[alpha] modulates murine tracheal rings responsiveness to G-protein-coupled receptor agonists and KCl.
Topics: Animals; Antigens, CD; Carbachol; Cholera Toxin; Colforsin; Dinoprostone; Drug Synergism; Female; In Vitro Techniques; Mice; Mice, Inbred BALB C; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Pertussis Toxin; Potassium Chloride; Receptors, G-Protein-Coupled; Receptors, Tumor Necrosis Factor; Receptors, Tumor Necrosis Factor, Type I; Trachea; Tumor Necrosis Factor-alpha | 2003 |
The small heat shock protein (HSP) 20 is dynamically associated with the actin cross-linking protein actinin.
Topics: Actinin; Actins; Animals; Carotid Arteries; Cattle; Colforsin; Heat-Shock Proteins; HSP20 Heat-Shock Proteins; Immunohistochemistry; Immunosorbent Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phosphoproteins; Phosphorylation; Serotonin | 2003 |
Pharmacological profile of the cyclic nociceptin/orphanin FQ analogues c[Cys10,14]N/OFQ(1-14)NH2 and c[Nphe1,Cys10,14]N/OFQ(1-14)NH2.
Topics: Animals; Binding, Competitive; Cell Membrane; Cerebral Cortex; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cysteine; Dose-Response Relationship, Drug; Electric Stimulation; Female; GTP-Binding Proteins; Male; Mice; Muscle Contraction; Naloxone; Narcotic Antagonists; Nociceptin; Opioid Peptides; Phenylalanine; Radioligand Assay; Rats; Rats, Wistar; Receptors, Opioid; Recombinant Proteins; Vas Deferens | 2003 |
Experimental strategies to promote functional recovery after peripheral nerve injuries.
Topics: Animals; Autonomic Denervation; Axons; Axotomy; Brain-Derived Neurotrophic Factor; Cell Count; Colforsin; Dextrans; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Evoked Potentials, Motor; Humans; In Vitro Techniques; Mice; Mice, Knockout; Motor Neurons; Muscle Contraction; Nerve Degeneration; Nerve Growth Factors; Nerve Regeneration; Peripheral Nerve Injuries; Peripheral Nerves; Rats; Receptor, Nerve Growth Factor; Receptor, trkB; Receptors, Nerve Growth Factor; Recovery of Function; Rhodamines; Schwann Cells; Tacrolimus; Time Factors; Transforming Growth Factor beta | 2003 |
Correlation between spontaneous electrical, calcium and mechanical activity in detrusor smooth muscle of the guinea-pig bladder.
Topics: Action Potentials; Amides; Animals; Apamin; Boron Compounds; Calcium; Calcium Signaling; Carbachol; Charybdotoxin; Colforsin; Cromakalim; Cyclic GMP; Dose-Response Relationship, Drug; Drug Synergism; Female; Fura-2; Guinea Pigs; Isotonic Contraction; Male; Mechanotransduction, Cellular; Microelectrodes; Muscle Contraction; Muscle, Smooth; Nifedipine; Pyridines; Transducers; Urinary Bladder | 2004 |
(S)-Albuterol activates pro-constrictory and pro-inflammatory pathways in human bronchial smooth muscle cells.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Albuterol; Bronchi; Calcium; Cells, Cultured; Colforsin; GTP-Binding Protein alpha Subunits; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; Inflammation; Muscle Contraction; Muscle, Smooth; NF-kappa B; Phosphatidylinositol 3-Kinases; Stereoisomerism | 2004 |
Evidence for nonadrenoceptor responses to imidazoline derivatives in the porcine isolated rectal artery.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-Antagonists; Animals; Arteries; Benzofurans; Colforsin; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Phenoxybenzamine; Receptors, Drug; Rectum; Swine; Vasoconstrictor Agents | 2003 |
Nickel inhibits urocortin-induced relaxation in the rat pulmonary artery.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Atrial Natriuretic Factor; Colforsin; Corticotropin-Releasing Hormone; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nickel; Potassium; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Sodium-Calcium Exchanger; Urocortins; Vasoconstrictor Agents | 2004 |
Evidence for a possible neurotransmitter/neuromodulator role of tyramine on the locust oviducts.
Topics: Adrenergic alpha-Antagonists; Animals; Calcium; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Electric Stimulation; Female; Grasshoppers; Immunohistochemistry; Membrane Potentials; Muscle Contraction; Neuromuscular Junction; Neuropeptides; Neurotransmitter Agents; Oligopeptides; Oviducts; Potassium; Tyramine | 2004 |
Phosphodiesterase-linked inhibition of nonmicturition activity in the isolated bladder.
Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Animals; Colforsin; Cyclic AMP; Female; Guinea Pigs; Muscle Contraction; Phosphodiesterase Inhibitors; Pressure; Urinary Bladder; Urination | 2004 |
Novel phosphospecific antibodies for monitoring phosphorylation of proteins encoded by the myosin light chain kinase genetic locus.
Topics: Amino Acid Sequence; Animals; Calcium; Colforsin; Cyclic AMP-Dependent Protein Kinases; Male; Mitogen-Activated Protein Kinases; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Myosin-Light-Chain Kinase; Peptide Fragments; Phorbol 12,13-Dibutyrate; Phosphorylation; Rats; Sequence Homology, Amino Acid; Serine; Signal Transduction | 2004 |
Effects of various selective phosphodiesterase inhibitors on carbachol-induced contraction and cyclic nucleotide contents in guinea pig taenia coli.
Topics: Adenine; Animals; Carbachol; Colforsin; Colon; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Guinea Pigs; Male; Milrinone; Muscle Contraction; Nitroprusside; Nucleotides, Cyclic; Phosphodiesterase Inhibitors; Purinones; Vinca Alkaloids | 2004 |
Heat shock protein 20-mediated force suppression in forskolin-relaxed swine carotid artery.
Topics: Actins; Amino Acid Sequence; Animals; Carotid Arteries; Colforsin; Heat-Shock Proteins; HSP20 Heat-Shock Proteins; Humans; Molecular Sequence Data; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nucleotides, Cyclic; Phosphoproteins; Phosphorylation; Sequence Alignment; Serine; Stress, Mechanical; Swine | 2005 |
The M2 muscarinic receptor mediates contraction through indirect mechanisms in mouse urinary bladder.
Topics: Adrenergic beta-Agonists; Animals; Binding, Competitive; Colforsin; Dinoprost; Diphenylacetic Acids; In Vitro Techniques; Isoproterenol; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscarinic Agonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Oxotremorine; Piperidines; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Urinary Bladder | 2005 |
Anxiolytic-like effect of a serotonergic ligand with high affinity for 5-HT1A, 5-HT2A and 5-HT3 receptors.
Topics: 3,4-Dihydroxyphenylacetic Acid; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Anti-Anxiety Agents; Behavior, Animal; Binding, Competitive; Body Temperature Regulation; Bradycardia; Colforsin; Dopamine; Dose-Response Relationship, Drug; Guinea Pigs; HeLa Cells; Humans; Hydroxyindoleacetic Acid; Hypothalamus; Ileum; In Vitro Techniques; Male; Membrane Potentials; Mice; Motor Activity; Muscle Contraction; Neurons; Piperazines; Pyrazines; Radioligand Assay; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Receptor Agonists; Social Behavior; Transfection | 2005 |
Insulin-induced changes in beta-adrenergic response: an experimental study in the isolated rat papillary muscle.
Topics: Adrenergic beta-Agonists; Animals; Calcium; Colforsin; Dose-Response Relationship, Drug; Drug Interactions; Hypoglycemic Agents; In Vitro Techniques; Insulin; Isoproterenol; Male; Muscle Contraction; Papillary Muscles; Rats; Rats, Inbred WKY; Receptors, Adrenergic, beta | 2005 |
Potentiation of beta-adrenoceptor function in bovine tracheal smooth muscle by inhibition of protein kinase C.
Topics: Adrenergic beta-Agonists; Animals; Cattle; Colforsin; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Histamine; In Vitro Techniques; Indoles; Isoproterenol; Maleimides; Methacholine Chloride; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Protein Kinase C; Receptors, Adrenergic, beta; Trachea | 2005 |
Enhanced oxidative stress impairs cAMP-mediated dilation by reducing Kv channel function in small coronary arteries of diabetic rats.
Topics: 4-Aminopyridine; Animals; Antioxidants; Blood Glucose; Body Weight; Colforsin; Coronary Vessels; Cyclic AMP; Diabetes Mellitus, Experimental; Male; Microscopy, Video; Muscle Contraction; NADPH Oxidases; Oxidative Stress; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Spectrometry, Fluorescence; Superoxides; Vasodilation | 2005 |
Absence of force suppression in rabbit bladder correlates with low expression of heat shock protein 20.
Topics: Adenylyl Cyclases; Animals; Carbachol; Carotid Arteries; Colforsin; Cyclic GMP; Enzyme Activation; HSP20 Heat-Shock Proteins; Immunologic Techniques; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Myosin Light Chains; Phosphorylation; Rabbits; Staining and Labeling; Swine; Urinary Bladder | 2005 |
Stimulation of soluble guanylyl cyclase by BAY 41-2272 relaxes anococcygeus muscle: interaction with nitric oxide.
Topics: Animals; Carbachol; Carbolines; Colforsin; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Drug Synergism; Electric Stimulation; Enzyme Activation; Enzyme Inhibitors; Guanylate Cyclase; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase; Nitroglycerin; Oxadiazoles; Pyrazoles; Pyridines; Quinoxalines; Rats; Rats, Wistar; Receptors, Cytoplasmic and Nuclear; Soluble Guanylyl Cyclase; Tadalafil; Tetrodotoxin | 2006 |
Convergence of Ca2+-desensitizing mechanisms activated by forskolin and phenylephrine pretreatment, but not 8-bromo-cGMP.
Topics: Animals; Blotting, Western; Calcium; Cells, Cultured; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Electrophoresis, Polyacrylamide Gel; Endothelium, Vascular; Femoral Artery; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Phenylephrine; Phosphorylation; Potassium Chloride; Rabbits; Vasoconstrictor Agents | 2006 |
Involvement of reduced sensitivity to Ca in beta-adrenergic action on airway smooth muscle.
Topics: Adrenergic beta-Agonists; Amides; Animals; Asthma; Bucladesine; Calcium; Calcium Channel Blockers; Colforsin; Cyclic AMP Receptor Protein; Cyclic AMP-Dependent Protein Kinases; Depression, Chemical; Fura-2; Guinea Pigs; Imidazoles; In Vitro Techniques; Indoles; Intracellular Signaling Peptides and Proteins; Isoproterenol; Male; Maleimides; Marine Toxins; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Myosin-Light-Chain Phosphatase; Oxazoles; Protein Kinase C; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Trachea | 2006 |
Modulation of the Ca2+ sensitivity of airway smooth muscle cells in murine lung slices.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Arterioles; Bronchoconstrictor Agents; Caffeine; Calcium; Central Nervous System Stimulants; Colforsin; Cyclic AMP; Enzyme Inhibitors; In Vitro Techniques; Male; Methacholine Chloride; Mice; Mice, Inbred BALB C; Muscle Contraction; Myocytes, Smooth Muscle; Protein Kinase C; Respiratory System; Ryanodine | 2006 |
Paradoxical effect of salbutamol in a model of acute organophosphates intoxication in guinea pigs: role of substance P release.
Topics: Albuterol; Animals; Calcium; Cholinesterase Inhibitors; Colforsin; Diamines; Guinea Pigs; Lung; Male; Muscle Contraction; omega-Conotoxins; Parathion; Physostigmine; Pirenzepine; Plethysmography, Whole Body; Substance P; Tetrodotoxin; Tryptophan | 2007 |
Involvement of Na+-Ca2+ exchanger in cAMP-mediated relaxation in mice aorta: evaluation using transgenic mice.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Aniline Compounds; Animals; Aorta; Aorta, Thoracic; Calcium; Colforsin; Cyclic AMP; Dinoprost; Dogs; Fluorescent Dyes; Fluorometry; Fura-2; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phenyl Ethers; Sodium; Sodium-Calcium Exchanger; Vasoconstrictor Agents | 2007 |
Antagonistic effects of vasotocin and isotocin on the upper esophageal sphincter muscle of the eel acclimated to seawater.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Acclimatization; Anguilla; Animals; Antidiuretic Hormone Receptor Antagonists; Colforsin; Drinking Behavior; Esophageal Sphincter, Upper; Muscle Contraction; Oxytocin; Receptors, Oxytocin; Seawater; Vasotocin | 2007 |
Post- and pre-synaptic action of isotocin in the upper esophageal sphincter muscle of the eel: its role in water drinking.
Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Anesthetics, Local; Anguilla; Animals; Colforsin; Dose-Response Relationship, Drug; Drinking Behavior; Esophageal Sphincter, Upper; Muscle Contraction; Oxytocin; Phosphodiesterase Inhibitors; Presynaptic Terminals; Synapses; Tetrodotoxin | 2007 |
[Recent progress in basic research concerning the management of benign prostatic hyperplasia].
Topics: Colforsin; Humans; Male; Muscle Contraction; Muscle, Skeletal; Phenylephrine; Piperazines; Prostatic Hyperplasia; Purines; Rolipram; Sildenafil Citrate; Sulfones | 2007 |
Stimulatory phosphorylation of cAMP-specific PDE4D5 by contractile agonists is mediated by PKC-dependent inactivation of protein phosphatase 2A.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Cells, Cultured; Cholecystokinin; Colforsin; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Enzyme Activation; Enzyme Activators; Enzyme Inhibitors; Gastric Mucosa; GTP-Binding Protein alpha Subunits, Gq-G11; Muscle Contraction; Myocytes, Smooth Muscle; Okadaic Acid; Phospholipase C beta; Phosphorylation; Protein Kinase C; Protein Phosphatase 2; Rabbits; Signal Transduction; Stomach; Transfection | 2008 |
PDE4 and PDE5 regulate cyclic nucleotides relaxing effects in human umbilical arteries.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Colforsin; Cyclic AMP; Cyclic GMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Cyclic Nucleotide Phosphodiesterases, Type 5; Dipyridamole; Female; Guanylate Cyclase; Histamine; Humans; In Vitro Techniques; Isoenzymes; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Naphthyridines; Nitroprusside; Phosphodiesterase 4 Inhibitors; Phosphodiesterase 5 Inhibitors; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; Rolipram; Serotonin; Umbilical Arteries; Vasodilator Agents | 2008 |
Sildenafil inhibits duodenal contractility via activation of the NO-K+ channel pathway.
Topics: Animals; Colforsin; Diazoxide; Duodenum; In Vitro Techniques; Male; Muscle Contraction; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase Type II; Nitric Oxide Synthase Type III; Nitroprusside; Phosphodiesterase Inhibitors; Piperazines; Potassium Channel Blockers; Potassium Channels; Purines; Rats; Rats, Wistar; Sildenafil Citrate; Sulfones; Vasodilator Agents | 2008 |
Prolonged heterologous beta2-adrenoceptor desensitization promotes proasthmatic airway smooth muscle function via PKA/ERK1/2-mediated phosphodiesterase-4 induction.
Topics: Adrenergic beta-2 Receptor Agonists; Animals; Asthma; Butadienes; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Cyclic Nucleotide Phosphodiesterases, Type 4; Dinoprostone; Enzyme Induction; Humans; Isoquinolines; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Muscle Contraction; Muscle Relaxation; Nitriles; Pertussis Toxin; Phosphodiesterase 4 Inhibitors; Rabbits; Receptors, G-Protein-Coupled; Rolipram; Signal Transduction; Sulfonamides; Trachea | 2008 |
Effects of isoproterenol and forskolin on tension, cyclic AMP levels, and cyclic AMP dependent protein kinase activity in bovine coronary artery.
Topics: Animals; Cardiotonic Agents; Cattle; Colforsin; Coronary Vessels; Cyclic AMP; Diterpenes; In Vitro Techniques; Isoproterenol; Muscle Contraction; Protein Kinases | 1984 |
Role of cAMP for regulation of impulse-evoked noradrenaline release from the rabbit pulmonary artery and its possible relationship to presynaptic ACTH receptors.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Bucladesine; Colforsin; Cyclic AMP; Diterpenes; Electric Stimulation; Enzyme Activation; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Naphthyridines; Norepinephrine; Phosphodiesterase Inhibitors; Pulmonary Artery; Rabbits; Receptors, Cell Surface; Receptors, Corticotropin | 1984 |
Effects of forskolin in rat vas deferens--evidence for facilitatory beta-adrenoceptors.
Topics: Adrenergic beta-Agonists; Animals; Colforsin; Diterpenes; Electric Stimulation; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Rats; Rats, Inbred Strains; Vas Deferens | 1983 |
Serotonin and forskolin enhance both magnitude of contraction and relaxation rate of Aplysia dorsal extrinsic muscle independently of acetylcholine receptor.
Topics: Acetylcholine; Animals; Aplysia; Colforsin; Cyclic AMP; Diterpenes; Electric Stimulation; Ethanol; Hexamethonium Compounds; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscles; Receptors, Cholinergic; Serotonin | 1984 |
Effects of selected bronchodilators on antigen- and A23187-induced contraction of guinea-pig trachea.
Topics: Aminophylline; Animals; Anti-Bacterial Agents; Antigens; Bronchodilator Agents; Bucladesine; Calcimycin; Colforsin; Dinoprostone; Diterpenes; Guinea Pigs; Indomethacin; Isoproterenol; Male; Muscle Contraction; Ovalbumin; Prostaglandins E; Trachea | 1983 |
Relaxant effects of forskolin in smooth muscle. Role of cyclic AMP.
Topics: Adenylyl Cyclases; Animals; Cattle; Colforsin; Cyclic AMP; Diterpenes; Dogs; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Muscle, Smooth, Vascular; Phosphodiesterase Inhibitors; Rabbits; Rats; Rats, Inbred Strains; Species Specificity | 1983 |
Comparison of the effects of forskolin and isoproterenol on cyclic AMP levels and tension in bovine coronary artery.
Topics: Animals; Cattle; Colforsin; Cyclic AMP; Diterpenes; Isoproterenol; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular | 1983 |
The action of forskolin on muscle cells is modified by hormones, calcium ions and calcium antagonists.
Topics: Adenylyl Cyclases; Animals; Calcium; Calcium Channel Blockers; Colforsin; Diterpenes; Electric Stimulation; Guinea Pigs; Hormones; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Myocardium; Protein Kinases; Proteins; Rats; Rats, Inbred Strains; Sodium-Potassium-Exchanging ATPase | 1983 |
Myosin phosphorylation and cyclic adenosine 3',5'-monophosphate in relaxation of arterial smooth muscle by vasodilators.
Topics: Animals; Carotid Arteries; Colforsin; Cyclic AMP; Diterpenes; Dose-Response Relationship, Drug; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Myosins; Phosphorylation; Swine; Time Factors; Vasodilator Agents | 1984 |
cAMP-dependent reduction in membrane fluxes during relaxation of arterial smooth muscle.
Topics: Angiotensin II; Animals; Arteries; Colforsin; Cyclic AMP; Diterpenes; Male; Membranes; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Potassium Radioisotopes; Rats; Rats, Inbred Strains; Time Factors | 1984 |
Inhibition of antigen and calcium ionophore A23187 induced contractions of guinea pig airways by isoprenaline and forskolin.
Topics: Animals; Anti-Bacterial Agents; Calcimycin; Cardiotonic Agents; Colforsin; Diterpenes; Guinea Pigs; Immunization; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle, Smooth; Ovalbumin; Trachea | 1983 |
TPA-induced contraction of isolated rabbit vascular smooth muscle.
Topics: Animals; Arteries; Calcimycin; Calcium; Colforsin; Diterpenes; Kinetics; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Phorbols; Phosphorylation; Protein Kinases; Rabbits; Tetradecanoylphorbol Acetate | 1984 |
Pharmacological studies on coleonol, a hypotensive diterpene from Coleus forskohlii.
Topics: Animals; Antihypertensive Agents; Behavior, Animal; Blood Pressure; Cats; Colforsin; Diterpenes; Dogs; Guinea Pigs; Hemodynamics; In Vitro Techniques; Lethal Dose 50; Mice; Muscle Contraction; Muscle, Smooth; Rabbits; Rats | 1981 |
Alpha 2-adrenoceptor mediated inhibition of forskolin-stimulated cyclic AMP accumulation in isolated porcine palmar lateral veins.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenine; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Colforsin; Cyclic AMP; Enzyme Inhibitors; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Prazosin; Pyrrolidinones; Receptors, Adrenergic, alpha-2; Rolipram; Swine; Veins; Yohimbine | 1995 |
Serotoninergic 5-HT1-like receptors of the rabbit ear artery: how silent are they?
Topics: Adenylyl Cyclases; Animals; Arteries; Colforsin; Ear, External; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Rabbits; Receptors, Serotonin | 1995 |
Serotonin and acetylcholine: further analysis of praziquantel-induced contraction of magnesium-paralysed Schistosoma mansoni.
Topics: 1-Methyl-3-isobutylxanthine; 4-Aminopyridine; Amifampridine; Animals; Arecoline; Carbachol; Colforsin; Dose-Response Relationship, Drug; In Vitro Techniques; Ions; Magnesium; Male; Muscle Contraction; Paralysis; Phorbol 12,13-Dibutyrate; Praziquantel; Schistosoma mansoni; Serotonin | 1993 |
Relaxant mechanisms of cyclic AMP-increasing agents in porcine coronary artery.
Topics: 1-Methyl-3-isobutylxanthine; 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic beta-Agonists; Animals; Calcium; Colforsin; Coronary Vessels; Cyclic AMP; Cyclic GMP; Ethanolamines; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Potassium Chloride; Prostaglandin Endoperoxides, Synthetic; Ryanodine; Swine; Thromboxane A2; Vasodilator Agents | 1994 |
Identification of PDE isozymes in human pulmonary artery and effect of selective PDE inhibitors.
Topics: 1-Methyl-3-isobutylxanthine; Adult; Aged; Antihypertensive Agents; Carbachol; Colforsin; Cytosol; Dinoprost; Dose-Response Relationship, Drug; Female; Humans; Isoenzymes; Kinetics; Lung Neoplasms; Male; Middle Aged; Muscle Contraction; Muscle Relaxation; Muscle Tonus; Muscle, Smooth, Vascular; Nitroprusside; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Pulmonary Artery; Purinones; Pyridazines; Pyrrolidinones; Rolipram | 1994 |
Smooth muscle contractility in prostatic hyperplasia: role of cyclic adenosine monophosphate.
Topics: Bucladesine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Humans; Male; Milrinone; Muscle Contraction; Muscle, Smooth; Papaverine; Phenylephrine; Prostatic Hyperplasia; Pyridones; Theophylline | 1994 |
Galanin induces opposite effects via different intracellular pathways in smooth muscle cells from dog colon.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cholecystokinin; Colforsin; Colon; Cyclic AMP; Dogs; Ethylmaleimide; Galanin; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neuropeptides; Peptides; Pertussis Toxin; Somatostatin; Thionucleotides; Vasoactive Intestinal Peptide; Virulence Factors, Bordetella | 1994 |
Pathways involved in muscarinic M1 and M2 receptor stimulation in rabbit vas deferens.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Adenylyl Cyclase Inhibitors; Animals; Carbachol; Colforsin; Dose-Response Relationship, Drug; Electric Stimulation; In Vitro Techniques; Lithium Chloride; Male; Muscle Contraction; Muscle, Smooth; Parasympathomimetics; Phosphatidylinositols; Rabbits; Receptors, Muscarinic; Signal Transduction; Stereoisomerism; Tetradecanoylphorbol Acetate; Vas Deferens | 1994 |
Potentiation of P1075-induced K+ channel opening by stimulation of adenylate cyclase in rat isolated aorta.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Aorta; Binding, Competitive; Bucladesine; Colforsin; Cyclic AMP-Dependent Protein Kinases; Drug Interactions; Enzyme Activation; Enzyme Inhibitors; Guanidines; In Vitro Techniques; Isoquinolines; Isotope Labeling; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phosphodiesterase Inhibitors; Potassium Channels; Pyridines; Rats; Rats, Sprague-Dawley; Rubidium; Sulfonamides; Vasodilator Agents | 1995 |
Sustained contraction produced by caffeine after ryanodine treatment in the circular muscle of the guinea-pig gastric antrum and rabbit portal vein.
Topics: Animals; Caffeine; Calcium; Carbachol; Colforsin; Female; Fura-2; Guinea Pigs; Indomethacin; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Portal Vein; Pyloric Antrum; Rabbits; Ryanodine | 1995 |
Myosin light chain kinase phosphorylation in swine carotid artery contraction and relaxation.
Topics: Animals; Calcium; Carotid Artery, Common; Colforsin; Histamine; In Vitro Techniques; Kinetics; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Myosins; Peptide Mapping; Phosphates; Phosphopeptides; Phosphorus Radioisotopes; Phosphorylation; Potassium Chloride; Swine | 1995 |
Pharmacological natures of caffeine-induced endothelium-dependent and -independent contraction in canine mesenteric artery.
Topics: Adenylyl Cyclases; Animals; Benzopyrans; Caffeine; Calcium; Calcium Channel Blockers; Colforsin; Cromakalim; Dogs; Edetic Acid; Egtazic Acid; Endothelium, Vascular; Female; In Vitro Techniques; Magnesium; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Nitroglycerin; Potassium Channels; Pyrroles; Vasodilator Agents | 1995 |
Age-dependent alterations in beta-adrenergic responsiveness of rat detrusor smooth muscle.
