Page last updated: 2024-08-17

carbostyril and HIV Coinfection

carbostyril has been researched along with HIV Coinfection in 245 studies

Research

Studies (245)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (1.63)18.2507
2000's25 (10.20)29.6817
2010's183 (74.69)24.3611
2020's33 (13.47)2.80

Authors

AuthorsStudies
Calcagno, A; Calza, S; Castelli, F; Cattelan, AM; Celesia, BM; Chiesa, A; De Socio, G; Ferrara, M; Focà, E; Guaraldi, G; Madeddu, G; Milic, J; Nozza, S; Orofino, G; Piconi, S; Renzetti, S; Siano, M1
Gao, LY; Hu, Y; Huang, XJ; Ma, P; Wu, H; Wu, Y; Xia, H; Yan, ZF1
Chang, SF; Chang, SY; Chuang, YC; Hsiao, CY; Hsieh, TW; Hsu, JY; Huang, YS; Hung, CC; Liu, WC; Su, YC; Sun, HY1
Aydin, OA; Bilge, B; Bolukcu, S; Dokmetas, I; Gumuser, F; Gunduz, A; Karaosmanoglu, HK; Mete, B; Tabak, F; Yildiz, DS1
Barry, S; Chopra, A; Ibrahim, A; Pokhrel, K; Smith, T1
Dee, N; Dewar, R; George, J; Grossman, Z; Hill, S; Huik, K; Khan, M; Kuriakose, S; Lange, CM; Maldarelli, F; Pau, A; Rehm, CA; Rehman, T; Stoll, P1
Brummel, SS; Chadwick, EG; Huo, Y; Jacobson, DL; Jao, J; Kacanek, D; Kahlert, CR; Patel, K; Powis, KM; Seage, GR; Shiau, S; Sultan-Beyer, L; Williams, PL; Yee, LM; Zash, R1
Cao, T; He, Y; Jia, X; Ju, B; Liu, J; Liu, X; Peng, Q; Rao, M; Song, Y; Sun, L; Wang, H; Wang, S; Xu, L; Zhang, H; Zhang, L; Zhang, Q; Zhao, F; Zhou, J; Zhou, Y1
Brehm, TT; Degen, O; Franz, M; Hertling, S; Hüfner, A; Kreuels, B; Schmiedel, S; Schulze Zur Wiesch, J1
Chen, SQ; Li, Q; Yang, LL; Zhou, LB1
Burgi, A; Letendre, SL; Little, SJ; Ma, Q; Morse, GD; Ocque, AJ; Sanders, C1
Castagna, A; Gianotti, N1
Das, M; Haubrich, R; Maggiolo, F; Mateo-Garcia, MG; McNicholl, I; Molina, JM; Ong, E; Piontkowsky, D; Pulido, F; Raffi, F; Rizzardini, G; Shao, Y1
Bezenchek, A; Borghetti, A; Callegaro, A; Colafigli, M; Costantini, A; De Luca, A; Di Carlo, D; Farinacci, D; Ferrara, SM; Gagliardini, R; Gianotti, N; Giombini, E; Gismondo, MR; Lombardi, F; Maggiolo, F; Modica, S; Redi, D; Rossetti, B; Rusconi, S; Sterrantino, G; Zazzi, M1
Albanesi, E; Appendino, A; Boccuto, A; Dragoni, F; Giannini, A; Saladini, F; Vicenti, I; Zazzi, M1
Hollenbeck, BL; Kishore, S; Lee, MSL; Padival, S1
Biasiotto, G; Bonito, A; Calza, S; Castelli, F; Quiros-Roldan, E; Vezzoli, M; Zanella, I1
Ajana, F; Bani-Sadr, F; Bouvet, E; Cotte, L; Galempoix, JM; Gantner, P; Hessamfar, M; Hustache-Mathieu, L; Lebrette, MG; Muret, P; Pellissier, G; Piroth, L; Rey, D; Rouveix, E; Simon, A; Souala, MF; Truchetet, F; Valin, N1
Butler, AM; O'Halloran, JA; Olsen, MA; Powderly, WG; Sahrmann, J1
Bukkems, V; Burger, D; Colbers, A; Garcia, C; Konopnicki, D; Lambert, JS; Necsoi, C; Rockstroh, J; Schwarze-Zander, C; Tenorio, CH1
Chitongo, R; Cloete, R; Jacobs, GB; Mikasi, SG; Obasa, AE1
Dicker, I; Higley, H; Jenkins, S; Krystal, M; Lin, Z; Mathur, A; Meanwell, NA; Naidu, BN; Panja, C; Parker, D; Patel, M; Protack, T; Rampulla, R; Terry, B; Walker, MA1
Chen, H; Chowdhury, P; Gong, Y; Gorantla, S; Kumar, S; Nagesh, PKB; Sinha, N; Yallapu, MM; Zhi, K1
Castagna, A; Fornabaio, C; Galli, L; Malena, M; Menozzi, M; Poli, A; Santoro, MM; White, KL; Zazzi, M1
Amador, C; de Zárraga, MA; Díez Martínez, M; Górgolas, M; Jarrín, I; Moreno, C; Navarro, M; Pérez-Elías, MJ; Pérez-Martínez, L; Ruiz-Algueró, M; Suárez-García, I; Viciana, P1
Cong, ME; Dinh, C; García-Lerma, JG; Haaland, R; Heneine, W; Holder, A; Johnson, R; Kelley, CF; Kelley, K; Khalil, G; Massud, I; Mills, P; Pan, Y; Ruone, S; Sanchez, T; Zlotorzynska, M1
Chang, SF; Chang, SY; Chen, GJ; Cheng, CY; Chuang, YC; Hsieh, MH; Huang, SH; Hung, CC; Lee, CH; Lee, YC; Lee, YL; Su, LS; Sun, HY; Tang, HJ; Tsai, HC1
Cloete, R; Ikomey, GM; Isaacs, D; Jacobs, GB; Mikasi, SG; Obasa, AE; Shityakov, S1
Festa, L; Grinspan, JB; Jordan-Sciutto, KL; Monnerie, H; Putatunda, R; Romer, M; Roth, LM; Zidane, B1
Amano, K; Hachiya, A; Ichiki, A; Kinai, E; Yotsumoto, M1
Adams, JL; Baxter, J; Choi, YC; George, J; Pontiggia, L; West, M1
DeMarais, P; Max, B1
Cheng, CY; Cheng, SH; Ho, MW; Huang, SH; Huang, YS; Hung, CC; Lee, CH; Lee, YT; Lin, SP; Liou, BH; Liu, CE; Lu, PL; Sun, HY; Tang, HJ; Tsai, HC; Yang, CJ1
Ma, R; Tong, ZW; Xu, B; Zhang, Q; Zhang, YS; Zhao, CS; Zhao, RG1
Castagna, A; Esser, S; Haubrich, R; Llibre, JM; Margot, N; McNicholl, IR; Molina, JM; Perez-Valero, I; Piontkowsky, D; Pulido, F; Shao, Y; Temme, L1
Adimora, AA; Dastgheyb, R; Fischl, MA; Fitzgerald, KC; Gustafson, DR; Kamkwalala, AR; Konkle-Parker, D; Lahiri, CD; Maki, PM; Milam, J; O'Halloran, JA; Ofotokun, I; Rubin, LH; Sharma, A; Sheth, AN; Spence, AB; Wang, K; Weber, KM; Williams, DW; Xu, Y1
Bendtsen, F; Benfield, T; Gelpi, M; Kirkegaard-Klitbo, DM; Nielsen, SD; Thomsen, MT1
Chimukangara, B; Gordon, M; Mbhele, N1
Blanch, J; Blanco, JL; de Lazzari, E; Gatell, JM; Gonzalez-Cordon, A; Laguno, M; Lonca, M; Mallolas, J; Marcos, MA; Martinez, E; Martinez-Rebollar, M; Padilla, M; Peñafiel, J; Rodriguez, A; Rojas, J; Tricas, A1
Castagna, A; Chiappetta, S; Galli, L; Lazzarin, A; Nozza, S; Poli, A; Ripa, M; Rovelli, C; Spagnuolo, V; Tambussi, G2
Al Tabaa, O; Audren, V; Blum, L; Hayton, E; Pertuiset, E1
Aitken, C; Bradley-Stewart, A; Gunson, R; MacLean, A; Urcia, C1
Buclin, T; Decosterd, L; Francini, K; Livio, F; Marzolini, C; Tissot, F; Winterfeld, U1
Angione, SA; Cherian, SM; Özdener, AE1
Avettand-Fenoel, V; Bellecave, P; Bonnet, F; Caldato, S; Hessamfar, M; Morlat, P; Ngo Bell, EC; Saunier, A; Tumiotto, C; Vandenhende, MA1
Hughes, CA; Phillips, EJ; Seet, J; Tseng, A; Wu, J1
