Page last updated: 2024-08-17

carbostyril and Malaria, Falciparum

carbostyril has been researched along with Malaria, Falciparum in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's12 (80.00)24.3611
2020's3 (20.00)2.80

Authors

AuthorsStudies
Anas, M; Chaluvalappil, SV; Kalluruttimmal, R; Kumar, N; Kumari, V; Kurian, J; Manhas, A; Manheri, MK1
Awalt, JK; Bailey, BL; Baud, D; Baum, J; Brand, S; Chakraborty, A; Churchyard, A; Cowman, AF; Currie, I; Dans, MG; Favuzza, P; Jackson, PF; Jarman, KE; Lumb, C; Maier, AG; Mukherjee, P; Ngo, A; Nguyen, W; Palandri, J; Papenfuss, T; Penington, J; Ramesh, S; Sleebs, BE; van Dooren, GG; Winzeler, EA; Wittlin, S1
Chinigo, G; Clark, RD; Ferrer, S; Gadwood, R; Gamo, FJ; Lafuente, MJ; Lawless, MS; Le Roch, KG; Morris, DN; Prudhomme, J; Woltosz, WS1
Bruzual, I; Dodean, RA; Doggett, JS; Krollenbrock, A; McConnell, EV; Nilsen, A; Pou, S; Riscoe, MK; Smilkstein, MJ; Winter, R; Zakharov, LN1
Romero, AH1
Dass, S; Ganesan, SM; Ke, H; Mather, MW; Morrisey, JM; Nilsen, A; Pou, S; Riscoe, MK; Vaidya, AB1
Beteck, RM; Hoppe, HC; Jordaan, A; Khanye, SD; Laming, D; Seldon, R; Warner, DF1
Angulo-Barturen, I; Avery, VM; Bathurst, I; Burrows, JN; Charman, SA; Cross, RM; Delves, MJ; Duffy, S; Ferrer, S; Forquer, IP; Gamo, FJ; Guy, RK; Herreros, E; Jiménez-Díaz, MB; Kelly, JX; Kocken, CHM; Kyle, DE; LaCrue, AN; Li, Y; Manetsch, R; Marfurt, J; Mather, MW; Morrisey, JM; Mutka, T; Nilsen, A; Noviyanti, R; Price, RN; Riscoe, MK; Ryan, E; Saenz, FE; Sanz, LM; Sebayang, BF; Shackleford, DM; Siegl, P; Sinden, RE; Steuten, J; Vaidya, AB; White, KL; Winter, RW; Wirjanata, G; Zeeman, AM1
Harrington, M1
Cross, RM; Kyle, DE; Lacrue, AN; Maignan, JR; Manetsch, R; Sáenz, FE; Udenze, KO1
Aher, RB; Roy, K1
Forquer, IP; Hinrichs, DJ; Kelly, JX; Kim, K; Li, Y; Mather, MW; Meermeier, E; Miley, GP; Morrisey, JM; Nilsen, A; Pershing, AM; Pou, S; Riscoe, MK; Stickles, AM; Ting, LM; Vaidya, AB; Winter, RW1
Ha, YR; Hong, Y; Hwang, BG; Lee, SJ; Yang, HW1
Forquer, IP; Kelly, JX; Li, Y; Morrisey, JM; Nilsen, A; Pou, S; Riscoe, MK; Smilkstein, MJ; Stickles, AM; Vaidya, AB; Winter, RW1
Amewu, RK; Antoine, T; Berger, O; Berry, NG; Biagini, GA; Chadwick, J; Charoensutthivarakul, S; Davies, J; Delves, MJ; Fisher, N; Gibbons, P; Hemingway, J; Hill, A; Hong, DW; Kocken, CH; Lawrenson, AS; Leung, SC; Mbekeani, A; Mubaraki, MA; Nixon, GL; O'Neill, PM; Pacorel, B; Pidathala, C; Sharma, R; Shone, AE; Sinden, RE; Srivastava, A; Stocks, PA; Taylor, L; Ward, SA; Warman, AJ; Zeeman, AM1

Reviews

1 review(s) available for carbostyril and Malaria, Falciparum

ArticleYear
Role of Trifluoromethyl Substitution in Design of Antimalarial Quinolones: a Comprehensive Review.
    Topics in current chemistry (Cham), 2019, Mar-05, Volume: 377, Issue:2

    Topics: Antimalarials; Drug Design; Hydrocarbons, Fluorinated; Malaria, Falciparum; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolones

2019

Other Studies

14 other study(ies) available for carbostyril and Malaria, Falciparum

ArticleYear
Adenine Modification at C7 as a Viable Strategy to Potentiate the Antimalarial Activity of Quinolones.
    ChemMedChem, 2022, 01-19, Volume: 17, Issue:2

    Topics: Adenine; Animals; Antimalarials; Chlorocebus aethiops; Dose-Response Relationship, Drug; Malaria, Falciparum; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolones; Structure-Activity Relationship; Vero Cells

2022
7-
    ACS infectious diseases, 2023, 03-10, Volume: 9, Issue:3

    Topics: Animals; Antimalarials; Cytochromes b; Folic Acid Antagonists; Malaria, Falciparum; Mice; Plasmodium falciparum; Quinolones

2023
Design and tests of prospective property predictions for novel antimalarial 2-aminopropylaminoquinolones.
    Journal of computer-aided molecular design, 2020, Volume: 34, Issue:11