Topics: Aging; Animals; Bucladesine; Cholera Toxin; Colforsin; Cyclic AMP; Electric Stimulation; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Potassium Chloride; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta; Urinary Bladder | 1995 |
Contractile effects of prostanoids on fetal rabbit ductus arteriosus.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Analysis of Variance; Animals; Colforsin; Dinoprost; Dinoprostone; Dose-Response Relationship, Drug; Ductus Arteriosus; Female; In Vitro Techniques; Indomethacin; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Pregnancy; Prostaglandin Endoperoxides, Synthetic; Prostaglandins E, Synthetic; Rabbits; Receptors, Prostaglandin; Thromboxane A2; Thromboxanes; Vasoconstrictor Agents | 1995 |
The effects of aldose reductase inhibition with ponalrestat on changes in vascular function in streptozotocin diabetic rats.
Topics: Aldehyde Reductase; Animals; Aorta, Thoracic; Carbachol; Colforsin; Diabetes Mellitus, Experimental; Endothelium, Vascular; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroprusside; Phenylephrine; Phthalazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1 | 1994 |
Multiple mechanisms in the smooth muscle relaxant action of calcitonin gene-related peptide (CGRP) in the guinea-pig ureter.
Topics: Action Potentials; Animals; Arginine; Benzopyrans; Calcitonin Gene-Related Peptide; Colforsin; Cromakalim; Dose-Response Relationship, Drug; Electric Stimulation; Glyburide; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Nitroarginine; Parasympatholytics; Pyrroles; Ureter | 1994 |
Mechanisms of cyclic nucleotide-induced relaxation in canine tracheal smooth muscle.
Topics: Adenylyl Cyclases; Animals; Calcium Channels; Calcium-Transporting ATPases; Carbachol; Colforsin; Cyclic AMP; Cyclic GMP; Dogs; Female; Indoles; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Potassium Chloride; Sarcoplasmic Reticulum; Trachea | 1995 |
Augmented agonist-induced Ca(2+)-sensitization of coronary artery contraction in genetically hypertensive rats. Evidence for altered signal transduction in the coronary smooth muscle cells.
Topics: Actin Cytoskeleton; Animals; Calcium; Cell Membrane Permeability; Colforsin; Coronary Vessels; Escin; Guanosine 5'-O-(3-Thiotriphosphate); Hypertension; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Potassium Chloride; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Serotonin; Signal Transduction | 1994 |
Regulation of PI hydrolysis and cAMP formation by muscarinic M3 receptor in guinea pig gallbladder.
Topics: Animals; Carbachol; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Gallbladder; Guinea Pigs; Hydrolysis; Male; Muscarinic Antagonists; Muscle Contraction; Phosphatidylinositols; Receptors, Muscarinic; Sincalide | 1994 |
Serotonin and its requirement for maintenance of contractility in muscle fibres isolated from Schistosoma mansoni.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Antimony Potassium Tartrate; Calcium; Cobalt; Colforsin; Culture Media; Dose-Response Relationship, Drug; Muscle Contraction; Nicardipine; Potassium; Protein Kinase Inhibitors; Schistosoma mansoni; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1994 |
Aging and chloride channel regulation in rat fast-twitch muscle fibres.
Topics: Aging; Animals; Calcimycin; Chloride Channels; Chlorides; Cholera Toxin; Colforsin; Electric Conductivity; Male; Muscle Contraction; Muscles; Phorbol 12,13-Dibutyrate; Potassium; Rats; Rats, Wistar; Time Factors; Toes; Virulence Factors, Bordetella | 1994 |
Phorbol ester (PMA)-induced biphasic contraction of the rat aorta and effects of sodium nitroprusside and forskolin on the contraction.
Topics: Adenylyl Cyclases; Animals; Aorta, Thoracic; Calcium; Calcium Channels; Colforsin; Drug Interactions; Enzyme Activation; Guanylate Cyclase; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroprusside; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate | 1993 |
The effectiveness of beta-adrenoceptor stimulation and the contribution of beta 1-adrenoceptors increase from the proximal to the distal part of the canine saphenous vein.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atenolol; Colforsin; Dobutamine; Dogs; Epinephrine; Female; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Propanolamines; Receptors, Adrenergic, beta; Saphenous Vein; Terbutaline | 1993 |
Platelet-activating factor (PAF) induces a contraction of isolated smooth muscle cells from guinea pig ileum: intracellular pathway involved.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Animals; Calcium; Cholera Toxin; Colforsin; GTP-Binding Proteins; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Pertussis Toxin; Platelet Activating Factor; Platelet Membrane Glycoproteins; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Signal Transduction; Sincalide; Vasoactive Intestinal Peptide; Virulence Factors, Bordetella | 1993 |
Inhibition of myosin light chain phosphatase during Ca(2+)-independent vasocontraction.
Topics: Animals; Aorta, Thoracic; Calcium; Colforsin; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Phosphatase; Norepinephrine; Phorbol 12,13-Dibutyrate; Phorbols; Phosphates; Phosphoprotein Phosphatases; Phosphorus Radioisotopes; Rats; Rats, Wistar; Vasoconstriction; Vasodilator Agents | 1993 |
Synergistic effects of cyclic AMP-related vasodilators and the phosphatase inhibitor okadaic acid.
Topics: Animals; Aorta; Atrial Natriuretic Factor; Bucladesine; Colforsin; Drug Synergism; Ethers, Cyclic; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nicardipine; Nitroglycerin; Nitroprusside; Okadaic Acid; Phosphoprotein Phosphatases; Potassium; Rats; Rats, Wistar; Vasodilator Agents; Verapamil | 1993 |
Effects of a water-soluble forskolin derivative (NKH477) and a membrane-permeable cyclic AMP analogue on noradrenaline-induced Ca2+ mobilization in smooth muscle of rabbit mesenteric artery.
Topics: Animals; Bucladesine; Calcium; Cell Membrane Permeability; Colforsin; Escin; Inositol 1,4,5-Trisphosphate; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Potassium; Rabbits; Solubility; Vasodilator Agents; Water | 1993 |
Beta-adrenergic inhibition of electrical and mechanical activity in canine colon: role of cAMP.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Animals; Bacterial Toxins; Calcium; Colforsin; Colon; Cyclic AMP; Dogs; Electric Stimulation; Female; Fura-2; Hemolysin Proteins; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Neurotoxins; Receptors, Adrenergic, beta; Spectrometry, Fluorescence; Tetrodotoxin; Time Factors | 1993 |
Impaired beta-adrenergic receptor activation of adenylyl cyclase in airway smooth muscle in the basenji-greyhound dog model of airway hyperresponsiveness.
Topics: Adenylyl Cyclases; Analysis of Variance; Animals; Bronchial Hyperreactivity; Bucladesine; Cholera Toxin; Colforsin; Dinoprostone; Disease Models, Animal; Dogs; Enzyme Activation; Immunoblotting; Isoproterenol; Lung; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Radioimmunoassay; Receptors, Adrenergic, beta; Trachea | 1993 |
Inhibitory effect of forskolin on myosin phosphorylation-dependent and independent contractions in bovine tracheal smooth muscle.
Topics: Animals; Calcium; Cattle; Colforsin; Cyclic AMP; Depression, Chemical; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Myosin Light Chains; Phosphorylation; Trachea | 1995 |
Endothelin receptors in the cornea, iris and ciliary processes. Evidence from binding, secondary messenger and PCR studies.
Topics: Animals; Autoradiography; Base Sequence; Binding Sites; Ciliary Body; Colforsin; Cornea; Cyclic AMP; DNA Primers; Endothelins; Inositol Phosphates; Iris; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Polymerase Chain Reaction; Rabbits; Receptors, Endothelin; Second Messenger Systems | 1993 |
Involvement of the M2 muscarinic receptor in contractions of the guinea pig trachea, guinea pig esophagus, and rat fundus.
Topics: Adrenergic beta-Agonists; Animals; Colforsin; Cyclic AMP; Esophagus; Gastric Fundus; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Pertussis Toxin; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Serotonin; Trachea; Virulence Factors, Bordetella | 1996 |
beta-Adrenergic relaxation in mesenteric resistance arteries of spontaneously hypertensive and Wistar-Kyoto rats: the role of precontraction and intracellular Ca2+.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Calcium; Colforsin; Isoproterenol; Male; Mesenteric Arteries; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phenylephrine; Potassium; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Vascular Resistance | 1996 |
Effects of various phosphodiesterase-inhibitors, forskolin, and sodium nitroprusside on porcine detrusor smooth muscle tonic responses to muscarinergic stimulation and cyclic nucleotide levels in vitro.
Topics: Adenylyl Cyclases; Animals; Colforsin; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Guanylate Cyclase; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nitroprusside; Nucleotides, Cyclic; Phosphodiesterase Inhibitors; Receptors, Muscarinic; Signal Transduction; Swine; Urinary Bladder; Vasodilator Agents | 1996 |
Modulation of agonist-induced phosphoinositide metabolism, Ca2+ signalling and contraction of airway smooth muscle by cyclic AMP-dependent mechanisms.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic beta-Agonists; Animals; Calcium; Cattle; Cells, Cultured; Cholinergic Agents; Colforsin; Cyclic AMP; Histamine; Isoproterenol; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Phosphatidylinositols; Signal Transduction; Trachea | 1996 |
Cardiovascular effects of a novel, potent and selective phosphodiesterase 5 inhibitor, DMPPO: in vitro and in vivo characterization.
Topics: 3',5'-Cyclic-GMP Phosphodiesterases; Adrenergic alpha-Agonists; Allopurinol; Animals; Aorta, Thoracic; Atrial Natriuretic Factor; Blood Pressure; Colforsin; Cyclic AMP; Cyclic GMP; Cyclic Nucleotide Phosphodiesterases, Type 5; Hemodynamics; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nitroprusside; Phenylephrine; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Rats; Rats, Inbred SHR; Rats, Sprague-Dawley; Vasodilator Agents | 1996 |
The effect of prostaglandin E2 and prostaglandin F2 alpha on ovarian tissue in the Florida crayfish Procambarus paeninsulanus.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Arachidonic Acid; Astacoidea; Colforsin; Cyclic AMP; Dinoprost; Dinoprostone; Female; Muscle Contraction; Ovary; Phosphorylation | 1995 |
Effects of cyclic GMP elevation on isoprenaline-induced increase in cyclic AMP and relaxation in rat aortic smooth muscle: role of phosphodiesterase 3.
Topics: Adrenergic beta-Agonists; Allopurinol; Animals; Aorta, Thoracic; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Drug Synergism; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitroprusside; Phosphodiesterase Inhibitors; Rats; Vasodilator Agents | 1996 |
The influence of hyperthyroidism on beta-adrenoceptor-mediated relaxation of isolated small mesenteric arteries.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Colforsin; Dose-Response Relationship, Drug; Hyperthyroidism; Imidazoles; Isoproterenol; Male; Mesenteric Arteries; Methoxamine; Muscle Contraction; Muscle Relaxation; Propanolamines; Prostaglandin Endoperoxides, Synthetic; Rats; Rats, Wistar; Thromboxane A2; Thyroxine; Vascular Resistance; Vasoconstrictor Agents | 1996 |
Pharmacological activation changes stiffness of cultured human airway smooth muscle cells.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Actins; Bradykinin; Bronchodilator Agents; Bucladesine; Carbachol; Cells, Cultured; Colforsin; Collagen; Cytoskeleton; Dinoprostone; Histamine; Humans; Isoproterenol; Kinetics; Magnetics; Muscarinic Agonists; Muscle Contraction; Muscle, Smooth; Myosins; Potassium Chloride; Substance P; Time Factors; Trachea | 1996 |
Pharmacological nature of TP receptor mediated contraction in human intrapulmonary artery.
Topics: Adult; Aged; Calcium; Colforsin; Female; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Nifedipine; Nitroglycerin; Pulmonary Artery; Receptors, Prostaglandin; Receptors, Thromboxane A2, Prostaglandin H2; Thromboxane A2; Type C Phospholipases | 1996 |
Effects of putative K+ channel blockers on beta-adrenoceptor-mediated vasorelaxation of rat mesenteric artery.
Topics: Adenosine Triphosphate; Adrenergic beta-Agonists; Animals; Barium; Benzopyrans; Calcium; Charybdotoxin; Colforsin; Cromakalim; Cyclic AMP; Dose-Response Relationship, Drug; Fenoterol; Glyburide; Isoproterenol; Male; Mesenteric Arteries; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phenylephrine; Potassium Channel Blockers; Pyrroles; Rats; Rats, Sprague-Dawley; Vasoconstrictor Agents; Vasodilator Agents | 1997 |
Potentiation of the relaxing action of isoproterenol by forskolin in rabbit aortic rings: the involvement of beta 2-adrenoceptors.