Balboa-Barreiro, V; Castro-Iglesias, Á; Cid-Silva, P; Fernández-Bargiela, N; Llibre, JM; Margusino-Framiñán, L; Martín-Herranz, I; Pernas-Souto, B; Poveda, E1
Bandera, A; Bonfanti, P; Calza, L; Carenzi, L; Celesia, BM; Cordier, L; De Socio, GV; Di Biagio, A; Falasca, K; Gori, A; Madeddu, G; Maggi, P; Martinelli, C; Orofino, G; Pellicanò, GF; Quirino, T; Ricci, E; Rusconi, S; Squillace, N; Vichi, F1
Andreatta, K; Antinori, A; Berenguer, J; Bloch, M; Cote, P; Flamm, J; Garner, W; McColl, DJ; Nguyen-Cleary, T; Piontkowsky, D; Pozniak, A; Szwarcberg, J; Ward, D1
Baecke, C; Decoutere, L; Gyssens, IC; Messiaen, P; van der Hilst, JCH1
Clark, MR; Deng, Y; Mohideen, M; Panse, G; Quijano, E; Saltzman, WM; Song, E; Zhang, W1
Alessandri-Gradt, E; Bertine, M; Charpentier, C; Collin, G; Descamps, D; Leoz, M; Plantier, JC; Tourneroche, A; Unal, G1
Cao, H; Chang, S; Hodder, SL; Kulkarni, R; Miller, MD; White, KL1
Calvez, V; Charpentier, C; Collin, G; Delelis, O; Descamps, D; Malet, I; Marcelin, AG; Subra, F1
Baldelli, S; Cattaneo, D; Clementi, E; Galli, M; Gervasoni, C; Giacomelli, A; Mazzali, C; Meraviglia, P; Milazzo, L; Minisci, D; Resnati, C; Rizzardini, G1
Arnaiz, JA; Cruceta, A; García, F; Gatell, JM; González, E; González-Cordón, A; Inciarte, A; Laguno, M; Leal, L; León, A; Lucero, C; Mallolas, J; Martínez-Rebollar, M; Rojas, J; Torres, B1
Ganase, B; Harrigan, PR; Harris, M; Hull, MW; Montaner, JSG; Watson, B1
DeJesus, E; Haas, B; Liu, YP; Makadzange, T; Margot, N; McCallister, S; Mills, A; Ramgopal, MN; Segal-Maurer, S1
Akagi, L; Barrios, R; Guillemi, S; Lepik, KJ; Lima, VD; Montaner, JSG; Toy, J; Ulloa, AC; Wang, L; Yip, B1
Avihingsanon, A; Cao, H; Cheng, A; Hagins, D; Hodder, S; Jiang, S; Kido, A; Kityo, C; Kulkarni, R; Squires, K1
Domingo, JC; Domingo, P; Gallego-Escuredo, JM; Gasa, L; Giralt, M; Maroto, AF; Mateo, GM; Morón-Ros, S; Moure, R; Quesada-López, T; Villarroya, F; Villarroya, J1
Cogill, D; Hamers, RL; Lane, HC; Larder, BA; Montaner, JSG; Perez-Elias, MJ; Pozniak, A; Rehm, CA; Reiss, P; Revell, AD; Tempelman, H; van Sighem, AI; Wang, D; Wood, R1
Burger, DM; Colbers, A; Greupink, R; Schalkwijk, SJ; Ter Heine, R; van der Galiën, R; van Herwaarden, AE1
Adorni, F; Borghi, V; Bruzzone, B; Di Biagio, A; Francisci, D; Mancon, A; Maserati, R; Meraviglia, P; Micheli, V; Monno, L; Paolucci, S; Pecorari, M; Punzi, G; Rusconi, S; Tau, P; Zazzi, M1
Anstett, K; Brenner, BG; Ibanescu, RI; Mésplède, T; Oliveira, M; Robbins, MA; Routy, JP1
Acosta, EP; Badell, ML; Barr, E; Best, BM; Burchett, S; Capparelli, EV; Chakhtoura, N; Mirochnick, M; Momper, JD; Park, K; Purswani, M; Shapiro, DE; Smith, E; Stek, A; Wang, J1
Álvarez, H; Díaz-Cambre, H; García-González, J; Llibre, JM; Mariño, A; Valcarce, N1
Álvarez, H; Llibre, JM; Yzusqui, M1
Chauhan, M; Chokkar, N; Kalra, S; Kumar, R1
Cabot, JF; Denault, JS; Langlois, H; Marcotte, S; Sheehan, NL1
Bagella, P; Baldin, G; Capetti, A; Ciccullo, A; Cossu, MV; De Luca, A; Di Giambenedetto, S; Giacomelli, A; Lagi, F; Latini, A; Madeddu, G; Rusconi, S; Sterrantino, G1
Bruzzone, B; D'Autilia, R; De Luca, A; Di Biagio, A; Francisci, D; Lagi, F; Lombardi, F; Maffeo, M; Magnani, G; Modica, S; Paolucci, S; Pecorari, M; Penco, G; Rossetti, B; Sacchini, D; Vicenti, I; Zazzi, M1
Andreoni, M; Cerva, C; Maffongelli, G; Malagnino, V; Sarmati, L; Teti, E1
Cortina-Borja, M; Peters, H; Rasi, V; Sconza, R; Thorne, C1
Allavena, C; Bani-Sadr, F; Bregigeon, S; Cabié, A; Cuzin, L; Ferry, T; Katlama, C; Lourenco, J; Pugliese, P; Rey, D; Reynes, J1
Cottrell, ML; Garcia, B; Imaz, A; Kashuba, ADM; Morenilla, S; Niubó, J; Perez, E; Podzamczer, D; Tiraboschi, JM1
Capetti, AF; Cossu, MV; Giacomet, V; Rizzardini, G; Zuccotti, G1
Fujiwara, T; Kawauchi-Miki, S; Miki, S; Seki, T; Yoshinaga, T1
Brown, SD; Cluck, DB; Duffourc, MM; Harirforoosh, S; Moorman, JP; Murrell, DE; Wang, KS1
Abdulghani, N; Ambrosioni, J; Casabona, J; Curran, A; Domingo, P; Force, L; Homar, F; Llibre, JM; Miró, JM; Montoliu, A; Peraire, J; Riera, M; Tiraboschi, J1
Antinori, A; Castagna, A; Costantini, A; Cozzi-Lepri, A; d'Arminio Monforte, A; Di Biagio, A; Gianotti, N; Lo Caputo, S; Marchetti, G; Mazzarello, G; Mazzotta, V; Rusconi, S1
Bugnon, S; Godinho, R; Gracin, T; Tataw, J1
Alfaro, J; Bogdanov, AA; Bolotin, E; Castillo, G; Gottikh, MB; Gupta, S; Leporati, A1
Abo, YN; Foster, C; Lyall, H; Mackie, N; Refsum, E; Tudor-Williams, G1
Baldelli, S; Cattaneo, D; Gervasoni, C; Ridolfo, A1
Beeker, N; Chouchana, L; Treluyer, JM1
Cassetti, I; Castillo, S; Cecchini, DM; Copertari, G; Lacal, V; Rodriguez, CG1
Ambrosioni, J; de Lazzari, E; García, F; Marcos, MÁ; Miró, JM; Mosquera, MM; Nicolás, D; Rico, JÁF1
Kaplun, O; Psevdos, G1
Alteri, C; Andreoni, M; Antinori, A; Bezenchek, A; Borghi, V; Cascio, A; De Luca, A; Di Carlo, D; Incardona, F; Perno, CF; Santoro, MM; Scutari, R; Vicenti, I; Zazzi, M; Zuccaro, V1
Conway-Washington, C; Dinh, C; Fountain, J; Haaland, RE; Hall, L; Holder, A; Kelley, CF; Livermont, T; Lupo, LD; Martin, A1
Abram, ME; Callebaut, C; Margot, NA; Ram, RR; White, KL1
Karmon, SL; Markowitz, M1
Abram, ME; Andreatta, KN; Barnes, TL; Chen, X; Goodman, DD; Hluhanich, RM; Margot, NA; McColl, DJ; Miller, MD; Niedziela-Majka, A; Novikov, N; Svarovskaia, ES; White, KL; Ye, L1
Bruce, RD; Custodio, JM; Friedland, GH; Kearney, BP; Ramanathan, S; Rhee, MS; Wei, LX; Winkle, P1
Aouri, M; Buclin, T; Calmy, A; Cavassini, M; Decosterd, LA; Hirschel, B; Rauch, A; Telenti, A1
Fransen, S; Frantzell, A; Huang, W; Petropoulos, CJ1
