clobenpropit has been researched along with Active Hyperemia in 1 studies
clobenpropit: histamine H3 receptor antagonist
clobenpropit : An imidothiocarbamic ester that consists of isothiourea bearing S-3-(imidazol-4-yl)propyl and N-4-chlorobenzyl substituents. An extremely potent histamine H3 antagonist/inverse agonist (pA2 = 9.93). Also displays partial agonist activity at H4 receptors; induces eosinophil shape change with an EC50 of 3 nM.
| Excerpt | Relevance | Reference |
|---|---|---|
| "Pretreatment with clobenpropit was without any effect on control MBF and AP but significantly reduced most of RH responses." | 1.32 | Histamine H3 receptors modulate reactive hyperemia in rat gut. ( Biernat, J; Brzozowski, T; Konturek, SJ; Obuchowicz, R; Pawlik, MW; Pawlik, WW; Sendur, R, 2004) |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 1 (100.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Pawlik, WW | 1 |
| Obuchowicz, R | 1 |
| Pawlik, MW | 1 |
| Sendur, R | 1 |
| Biernat, J | 1 |
| Brzozowski, T | 1 |
| Konturek, SJ | 1 |
1 other study available for clobenpropit and Active Hyperemia
| Article | Year |
|---|---|
Histamine H3 receptors modulate reactive hyperemia in rat gut.
Topics: Animals; Blood Pressure; Female; Histamine Agonists; Histamine Antagonists; Hyperemia; Imidazoles; I | 2004 |