Topics: Adenylyl Cyclases; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Animals; Aorta, Thoracic; Bucladesine; Colforsin; Dobutamine; Drug Synergism; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Rabbits; Terbutaline | 1997 |
Discrepancy between inotropic response and cyclic AMP production induced by isoprenaline and forskolin in rat ventricle strips.
Topics: Adrenergic beta-Agonists; Animals; Colforsin; Cyclic AMP; Female; Isoproterenol; Male; Muscle Contraction; Myocardium; Rats; Rats, Sprague-Dawley; Ventricular Function, Right | 1997 |
Effect of contrast medium on corpus cavernosum smooth muscle.
Topics: Animals; Colforsin; Contrast Media; Cyclic AMP; Cyclic GMP; Diatrizoate; Dose-Response Relationship, Drug; In Vitro Techniques; Iohexol; Male; Muscle Contraction; Muscle, Smooth; Penis; Phosphodiesterase Inhibitors; Rabbits; Triiodobenzoic Acids | 1997 |
Interactions between neuropeptide Y and the adenylate cyclase pathway in rat mesenteric small arteries: role of membrane potential.
Topics: 4-Aminopyridine; Acetylcholine; Adenylyl Cyclases; Animals; Charybdotoxin; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dichlororibofuranosylbenzimidazole; Gadolinium; Glyburide; In Vitro Techniques; Isoproterenol; Male; Membrane Potentials; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Neuropeptide Y; Nifedipine; Potassium Channels; Rats; Rats, Wistar; Thionucleotides | 1997 |
The role of cyclic nucleotides in guinea-pig bladder contractility.
Topics: Animals; Carbachol; Colforsin; Cyclic AMP; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Ovalbumin; Purinones; Pyrrolidinones; Rolipram; Urinary Bladder | 1997 |
Expression of functional alpha2-adrenergic receptor subtypes in human corpus cavernosum and in cultured trabecular smooth muscle cells.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Binding, Competitive; Brimonidine Tartrate; Cells, Cultured; Colforsin; Cyclic AMP; Humans; Idazoxan; Male; Muscle Contraction; Muscle, Smooth; Penis; Quinoxalines; Radioisotopes; Receptors, Adrenergic, alpha-2; Ribonucleases; RNA, Messenger; Yohimbine | 1997 |
Motor responses in rat ileum evoked by nitric oxide donors vs. field stimulation: modulation by pituitary adenylate cyclase-activating peptide, forskolin and guanylate cyclase inhibitors.
Topics: Animals; Colforsin; Electric Stimulation; Female; Guanylate Cyclase; Ileum; Muscle Contraction; Neuropeptides; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitroprusside; Pituitary Adenylate Cyclase-Activating Polypeptide; Rats; Rats, Sprague-Dawley | 1997 |
[The effect of RU486 on contractility of rabbit oviduct smooth muscle].
Topics: Abortifacient Agents, Steroidal; Adrenergic alpha-Agonists; Animals; Calcium Channel Blockers; Colforsin; Endoplasmic Reticulum; Fallopian Tubes; Female; Mifepristone; Muscle Contraction; Muscle, Smooth; Norepinephrine; Rabbits; Verapamil | 1996 |
Cyclic AMP modulates part of the relaxant action of calcitonin gene-related peptide in guinea pig gallbladder strips.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclase Inhibitors; Animals; Bucladesine; Calcitonin Gene-Related Peptide; Cholecystokinin; Cholera Toxin; Colforsin; Cyclic AMP; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Gallbladder; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Rats; Thionucleotides | 1997 |
Small heat shock proteins and vasospasm in human umbilical artery smooth muscle.
Topics: Colforsin; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Heat-Shock Proteins; HSP20 Heat-Shock Proteins; Humans; Muscle Contraction; Muscle, Smooth, Vascular; Phosphoproteins; Phosphorylation; Umbilical Arteries | 1997 |
Contractile roles of the M2 and M3 muscarinic receptors in the guinea pig colon.
Topics: Animals; Colforsin; Colon; Cyclic AMP; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Oxotremorine; Pertussis Toxin; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Virulence Factors, Bordetella | 1998 |
Thrombin-induced vasospasm: cellular signaling mechanisms.
Topics: Animals; Calcium-Calmodulin-Dependent Protein Kinases; Carotid Arteries; Cattle; Colforsin; Endothelin-1; Hemostasis; In Vitro Techniques; Ischemic Attack, Transient; Muscle Contraction; Muscle, Smooth, Vascular; Myosin Light Chains; Myosin-Light-Chain Kinase; Phosphotyrosine; Potassium; Signal Transduction; Thrombin | 1998 |
Relaxant effects of NKH477, a new water-soluble forskolin derivative, on guinea-pig tracheal smooth muscle: the role of Ca2+-activated K+ channels.
Topics: Animals; Bronchodilator Agents; Calcium; Colforsin; Cyclic AMP; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nifedipine; Peptides; Potassium; Potassium Channels; Solubility; Trachea; Water | 1998 |
cAMP protects endothelial barrier function independent of inhibiting MLC20-dependent tension development.
Topics: Cells, Cultured; Colforsin; Cyclic AMP; Electric Impedance; Endothelium, Vascular; Humans; Molecular Weight; Muscle Contraction; Myosin Light Chains; Phosphorylation; Signal Transduction; Theophylline; Thrombin; Umbilical Veins | 1998 |
Human 5-HT1B receptor stimulated inositol phospholipid hydrolysis in CHO cells: synergy with Gq-coupled receptors.
Topics: Animals; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; DNA, Complementary; Dose-Response Relationship, Drug; GTP-Binding Proteins; Humans; Hydrolysis; Inositol Phosphates; Muscle Contraction; Muscle, Smooth, Vascular; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Second Messenger Systems; Serotonin Receptor Agonists; Sumatriptan | 1998 |
The role of cAMP in the actions of the peptide AF3 in the parasitic nematodes Ascaris suum and Ascaridia galli.
Topics: 1-Methyl-3-isobutylxanthine; Acetylcholine; Animals; Ascaridia; Ascaris suum; Colforsin; Cyclic AMP; In Vitro Techniques; Muscle Contraction; Muscles; Oligopeptides; Second Messenger Systems | 1998 |
Effect of cAMP- and cGMP-related drugs on porcine cultured ciliary muscle.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Antihypertensive Agents; Bucladesine; Carbachol; Cells, Cultured; Ciliary Body; Colforsin; Cyclic AMP; Cyclic GMP; Immunoenzyme Techniques; Intraocular Pressure; Microscopy, Electron; Muscle Contraction; Muscle, Smooth; Nitroprusside; Phosphodiesterase Inhibitors; Swine | 1998 |
Evidence that cannabinoid-induced inhibition of electrically evoked contractions of the myenteric plexus--longitudinal muscle preparation of guinea-pig small intestine can be modulated by Ca2+ and cAMP.
Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Adenylate Cyclase Toxin; Animals; Benzoxazines; Calcium; Calcium Channel Blockers; Cannabinoids; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Intestine, Small; Male; Morphine Derivatives; Morpholines; Muscle Contraction; Myenteric Plexus; Naphthalenes; Phosphodiesterase Inhibitors; Receptors, Cannabinoid; Receptors, Drug; Receptors, Opioid, mu; Virulence Factors, Bordetella | 1998 |
Alpha2-adrenoceptor-mediated contractions of the porcine isolated ear artery: evidence for a cyclic AMP-dependent and a cyclic AMP-independent mechanism.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-Agonists; Angiotensin II; Animals; Arteries; Brimonidine Tartrate; Colforsin; Cyclic AMP; Ear; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Nitroprusside; Quinoxalines; Receptors, Adrenergic, alpha-2; Swine | 1998 |
Vasorelaxant effect of olprinone, an inhibitor of phosphodiesterase 3, on mesenteric small artery and vein of rabbits.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Caffeine; Calcium; Colforsin; Cyclic Nucleotide Phosphodiesterases, Type 3; Imidazoles; Male; Mesenteric Arteries; Mesenteric Veins; Muscle Contraction; Nitroglycerin; Phosphodiesterase Inhibitors; Pyridones; Rabbits; Vasodilator Agents | 1998 |
Mechanisms of cardiomyocyte dysfunction in heart failure following myocardial infarction in rats.
Topics: Actin Cytoskeleton; Animals; Calcium; Calcium Channels; Calcium-Transporting ATPases; Colforsin; Fura-2; Heart Failure; Heart Ventricles; Hemodynamics; Male; Muscle Contraction; Myocardial Infarction; Myocardium; Patch-Clamp Techniques; Rats; Rats, Wistar; Sarcoplasmic Reticulum; Sodium; Thapsigargin | 1998 |
Relationship between decreased function and O2 consumption caused by cyclic GMP in cardiac myocytes and L-type calcium channels.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Analysis of Variance; Animals; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Colforsin; Cyclic GMP; Heart; Muscle Contraction; Myocardium; Nifedipine; Nitroprusside; Oxygen Consumption; Rabbits; Radioimmunoassay | 1998 |
Effects of halothane and isoflurane on beta-adrenoceptor-mediated responses in the vascular smooth muscle of rat aorta.
Topics: Adrenergic beta-Agonists; Anesthetics, Inhalation; Animals; Aorta, Thoracic; Colforsin; Cyclic AMP; Halothane; In Vitro Techniques; Isoflurane; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth, Vascular; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta | 1998 |
Muscarinic M2 receptor-mediated contraction in the guinea pig Taenia caeci: possible involvement of protein kinase C.
Topics: Animals; Cecum; Colforsin; Diphenylacetic Acids; Female; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Kinetics; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Parasympathomimetics; Piperidines; Pirenzepine; Protein Kinase C; Receptor, Muscarinic M2; Receptors, Muscarinic; Second Messenger Systems | 1998 |
Role of vasoactive intestinal polypeptide in the adaptation of intestinal smooth muscle cells to mechanical distension.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adaptation, Physiological; Animals; Cell Separation; Colforsin; Guinea Pigs; Ileum; In Vitro Techniques; Intestinal Diseases; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Receptors, Vasoactive Intestinal Peptide; Sincalide; Stress, Mechanical; Vasoactive Intestinal Peptide | 1998 |
Force, membrane potential and cytoplasmic Ca2+ responses to cyclic nucleotides in rat anococcygeus muscle.
Topics: Animals; Calcium; Colforsin; Cytoplasm; Drug Interactions; Male; Membrane Potentials; Muscle Contraction; Muscle, Smooth; Nitroprusside; Nucleotides, Cyclic; Phenylephrine; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Vasoconstrictor Agents; Vasodilator Agents | 1998 |
The involvement of protein kinase C and tyrosine kinase in vanadate-induced contraction.
Topics: Animals; Calcium Channel Blockers; Cats; Colforsin; Enzyme Inhibitors; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurotransmitter Agents; Nitroprusside; Protein Kinase C; Protein-Tyrosine Kinases; Stomach; Vanadates; Vasodilator Agents | 1998 |
Glicentin and oxyntomodulin modulate both the phosphoinositide and cyclic adenosine monophosphate signaling pathways in gastric myocytes.
Topics: Animals; Calcium; Carbachol; Colforsin; Cyclic AMP; Glicentin; Glucagon; Glucagon-Like Peptides; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Muscle Contraction; Muscle, Smooth; Oxyntomodulin; Peptide Fragments; Pertussis Toxin; Phosphatidylinositols; Protein Precursors; Pyloric Antrum; Rabbits; Signal Transduction; Type C Phospholipases; Virulence Factors, Bordetella | 1999 |
Cyclosporine-induced renal artery smooth muscle contraction is associated with increases in the phosphorylation of specific contractile regulatory proteins.
Topics: Animals; Cattle; Colforsin; Contractile Proteins; Cyclosporine; Heat-Shock Proteins; HSP20 Heat-Shock Proteins; Immunosuppressive Agents; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Myosin Light Chains; Phosphoproteins; Phosphorylation; Renal Artery | 1999 |
Pertussis toxin increases isoproterenol induced relaxation in field-stimulated ileum.
Topics: Animals; Colforsin; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Histamine; Histamine Agonists; Ileum; In Vitro Techniques; Isoproterenol; Male; Muscarinic Agonists; Muscle Contraction; Muscle Relaxation; Oxotremorine; Pertussis Toxin; Sympathomimetics; Virulence Factors, Bordetella | 1999 |
Identification of the G protein-activating domain of the natriuretic peptide clearance receptor (NPR-C).
Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Enzyme Activation; Enzyme Inhibitors; GTP-Binding Proteins; Guanosine Triphosphate; Guanylate Cyclase; Guinea Pigs; Isoenzymes; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Peptide Fragments; Phospholipase C beta; Protein Binding; Receptors, Atrial Natriuretic Factor; Type C Phospholipases | 1999 |
A study of NPY-mediated contractions of the porcine isolated ear artery.