Burioni, R; Canducci, F; Castagna, A; Ceresola, ER; Clementi, M; Gianotti, N; Lazzarin, A; Saita, D; Underwood, M1
Chuck, SL; Conway, B; Cooper, D; Elion, R; Liu, YP; Maggiolo, F; Margot, N; Molina, JM; Ramón Arribas López, J; Rhee, M; Szwarcberg, J; Wilkins, E1
Aldir, I; Horta, A; Serrado, M1
Perry, CM1
Ait-Khaled, M; Castagna, A; Chas, J; Doroana, M; Durant, J; Grossberg, R; Huang, J; Maggiolo, F; Mills, A; Min, S; Molina, JM; Moreno, S; Nichols, G; Penco, G; Song, I; Vavro, C; Wright, D; Yeo, JM1
Doyon, G; Huber, K; McMahon, D; Mellors, JW; Sluis-Cremer, N; Sobolewski, MD1
Gupta, S; Jayaswal, A; Mishra, H; Shah, K; Sharma, PK1
Hsiao, CB; Ma, Q; Sawyer, JR1
Deeks, ED1
Abraham, T; Saad, N; Wu, G1
Reviriego, C1
Alcaro, S; Artese, A; Calvez, V; Ceccherini-Silberstein, F; Costa, G; Delelis, O; Gimferrer Arriaga, L; Katlama, C; Malet, I; Marcelin, AG; Parrotta, L; Tmeizeh, A; Valantin, MA1
Ayala-Sims, VA; Fulco, PP1
Buskin, SE; Collier, AC; Frenkel, LM; Holte, S; Maenza, J; McKernan, J; Milne, R; Mullins, JI; Mykhalchenko, K; Stekler, JD; Stevens, CE; Tapia, KA1
Debyser, Z; Schrijvers, R2
Arribas, JR; Di Perri, G; Ebrahimi, R; Gathe, J; Nguyen, T; Pialoux, G; Piontkowsky, D; Reynes, J; Tebas, P; White, K1
Antela, A; Domingo, P; Garner, W; Girard, PM; Guyer, B; Henry, K; Markowitz, M; Mills, A; Nguyen, T; Piontkowsky, D; Pozniak, A; Stellbrink, HJ; White, K1
Bruzzone, B; Di Biagio, A; Gustinetti, G; Prinapori, R; Sticchi, L; Taramasso, L; Viscoli, C1
Miller, MD; Raffi, F; White, KL1
Arendt, V; Lambert, C; Seguin-Devaux, C; Zheng, Y1
Cheng, AK; Kulkarni, R; McColl, DJ; Miller, MD; Rhee, MS; Szwarcberg, J; White, KL1
Chan, CN; Connick, E; Folkvord, JM; Lee, CS; Levy, DN; Luo, Y; Mahajan, S; Muesing, MA; Pham, M; Trinité, B1
Fujiwara, T; Garvey, EP; Johns, BA; Kawasuji, T; Kawauchi-Miki, S; Kobayashi, M; Miki, S; Sato, A; Seki, T; Suyama-Kagitani, A; Taishi, T; Underwood, MR; Wakasa-Morimoto, C; Yoshinaga, T1
Abram, ME; Andrade-Villanueva, JF; Beraud, C; Cheng, AK; Fisher, M; Graham, H; Liu, Y; Post, FA; Rhee, MS; Szwarcberg, J; Winston, J1
Fisher, M; Raffe, S1
Amiel, C; Barin, F; Bettinger, D; Calvez, V; Charpentier, C; Delaugerre, C; Descamps, D; Flandre, P; Fourati, S; Jeulin, H; Le Guillou-Guillemette, H; Maillard, A; Marcelin, AG; Mirand, A; Montès, B; Morand-Joubert, L; Nicot, F; Reigadas, S; Rodallec, A; Signori-Schmuck, A; Trabaud, MA; Vallet, S1
Harirforoosh, S; Moorman, JP; Murrell, DE1
Clotet, B; Llibre, JM1
Baeten, JM; Wyatt, C1
Andrade-Villanueva, J; Callebaut, C; Cao, H; Cheng, AK; Crofoot, G; Custodio, JM; DeJesus, E; Fordyce, MW; Koenig, E; Martin, H; McCallister, S; Molina, JM; Oka, S; Plummer, A; Podzamczer, D; Post, F; Pozniak, A; Saag, M; Sax, PE; Thompson, M; Trottier, B; Wohl, D; Yin, MT; Zhong, L1
Fulco, PP; Gomes, DC; Good, BL1
Stone, L1
Blume, M; Brodt, HR; de Leuw, P; Kann, G; Schüttfort, G; Stephan, C; Wolf, T1
Chung, S; Cosconati, S; Costi, R; Cuzzucoli Crucitti, G; Di Leva, FS; Di Santo, R; Le Grice, SF; Madia, VN; Marchand, C; Marinelli, L; Masoaka, T; Messore, A; Métifiot, M; Novellino, E; Pescatori, L; Pommier, Y; Pupo, G; Saccoliti, F; Scipione, L; Tortorella, S1
Blanco, JL; Milinkovic, A; Moyle, G; Whitlock, G1
Bender, R; Berenguer, J; Garner, W; Mills, A; Nguyen, T; Pozniak, A; Speck, RM1
Abadi, J; Dehority, W; Viani, RM; Wiznia, A1
Anstett, K; Liang, J; Mesplède, T; Oliveira, M; Wainberg, MA1
Gauthier, TP; Schafer, JJ; Sherman, EM; Unger, NR; Worley, MV1
Custodio, JM; Gordi, T; Ling, KH; Ramanathan, S; Zhong, L1
Holguín, Á; Llácer Delicado, T; Torrecilla, E1
Abram, ME; Arribas, JR; Avihingsanon, A; Benson, P; Bloch, M; Cheng, A; Chetchotisakd, P; Crofoot, G; Custodio, JM; Fordyce, MW; Gathe, J; Gupta, SK; Lichtenstein, K; McCallister, S; Post, FA; Pozniak, A; Ramgopal, M; SenGupta, D; Wei, X1
Bonora, S; Calcagno, A; Di Perri, G; Trentalange, A1
Trustman, N; Wong, E; Yalong, A1
Arribas, JR; Brinson, C; Brunetta, J; Callebaut, C; Cheng, A; Cheret, A; Clarke, A; Clumeck, N; Das, M; Fordyce, M; Mussini, C; Oka, S; Rashbaum, B; Sax, PE; Stephens, J; Tashima, K; Tebas, P; Wohl, D; Zhong, L1
Callebaut, C; Fordyce, M; Kitrinos, KM; Margot, NA; McCallister, S; Miller, MD1
Burger, D; Colbers, A; Greupink, R; Konopnicki, D; Russel, FG; Schalkwijk, S1
Bertucci, R; Bonora, S; Calcagno, A; D'Avolio, A; Di Perri, G; Mornese Pinna, S; Motta, I; Simiele, M1
Klein, D; Pinsky, BA; Shafer, RW; Smith, DS; Varghese, V1
Godbole, S; Paranjape, R; Pawar, J; Shete, A; Suryawanshi, P; Thakar, M1
Aouri, M; Barceló, C; Buclin, T; Cavassini, M; Csajka, C; Decosterd, LA; Gaspar, F; Guidi, M; Panchaud, A; Rotger, M1
Benson, P; Brinson, C; Brunetta, J; Cheng, A; Crofoot, G; Das, M; Fordyce, M; Gallant, J; Garner, W; McCallister, S; Mills, A; Oka, S1
Deeks, ED; Greig, SL1
Jones, R; Levy, JB; Milburn, J1
Behrens, G; Borg, P; Bouee, S; M Llibre, J; Moyle, G; Piontkowsky, D; Raffi, F; Reilly, G; Rogatto, F1
Amara, A; Back, D; Boffito, M; Challenger, E; Egan, D; Elliot, E; Else, L; Fawcett, S; Khoo, S; Penchala, SD1
Fletcher, CV; Podany, AT; Scarsi, KK1
Cattaneo, D; Gervasoni, C; Invernizzi, A; Micheli, V; Resnati, C; Riva, A1
Han, YS; Mesplède, T; Wainberg, MA1
Destache, CJ; Mandal, S; Prathipati, PK1
Deng, Z; Huang, X; Li, M; Luo, J; Qin, Z; Wang, B; Wang, H; You, J1
Avihingsanon, A; Cao, H; Cheng, A; Hagins, D; Hodder, S; Jiang, S; Johnson, M; Kityo, C; Koenig, E; Squires, K; Szwarcberg, J; Voronin, E; White, K1
