Page last updated: 2024-09-02

cl 218872 and Absence Seizure

cl 218872 has been researched along with Absence Seizure in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19905 (71.43)18.7374
1990's2 (28.57)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barone, D; Gallico, L; Luzzani, F; Tarzia, G; Toja, E1
Cook, JM; Cox, ED; Diaz-Arauzo, H; Harris, B; Huang, Q; Ma, C; McKernan, R; Reddy, MS; Skolnick, P1
Garrett, KM; Melchior, CL; Tabakoff, B1
Corcoran, ME; McNamara, RK1
Beer, B; Coupet, J; Greenblatt, EN; Klepner, CA; Lippa, AS1
Stephens, DN; Weidmann, R1
Bates, JF; Hall, TW; Peake, L; Standish, LJ; Swearengen, ES1

Other Studies

7 other study(ies) available for cl 218872 and Absence Seizure

ArticleYear
Benzodiazepine receptor binding and anticonflict activity in a series of 3,6-disubstituted pyridazino[4,3-c]isoquinolines devoid of anticonvulsant properties.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:9

    Topics: Animals; Binding, Competitive; Chemical Phenomena; Chemistry; Conflict, Psychological; Diazepam; Isoquinolines; Male; Mice; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Structure-Activity Relationship

1985
Synthesis and evaluation of analogues of the partial agonist 6-(propyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (6-PBC) and the full agonist 6-(benzyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (Zk 93423)
    Journal of medicinal chemistry, 1998, Jul-02, Volume: 41, Issue:14

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Binding, Competitive; Carbolines; Cell Line; Cerebral Cortex; Drug Design; GABA Agonists; Humans; Male; Mice; Muscle Relaxation; Rats; Receptors, GABA-A; Recombinant Proteins; Seizures; Structure-Activity Relationship

1998
A benzodiazepine antagonist action of CL 218,872.
    Life sciences, 1984, May-28, Volume: 34, Issue:22

    Topics: Animals; Anticonvulsants; Benzodiazepines; Benzodiazepinones; Convulsants; Diazepam; Flumazenil; Male; Mice; Mice, Inbred C57BL; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1984
CL 218,872 a triazolopyridazine with a selective affinity for the benzodiazepine BZ1 receptor subtype, retards the development and expression of amygdaloid-kindled seizures: effects of flumazenil.
    Epilepsy research, 1993, Volume: 16, Issue:1

    Topics: Amygdala; Animals; Anti-Anxiety Agents; Drug Interactions; Flumazenil; Kindling, Neurologic; Male; Pyridazines; Rats; Receptors, GABA-A; Seizures

1993
A synthetic non-benzodiazepine ligand for benzodiazepine receptors: a probe for investigating neuronal substrates of anxiety.
    Pharmacology, biochemistry, and behavior, 1979, Volume: 11, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Body Temperature; Conflict, Psychological; gamma-Aminobutyric Acid; Glycine; Humans; Ligands; Male; Mice; Motor Activity; Neurons; Pentylenetetrazole; Pyridazines; Rats; Receptors, Drug; Seizures

1979
Blockade of FG 7142 kindling by anticonvulsants acting at sites distant from the benzodiazepine receptor.
    Brain research, 1989, Jul-17, Volume: 492, Issue:1-2

    Topics: Animals; Anticonvulsants; Carbolines; Clonazepam; Dibenzocycloheptenes; Dizocilpine Maleate; Female; Kindling, Neurologic; Mice; Pyridazines; Receptors, GABA-A; Seizures

1989
CL 218-872 pretreatment and intervention block kainate-induced convulsions and neuropathology.
    Behavioral neuroscience, 1988, Volume: 102, Issue:1

    Topics: Animals; Anticonvulsants; Brain; Diazepam; Kainic Acid; Male; Organ Specificity; Pyridazines; Rats; Rats, Inbred Strains; Seizures

1988