Topics: Adenylyl Cyclases; Adrenergic alpha-Agonists; Angiotensin II; Animals; Brimonidine Tartrate; Colforsin; Cyclic AMP; Ear, External; In Vitro Techniques; Isometric Contraction; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Neuropeptide Y; Nitroprusside; Quinoxalines; Receptors, Adrenergic, alpha-2; Receptors, Neuropeptide Y; Regional Blood Flow; Swine; Vasoconstrictor Agents; Vasodilator Agents | 1999 |
Structural determinants of the partial agonist-inverse agonist properties of 6'-azidohex-2'-yne-delta8-tetrahydrocannabinol at cannabinoid receptors.
Topics: Animals; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cyclohexanols; Dronabinol; Electric Stimulation; In Vitro Techniques; Male; Mice; Muscle Contraction; Receptors, Cannabinoid; Receptors, Drug; Structure-Activity Relationship; Vas Deferens | 1999 |
The mechanisms of alpha(2)-adrenoceptor agonist-induced contraction in longitudinal muscle of the porcine uterus.
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Calcium; Calcium Channel Blockers; Clonidine; Colforsin; Cyclic AMP; Female; Fluorescent Dyes; Fura-2; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Myometrium; Pertussis Toxin; Quinoxalines; Swine; Uterus; Verapamil; Virulence Factors, Bordetella | 2000 |
Role of cAMP in the short-term modulation of a neuromuscular system in aplysia.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclase Inhibitors; Animals; Aplysia; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electric Stimulation; Enzyme Inhibitors; Invertebrate Hormones; Motor Neurons; Muscle Contraction; Muscles; Neural Pathways; Neuromuscular Junction; Neuropeptides; Phorbol Esters; Serotonin | 2000 |
O-1057, a potent water-soluble cannabinoid receptor agonist with antinociceptive properties.
Topics: Analgesics; Analgesics, Non-Narcotic; Animals; Binding, Competitive; Cannabinoids; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cyclohexanols; Dronabinol; Drug Interactions; Guinea Pigs; Male; Mice; Mice, Inbred ICR; Muscle Contraction; Rats; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Solubility; Tritium; Vas Deferens; Water | 2000 |
Altered beta-adrenoceptor-mediated responses in the gastric smooth muscle of hypertensive rats.
Topics: Adrenergic beta-Agonists; Animals; Calcium; Calcium Channel Blockers; Colforsin; Electrophysiology; Gastric Emptying; Gastric Fundus; Gastric Mucosa; Hypertension; Isoproterenol; Male; Membrane Potentials; Microelectrodes; Muscle Contraction; Muscle, Smooth; Nicardipine; Nifedipine; Potassium; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta | 2000 |
K(ATP) channels mediate the beta(2)-adrenoceptor agonist-induced relaxation of rat detrusor muscle.
Topics: Adenosine Triphosphate; Adrenergic beta-Agonists; Animals; Clenbuterol; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Electric Stimulation; Female; Glyburide; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Pinacidil; Potassium Channels; Rats; Rats, Wistar; Urinary Bladder; Vasodilator Agents | 2000 |
Cyclic AMP regulates mRNA expression of alpha-1d and alpha-2a adrenergic receptors in cultured human corpus cavernosum smooth muscle cells.
Topics: Alprostadil; Cells, Cultured; Colforsin; Cyclic AMP; Gene Expression Regulation; Humans; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Penis; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Muscarinic; RNA, Messenger | 2000 |
Cyclic AMP-mediated inhibition of noradrenaline-induced contraction and Ca2+ influx in guinea-pig vas deferens.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Caffeine; Calcium; Calcium Channel Blockers; Colforsin; Cyclic AMP; Guinea Pigs; Intracellular Membranes; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Norepinephrine; Osmolar Concentration; Potassium; Vas Deferens | 2000 |
Regulation of coronary myoplasmic Ca(2+)-myosin light chain phosphorylation pathway and vasomotor tone: hyperpolarizing versus depolarizing cardioplegia.
Topics: Animals; Arterioles; Calcium; Cardioplegic Solutions; Colforsin; Coronary Vessels; Heart Arrest, Induced; Hypertonic Solutions; In Vitro Techniques; Isoproterenol; Magnesium; Male; Muscle Contraction; Muscle Tonus; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Phosphorylation; Pinacidil; Potassium; Rats; Rats, Sprague-Dawley | 2000 |
Functional characteristics of urinary tract smooth muscles in mice lacking cGMP protein kinase type I.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Carbachol; Cholinergic Agonists; Colforsin; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Electric Stimulation; Female; Gene Expression Regulation, Enzymologic; Immunohistochemistry; Male; Mice; Mice, Knockout; Muscle Contraction; Muscle, Smooth; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Urethra; Urinary Bladder | 2000 |
Sildenafil citrate on nitrergic transmission in anococcygeus muscles from the urogenital system of male and female mice.
Topics: Animals; Carbachol; Colforsin; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; Papaverine; Phosphodiesterase Inhibitors; Piperazines; Purines; Sex Factors; Sildenafil Citrate; Substrate Specificity; Sulfones; Synaptic Transmission; Urogenital System | 2000 |
Two independent pathways mediated by cAMP and protein kinase A enhance spontaneous transmitter release at Drosophila neuromuscular junctions.
Topics: Adenylyl Cyclases; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cobalt; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Drosophila; Drosophila Proteins; Electric Stimulation; Evoked Potentials; In Vitro Techniques; Insect Proteins; Muscle Contraction; Mutation; Myosin Heavy Chains; Neuromuscular Junction; Neuropeptides; Neurotransmitter Agents; Organ Specificity; Patch-Clamp Techniques; R-SNARE Proteins; Reaction Time; Signal Transduction; Synaptic Transmission; Tetrodotoxin; Vesicular Transport Proteins | 2000 |
Involvement of cyclic GMP in nitric-oxide-induced gastric relaxation Comparison of the actions of cyclic GMP and cyclic AMP.
Topics: Acetylcholine; Animals; Cats; Colforsin; Cyclic AMP; Cyclic GMP; Female; Inositol Phosphates; Isometric Contraction; Male; Muscle Contraction; Muscle, Smooth; Nitric Oxide; Nitroprusside; Stomach | 2001 |
Colforsin daropate improves contractility in fatigued canine diaphragm.
Topics: Animals; Cardiotonic Agents; Colforsin; Diaphragm; Dogs; Dose-Response Relationship, Drug; Hemodynamics; Muscle Contraction; Muscle Fatigue | 2001 |
HNS-32, a novel azulene-1-carboxamidine derivative, inhibits nifedipine-sensitive and -insensitive contraction of the isolated rabbit aorta.
Topics: Animals; Anti-Arrhythmia Agents; Aorta, Thoracic; Calcium Channel Blockers; Colforsin; Endothelium, Vascular; Enzyme Activation; In Vitro Techniques; Male; Membrane Potentials; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Nitroglycerin; Norepinephrine; Phorbol 12,13-Dibutyrate; Potassium Channel Blockers; Potassium Chloride; Protein Kinase C; Pyridines; Rabbits; Tetraethylammonium; Vasoconstrictor Agents; Vasodilator Agents | 2001 |
Loss of annexin A7 leads to alterations in frequency-induced shortening of isolated murine cardiomyocytes.
Topics: Animals; Annexin A7; Caffeine; Calcium; Cardiotonic Agents; Central Nervous System Stimulants; Colforsin; Embryo, Mammalian; Female; Gene Targeting; Glucose; Homeostasis; Hypoglycemic Agents; Immunoblotting; Insulin; Insulin Secretion; Islets of Langerhans; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Muscle Contraction; Myocardium; Patch-Clamp Techniques; Tolbutamide | 2001 |
Role of lysophosphatidylcholine in the desensitization of beta-adrenergic receptors by Ca(2+) sensitization in tracheal smooth muscle.
Topics: Adenylate Cyclase Toxin; Adrenergic beta-Agonists; Amides; Animals; Bucladesine; Calcium; Cholera Toxin; Colforsin; Dinoprostone; Dose-Response Relationship, Drug; Enzyme Inhibitors; Guinea Pigs; In Vitro Techniques; Indoles; Isoproterenol; Lysophosphatidylcholines; Male; Maleimides; Methacholine Chloride; Muscarinic Agonists; Muscle Contraction; Muscle, Smooth; Pyridines; Receptors, Adrenergic, beta; rho GTP-Binding Proteins; Spectrometry, Fluorescence; Theophylline; Trachea; Virulence Factors, Bordetella | 2001 |
Relaxation and modulation of cyclic AMP production in response to atrial natriuretic peptides in guinea pig tracheal smooth muscle.
Topics: Adenylyl Cyclases; Animals; Apamin; Atrial Natriuretic Factor; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Glyburide; Guanylate Cyclase; Guinea Pigs; Histamine; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Natriuretic Peptide, C-Type; Nitroprusside; Oxadiazoles; Peptide Fragments; Peptides; Phosphodiesterase Inhibitors; Potassium Channel Blockers; Quinoxalines; Rolipram; Trachea | 2001 |
Beta2-adrenoceptor-mediated inhibition of field stimulation induced contractile responses of the smooth muscle of the rat prostate gland.
Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Albuterol; Animals; Atenolol; Catechols; Colforsin; Electric Stimulation; Electrophysiology; Ethanolamines; Male; Muscle Contraction; Nitroprusside; Norepinephrine; Propanolamines; Propranolol; Prostate; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-2 | 2001 |
Identification and functional study of phosphodiesterases in rat urinary bladder.
Topics: Animals; Colforsin; Cyclic AMP; Cyclic GMP; Enzyme Activation; Female; Guanylate Cyclase; In Vitro Techniques; Isoenzymes; Male; Muscle Contraction; Nitric Oxide Donors; Nitroprusside; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Rats; Rats, Wistar; Urinary Bladder | 2001 |
Phosphorylation of kinase-related protein (telokin) in tonic and phasic smooth muscles.
Topics: Animals; Carotid Arteries; Chickens; Colforsin; Culture Techniques; Gizzard, Avian; Isometric Contraction; Muscle Contraction; Muscle Proteins; Muscle Relaxation; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Peptide Fragments; Peptide Mapping; Peptides; Phorbol 12,13-Dibutyrate; Phosphorylation; Potassium Chloride; Time Factors | 2001 |
Effects of various nitric oxide donating agents on the contractility and cyclic nucleotide turnover of human seminal vesicles in vitro.
Topics: Aged; Colforsin; Cyclic AMP; Cyclic GMP; Electric Stimulation; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Nitric Oxide Donors; Seminal Vesicles | 2002 |
Pharmacological profile of evodiamine in isolated rabbit corpus cavernosum.
Topics: Aging; Animals; Colforsin; Electric Stimulation; In Vitro Techniques; Isometric Contraction; Male; Muscle Contraction; Muscle Relaxation; Nitric Oxide Donors; Nitroprusside; Nucleotides, Cyclic; Penis; Plant Extracts; Potassium; Potassium Channel Blockers; Quinazolines; Rabbits | 2002 |
Different effects of beta-adrenoceptor desensitization on inhibitory actions in guinea-pig trachealis.
Topics: Adrenergic beta-Agonists; Animals; Colforsin; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neural Inhibition; Procaterol; Receptors, Adrenergic, beta; Theophylline; Trachea | 2002 |
Intracellular pathways triggered by galanin to induce contraction of pig ileum smooth muscle cells.
Topics: Acetylcholine; Animals; Cell Communication; Colforsin; Dose-Response Relationship, Drug; Galanin; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Neuropeptides; Nifedipine; Peptides; Pertussis Toxin; Sincalide; Swine; Vasoactive Intestinal Peptide; Virulence Factors, Bordetella | 1992 |
Calcium channel blocker-like action of 1,9-dideoxyforskolin in vascular smooth muscle.
Topics: Animals; Aorta, Thoracic; Calcium; Calcium Channel Blockers; Colforsin; Cytosol; Fura-2; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Potassium; Rats; Rats, Wistar | 1992 |
Action of alpha 2A-adrenergic receptors in circular smooth muscle of canine proximal colon.
Topics: Adenylate Cyclase Toxin; Animals; Binding, Competitive; Cell Membrane; Clonidine; Colforsin; Colon; Dogs; Epinephrine; Female; In Vitro Techniques; Isoproterenol; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Oxymetazoline; Pertussis Toxin; Prazosin; Receptors, Adrenergic, alpha; Tetrodotoxin; Virulence Factors, Bordetella; Yohimbine | 1992 |
Effects of isoproterenol and forskolin on carbachol- and fluoroaluminate-induced polyphosphoinositide hydrolysis, inositol trisphosphate production, and contraction in bovine iris sphincter smooth muscle: interaction between cAMP and IP3 second messenger
Topics: Aluminum; Animals; Carbachol; Cattle; Colforsin; Cyclic AMP; Deferoxamine; Fluorine; Hydrolysis; Inositol 1,4,5-Trisphosphate; Iris; Isoproterenol; Kinetics; Muscle Contraction; Muscle, Smooth; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositols; Phosphorylation; Second Messenger Systems; Sodium Fluoride | 1992 |
A novel cyclic analog of neuropeptide Y specific for the Y2 receptor.