Di Cristanziano, V; Esser, S; Heger, E; Jensen, B; Kaiser, R; Knops, E; Lübke, N; Pironti, A; Remmel, K; Theis, AA; Walter, H1
Batra, J; Chakraborty, R; Gaur, AH; Kizito, H; Kosalaraksa, P; Luesomboon, W; Myers, M; Porter, D; Prasitsueubsai, W; Quirk, E; Rakhmanina, N; Rassool, M; Rhee, MS; SenGupta, D; Shao, Y; Ting, L1
Childs-Kean, LM; Kisgen, JJ; Sherman, EM; Unger, NR; Worley, MV1
Boffito, M; Chirwa, M; Elliot, E1
Benmarzouk-Hidalgo, OJ; Espinosa, N; Fernandez-Magdaleno, T; Gutierrez-Valencia, A; Llaves, S; Lopez-Cortes, LF; Viciana, P1
Barin, F; Bernard, L; Capitao, M; Chaix, ML; Delaugerre, C; Maakaroun-Vermesse, Z; Néré, ML; Salmona, M; Splittgerber, M; Stefic, K1
Imaz, A; Podzamczer, D1
Destache, CJ; Fan, W; Kang, G; Li, Q; Mandal, S; Prathipati, PK; Yuan, Z; Zhou, Y1
Ambrosioni, J; Miró, JM; Mosquera, MM1
Blondel, L; Charpentier, C; Descamps, D; Joly, V; Landman, R; Lê, M; Matheron, S; Perrier, M; Peytavin, G; Pinto, A; Visseaux, B; Yazdanpanah, Y1
Kumar, S; Lukka, PB; Meibohm, B; Midde, NM; Sinha, N1
Arribas, JR; Callebaut, C; Cheng, A; Clarke, AE; Das, M; DeJesus, E; Guo, S; Haas, B; McCallister, S; McDonald, C; Plummer, A; Sax, PE; Thompson, M; Wang, H; Wohl, DA1
Tedaldi, EM1
Balzarini, J; Cecchetti, V; Daelemans, D; Fravolini, A; Manfroni, G; Massari, S; Pannecouque, C; Sabatini, S; Stevens, M; Tabarrini, O1
Bénard, A; Brun-Vézinet, F; Campa, P; Chêne, G; Collin, G; Damond, F; Descamps, D; Matheron, S; Peytavin, G; Roquebert, B1
Rondelez, E; Stuyver, LJ; Van Baelen, K; Van Eygen, V1
Grant, P; Zolopa, A1
Klibanov, OM1
Neamati, N; Odde, S; Ramkumar, K; Serrao, E1
Amellal, B; Calvez, V; Cissé, M; Delelis, O; Derache, A; Katlama, C; Koita, V; Maïga, AI; Malet, I; Marcelin, AG; Morand-Joubert, L; Mouscadet, JF; Murphy, R; Soulie, C; Tchertanov, L1
Alsina, M; Bennàssar, A; Guilabert, A; Mascaró, JM; Pintor, L1
Christ, F; Debyser, Z; McNeely, M; Thys, W1
Bellamy, R; Payne, B1
Ariën, K; Clynhens, M; Rondelez, E; Stuyver, LJ; Van Baelen, K; Van den Zegel, P; Van Eygen, V; Winters, B1
de Mendoza, C; Garrido, C; Soriano, V1
Abreu, P; Barbosa, JE; Batalha, PN; Bou-Habib, DC; Castro, HC; Cirne-Santos, CC; Cunha, AC; de Souza, MC; Ferreira, VF; Garrido, V; Giongo, V; Nogueira, CM; Paixão, IC; Rodrigues, CR; Santos, Fda C; Silva, Dde O; Simonetti, BR; Souza, TM; Temerozo, JR1
Fätkenheuer, G; Kümmerle, T; Lehmann, C; Meuer, K1
Schafer, JJ; Squires, KE1
Cooper, DA; Koelsch, KK1
Berger, DS; Cheng, AK; Chuck, SL; Enejosa, JV; Kearney, BP; Lampiris, H; Zhong, L; Zolopa, AR1
Fish, MQ; Hewer, R; Papathanasopoulos, MA; Stevens, WS; Venter, WD; Wallis, CL1
Anies, G; Breilh, D; da Silva, D; Dupon, M; Fleury, H; Masquelier, B; Morlat, P; Neau, D; Reigadas, S; Van Baelen, K; Van Wesenbeeck, L; Wittkop, L1
German, P; Hui, J; Kearney, BP; Warren, D; West, S1
Bottega, L; Cecchetti, V; Daelemans, D; Gatto, B; Manfroni, G; Massari, S; Meschini, F; Palumbo, M; Pannecouque, C; Tabarrini, O1
Aung, GL; Kawamoto, LS; O'Brien, JG; Tien, PG1
German, P; Kearney, BP; Mathias, AA; Ramanathan, S1
Chuck, SL; Cohen, C; DeJesus, E; Elion, R; Kearney, BP; Liu, HC; Ramanathan, S; Rashbaum, B; Ruane, P; Shamblaw, D; Warren, DR; Yale, K1
Chen, FE; Gu, SX; He, QQ; Liu, J; Wu, HQ; Yang, LM; Zhang, X; Zheng, YT1
Chimirri, A; De Luca, L; Debyzer, Z; Faliti, CE; Ferro, S; Gitto, R; Grazia, SD1
Debyser, Z; Desimmie, BA; Schrijvers, R1
Andrade-Villanueva, J; Cheng, AK; Chuck, SL; Clotet, B; Clumeck, N; Lamarca, A; Liu, YP; Margot, N; Molina, JM; Zhong, L1
Hughes, SH; Johnson, BC; Métifiot, M; Pommier, Y1
Lampiris, HW1
Andreatta, KN; Hluhanich, RM; Jones, GS; Margot, NA; McColl, DJ; Miller, MD; Tsiang, M; White, KL1
Vega, V; Wills, T1
Caballero, E; de Mendoza, C; Garcia, F; Garrido, C; Gutierrez, F; Pattery, T; Soriano, V; Van Houtte, M; Villacian, J; Zahonero, N1
Delaugerre, C; Nguyen, HL; Ruxrungtham, K1
Marchand, C1
Cheng, AK; DeJesus, E; Gathe, J; Henry, K; Kearney, BP; Molina, JM; Ramanathan, S; Rockstroh, JK; Szwarcberg, J; Wei, X; White, K; Yale, K1
Cheng, AK; Cohen, C; DeJesus, E; Gallant, JE; Kearney, BP; Liu, HC; Mills, A; Quirk, E; Sax, PE; Szwarcberg, J; White, K; Wohl, D; Yale, K; Zhong, L; Zolopa, A1
Bookstaver, PB; Rokas, KE; Shamroe, CL; Weissman, SB1
Lennox, JL1
Adams, JL; Greener, BN; Kashuba, AD1
Blanco, JL; Martinez-Picado, J1
Carr, A; Lee, FJ1
Pommer, P1
Klibanov, OM; Olin, JL; Spooner, LM1
Hussar, DA; Martinez, LN1
Breeze, S1
Morrow, T1
Temesgen, Z1
Raffi, F; Wainberg, MA1
Bourgeois, A; Caldwell, D; Newsom, D; Womack, S1
Abram, M; Cheng, AK; DeJesus, E; Fordyce, MW; Gathe, J; Henry, K; Molina, JM; Plummer, A; Ramanathan, S; Rockstroh, JK; Szwarcberg, J; Wei, X1
Cheng, AK; Cohen, C; DeJesus, E; Gallant, JE; Liu, HC; Mills, A; Plummer, A; Rhee, MS; Sax, PE; Szwarcberg, J; White, KL; Wohl, D; Zolopa, A1
Aïdara-Kane, A; Gassama-Sow, A; Guèye, M; Guèye-N'diaye, A; M'boup, S; Perret, JL; Sow, PS1
Antoniades, C; Knisely, A; Macdonald, C; Norris, S; Taylor, C1
Berger, D; Cheng, AK; Cohen, C; DeJesus, E; Elion, R; Farthing, C; Hawkins, T; Kearney, BP; Markowitz, M; McColl, D; Ruane, P; Zhong, L1
Aquaro, S; Balzarini, J; Cecchetti, V; De Clercq, E; Fravolini, A; Pannecouque, C; Perno, CF; Pollicita, M; Schols, D; Stevens, M; Tabarrini, O; Verbeken, E1
Correll, T; Klibanov, OM1
Miller, M1
Chaisson, RE; Moore, RD; Styrt, BA1
Cecchetti, V; Cruciani, G; Filipponi, E; Fravolini, A; Tabarrini, O1
Evans, TG; Riley, D1
Catalán, S; Chaves, F; de Rafael, L; Dronda, F1
Archambaud, M; Clavé, D; Massip, P; Moatti, N; Rouquet, RM1

