carbostyril has been researched along with Malaria, Falciparum in 15 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 12 (80.00) | 24.3611 |
2020's | 3 (20.00) | 2.80 |
Authors | Studies |
---|---|
Anas, M; Chaluvalappil, SV; Kalluruttimmal, R; Kumar, N; Kumari, V; Kurian, J; Manhas, A; Manheri, MK | 1 |
Awalt, JK; Bailey, BL; Baud, D; Baum, J; Brand, S; Chakraborty, A; Churchyard, A; Cowman, AF; Currie, I; Dans, MG; Favuzza, P; Jackson, PF; Jarman, KE; Lumb, C; Maier, AG; Mukherjee, P; Ngo, A; Nguyen, W; Palandri, J; Papenfuss, T; Penington, J; Ramesh, S; Sleebs, BE; van Dooren, GG; Winzeler, EA; Wittlin, S | 1 |
Chinigo, G; Clark, RD; Ferrer, S; Gadwood, R; Gamo, FJ; Lafuente, MJ; Lawless, MS; Le Roch, KG; Morris, DN; Prudhomme, J; Woltosz, WS | 1 |
Bruzual, I; Dodean, RA; Doggett, JS; Krollenbrock, A; McConnell, EV; Nilsen, A; Pou, S; Riscoe, MK; Smilkstein, MJ; Winter, R; Zakharov, LN | 1 |
Romero, AH | 1 |
Dass, S; Ganesan, SM; Ke, H; Mather, MW; Morrisey, JM; Nilsen, A; Pou, S; Riscoe, MK; Vaidya, AB | 1 |
Beteck, RM; Hoppe, HC; Jordaan, A; Khanye, SD; Laming, D; Seldon, R; Warner, DF | 1 |
Angulo-Barturen, I; Avery, VM; Bathurst, I; Burrows, JN; Charman, SA; Cross, RM; Delves, MJ; Duffy, S; Ferrer, S; Forquer, IP; Gamo, FJ; Guy, RK; Herreros, E; Jiménez-Díaz, MB; Kelly, JX; Kocken, CHM; Kyle, DE; LaCrue, AN; Li, Y; Manetsch, R; Marfurt, J; Mather, MW; Morrisey, JM; Mutka, T; Nilsen, A; Noviyanti, R; Price, RN; Riscoe, MK; Ryan, E; Saenz, FE; Sanz, LM; Sebayang, BF; Shackleford, DM; Siegl, P; Sinden, RE; Steuten, J; Vaidya, AB; White, KL; Winter, RW; Wirjanata, G; Zeeman, AM | 1 |
Harrington, M | 1 |
Cross, RM; Kyle, DE; Lacrue, AN; Maignan, JR; Manetsch, R; Sáenz, FE; Udenze, KO | 1 |
Aher, RB; Roy, K | 1 |
Forquer, IP; Hinrichs, DJ; Kelly, JX; Kim, K; Li, Y; Mather, MW; Meermeier, E; Miley, GP; Morrisey, JM; Nilsen, A; Pershing, AM; Pou, S; Riscoe, MK; Stickles, AM; Ting, LM; Vaidya, AB; Winter, RW | 1 |
Ha, YR; Hong, Y; Hwang, BG; Lee, SJ; Yang, HW | 1 |
Forquer, IP; Kelly, JX; Li, Y; Morrisey, JM; Nilsen, A; Pou, S; Riscoe, MK; Smilkstein, MJ; Stickles, AM; Vaidya, AB; Winter, RW | 1 |
Amewu, RK; Antoine, T; Berger, O; Berry, NG; Biagini, GA; Chadwick, J; Charoensutthivarakul, S; Davies, J; Delves, MJ; Fisher, N; Gibbons, P; Hemingway, J; Hill, A; Hong, DW; Kocken, CH; Lawrenson, AS; Leung, SC; Mbekeani, A; Mubaraki, MA; Nixon, GL; O'Neill, PM; Pacorel, B; Pidathala, C; Sharma, R; Shone, AE; Sinden, RE; Srivastava, A; Stocks, PA; Taylor, L; Ward, SA; Warman, AJ; Zeeman, AM | 1 |
1 review(s) available for carbostyril and Malaria, Falciparum
Article | Year |
---|---|
Role of Trifluoromethyl Substitution in Design of Antimalarial Quinolones: a Comprehensive Review.
Topics: Antimalarials; Drug Design; Hydrocarbons, Fluorinated; Malaria, Falciparum; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolones | 2019 |
14 other study(ies) available for carbostyril and Malaria, Falciparum
Article | Year |
---|---|
Adenine Modification at C7 as a Viable Strategy to Potentiate the Antimalarial Activity of Quinolones.
Topics: Adenine; Animals; Antimalarials; Chlorocebus aethiops; Dose-Response Relationship, Drug; Malaria, Falciparum; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolones; Structure-Activity Relationship; Vero Cells | 2022 |
7-
Topics: Animals; Antimalarials; Cytochromes b; Folic Acid Antagonists; Malaria, Falciparum; Mice; Plasmodium falciparum; Quinolones | 2023 |
Design and tests of prospective property predictions for novel antimalarial 2-aminopropylaminoquinolones.