Topics: Amino Acid Sequence; Animals; Blood Pressure; Cell Membrane; Colforsin; Cyclic AMP; Electric Stimulation; Humans; Kidney Cortex; Male; Molecular Sequence Data; Muscle Contraction; Neuropeptide Y; Peptide Fragments; Peptides, Cyclic; Rabbits; Rats; Receptors, Neuropeptide Y; Receptors, Neurotransmitter; Synapses; Tumor Cells, Cultured; Vas Deferens | 1992 |
Studies on the mechanism of 5-HT1 receptor-induced smooth muscle contraction in dog saphenous vein.
Topics: Adenylyl Cyclase Inhibitors; Animals; Brain Chemistry; Calcium; Colforsin; Cyclic AMP; Dinoprostone; Dogs; Female; In Vitro Techniques; Indoles; Isometric Contraction; Male; Muscle Contraction; Muscle, Smooth, Vascular; Receptors, Serotonin; Saphenous Vein; Serotonin; Serotonin Antagonists; Sulfonamides; Sumatriptan; Vasoconstrictor Agents | 1992 |
Direct inhibitory mechanisms of halothane on canine tracheal smooth muscle contraction.
Topics: Animals; Calcium; Colforsin; Cyclic AMP; Dogs; Halothane; Muscle Contraction; Muscle, Smooth; Protein Kinase C; Signal Transduction; Trachea | 1992 |
Dibutyryl cyclic AMP and forskolin inhibit phosphatidylinositol hydrolysis, Ca2+ influx and contraction in vascular smooth muscle.
Topics: Animals; Bucladesine; Calcium; Colforsin; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phosphatidylinositols; Potassium; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Signal Transduction | 1992 |
Possible mechanisms of action of the antispasmodic agent tiropramide in the isolated detrusor from rats.
Topics: Animals; Calcium; Carbachol; Colforsin; Cyclic AMP; Cytosol; Fura-2; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Papaverine; Parasympatholytics; Rats; Rats, Wistar; Tyrosine; Urinary Bladder | 1992 |
Pharmacological characterization of alpha 2-adrenoceptors in isolated jejunum of rabbits.
Topics: Animals; Clonidine; Colforsin; GTP-Binding Proteins; Guanabenz; In Vitro Techniques; Jejunum; Muscle Contraction; Norepinephrine; Rabbits; Receptors, Adrenergic, alpha | 1992 |
Relaxation of soman-induced contracture of airway smooth muscle in vitro.
Topics: Acetylcholine; Adrenergic beta-Agonists; Albuterol; Animals; Colforsin; Dogs; Dose-Response Relationship, Drug; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Soman; Theophylline; Trachea | 1992 |
The role of cyclic AMP in non-adrenergic non-cholinergic contraction in guinea-pig bronchi.
Topics: Animals; Autonomic Nervous System; Benzopyrans; Bronchi; Bronchodilator Agents; Bucladesine; Colforsin; Cromakalim; Cyclic AMP; Electric Stimulation; Ethanolamines; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurons, Afferent; Nitroprusside; Procaterol; Pyrroles; Substance P; Theophylline | 1992 |
On the pharmacological and physiological role of glibenclamide-sensitive potassium channels in colonic smooth muscle.
Topics: Animals; Benzopyrans; Carbachol; Colforsin; Colon; Cromakalim; Dogs; Drug Interactions; Electric Stimulation; Female; Gallopamil; Glyburide; Male; Muscle Contraction; Muscle, Smooth; Potassium Channels; Pyrroles; Stereoisomerism | 1992 |
Involvement of a pertussis toxin-sensitive G-protein in excitation-contraction coupling of intact and cut-end voltage-clamped skeletal muscle fibres.
Topics: Animals; Colforsin; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Membrane Potentials; Muscle Contraction; Muscles; Neurons; Pertussis Toxin; Rana ridibunda; Virulence Factors, Bordetella | 1992 |
Characteristics of the contractile response of rabbit aorta produced by cromakalim in calcium-free solution.
Topics: Animals; Aorta; Benzopyrans; Calcium; Colforsin; Cromakalim; Guanidines; Male; Microelectrodes; Minoxidil; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Nitroglycerin; Pinacidil; Potassium; Potassium Channels; Pyridines; Pyrroles; Rabbits; Vasoconstriction | 1992 |
Acute endothelial cell contraction in vitro: a comparison with vascular smooth muscle cells and fibroblasts.
Topics: Actin Cytoskeleton; Animals; Aorta; Bradykinin; Cattle; Colforsin; Culture Techniques; Cytochalasin B; Endothelium; Fibroblasts; Histamine; Muscle Contraction; Muscle, Smooth, Vascular; Rats; Serotonin; Thrombin; Vasoconstriction | 1992 |
Hydrogen peroxide reduces beta-adrenoceptor function in the rat small intestine.
Topics: Animals; Bucladesine; Colforsin; Duodenum; Hydrogen Peroxide; Ileum; Intestine, Small; Isoproterenol; Jejunum; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Oxidation-Reduction; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1991 |
Functional antagonism in rabbit pulmonary veins contracted by endothelin.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Colforsin; Cyclic AMP; Cyclic GMP; Endothelins; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle, Smooth, Vascular; Nitroprusside; Norepinephrine; Phenylephrine; Prostaglandin Endoperoxides, Synthetic; Pulmonary Artery; Pulmonary Veins; Rabbits; Receptors, Cell Surface | 1991 |
Inositol phosphates formed in rat aorta after alpha 1-adrenoceptor stimulation are inhibited by forskolin.
Topics: Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Colforsin; Cyclic AMP; In Vitro Techniques; Inositol Phosphates; Isometric Contraction; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Rats; Rats, Inbred Strains | 1991 |
Response of the rat tail artery to prolonged exposure to noradrenaline.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Arteries; Colforsin; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Rats; Regional Blood Flow; Tail; Temperature | 1990 |
Effects of pimobendan, a cardiotonic and vasodilating agent with phosphodiesterase inhibiting properties, on isolated arteries and veins of rats.
Topics: 1-Methyl-3-isobutylxanthine; Aminophylline; Animals; Arteries; Cardiotonic Agents; Colforsin; Drug Interactions; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phosphodiesterase Inhibitors; Pyridazines; Rats; Rats, Inbred Strains; Vasodilator Agents; Veins | 1990 |
Endothelium reduces DNA synthesis in isolated arteries.
Topics: Acetylcholine; Animals; Atrial Natriuretic Factor; Bromodeoxyuridine; Colforsin; Culture Techniques; Cyclic AMP; Cyclic GMP; Dinoprostone; DNA; Endothelium, Vascular; Iloprost; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nitroprusside; Potassium; Rats; Rats, Inbred WKY; Renal Artery; Sympathectomy | 1991 |
Effects of cyclic AMP-affecting agents on contractile reactivity of isolated mesenteric and renal resistance arteries of the rat.
Topics: 1-Methyl-3-isobutylxanthine; Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Arteries; Bucladesine; Colforsin; Cyclic AMP; Dinoprostone; Enzyme Activation; In Vitro Techniques; Isometric Contraction; Isoproterenol; Male; Mesenteric Arteries; Milrinone; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Pertussis Toxin; Pyridones; Rats; Rats, Inbred WKY; Receptors, Adrenergic, beta; Renal Circulation; Sodium Fluoride; Sympathectomy; Vascular Resistance; Vasodilator Agents; Virulence Factors, Bordetella | 1990 |
Relaxation response of isolated canine veins to agents that act on the adenylate cyclase-cyclic AMP system: further investigation.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Adrenergic alpha-Agonists; Animals; Colforsin; Cyclic AMP; Dogs; Female; In Vitro Techniques; Isoproterenol; Male; Methoxamine; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Papaverine; Veins | 1990 |
Prevention of cyclosporine A-induced vascular toxicity by pentoxifylline.
Topics: Acetylcholine; Animals; Arginine; Colforsin; Cyclosporine; Endothelium, Vascular; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Neuromuscular Depolarizing Agents; Nitric Oxide; Nitroprusside; omega-N-Methylarginine; Pentoxifylline; Phenylephrine; Rats; Rats, Inbred Strains; Vascular Diseases | 1991 |
Involvement of nitric oxide in nerve-mediated inhibition and action of vasoactive intestinal peptide in colonic smooth muscle.
Topics: Animals; Arginine; Colforsin; Colon; Dogs; Female; In Vitro Techniques; Male; Membrane Potentials; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nitric Oxide; Nitroarginine; Stereoisomerism; Vasoactive Intestinal Peptide | 1992 |
Aminoalkylindoles: actions on specific G-protein-linked receptors.
Topics: Adenylyl Cyclase Inhibitors; Analgesics; Animals; Brain; Colforsin; GTP-Binding Proteins; Guanosine Triphosphate; Hydrogen-Ion Concentration; In Vitro Techniques; Indoles; Male; Mice; Muscle Contraction; Receptors, Drug; Vas Deferens | 1991 |
Endothelium-dependent effects of pentoxifylline in rat aorta.
Topics: Acetylcholine; Animals; Aorta, Thoracic; Colforsin; Endothelium, Vascular; In Vitro Techniques; Indomethacin; Male; Methylene Blue; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Pentoxifylline; Rats; Rats, Inbred Strains; Serotonin | 1991 |
Peptidergic and serotonergic facilitation of a neuromuscular synapse in Aplysia.
Topics: Animals; Aplysia; Colforsin; Evoked Potentials; Membrane Potentials; Motor Neurons; Muscle Contraction; Neuromuscular Junction; Neuropeptides; Serotonin; Synapses | 1990 |
Identification of neurotransmitters by selective protection of postjunctional receptors.
Topics: Adenosine Triphosphate; Animals; Bucladesine; Colforsin; Electric Stimulation; Ethylmaleimide; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Myenteric Plexus; Receptors, Neurotransmitter; Stomach; Vasoactive Intestinal Peptide | 1990 |
Direct inhibition of chicken gizzard smooth muscle contractile apparatus by caffeine.
Topics: Actomyosin; Animals; Ca(2+) Mg(2+)-ATPase; Caffeine; Calcium-Transporting ATPases; Chickens; Colforsin; Cyclic AMP; Erythrocyte Membrane; Gizzard, Avian; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Myosin-Light-Chain Kinase; Phosphoric Monoester Hydrolases; Phosphorylation; Potassium Chloride | 1990 |
Neuropeptide Y stimulation of myosin light chain phosphorylation in cultured aortic smooth muscle cells.
Topics: Adenylate Cyclase Toxin; Animals; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic GMP; Enzyme Activation; In Vitro Techniques; Inositol Phosphates; Muscle Contraction; Muscle, Smooth, Vascular; Myosins; Neuropeptide Y; Pertussis Toxin; Phosphorylation; Protein Kinase C; Signal Transduction; Swine; Virulence Factors, Bordetella | 1990 |
Endothelin modulation of neuroeffector transmission in rat and guinea pig vas deferens.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Adenosine Triphosphate; Animals; Autonomic Nervous System; Colforsin; Electric Stimulation; Endothelins; Felodipine; Guinea Pigs; In Vitro Techniques; Indomethacin; Male; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Neuroeffector Junction; Norepinephrine; Rats; Sympathetic Nervous System; Synaptic Transmission; Vas Deferens | 1990 |
Epithelium, contractile tone, and responses to relaxing agonists in canine bronchi.
Topics: Acetylcholine; Animals; Bronchi; Colforsin; Cyclic AMP; Cyclic GMP; Dogs; Epithelium; Female; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Nitric Oxide; Nitroprusside; Serotonin | 1990 |
Characterization of the adenosine receptor in porcine coronary arteries.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Colforsin; Coronary Vessels; Dinoprost; In Vitro Techniques; Kinetics; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Receptors, Purinergic; Swine | 1990 |
Changes in cytosolic CA2+ and contraction induced by various stimulants and relaxants in canine tracheal smooth muscle.
Topics: Animals; Benzofurans; Calcium; Carbachol; Colforsin; Cytosol; Dogs; Fura-2; Isoproterenol; Muscle Contraction; Muscle, Smooth; Phorbol Esters; Potassium; Trachea; Verapamil | 1990 |
Bronchodilator and antiallergy activity of forskolin.