Reviews

50 review(s) available for carbostyril and HIV Coinfection

ArticleYear
Meta-analysis and systematic review of the efficacy and resistance for human immunodeficiency virus type 1 integrase strand transfer inhibitors.
    International journal of antimicrobial agents, 2019, Volume: 54, Issue:5

    Topics: Amides; Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; Heterocyclic Compounds, 4 or More Rings; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Microbial Sensitivity Tests; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Virus Replication

2019
HIV-1 integrase strand transfer inhibitors: a review of current drugs, recent advances and drug resistance.
    International journal of antimicrobial agents, 2021, Volume: 57, Issue:5

    Topics: Amides; Anti-Retroviral Agents; Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Virus Replication

2021
A Review of the Efficacy and Safety of Genvoya® (Elvitegravir, Cobicistat, Emtricitabine, and Tenofovir Alafenamide) in the Management of HIV-1 Infection.
    Journal of pharmacy practice, 2018, Volume: 31, Issue:2

    Topics: Anti-HIV Agents; Clinical Trials, Phase III as Topic; Cobicistat; Diarrhea; Disease Management; Drug Combinations; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; Emtricitabine; Headache; HIV Infections; HIV-1; Humans; Nausea; Quinolones; Randomized Controlled Trials as Topic; Tenofovir; Treatment Outcome

2018
Cobicistat Versus Ritonavir: Similar Pharmacokinetic Enhancers But Some Important Differences.
    The Annals of pharmacotherapy, 2017, Volume: 51, Issue:11

    Topics: Anti-HIV Agents; Atazanavir Sulfate; Cobicistat; Darunavir; Drug Interactions; HIV Infections; Humans; Quinolones; Ritonavir

2017
Pharmacokinetics of HIV-Integrase Inhibitors During Pregnancy: Mechanisms, Clinical Implications and Knowledge Gaps.
    Clinical pharmacokinetics, 2019, Volume: 58, Issue:3

    Topics: Amides; Anti-Retroviral Agents; Female; Heterocyclic Compounds, 3-Ring; Heterocyclic Compounds, 4 or More Rings; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Infectious Disease Transmission, Vertical; Knowledge; Oxazines; Piperazines; Pregnancy; Pyridones; Quinolones; Raltegravir Potassium

2019
Clinical Impact of Virological Failure and Resistance Analysis Definitions used in Pivotal Clinical Trials of Initial Antiretroviral Treatment: A Systematic Review
    AIDS reviews, 2018, Volume: 20, Issue:3

    Topics: Amides; Anti-Retroviral Agents; Clinical Trials as Topic; Cobicistat; Darunavir; Drug Resistance, Viral; Genotype; Heterocyclic Compounds, 3-Ring; Heterocyclic Compounds, 4 or More Rings; HIV Infections; Humans; Oxazines; Piperazines; Pyridones; Quinolones; Rilpivirine; RNA, Viral; Triazoles; Viral Load

2018
A Review on Quinoline Derived Scaffolds as Anti-HIV Agents.
    Mini reviews in medicinal chemistry, 2019, Volume: 19, Issue:6

    Topics: Animals; Anti-HIV Agents; Drug Discovery; HIV; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; Humans; Models, Molecular; Quinolones

2019
An evaluation of elvitegravir plus cobicistat plus tenofovir alafenamide plus emtricitabine as a single-tablet regimen for the treatment of HIV in children and adolescents.
    Expert opinion on pharmacotherapy, 2019, Volume: 20, Issue:3

    Topics: Adenine; Adolescent; Alanine; Anti-HIV Agents; Child; Cobicistat; Emtricitabine; HIV Infections; Humans; Quinolones; Tablets; Tenofovir; United States; United States Food and Drug Administration

2019
Next-generation integrase inhibitors : where to after raltegravir?
    Drugs, 2013, Volume: 73, Issue:3

    Topics: Clinical Trials as Topic; Drug Discovery; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Oxazines; Piperazines; Pyridones; Pyrrolidinones; Quinolones; Raltegravir Potassium

2013
Single-tablet regimens in HIV: does it really make a difference?
    Current medical research and opinion, 2014, Volume: 30, Issue:1

    Topics: Adenine; Anti-HIV Agents; Carbamates; Cobicistat; Deoxycytidine; Drug Administration Schedule; Drug Combinations; Emtricitabine; HIV Infections; HIV-1; Humans; Nitriles; Organophosphonates; Pyrimidines; Quinolones; Reverse Transcriptase Inhibitors; Rilpivirine; Tablets; Tenofovir; Thiazoles

2014
Elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate single-tablet regimen (Stribild®): a review of its use in the management of HIV-1 infection in adults.
    Drugs, 2014, Volume: 74, Issue:1

    Topics: Adenine; Anti-HIV Agents; Carbamates; Deoxycytidine; Drug Combinations; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV Infections; HIV-1; Humans; Organophosphonates; Quinolones; Tablets; Thiazoles

2014
Elvitegravir: a review of its use in adults with HIV-1 infection.
    Drugs, 2014, Volume: 74, Issue:6

    Topics: Adult; Drug Administration Schedule; Drug Resistance, Viral; Drug Therapy, Combination; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Quinolones

2014
Dolutegravir for the treatment of adult patients with HIV-1 infection.
    Expert review of anti-infective therapy, 2014, Volume: 12, Issue:5

    Topics: Adult; Clinical Trials as Topic; Dideoxynucleosides; Drug Administration Schedule; Drug Combinations; Drug Interactions; Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Lamivudine; Oxazines; Piperazines; Pyridones; Pyrrolidinones; Quinolones; Raltegravir Potassium

2014
Which patients have greatest need for elvitegravir/cobicistat/ emtricitabine/tenofovirDF-based therapy?
    Recent patents on anti-infective drug discovery, 2014, Volume: 9, Issue:1

    Topics: Adenine; Anti-HIV Agents; Carbamates; Cobicistat; Deoxycytidine; Drug Combinations; Emtricitabine; HIV Infections; HIV-1; Humans; Patents as Topic; Phosphorous Acids; Quinolones; Thiazoles

2014
Resistance analyses of integrase strand transfer inhibitors within phase 3 clinical trials of treatment-naive patients.
    Viruses, 2014, Jul-22, Volume: 6, Issue:7

    Topics: Clinical Trials, Phase III as Topic; Drug Resistance, Viral; Drug Therapy, Combination; Endpoint Determination; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Male; Oxazines; Piperazines; Pyridones; Pyrrolidinones; Quinolones; Raltegravir Potassium; Treatment Outcome; Viral Load

2014
The pharmacokinetics, pharmacodynamics and clinical efficacy of elvitegravir + cobicistat + emtricitabine + tenofovir combination therapy for the treatment of HIV.
    Expert opinion on drug metabolism & toxicology, 2015, Volume: 11, Issue:3

    Topics: Adenine; Adult; Anti-HIV Agents; Carbamates; Deoxycytidine; Drug Approval; Drug Combinations; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; European Union; HIV Infections; HIV-1; Humans; Organophosphonates; Quinolones; Tablets; Thiazoles

2015
Stribild: a review of component characteristics and combination drug efficacy.
    European review for medical and pharmacological sciences, 2015, Volume: 19, Issue:5

    Topics: Adenine; Anti-HIV Agents; Carbamates; Deoxycytidine; Drug Combinations; Drug Synergism; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV Infections; Humans; Organophosphonates; Quinolones; Thiazoles

2015
[Resistance profile and genetic barrier of dolutegravir].
    Enfermedades infecciosas y microbiologia clinica, 2015, Volume: 33 Suppl 1

    Topics: Amino Acid Substitution; Clinical Trials as Topic; Drug Resistance, Multiple, Viral; Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Mutation, Missense; Oxazines; Piperazines; Point Mutation; Pyridones; Quinolones; Raltegravir Potassium; Virus Replication

2015
HIV integrase inhibitors: a new era in the treatment of HIV.
    Expert opinion on pharmacotherapy, 2015, Volume: 16, Issue:9

    Topics: Clinical Trials as Topic; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Oxazines; Piperazines; Pyridones; Pyrrolidinones; Quinolones; Raltegravir Potassium

2015
Use of Integrase Inhibitors in HIV-Infected Children and Adolescents.
    Drugs, 2015, Volume: 75, Issue:13

    Topics: Adolescent; Adult; Age Factors; Child; Drug Approval; Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium

2015
Cobicistat: Review of a Pharmacokinetic Enhancer for HIV Infection.
    Clinical therapeutics, 2015, Sep-01, Volume: 37, Issue:9

    Topics: Anti-HIV Agents; Cobicistat; Cytochrome P-450 CYP3A Inhibitors; Darunavir; Drug Interactions; Drug Therapy, Combination; HIV Infections; HIV-1; Humans; Quinolones

2015
Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide for the treatment of HIV in adults.
    Expert opinion on pharmacotherapy, 2016, Volume: 17, Issue:3

    Topics: Anti-HIV Agents; Bone Density; Clinical Trials as Topic; Cobicistat; Drug Combinations; Drug Resistance, Viral; Emtricitabine; HIV Infections; Humans; Quinolones; Tablets; Tenofovir

2016
HIV pharmacotherapy: A review of integrase inhibitors.
    JAAPA : official journal of the American Academy of Physician Assistants, 2016, Volume: 29, Issue:2

    Topics: Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Randomized Controlled Trials as Topic

2016
Elvitegravir/Cobicistat/Emtricitabine/Tenofovir Alafenamide: A Review in HIV-1 Infection.
    Drugs, 2016, Volume: 76, Issue:9