Topics: Antimalarials; Dihydroorotate Dehydrogenase; Drug Design; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Molecular Docking Simulation; Molecular Structure; Oxidoreductases Acting on CH-CH Group Donors; Plasmodium falciparum; Quantitative Structure-Activity Relationship; Quinolones | 2020 |
Targeted Structure-Activity Analysis of Endochin-like Quinolones Reveals Potent Qi and Qo Site Inhibitors of Toxoplasma gondii and Plasmodium falciparum Cytochrome bc
Topics: Animals; Antiprotozoal Agents; Cells, Cultured; Drug Discovery; Drug Resistance; Electron Transport Complex III; Humans; Malaria, Falciparum; Mice; Molecular Structure; Phenyl Ethers; Plasmodium falciparum; Quinolones; Structure-Activity Relationship; Toxoplasma; Toxoplasmosis | 2018 |
Mitochondrial type II NADH dehydrogenase of Plasmodium falciparum (PfNDH2) is dispensable in the asexual blood stages.
Topics: Animals; Antimalarials; Cells, Cultured; CRISPR-Cas Systems; Drug Resistance; Electron Transport Complex I; Electron Transport Complex III; Erythrocytes; Gene Knockout Techniques; Humans; Malaria, Falciparum; Mitochondria; NADH Dehydrogenase; Plasmodium falciparum; Protozoan Proteins; Quinolones | 2019 |
New Quinolone-Based Thiosemicarbazones Showing Activity Against
Topics: Animals; Anti-Infective Agents; Candy; Drug Interactions; HeLa Cells; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Molecular Structure; Mycobacterium tuberculosis; Plasmodium falciparum; Quinolones; Small Molecule Libraries; Thiosemicarbazones; Tuberculosis | 2019 |
Quinolone-3-diarylethers: a new class of antimalarial drug.
Topics: Animals; Antimalarials; Atovaquone; Drug Resistance; Drug Synergism; Life Cycle Stages; Malaria; Malaria, Falciparum; Mice; Plasmodium falciparum; Plasmodium vivax; Proguanil; Pyridones; Quinolones | 2013 |
A new twist in targeting malaria parasites.
Topics: Administration, Oral; Animals; Antimalarials; Humans; Malaria, Falciparum; Mice; Plasmodium falciparum; Quinolones | 2013 |
4-(1H)-Quinolones and 1,2,3,4-Tetrahydroacridin-9(10H)-ones prevent the transmission of Plasmodium falciparum to Anopheles freeborni.
Topics: Acridines; Animals; Anopheles; Antimalarials; Female; Humans; Insect Vectors; Life Cycle Stages; Malaria; Malaria, Falciparum; Male; Mice; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Quinolones; Salivary Glands; Structure-Activity Relationship | 2013 |
Classification SAR modeling of diverse quinolone compounds for antimalarial potency against Plasmodium falciparum.
Topics: Antimalarials; Computer Simulation; Discriminant Analysis; Drug Design; Humans; Malaria, Falciparum; Models, Biological; Models, Molecular; Plasmodium falciparum; Quantitative Structure-Activity Relationship; Quinolones | 2014 |
Inhibition of cytochrome bc1 as a strategy for single-dose, multi-stage antimalarial therapy.
Topics: Animals; Antimalarials; Drug Resistance; Electron Transport Complex III; Female; Malaria, Falciparum; Mice; Parasitemia; Phenyl Ethers; Plasmodium falciparum; Plasmodium yoelii; Quinolones | 2015 |
Effect of Farnesyltransferase Inhibitor R115777 on Mitochondria of Plasmodium falciparum.
Topics: Antimalarials; Enzyme Inhibitors; Farnesyltranstransferase; Humans; Malaria, Falciparum; Mitochondria; Plasmodium falciparum; Protozoan Proteins; Quinolones | 2015 |
Atovaquone and ELQ-300 Combination Therapy as a Novel Dual-Site Cytochrome bc1 Inhibition Strategy for Malaria.
Topics: Animals; Antimalarials; Atovaquone; Drug Combinations; Drug Therapy, Combination; Electron Transport Complex III; Female; Malaria, Falciparum; Mice; Parasitemia; Plasmodium falciparum; Proguanil; Quinolones | 2016 |
Generation of quinolone antimalarials targeting the Plasmodium falciparum mitochondrial respiratory chain for the treatment and prophylaxis of malaria.
Topics: Animals; Antimalarials; Cells, Cultured; Electron Transport; Electron Transport Complex I; Electron Transport Complex III; Hepatocytes; Macaca mulatta; Malaria, Falciparum; Male; Mice; Mice, Inbred Strains; Mitochondria; Plasmodium berghei; Plasmodium cynomolgi; Plasmodium falciparum; Pyridines; Quinolones | 2012 |