Topics: Animals; Bronchial Spasm; Bronchodilator Agents; Colforsin; Cyclic AMP; Diterpenes; Guinea Pigs; Histamine Release; Hypersensitivity; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Secretory Rate; SRS-A | 1985 |
Plasma membrane calcium flux, protein kinase C activation and smooth muscle contraction.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Cell Membrane; Colforsin; Drug Synergism; Enzyme Activation; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Nitrendipine; Ouabain; Perfusion; Phospholipids; Potassium; Protein Kinase C; Rabbits; Tetradecanoylphorbol Acetate; Vasoconstriction | 1985 |
Activation of tracheal smooth muscle contraction: synergism between Ca2+ and activators of protein kinase C.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcimycin; Calcium; Cattle; Colforsin; Diterpenes; Drug Synergism; Enzyme Activation; Ethers; In Vitro Techniques; Ionomycin; Muscle Contraction; Muscle, Smooth; Nifedipine; Protein Kinase C; Terpenes; Tetradecanoylphorbol Acetate; Trachea | 1985 |
Identified octopaminergic neurons modulate contractions of locust visceral muscle via adenosine 3',5'-monophosphate (cyclic AMP).
Topics: 1-Methyl-3-isobutylxanthine; Animals; Biogenic Amines; Colforsin; Cyclic AMP; Female; Grasshoppers; In Vitro Techniques; Muscle Contraction; Muscles; Octopamine; Oviducts; Synaptic Transmission | 1986 |
Effects of forskolin on contractility and cyclic AMP levels in rabbit detrusor muscle.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Colforsin; Cyclic AMP; In Vitro Techniques; Muscle Contraction; Muscles; Propranolol; Rabbits | 1986 |
Age-related decrease in beta adrenergic receptor-mediated vascular smooth muscle relaxation.
Topics: 1-Methyl-3-isobutylxanthine; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Acetylcholine; Aging; Bucladesine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Iodocyanopindolol; Isoproterenol; Mesenteric Arteries; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroglycerin; Pindolol; Receptors, Adrenergic, beta; Serotonin | 1986 |
Parathyroid hormone-induced changes in cyclic nucleotide levels during relaxation of the rabbit [correction of rat] aorta.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Aorta, Thoracic; Colforsin; Cyclic AMP; Cyclic GMP; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroprusside; Parathyroid Hormone; Rabbits | 1987 |
Recovery of free muscle grafts in rat: improvement is associated with an increase in cyclic adenosine monophosphate concentration or use of the condition/test paradigm.
Topics: Animals; Colforsin; Cyclic AMP; Female; Muscle Contraction; Muscles; Neovascularization, Pathologic; Rats; Rats, Inbred Strains | 1987 |
Stimulation of acetylcholine release from myenteric neurons of guinea pig small intestine by forskolin and cyclic AMP.
Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Animals; Bucladesine; Colforsin; Cyclic AMP; Guinea Pigs; In Vitro Techniques; Intestine, Small; Muscle Contraction; Myenteric Plexus; Theophylline | 1987 |
Inhibitory effects of caffeine on contractions and calcium movement in vascular and intestinal smooth muscle.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Caffeine; Calcium; Calcium Radioisotopes; Colforsin; Cyclic AMP; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Norepinephrine; Rabbits | 1988 |
Inhibition of atrial natriuretic peptide secretion by forskolin in noncontracting cultured atrial myocytes.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Atrial Natriuretic Factor; Bucladesine; Calcium; Cells, Cultured; Colforsin; Cyclic GMP; Egtazic Acid; Muscle Contraction; Muscle, Smooth, Vascular; Protein Kinase C; Ryanodine; Sarcoplasmic Reticulum; Secretory Rate; Tetradecanoylphorbol Acetate | 1988 |
Cyclic AMP only partially mediates the actions of serotonin at lobster neuromuscular junctions.
Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Colforsin; Cyclic AMP; Electrophysiology; Muscle Contraction; Nephropidae; Neuromuscular Junction; Serotonin; Time Factors | 1989 |
Role of stimulatory GTP-binding protein (Gs) in reduced beta-adrenoceptor coupling in the femoral artery of spontaneously hypertensive rats.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic alpha-Antagonists; Animals; Bucladesine; Cholera Toxin; Colforsin; Femoral Artery; GTP-Binding Proteins; Guanosine Triphosphate; Hypertension; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Timolol | 1988 |
Effects of atrial natriuretic factor (ANF) on phenylephrine-triggered intra- and extracellular calcium dependent contraction in rat aorta.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Atrial Natriuretic Factor; Calcium; Colforsin; Cyclic AMP; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Phenylephrine; Rats; Rats, Inbred Strains | 1989 |
Beta-adrenergic relaxation of dog trachealis: contractile agonist-specific interaction.
Topics: 1-Methyl-3-isobutylxanthine; Acetylcholine; Adrenergic beta-Agonists; Animals; Bucladesine; Colforsin; Dogs; Histamine; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle, Smooth; Potassium Chloride; Serotonin; Trachea | 1989 |
Neuropeptide Y-induced intracellular Ca2+ increases in vascular smooth muscle cells.
Topics: 1-Methyl-3-isobutylxanthine; Angiotensin II; Animals; Bradykinin; Calcium; Cells, Cultured; Colforsin; Cytoplasm; GTP-Binding Proteins; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Muscle Contraction; Muscle, Smooth, Vascular; Neuropeptide Y; Pertussis Toxin; Receptors, Neuropeptide Y; Receptors, Neurotransmitter; Swine; Virulence Factors, Bordetella | 1989 |
Effects of intracellular alkalinization on resting and agonist-induced vascular tone.
Topics: Acetates; Ammonium Chloride; Angiotensin II; Animals; Aorta; Calcimycin; Calcium; Choline; Colforsin; Egtazic Acid; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Models, Cardiovascular; Muscle Contraction; Muscle Tonus; Muscle, Smooth, Vascular; Rats; Reference Values | 1989 |
Influence of stimulators and inhibitors of cyclic nucleotides on lower esophageal sphincter.
Topics: Animals; Colforsin; Cyclic AMP; Cyclic GMP; Electric Stimulation; Esophagogastric Junction; Ethylmaleimide; Female; In Vitro Techniques; Male; Methylene Blue; Muscle Contraction; Nitroprusside; Opossums; Phosphodiesterase Inhibitors; Vasoactive Intestinal Peptide | 1989 |
A comparison of vasodilator activity of agents activating cyclic nucleotides with those inhibiting their metabolism in rabbit isolated ear artery.
Topics: Animals; Colforsin; Cyclic AMP; Cyclic GMP; Ear, External; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nitroprusside; Phosphodiesterase Inhibitors; Regional Blood Flow; Sympathetic Nervous System; Vasodilation | 1989 |
Involvement of endothelial cells in relaxation and contraction responses of the aorta to isoproterenol in naive and streptozotocin-induced diabetic rats.
Topics: Animals; Aorta; Colforsin; Diabetes Mellitus, Experimental; Drug Interactions; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroprusside; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1989 |
Contractile force and intracellular Ca2+ during relaxation of canine tracheal smooth muscle.
Topics: Acetylcholine; Aequorin; Animals; Calcium; Carbachol; Colforsin; Dogs; In Vitro Techniques; Indicators and Reagents; Isometric Contraction; Isoproterenol; Kinetics; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Ouabain; Potassium; Serotonin; Sodium-Potassium-Exchanging ATPase; Trachea | 1989 |
Direct regulation of smooth muscle contractile elements by second messengers.
Topics: Animals; Calcium; Colforsin; Cyclic AMP; Cyclic GMP; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Phorbol 12,13-Dibutyrate; Rats; Rats, Inbred WKY; Second Messenger Systems | 1989 |
Calcium-force coupling mechanisms during vasodilator-induced relaxation of ferret aorta.
Topics: Animals; Aorta, Thoracic; Calcium; Carnivora; Colforsin; Ferrets; Hydralazine; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Nifedipine | 1989 |
Effect of forskolin on cytosolic Ca++ level and contraction in vascular smooth muscle.
Topics: Animals; Calcium; Colforsin; Cytosol; Drug Interactions; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Potassium Chloride; Rats; Rats, Inbred Strains | 1989 |
The effect of relaxants working through different transduction mechanisms on the tonic contraction produced in rat aorta by 4 beta-phorbol dibutyrate.
Topics: Animals; Aorta, Thoracic; Benzopyrans; Colforsin; Cromakalim; In Vitro Techniques; Isoproterenol; Male; Methoxamine; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroprusside; Parasympatholytics; Phorbol 12,13-Dibutyrate; Pyrroles; Rats; Rats, Inbred Strains; Xanthines | 1989 |
Synthetic tumor-derived human hypercalcemic factor exhibits parathyroid hormone-like vasorelaxation in renal arteries.
Topics: Animals; Colforsin; Cyclic AMP; Humans; Male; Methoxamine; Muscle Contraction; Muscle Relaxation; Neoplasm Proteins; Parathyroid Hormone; Parathyroid Hormone-Related Protein; Peptide Fragments; Proteins; Rabbits; Renal Artery | 1987 |
Co-regulation of tracheal tone by cyclic AMP- and cyclic GMP-dependent mechanisms.
Topics: Animals; Bucladesine; Carbachol; Colforsin; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Guinea Pigs; Male; Muscle Contraction; Nitroprusside; Trachea | 1987 |
Effects of several in vitro systems on the potencies of putative adrenocorticotropin secretagogues on rat anterior pituitary cells.
Topics: Acetylcholine; Adrenocorticotropic Hormone; Angiotensin II; Animals; Arginine Vasopressin; Cells, Cultured; Colforsin; Corticotropin-Releasing Hormone; Diglycerides; Epinephrine; Kinetics; Male; Muscle Contraction; Oxytocin; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains | 1988 |
Effects of colforsin, trequinsin and isoprenaline on norepinephrine-induced contractions and cyclic nucleotide levels of isolated vascular tissue.
Topics: Acetylcholine; Animals; Aorta, Thoracic; Colforsin; Cyclic AMP; Cyclic GMP; Female; In Vitro Techniques; Isoproterenol; Isoquinolines; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Platelet Aggregation Inhibitors; Rabbits; Tetrahydroisoquinolines | 1988 |
Effect of Na-K adenosinetriphosphatase activity on relaxation of canine tracheal smooth muscle.
Topics: Animals; Calcium Channel Blockers; Colforsin; Dinoprostone; Dogs; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nitroprusside; Potassium; Prostaglandins E; Sodium-Potassium-Exchanging ATPase; Trachea | 1988 |
Does the hydrolysis of inositol phospholipids lead to the opening of voltage operated Ca2+ channels in guinea-pig ileum? Studies with fluoride ions and caffeine.
Topics: Animals; Caffeine; Calcium; Carbachol; Colforsin; Cyclic AMP; Fluorides; Guinea Pigs; Ileum; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Phosphatidylinositols | 1988 |
Inhibitory effects of forskolin on vascular smooth muscle of rabbit aorta.
Topics: Animals; Aorta, Thoracic; Caffeine; Calcium; Calcium Radioisotopes; Colforsin; Cyclic AMP; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Rabbits | 1988 |
Effects of cilostazol, a selective cAMP phosphodiesterase inhibitor on the contraction of vascular smooth muscle.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Aorta, Thoracic; Azoles; Bucladesine; Calcium; Cilostazol; Colforsin; Cyclic AMP; Cyclic GMP; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Rabbits; Tetrazoles; Vasodilator Agents | 1988 |
Differential inhibitory effects of forskolin, isoproterenol, and dibutyryl cyclic adenosine monophosphate on phosphoinositide hydrolysis in canine tracheal smooth muscle.
Topics: Animals; Bucladesine; Colforsin; Dogs; Histamine; Hydrolysis; Isoproterenol; Methacholine Chloride; Methacholine Compounds; Muscle Contraction; Muscle, Smooth; Phosphatidylinositols; Trachea | 1988 |
Pharmacologic enhancement of functional recovery in free muscle transfers.
Topics: Animals; Colforsin; Cyclic AMP; Electromyography; Muscle Contraction; Muscles; Nerve Regeneration; Rabbits; Stimulation, Chemical | 1988 |
[Effect of beta-agonists on membrane potentials of isolated smooth muscle of the guinea pig trachea].
Topics: Adrenergic beta-Agonists; Animals; Bucladesine; Catecholamines; Colforsin; Guinea Pigs; In Vitro Techniques; Membrane Potentials; Muscle Contraction; Muscle, Smooth; Theophylline; Trachea | 1985 |
Beta agonist-induced desensitization in pig bronchus.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Airway Resistance; Animals; Bronchi; Colforsin; Fenoterol; Hydrocortisone; In Vitro Techniques; Indomethacin; Isoproterenol; Muscle Contraction; Muscle Relaxation; Norepinephrine; Phenylephrine; Quinacrine; Receptors, Adrenergic, beta; Stereoisomerism; Swine; Theophylline | 1986 |
Beta-adrenergic agonists and cyclic AMP decrease intracellular resting free-calcium concentration in ileum smooth muscle.