    Topics: Adenine; Adolescent; Adult; Alanine; Anti-HIV Agents; Clinical Trials, Phase III as Topic; Cobicistat; Drug Combinations; Emtricitabine; HIV Infections; HIV-1; Humans; Quinolones; Randomized Controlled Trials as Topic; Reverse Transcriptase Inhibitors; Tenofovir

2016
Renal effects of novel antiretroviral drugs.
    Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association, 2017, 03-01, Volume: 32, Issue:3

    Topics: Adenine; Alanine; Anti-HIV Agents; Atazanavir Sulfate; Cobicistat; Creatinine; Disease Progression; Heterocyclic Compounds, 3-Ring; HIV Infections; Humans; Oxazines; Piperazines; Proteinuria; Pyridones; Quinolones; Raltegravir Potassium; Renal Insufficiency, Chronic; Tenofovir

2017
Comparative Clinical Pharmacokinetics and Pharmacodynamics of HIV-1 Integrase Strand Transfer Inhibitors.
    Clinical pharmacokinetics, 2017, Volume: 56, Issue:1

    Topics: Anti-Retroviral Agents; Area Under Curve; Coinfection; Cytochrome P-450 CYP3A; Drug Combinations; Drug Interactions; Female; Half-Life; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; Humans; Liver Failure; Metabolic Clearance Rate; Oxazines; Piperazines; Pregnancy; Protein Binding; Pyridones; Quinolones; Raltegravir Potassium; Renal Insufficiency

2017
Differences among HIV-1 subtypes in drug resistance against integrase inhibitors.
    Infection, genetics and evolution : journal of molecular epidemiology and evolutionary genetics in infectious diseases, 2016, Volume: 46

    Topics: Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium

2016
Therapy-Emergent Drug Resistance to Integrase Strand Transfer Inhibitors in HIV-1 Patients: A Subgroup Meta-Analysis of Clinical Trials.
    PloS one, 2016, Volume: 11, Issue:8

    Topics: Clinical Trials as Topic; Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Virus Replication

2016
Elvitegravir for the treatment of HIV.
    Expert opinion on pharmacotherapy, 2016, Volume: 17, Issue:17

    Topics: Anti-HIV Agents; Clinical Trials as Topic; Cobicistat; Cytochrome P-450 CYP3A Inhibitors; Drug Interactions; Drug Therapy, Combination; HIV Infections; HIV-1; Humans; Quinolones; Ritonavir; Treatment Outcome

2016
How recent findings on the pharmacokinetics and pharmacodynamics of integrase inhibitors can inform clinical use.
    Current opinion in infectious diseases, 2017, Volume: 30, Issue:1

    Topics: Cobicistat; Drug Interactions; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Viral Load

2017
Emerging therapies for hepatitis C and HIV in drug abusers: drugs and strategies.
    Journal of addictive diseases, 2008, Volume: 27, Issue:2

    Topics: Anti-Retroviral Agents; Antiviral Agents; Comorbidity; Hepatitis C, Chronic; HIV Infections; Humans; Pyrimidine Nucleosides; Pyrrolidinones; Quinolones; Raltegravir Potassium; Substance Abuse, Intravenous

2008
Integrase inhibitors: a clinical review of raltegravir and elvitegravir.
    Journal of HIV therapy, 2008, Volume: 13, Issue:2

    Topics: Clinical Trials, Phase III as Topic; Dose-Response Relationship, Drug; Drug Interactions; Drug Resistance, Viral; Drug Therapy, Combination; HIV; HIV Infections; HIV Integrase; HIV Protease Inhibitors; Humans; Pyrrolidinones; Quinolones; Raltegravir Potassium

2008
Raltegravir, elvitegravir, and metoogravir: the birth of "me-too" HIV-1 integrase inhibitors.
    Retrovirology, 2009, Mar-05, Volume: 6

    Topics: Antiviral Agents; Drug Discovery; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Pyrrolidinones; Quinolones; Raltegravir Potassium

2009
Targeting the HIV integration process in antiviral therapy.
    Journal of HIV therapy, 2008, Volume: 13, Issue:4

    Topics: HIV; HIV Infections; HIV Integrase Inhibitors; Humans; Pyrrolidinones; Quinolones; Raltegravir Potassium; Virus Integration

2008
Tuberculosis in people with HIV.
    BMJ clinical evidence, 2007, Jun-01, Volume: 2007

    Topics: Disease Progression; HIV Infections; Humans; Meta-Analysis as Topic; Quinolones; Survival Analysis; Time Factors; Tuberculosis; United States Food and Drug Administration

2007
[Resistance to integrase inhibitors].
    Enfermedades infecciosas y microbiologia clinica, 2008, Volume: 26 Suppl 12

    Topics: Amino Acid Substitution; Clinical Trials as Topic; Drug Resistance, Multiple, Viral; Drug Resistance, Viral; Genetic Variation; HIV; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; Humans; Models, Molecular; Mutation, Missense; Point Mutation; Protein Conformation; Pyrrolidinones; Quinolones; Raltegravir Potassium

2008
Integrase inhibitors: a novel class of antiretroviral agents.
    The Annals of pharmacotherapy, 2010, Volume: 44, Issue:1

    Topics: Anti-HIV Agents; HIV Infections; Humans; Integrase Inhibitors; Pyrrolidinones; Quinolones; Raltegravir Potassium

2010
Integrase inhibitors in salvage therapy regimens for HIV-1 infection.
    Current opinion in HIV and AIDS, 2009, Volume: 4, Issue:6

    Topics: HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Quinolones; Salvage Therapy

2009
Clinical pharmacokinetic and pharmacodynamic profile of the HIV integrase inhibitor elvitegravir.
    Clinical pharmacokinetics, 2011, Volume: 50, Issue:4

    Topics: Animals; Drug Interactions; Drug Therapy, Combination; HIV Infections; HIV Integrase Inhibitors; Humans; Quinolones

2011
Elvitegravir: a once-daily, boosted, HIV-1 integrase inhibitor.
    Expert review of anti-infective therapy, 2012, Volume: 10, Issue:1

    Topics: Adenine; Carbamates; Clinical Trials, Phase I as Topic; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Deoxycytidine; Drug Combinations; Drug Interactions; Drug Resistance, Viral; Drug-Related Side Effects and Adverse Reactions; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Organophosphonates; Quinolones; Randomized Controlled Trials as Topic; Thiazoles

2012
Elvitegravir: a once-daily inhibitor of HIV-1 integrase.
    Expert opinion on investigational drugs, 2012, Volume: 21, Issue:3

    Topics: Anti-HIV Agents; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Drug Administration Schedule; Drug Combinations; Drug Resistance, Viral; Drug Therapy, Combination; HIV Infections; HIV Integrase Inhibitors; Humans; Quinolones

2012
Update on raltegravir and the development of new integrase strand transfer inhibitors.
    Southern medical journal, 2012, Volume: 105, Issue:7

    Topics: Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Oxazines; Piperazines; Pyridones; Pyrrolidinones; Quinolones; Raltegravir Potassium

2012
The use of HIV-1 integrase inhibitors in antiretroviral naive patients.
    Current opinion in HIV and AIDS, 2012, Volume: 7, Issue:5

    Topics: Antiretroviral Therapy, Highly Active; Clinical Trials as Topic; Coinfection; Hepatitis C; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Oxazines; Piperazines; Pyridones; Pyrrolidinones; Quinolones; Raltegravir Potassium; Treatment Outcome

2012
Pharmacology of HIV integrase inhibitors.
    Current opinion in HIV and AIDS, 2012, Volume: 7, Issue:5

    Topics: Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Oxazines; Piperazines; Pyridones; Pyrrolidinones; Quinolones; Raltegravir Potassium; United States

2012
Combinational therapies for HIV: a focus on EVG/COBI/FTC/TDF.
    Expert opinion on pharmacotherapy, 2012, Volume: 13, Issue:13

    Topics: Adenine; Anti-HIV Agents; Carbamates; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Cobicistat; Deoxycytidine; Drug Combinations; Drug Resistance, Multiple, Viral; Emtricitabine; HIV Infections; Humans; Organophosphonates; Quinolones; Tenofovir; Thiazoles

2012
HIV integrase inhibitors in ART-experienced patients.
    Current opinion in HIV and AIDS, 2012, Volume: 7, Issue:5

    Topics: Antiretroviral Therapy, Highly Active; Clinical Trials as Topic; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Oxazines; Piperazines; Pyridones; Pyrrolidinones; Quinolones; Raltegravir Potassium; Salvage Therapy; Treatment Outcome

2012
Tolerability of HIV integrase inhibitors.
    Current opinion in HIV and AIDS, 2012, Volume: 7, Issue:5

    Topics: Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Drug-Related Side Effects and Adverse Reactions; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Kidney; Lipid Metabolism; Oxazines; Piperazines; Pyridones; Pyrrolidinones; Quinolones; Raltegravir Potassium