    Topics: Antimalarials; Dihydroorotate Dehydrogenase; Drug Design; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Molecular Docking Simulation; Molecular Structure; Oxidoreductases Acting on CH-CH Group Donors; Plasmodium falciparum; Quantitative Structure-Activity Relationship; Quinolones

2020
Targeted Structure-Activity Analysis of Endochin-like Quinolones Reveals Potent Qi and Qo Site Inhibitors of Toxoplasma gondii and Plasmodium falciparum Cytochrome bc
    ACS infectious diseases, 2018, 11-09, Volume: 4, Issue:11

    Topics: Animals; Antiprotozoal Agents; Cells, Cultured; Drug Discovery; Drug Resistance; Electron Transport Complex III; Humans; Malaria, Falciparum; Mice; Molecular Structure; Phenyl Ethers; Plasmodium falciparum; Quinolones; Structure-Activity Relationship; Toxoplasma; Toxoplasmosis

2018
Mitochondrial type II NADH dehydrogenase of Plasmodium falciparum (PfNDH2) is dispensable in the asexual blood stages.
    PloS one, 2019, Volume: 14, Issue:4

    Topics: Animals; Antimalarials; Cells, Cultured; CRISPR-Cas Systems; Drug Resistance; Electron Transport Complex I; Electron Transport Complex III; Erythrocytes; Gene Knockout Techniques; Humans; Malaria, Falciparum; Mitochondria; NADH Dehydrogenase; Plasmodium falciparum; Protozoan Proteins; Quinolones

2019
New Quinolone-Based Thiosemicarbazones Showing Activity Against
    Molecules (Basel, Switzerland), 2019, May-04, Volume: 24, Issue:9

    Topics: Animals; Anti-Infective Agents; Candy; Drug Interactions; HeLa Cells; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Molecular Structure; Mycobacterium tuberculosis; Plasmodium falciparum; Quinolones; Small Molecule Libraries; Thiosemicarbazones; Tuberculosis

2019
Quinolone-3-diarylethers: a new class of antimalarial drug.
    Science translational medicine, 2013, Mar-20, Volume: 5, Issue:177

    Topics: Animals; Antimalarials; Atovaquone; Drug Resistance; Drug Synergism; Life Cycle Stages; Malaria; Malaria, Falciparum; Mice; Plasmodium falciparum; Plasmodium vivax; Proguanil; Pyridones; Quinolones

2013
A new twist in targeting malaria parasites.
    Lab animal, 2013, Volume: 42, Issue:5

    Topics: Administration, Oral; Animals; Antimalarials; Humans; Malaria, Falciparum; Mice; Plasmodium falciparum; Quinolones

2013
4-(1H)-Quinolones and 1,2,3,4-Tetrahydroacridin-9(10H)-ones prevent the transmission of Plasmodium falciparum to Anopheles freeborni.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:12

    Topics: Acridines; Animals; Anopheles; Antimalarials; Female; Humans; Insect Vectors; Life Cycle Stages; Malaria; Malaria, Falciparum; Male; Mice; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Quinolones; Salivary Glands; Structure-Activity Relationship

2013
Classification SAR modeling of diverse quinolone compounds for antimalarial potency against Plasmodium falciparum.
    Combinatorial chemistry & high throughput screening, 2014, Volume: 17, Issue:5

    Topics: Antimalarials; Computer Simulation; Discriminant Analysis; Drug Design; Humans; Malaria, Falciparum; Models, Biological; Models, Molecular; Plasmodium falciparum; Quantitative Structure-Activity Relationship; Quinolones

2014
Inhibition of cytochrome bc1 as a strategy for single-dose, multi-stage antimalarial therapy.
    The American journal of tropical medicine and hygiene, 2015, Volume: 92, Issue:6

    Topics: Animals; Antimalarials; Drug Resistance; Electron Transport Complex III; Female; Malaria, Falciparum; Mice; Parasitemia; Phenyl Ethers; Plasmodium falciparum; Plasmodium yoelii; Quinolones

2015
Effect of Farnesyltransferase Inhibitor R115777 on Mitochondria of Plasmodium falciparum.
    The Korean journal of parasitology, 2015, Volume: 53, Issue:4

    Topics: Antimalarials; Enzyme Inhibitors; Farnesyltranstransferase; Humans; Malaria, Falciparum; Mitochondria; Plasmodium falciparum; Protozoan Proteins; Quinolones

2015
Atovaquone and ELQ-300 Combination Therapy as a Novel Dual-Site Cytochrome bc1 Inhibition Strategy for Malaria.
    Antimicrobial agents and chemotherapy, 2016, Volume: 60, Issue:8

    Topics: Animals; Antimalarials; Atovaquone; Drug Combinations; Drug Therapy, Combination; Electron Transport Complex III; Female; Malaria, Falciparum; Mice; Parasitemia; Plasmodium falciparum; Proguanil; Quinolones

2016
Generation of quinolone antimalarials targeting the Plasmodium falciparum mitochondrial respiratory chain for the treatment and prophylaxis of malaria.
    Proceedings of the National Academy of Sciences of the United States of America, 2012, May-22, Volume: 109, Issue:21

    Topics: Animals; Antimalarials; Cells, Cultured; Electron Transport; Electron Transport Complex I; Electron Transport Complex III; Hepatocytes; Macaca mulatta; Malaria, Falciparum; Male; Mice; Mice, Inbred Strains; Mitochondria; Plasmodium berghei; Plasmodium cynomolgi; Plasmodium falciparum; Pyridines; Quinolones

2012