Page last updated: 2024-08-17

carbostyril and Muscle Relaxation

carbostyril has been researched along with Muscle Relaxation in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19901 (8.33)18.7374
1990's5 (41.67)18.2507
2000's4 (33.33)29.6817
2010's2 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Durgin, BG; Galley, JC; Hahn, SA; Miller, MP; Straub, AC; Wood, KC; Yuan, S1
Chen, Y; Hegde, SS; Hughes, AD; Jasper, JR; Lee, TW; Mammen, M; Martin, WJ; McNamara, A; Pulido-Rios, MT; Steinfeld, T1
Gündüz, MG; Oztürk, GS; Safak, C; Sarioğlu, Y; Simşek, R; Vural, M1
Brioni, JD; Buckner, SA; Carroll, WA; Chapple, CR; Chess-Williams, R; Coghlan, MJ; Davis-Taber, R; Daza, AV; Gopalakrishnan, M; Liu, D; Liu, Y; Milicic, I; Molinari, EJ; Scott, VE; Sellers, D; Shieh, CC; Sullivan, JP; Whiteaker, KL; Williams, M1
Boissard, CG; Cook, D; Ding, M; Dworetzky, SI; Fan, W; Flint, K; Goggins, GD; Gribkoff, VK; Hewawasam, P; Lodge, NJ; Myers, RA; Starrett, JE1
Aydin, F; Erol, K; Linden, A; Safak, C; Simşek, R; Ulgen, M1
Kuo, SC; Yu, SM1
Bast, A; Donnell, D; Voss, HP1
Andersson, KE; Degerman, E; Lindgren, S; Manganiello, V; Rascón, A1
Ikezawa, K; Kikkawa, H; Naito, K1
Crankshaw, D; Haslam, RJ; Maurice, DH1
Fujimura, H; Kobayashi, G; Matsuda, H; Yamahara, J1

Other Studies

12 other study(ies) available for carbostyril and Muscle Relaxation

ArticleYear
Antagonism of Forkhead Box Subclass O Transcription Factors Elicits Loss of Soluble Guanylyl Cyclase Expression.
    Molecular pharmacology, 2019, Volume: 95, Issue:6

    Topics: Animals; Aorta, Thoracic; Cell Cycle Proteins; Cells, Cultured; Dose-Response Relationship, Drug; Down-Regulation; Forkhead Transcription Factors; Gene Expression Regulation; Mice; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Quinolones; Rats; Soluble Guanylyl Cyclase

2019
Pharmacologic characterization of GSK-961081 (TD-5959), a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties.
    The Journal of pharmacology and experimental therapeutics, 2014, Volume: 351, Issue:1

    Topics: Adrenergic beta-2 Receptor Antagonists; Albuterol; Animals; Bronchodilator Agents; Carbamates; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Drug Evaluation, Preclinical; Guinea Pigs; HEK293 Cells; Humans; Lung; Muscarinic Antagonists; Muscle Relaxation; Muscle, Smooth; Protein Binding; Quinolones; Receptors, Adrenergic, beta; Receptors, Muscarinic; Salmeterol Xinafoate; Scopolamine Derivatives; Tiotropium Bromide; Tissue Distribution; Trachea

2014
Synthesis of 2-methyl-4-aryl-4,6,7,8-tetrahydro-5(1H)-quinolone derivatives and their effects on potassium channels.
    Arzneimittel-Forschung, 2008, Volume: 58, Issue:12

    Topics: Animals; In Vitro Techniques; Indicators and Reagents; Magnetic Resonance Spectroscopy; Muscle Relaxation; Muscle, Smooth; Pinacidil; Potassium Channels; Potassium Chloride; Quinolones; Rabbits; Spectrophotometry, Infrared; Urinary Bladder

2008
(-)-(9S)-9-(3-Bromo-4-fluorophenyl)-2,3,5,6,7,9-hexahydrothieno[3,2-b]quinolin-8(4H)-one 1,1-dioxide (A-278637): a novel ATP-sensitive potassium channel opener efficacious in suppressing urinary bladder contractions. I. In vitro characterization.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 303, Issue:1

    Topics: Amides; Animals; Aorta, Thoracic; ATP-Binding Cassette Transporters; Benzophenones; Cyclic S-Oxides; Cyclobutanes; Guinea Pigs; Humans; In Vitro Techniques; Ion Channel Gating; KATP Channels; Kinetics; Male; Membrane Potentials; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Muscle, Smooth, Vascular; Nitriles; Patch-Clamp Techniques; Portal Vein; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Quinolones; Rats; Rats, Sprague-Dawley; Urinary Bladder