2012
Elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate single tablet for HIV-1 infection treatment.
    The Annals of pharmacotherapy, 2012, Volume: 46, Issue:12

    Topics: Adenine; Anti-HIV Agents; Carbamates; Clinical Trials, Phase III as Topic; Deoxycytidine; Drug Combinations; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV Infections; HIV Integrase Inhibitors; Humans; Organophosphonates; Quinolones; Tablets; Thiazoles; Viral Load

2012
Cobicistat-boosted elvitegravir-based fixed-dose combination antiretroviral therapy for HIV infection.
    Drugs of today (Barcelona, Spain : 1998), 2012, Volume: 48, Issue:12

    Topics: Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Carbamates; Cobicistat; Drug Approval; Drug Combinations; Drug Interactions; Drug Resistance, Viral; HIV Infections; HIV Integrase Inhibitors; Humans; Patient Safety; Quinolones; Thiazoles

2012
Integrase inhibitors: a new treatment option for patients with human immunodeficiency virus infection.
    Pharmacotherapy, 2008, Volume: 28, Issue:1

    Topics: Dose-Response Relationship, Drug; HIV Infections; HIV Integrase Inhibitors; Humans; Organic Chemicals; Pyrrolidinones; Quinolones; Raltegravir Potassium; Randomized Controlled Trials as Topic

2008

Trials

38 trial(s) available for carbostyril and HIV Coinfection

ArticleYear
Safety and efficacy of elvitegravir, dolutegravir, and raltegravir in a real-world cohort of treatment-naïve and -experienced patients.
    Medicine, 2019, Volume: 98, Issue:32

    Topics: Adult; Aged; Anti-Retroviral Agents; Antiretroviral Therapy, Highly Active; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Male; Middle Aged; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Retrospective Studies; Viral Load; Young Adult

2019
Bone mineral density in virologically suppressed people aged 60 years or older with HIV-1 switching from a regimen containing tenofovir disoproxil fumarate to an elvitegravir, cobicistat, emtricitabine, and tenofovir alafenamide single-tablet regimen: a m
    The lancet. HIV, 2019, Volume: 6, Issue:10

    Topics: Adenine; Aged; Aged, 80 and over; Alanine; Anti-HIV Agents; Bone Density; Cobicistat; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Middle Aged; Quinolones; Tablets; Tenofovir

2019
Elvitegravir-Cobicistat-Emtricitabine-Tenofovir Alafenamide Single-tablet Regimen for Human Immunodeficiency Virus Postexposure Prophylaxis.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2020, 02-14, Volume: 70, Issue:5

    Topics: Adenine; Alanine; Anti-HIV Agents; Cobicistat; Drug Combinations; Emtricitabine; HIV Infections; HIV-1; Humans; Quinolones; Tablets; Tenofovir

2020
Switching to the single-tablet regimen of elvitegravir, cobicistat, emtricitabine, and tenofovir DF from non-nucleoside reverse transcriptase inhibitor plus coformulated emtricitabine and tenofovir DF regimens: Week 96 results of STRATEGY-NNRTI.
    HIV clinical trials, 2017, Volume: 18, Issue:4

    Topics: Adult; Antiretroviral Therapy, Highly Active; Cobicistat; Drug Combinations; Drug Substitution; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Patient Reported Outcome Measures; Quinolones; Tablets; Tenofovir; Time Factors; Treatment Outcome

2017
Week 48 resistance analysis of Elvitegravir/Cobicistat/Emtricitabine/Tenofovir DF versus Atazanavir + Ritonavir + Emtricitabine/Tenofovir DF in HIV-1 infected women (WAVES study GS-US-236-0128).
    HIV clinical trials, 2017, Volume: 18, Issue:4

    Topics: Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Cobicistat; Drug Resistance, Viral; Emtricitabine; Female; Genotype; HIV Infections; HIV-1; Humans; Microbial Sensitivity Tests; Mutation; Quinolones; Sequence Analysis, DNA; Tenofovir; Time Factors; Treatment Failure; Treatment Outcome; Viral Load

2017
Tenofovir disoproxil fumarate/emtricitabine plus ritonavir-boosted lopinavir or cobicistat-boosted elvitegravir as a single-tablet regimen for HIV post-exposure prophylaxis.
    The Journal of antimicrobial chemotherapy, 2017, 10-01, Volume: 72, Issue:10

    Topics: Adult; Anti-HIV Agents; Cobicistat; Drug Therapy, Combination; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Lopinavir; Male; Medication Adherence; Post-Exposure Prophylaxis; Prospective Studies; Quinolones; Reverse Transcriptase Inhibitors; Ritonavir; Tablets; Tenofovir

2017
HIV treatment simplification to elvitegravir/cobicistat/emtricitabine/tenofovir disproxil fumarate (E/C/F/TDF) plus darunavir: a pharmacokinetic study.
    AIDS research and therapy, 2017, Nov-02, Volume: 14, Issue:1

    Topics: Adult; Aged; Anti-HIV Agents; Cobicistat; Darunavir; Drug Therapy, Combination; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Integrase Inhibitors; Male; Middle Aged; Protease Inhibitors; Quinolones; Reverse Transcriptase Inhibitors; Ritonavir; Tenofovir; Viral Load

2017
Superior Efficacy and Improved Renal and Bone Safety After Switching from a Tenofovir Disoproxil Fumarate- to a Tenofovir Alafenamide-Based Regimen Through 96 Weeks of Treatment.
    AIDS research and human retroviruses, 2018, Volume: 34, Issue:4

    Topics: Adenine; Alanine; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Bone Density; Cobicistat; Drug Combinations; Drug Substitution; Emtricitabine; HIV Infections; HIV-1; Humans; Kidney; Quinolones; RNA, Viral; Tenofovir; Treatment Outcome

2018
Brief Report: Efficacy and Safety of Switching to Coformulated Elvitegravir, Cobicistat, Emtricitabine, and Tenofovir Alafenamide (E/C/F/TAF) in Virologically Suppressed Women.
    Journal of acquired immune deficiency syndromes (1999), 2018, 06-01, Volume: 78, Issue:2

    Topics: Adenine; Adult; Alanine; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Cobicistat; Double-Blind Method; Drug Combinations; Drug Resistance, Viral; Drug-Related Side Effects and Adverse Reactions; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Integrase Inhibitors; Protease Inhibitors; Quinolones; RNA, Viral; Tenofovir

2018
Elvitegravir/cobicistat pharmacokinetics in pregnant and postpartum women with HIV.
    AIDS (London, England), 2018, 11-13, Volume: 32, Issue:17

    Topics: Administration, Oral; Adult; Anti-HIV Agents; Chromatography, Liquid; Cobicistat; Female; HIV Infections; Humans; Infant, Newborn; Middle Aged; Plasma; Postpartum Period; Pregnancy; Pregnancy Complications, Infectious; Prospective Studies; Quinolones; Tandem Mass Spectrometry; United States; Young Adult

2018
Seminal Tenofovir Concentrations, Viral Suppression, and Semen Quality With Tenofovir Alafenamide, Compared With Tenofovir Disoproxil Fumarate (Spanish HIV/AIDS Research Network, PreEC/RIS 40).
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2019, 09-27, Volume: 69, Issue:8

    Topics: Adenine; Adult; Alanine; Anti-Retroviral Agents; Cobicistat; Emtricitabine; HIV Infections; HIV-1; Humans; Male; Middle Aged; Prospective Studies; Quinolones; RNA, Viral; Semen; Semen Analysis; Tenofovir

2019
A randomized phase 3 study comparing once-daily elvitegravir with twice-daily raltegravir in treatment-experienced subjects with HIV-1 infection: 96-week results.
    Journal of acquired immune deficiency syndromes (1999), 2013, Aug-01, Volume: 63, Issue:4

    Topics: Double-Blind Method; Drug Resistance, Viral; Drug Therapy, Combination; HIV Infections; HIV Integrase Inhibitors; HIV Protease Inhibitors; HIV-1; Humans; Longitudinal Studies; Pyrrolidinones; Quinolones; Raltegravir Potassium; Ritonavir; RNA, Viral; Viral Load

2013
Dolutegravir in antiretroviral-experienced patients with raltegravir- and/or elvitegravir-resistant HIV-1: 24-week results of the phase III VIKING-3 study.
    The Journal of infectious diseases, 2014, Aug-01, Volume: 210, Issue:3

    Topics: Adult; Anti-HIV Agents; Drug Resistance, Viral; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV-1; Humans; Male; Middle Aged; Oxazines; Pilot Projects; Piperazines; Pyridones; Pyrrolidinones; Quinolones; Raltegravir Potassium; RNA, Viral; Viral Load