Topics: Animals; Bucladesine; Calcium; Colforsin; Cyclic AMP; Guinea Pigs; Ileum; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle, Smooth | 1987 |
Effect of methylene blue and N-ethylmaleimide on internal anal sphincter relaxation.
Topics: Adenylyl Cyclase Inhibitors; Anal Canal; Animals; Colforsin; Electric Stimulation; Female; Guanylate Cyclase; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nitroprusside | 1988 |
Effects of BN 52063 and other agents inhibiting platelet-activating factor-induced contractile responses in rat portal vein.
Topics: Albuterol; Animals; Colforsin; In Vitro Techniques; Lactones; Male; Muscle Contraction; Muscle, Smooth, Vascular; Plant Extracts; Platelet Activating Factor; Portal Vein; Rats; Rats, Inbred Strains; Theophylline | 1988 |
Cyclic nucleotides and contractility of isolated soleus muscle.
Topics: Animals; Colforsin; Cyclic AMP; Cyclic GMP; Diterpenes; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscles; Terbutaline | 1985 |
Characterization of pre- and post-junctional adenosine receptors in guinea-pig ileum.
Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cholinergic Fibers; Colforsin; Cyclic AMP; Diterpenes; Electric Stimulation; Gastrointestinal Motility; Guinea Pigs; Ileum; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Phenylisopropyladenosine; Pyrrolidinones; Receptors, Cell Surface; Receptors, Neurotransmitter; Receptors, Purinergic; Rolipram; Synaptic Transmission | 1985 |
Increases in muscle Ca2+ mediate changes in acetylcholinesterase and acetylcholine receptors caused by muscle contraction.
Topics: Acetylcholinesterase; Animals; Bucladesine; Calcium; Cells, Cultured; Colforsin; Muscle Contraction; Muscles; Nitroprusside; Rats; Receptors, Cholinergic; Tetrodotoxin; Veratridine | 1985 |
Neuropeptide Y is a potent inhibitor of cyclic AMP accumulation in feline cerebral blood vessels.
Topics: Animals; Cats; Cerebral Arteries; Clonidine; Colforsin; Cyclic AMP; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Nerve Tissue Proteins; Neuropeptide Y; Vascular Resistance | 1985 |
A role for adenylate cyclase in the subsensitivity to isoproterenol during ontogenesis of the embryonic chick ventricle.
Topics: Adenylyl Cyclases; Animals; Chick Embryo; Chickens; Chlorides; Colforsin; Cyclic AMP; Dihydroalprenolol; Dose-Response Relationship, Drug; Drug Interactions; Guanylyl Imidodiphosphate; Heart; Isoproterenol; Kinetics; Magnesium; Manganese; Manganese Compounds; Muscle Contraction; Myocardium; Receptors, Adrenergic, beta; Sodium Fluoride | 1985 |
[Effect of isoprenaline and the barium ion on the relaxation of the smooth muscle of the guinea pig trachea].
Topics: Animals; Barium; Colforsin; Cyclic AMP; Guinea Pigs; In Vitro Techniques; Ions; Isoproterenol; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Trachea | 1985 |
Effects of forskolin and cyclic nucleotides on isometric force in rat aorta.
Topics: Animals; Aorta, Thoracic; Bucladesine; Colforsin; Cyclic GMP; Isometric Contraction; Male; Muscle Contraction; Muscle, Smooth, Vascular; Rats; Rats, Inbred Strains; Vasomotor System | 1986 |
Influence of the epithelium on responsiveness of guinea-pig isolated trachea to contractile and relaxant agonists.
Topics: Acetylcholine; Animals; Asthma; Autoradiography; Carbachol; Cimetidine; Colforsin; Dose-Response Relationship, Drug; Epithelium; Female; Guinea Pigs; Histamine; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Kinetics; Male; Muscle Contraction; Nitroglycerin; Pindolol; Potassium; Receptors, Adrenergic, beta; Theophylline; Trachea | 1986 |
[Cyclic nucleotides].
Topics: Animals; Bronchi; Colforsin; Cyclic AMP; Cyclic GMP; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Nitro Compounds | 1985 |
Effects of relaxants on electrical and mechanical activities in the guinea-pig tracheal muscle.
Topics: Animals; Bucladesine; Colforsin; Epinephrine; Female; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Membrane Potentials; Muscle Contraction; Muscle Relaxants, Central; Muscle, Smooth; Norepinephrine; Terbutaline; Theophylline; Trachea | 1986 |
Relaxant effect of forskolin in rabbit detrusor smooth muscle: role of cyclic AMP.
Topics: Adenine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Colforsin; Cyclic AMP; Drug Synergism; Enzyme Activation; Imidazoles; Male; Muscle Contraction; Muscle, Smooth; Propranolol; Rabbits; Urinary Bladder | 1986 |
Further evidence for the involvement of cyclic AMP in Ca2+-dependent, but not Ca2+-independent, noradrenaline release in the rabbit pulmonary artery.
Topics: Acetylcholine; Animals; Calcium; Colforsin; Cyclic AMP; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Naphthyridines; Norepinephrine; Perfusion; Phosphodiesterase Inhibitors; Pulmonary Artery; Rabbits; Veratridine | 1986 |
Effect of dB-c-AMP and forskolin on the 45Ca influx, net Ca uptake and tension in rabbit aortic smooth muscle.
Topics: Animals; Aorta, Thoracic; Bucladesine; Calcium; Calcium Radioisotopes; Colforsin; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Phentolamine; Propranolol; Rats | 1987 |
The time course of changes in force and cyclic AMP levels produced by isoproterenol and forskolin in isolated rabbit detrusor muscle.
Topics: Animals; Colforsin; Cyclic AMP; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Rabbits; Time Factors; Urinary Bladder | 1987 |
Relationship of urotensin I induced vasodilatory action in rat thoracic aorta to Ca2+ regulation.
Topics: Animals; Aorta, Thoracic; Binding, Competitive; Bucladesine; Calcimycin; Calcium; Colforsin; Endothelium; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Papaverine; Peptides; Rats; Rats, Inbred Strains; Urotensins; Vasodilation; Verapamil | 1987 |
Relaxant effects of forskolin on guinea pig tracheal smooth muscle.
Topics: Animals; Colforsin; Cyclic AMP; Differential Threshold; Ethanol; Guinea Pigs; Histamine; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Respiration; Trachea | 1987 |
The relaxant and spasmogenic effects of some xanthine derivatives acting on guinea-pig isolated trachealis muscle.
Topics: Acetylcholine; Animals; Caffeine; Calcium; Colforsin; Egtazic Acid; Female; Guinea Pigs; In Vitro Techniques; Indomethacin; Male; Muscle Contraction; Muscle Relaxation; Muscle Tonus; Muscle, Smooth; Potassium Chloride; Temperature; Xanthines | 1988 |
The intracellular calcium stores in the rabbit trachealis.
Topics: Animals; Caffeine; Calcium; Carbachol; Colforsin; Egtazic Acid; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Rabbits; Trachea | 1988 |
Protein phosphorylation changes in bovine carotid artery smooth muscle during contraction and relaxation.
Topics: Angiotensin II; Animals; Calcium; Carotid Arteries; Cattle; Colforsin; Cytoplasm; Diglycerides; Histamine; Muscle Contraction; Muscle Proteins; Muscle Relaxation; Muscle, Smooth, Vascular; Phorbol Esters; Phosphoproteins; Phosphorylation; Potassium; Trachea | 1988 |
The role of adenylate cyclase in relaxation of brain arteries: studies with forskolin.
Topics: Adenylyl Cyclases; Animals; Basilar Artery; Brain Chemistry; Cattle; Cerebral Arteries; Colforsin; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Swine | 1988 |
The effects of isoproterenol on intracellular calcium concentration.
Topics: Animals; Atropine; Calcium; Carbachol; Cattle; Colforsin; Isoproterenol; Muscle Contraction; Muscle, Smooth; Phorbol Esters; Propranolol; Trachea; Vasoactive Intestinal Peptide | 1988 |
Effects of adenylate cyclase activators on porcine skeletal muscle in malignant hyperpyrexia.
Topics: Adenylyl Cyclases; Animals; Colforsin; Disease Susceptibility; In Vitro Techniques; Malignant Hyperthermia; Molybdenum; Muscle Contraction; Muscles; Norepinephrine; Sodium Fluoride; Swine | 1987 |
Forskolin counteracts the effects of the organophosphate soman at the neuromuscular junction.
Topics: Action Potentials; Animals; Colforsin; Diaphragm; Muscle Contraction; Neuromuscular Junction; Rats; Soman | 1987 |
Phorbol ester contracts rabbit thoracic aorta by increasing intracellular calcium and by activating calcium influx.
Topics: Animals; Biological Transport; Calcium; Colforsin; Cytoplasm; Extracellular Space; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Prazosin; Protein Kinase C; Rabbits; Time Factors | 1986 |
The effect of forskolin on the isometric contraction of the isolated hemidiaphragm of the rat.
Topics: Aminophylline; Animals; Calcium; Colforsin; Dose-Response Relationship, Drug; Drug Synergism; Electric Stimulation; Female; Isometric Contraction; Isoproterenol; Male; Muscle Contraction; Rats | 1986 |
Age dependence of adenylate cyclase in guinea pig ureter homogenate.
Topics: Adenylyl Cyclases; Aging; Alprostadil; Animals; Colforsin; Enzyme Activation; Ethanol; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Guinea Pigs; Isoproterenol; Male; Muscle Contraction; Propranolol; Sodium Fluoride; Ureter | 1986 |
Activation of cyclic AMP dependent protein kinase in rabbit aortic rings by prostaglandin E1 and forskolin is accompanied by contraction and relaxation, respectively.
Topics: Alprostadil; Animals; Aorta; Colforsin; Enzyme Activation; In Vitro Techniques; Muscle Contraction; Protein Kinases; Rabbits | 1986 |
Carbachol-induced protein phosphorylation changes in bovine tracheal smooth muscle.
Topics: Animals; Calcium; Calmodulin-Binding Proteins; Carbachol; Cattle; Colforsin; Cytosol; Desmin; Intermediate Filament Proteins; Isoelectric Point; Kinetics; Muscle Contraction; Muscle Proteins; Muscle, Smooth; Myosins; Phorbol Esters; Phosphoproteins; Phosphorylation; Trachea | 1986 |
Airway reactivity in chronic obstructive pulmonary disease. Failure of in vivo methacholine responsiveness to correlate with cholinergic, adrenergic, or nonadrenergic responses in vitro.
Topics: Aged; Albuterol; Bronchi; Bronchial Provocation Tests; Colforsin; Diterpenes; Female; Forced Expiratory Volume; Humans; In Vitro Techniques; Lung Diseases, Obstructive; Male; Methacholine Chloride; Methacholine Compounds; Middle Aged; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Pneumonectomy | 1985 |
Forskolin suppresses sympathetic neuron function and causes ocular hypotension.
Topics: Administration, Topical; Animals; Blood Pressure; Cats; Colforsin; Diterpenes; Dose-Response Relationship, Drug; Electric Stimulation; Eye; Hypotension; Intraocular Pressure; Muscle Contraction; Neurons; Nictitating Membrane; Norepinephrine; Sympathectomy; Sympathetic Nervous System; Water | 1985 |
Comparison of the effects of forskolin and isoprenaline on tracheal, cardiac and skeletal muscles from guinea-pig.
Topics: Animals; Cardiotonic Agents; Colforsin; Diterpenes; Guinea Pigs; Heart; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Muscles; Myocardial Contraction; Papillary Muscles; Practolol; Prenalterol; Trachea | 1985 |
Ca2+-dependent inhibition of smooth muscle adenylate cyclase activity.
Topics: Adenylyl Cyclase Inhibitors; Animals; Calcium; Calmodulin; Cattle; Colforsin; Diterpenes; Enzyme Activation; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Magnesium; Muscle Contraction; Muscle, Smooth, Vascular; Troponin; Troponin C | 1985 |
Phorbol myristate acetate causes in guinea-pig lung parenchymal strip a maintained spasm which is relatively resistant to isoprenaline.
Topics: Aminophylline; Animals; Colforsin; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Lung; Male; Muscle Contraction; Muscle, Smooth; Nitroprusside; Phorbols; Tetradecanoylphorbol Acetate | 1985 |
The effects of small cardioactive peptide B on the isolated heart and gill of Aplysia californica.
Topics: Adenylyl Cyclases; Animals; Aplysia; Colforsin; FMRFamide; Gills; Heart; In Vitro Techniques; Kinetics; Muscle Contraction; Myocardial Contraction; Neuropeptides; Oligopeptides; Perfusion; Serotonin; Sincalide; Vasoactive Intestinal Peptide; Vasotocin | 1985 |