2002
4-Aryl-3-(hydroxyalkyl)quinolin-2-ones: novel maxi-K channel opening relaxants of corporal smooth muscle targeted for erectile dysfunction.
    Journal of medicinal chemistry, 2003, Jul-03, Volume: 46, Issue:14

    Topics: Animals; Blood Pressure; Electric Stimulation; Erectile Dysfunction; In Vitro Techniques; Large-Conductance Calcium-Activated Potassium Channels; Male; Muscle Relaxation; Muscle, Smooth; Penile Erection; Penis; Potassium Channels, Calcium-Activated; Pressure; Quinolones; Rabbits; Rats; Rats, Inbred F344; Structure-Activity Relationship

2003
Studies on condensed 1,4-dihydropyridine derivatives and their calcium modulatory activities.
    Die Pharmazie, 2006, Volume: 61, Issue:8

    Topics: Animals; Biotransformation; Calcium Channel Blockers; Chromatography, High Pressure Liquid; Dihydropyridines; Female; In Vitro Techniques; Indicators and Reagents; Magnetic Resonance Spectroscopy; Male; Microsomes, Liver; Models, Molecular; Muscle Relaxation; Muscle, Smooth, Vascular; Quinolones; Rats; Sheep; Spectrophotometry, Infrared; X-Ray Diffraction

2006
Vasorelaxant effect of isoliquiritigenin, a novel soluble guanylate cyclase activator, in rat aorta.
    British journal of pharmacology, 1995, Volume: 114, Issue:8

    Topics: Aldehyde Reductase; Animals; Aorta; Chalcone; Chalcones; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Female; Guanylate Cyclase; Male; Methylene Blue; Muscle Relaxation; Muscle, Smooth, Vascular; Phenylephrine; Platelet Aggregation Inhibitors; Pyrrolidinones; Quinolones; Rats; Rats, Wistar; Rolipram

1995
Atypical molecular pharmacology of a new long-acting beta 2-adrenoceptor agonist, TA 2005.
    European journal of pharmacology, 1992, Dec-01, Volume: 227, Issue:4

    Topics: Adrenergic beta-Agonists; Amphetamines; Animals; Binding, Competitive; Bronchodilator Agents; Cattle; GTP-Binding Proteins; Guinea Pigs; Hydroxyquinolines; Iodocyanopindolol; Isoproterenol; Magnesium; Male; Muscle Relaxation; Muscle, Smooth; Pindolol; Quinolones; Receptors, Adrenergic, beta; Trachea

1992
Selective inhibition of cGMP-inhibited and cGMP-noninhibited cyclic nucleotide phosphodiesterases and relaxation of rat aorta.
    Biochemical pharmacology, 1991, Jul-15, Volume: 42, Issue:3

    Topics: 2',3'-Cyclic-Nucleotide Phosphodiesterases; Animals; Aorta; Cyclic AMP; Cyclic GMP; Drug Interactions; Isoenzymes; Milrinone; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phenylephrine; Pyridones; Pyrrolidinones; Quinolones; Rats; Rolipram; Serotonin; Vasodilator Agents

1991
Tracheal relaxing effects and beta 2-selectivity of TA-2005, a newly developed bronchodilating agent, in isolated guinea pig tissues.
    Japanese journal of pharmacology, 1991, Volume: 57, Issue:2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Amphetamines; Animals; Bronchodilator Agents; Ethanolamines; Formoterol Fumarate; Guanosine Triphosphate; Guinea Pigs; Heart Ventricles; Histamine; Hydroxyquinolines; In Vitro Techniques; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Kinetics; Lung; Male; Membranes; Muscle Contraction; Muscle Relaxation; Pindolol; Procaterol; Quinolones; Radioligand Assay; Receptors, Adrenergic, beta; Trachea

1991
Synergistic actions of nitrovasodilators and isoprenaline on rat aortic smooth muscle.
    European journal of pharmacology, 1991, Jan-10, Volume: 192, Issue:2

    Topics: Adenylyl Cyclases; Animals; Aorta; Dose-Response Relationship, Drug; Drug Synergism; In Vitro Techniques; Isoproterenol; Male; Molsidomine; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroprusside; Quinolones; Rats; Rats, Inbred Strains; Vasodilator Agents

1991
The vasorelaxant effect of evocarpine in isolated aortic strips: mode of action.
    European journal of pharmacology, 1988, Oct-11, Volume: 155, Issue:1-2

    Topics: Alkaloids; Animals; Aorta, Thoracic; Biological Transport, Active; Calcium Radioisotopes; Carotid Arteries; Cyclic AMP; Cyclic GMP; Guinea Pigs; In Vitro Techniques; Isometric Contraction; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Potassium; Quinolones; Rabbits; Rats; Rats, Inbred Strains; Sodium

1988