2014
Simplification to coformulated elvitegravir, cobicistat, emtricitabine, and tenofovir versus continuation of ritonavir-boosted protease inhibitor with emtricitabine and tenofovir in adults with virologically suppressed HIV (STRATEGY-PI): 48 week results o
    The Lancet. Infectious diseases, 2014, Volume: 14, Issue:7

    Topics: Adenine; Adult; Anti-HIV Agents; Carbamates; Cobicistat; Deoxycytidine; Drug Therapy, Combination; Emtricitabine; Female; HIV; HIV Infections; Humans; Male; Middle Aged; Organophosphonates; Protease Inhibitors; Quinolones; Ritonavir; Tenofovir; Thiazoles; Viral Load

2014
Switching to coformulated elvitegravir, cobicistat, emtricitabine, and tenofovir versus continuation of non-nucleoside reverse transcriptase inhibitor with emtricitabine and tenofovir in virologically suppressed adults with HIV (STRATEGY-NNRTI): 48 week r
    The Lancet. Infectious diseases, 2014, Volume: 14, Issue:7

    Topics: Adenine; Adult; Anti-HIV Agents; Carbamates; Cobicistat; Deoxycytidine; Emtricitabine; Female; HIV; HIV Infections; Humans; Male; Middle Aged; Organophosphonates; Quinolones; Reverse Transcriptase Inhibitors; Tenofovir; Thiazoles; Viral Load

2014
Week 144 resistance analysis of elvitegravir/cobicistat/emtricitabine/tenofovir DF versus efavirenz/emtricitabine/tenofovir DF in antiretroviral-naive patients.
    Antiviral therapy, 2015, Volume: 20, Issue:3

    Topics: Alkynes; Antiretroviral Therapy, Highly Active; Benzoxazines; Cobicistat; Cyclopropanes; Drug Resistance, Viral; Emtricitabine; Female; Genotype; HIV Infections; HIV-1; Humans; Male; Microbial Sensitivity Tests; Mutation; Quinolones; Tenofovir; Time Factors; Treatment Outcome; Viral Load

2015
Tenofovir alafenamide versus tenofovir disoproxil fumarate, coformulated with elvitegravir, cobicistat, and emtricitabine, for initial treatment of HIV-1 infection: two randomised, double-blind, phase 3, non-inferiority trials.
    Lancet (London, England), 2015, Jun-27, Volume: 385, Issue:9987

    Topics: Adenine; Adult; Alanine; Anti-HIV Agents; Arthralgia; Bone Density; Carbamates; CD4 Lymphocyte Count; Cobicistat; Deoxycytidine; Double-Blind Method; Drug Combinations; Emtricitabine; Female; Headache; HIV Infections; Humans; Kidney; Male; Nausea; Organophosphonates; Quinolones; Respiration Disorders; Sleep Initiation and Maintenance Disorders; Tenofovir; Thiazoles; Treatment Outcome; Viral Load

2015
Patient-Reported Symptoms Over 48 Weeks in a Randomized, Open-Label, Phase IIIb Non-Inferiority Trial of Adults with HIV Switching to Co-Formulated Elvitegravir, Cobicistat, Emtricitabine, and Tenofovir DF versus Continuation of Non-Nucleoside Reverse Tra
    The patient, 2015, Volume: 8, Issue:4

    Topics: Adult; Anti-HIV Agents; Cobicistat; Drug Combinations; Emtricitabine; Female; HIV Infections; Humans; Male; Middle Aged; Patient Outcome Assessment; Quality of Life; Quinolones; Tenofovir

2015
Population Pharmacokinetics of Boosted-Elvitegravir in HIV-Infected Patients.
    Journal of clinical pharmacology, 2016, Volume: 56, Issue:6

    Topics: Adolescent; Adult; Aged; Anti-HIV Agents; Child; Drug Therapy, Combination; Female; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; Humans; Male; Middle Aged; Quinolones; Young Adult

2016
Switching to Tenofovir Alafenamide, Coformulated With Elvitegravir, Cobicistat, and Emtricitabine, in HIV-Infected Patients With Renal Impairment: 48-Week Results From a Single-Arm, Multicenter, Open-Label Phase 3 Study.
    Journal of acquired immune deficiency syndromes (1999), 2016, Apr-15, Volume: 71, Issue:5

    Topics: Adult; Albuminuria; Bone Density; Cobicistat; Drug Substitution; Drug Therapy, Combination; Emtricitabine; Female; Glomerular Filtration Rate; HIV Infections; Humans; Male; Middle Aged; Proteinuria; Quinolones; Renal Insufficiency; Tenofovir

2016
Brief Report: A Randomized, Double-Blind Comparison of Tenofovir Alafenamide Versus Tenofovir Disoproxil Fumarate, Each Coformulated With Elvitegravir, Cobicistat, and Emtricitabine for Initial HIV-1 Treatment: Week 96 Results.
    Journal of acquired immune deficiency syndromes (1999), 2016, May-01, Volume: 72, Issue:1

    Topics: Adenine; Alanine; Albuminuria; Anti-HIV Agents; Bone Density; CD4 Lymphocyte Count; Cobicistat; Double-Blind Method; Drug Combinations; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Proteinuria; Quinolones; RNA, Viral; Tenofovir

2016
Rare emergence of drug resistance in HIV-1 treatment-naïve patients after 48 weeks of treatment with elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide.
    HIV clinical trials, 2016, Volume: 17, Issue:2

    Topics: Adenine; Adult; Alanine; Anti-HIV Agents; CD4 Lymphocyte Count; Cobicistat; Drug Resistance, Viral; Drug Therapy, Combination; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Middle Aged; Quinolones; Tenofovir; Young Adult

2016
Brief Report: Efficacy and Safety of Switching to a Single-Tablet Regimen of Elvitegravir/Cobicistat/Emtricitabine/Tenofovir Alafenamide in HIV-1/Hepatitis B-Coinfected Adults.
    Journal of acquired immune deficiency syndromes (1999), 2016, 11-01, Volume: 73, Issue:3

    Topics: Adenine; Alanine; Anti-HIV Agents; Cobicistat; Coinfection; Drug Combinations; Drug Substitution; Emtricitabine; Female; Hepatitis B; HIV Infections; Humans; Male; Middle Aged; Quinolones; Tenofovir; Treatment Outcome

2016
An Indirect Comparison of Efficacy and Safety of Elvitegravir/Cobicistat/Emtricitabine/Tenofovir Disoproxil Fumarate and Abacavir/Lamivudine + Dolutegravir in Initial Therapy.
    PloS one, 2016, Volume: 11, Issue:5

    Topics: Adult; Algorithms; Anti-HIV Agents; Cobicistat; Dideoxynucleosides; Drug Combinations; Emtricitabine; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV-1; Humans; Lamivudine; Male; Oxazines; Patient Safety; Piperazines; Pyridones; Quinolones; Risk; Tenofovir

2016
Integrase inhibitor versus protease inhibitor based regimen for HIV-1 infected women (WAVES): a randomised, controlled, double-blind, phase 3 study.
    The lancet. HIV, 2016, Volume: 3, Issue:9

    Topics: Adult; Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; Cobicistat; Double-Blind Method; Emtricitabine; Female; HIV Infections; HIV Integrase Inhibitors; HIV Protease Inhibitors; Humans; International Cooperation; Quinolones; Ritonavir; RNA, Viral; Tenofovir; Viral Load

2016
Safety, efficacy, and pharmacokinetics of a single-tablet regimen containing elvitegravir, cobicistat, emtricitabine, and tenofovir alafenamide in treatment-naive, HIV-infected adolescents: a single-arm, open-label trial.
    The lancet. HIV, 2016, Volume: 3, Issue:12

    Topics: Adenine; Adolescent; Alanine; Anti-HIV Agents; Area Under Curve; CD4 Lymphocyte Count; Child; Cobicistat; Drug Therapy, Combination; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Lost to Follow-Up; Male; Quinolones; RNA, Viral; South Africa; Tablets; Tenofovir; Thailand; Uganda; United States; Viral Load

2016
Switch as maintenance to elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate: week 48 results in a clinical cohort.
    The Journal of antimicrobial chemotherapy, 2017, 06-01, Volume: 72, Issue:6

    Topics: Adult; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; CD4 Lymphocyte Count; Cobicistat; Cohort Studies; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Maintenance Chemotherapy; Male; Middle Aged; Polymerase Chain Reaction; Quinolones; RNA, Viral; Tablets; Tenofovir; Viral Load; Viremia

2017
Brief Report: Randomized, Double-Blind Comparison of Tenofovir Alafenamide (TAF) vs Tenofovir Disoproxil Fumarate (TDF), Each Coformulated With Elvitegravir, Cobicistat, and Emtricitabine (E/C/F) for Initial HIV-1 Treatment: Week 144 Results.
    Journal of acquired immune deficiency syndromes (1999), 2017, 06-01, Volume: 75, Issue:2

    Topics: Adenine; Alanine; Anti-HIV Agents; Bone Density; CD4 Lymphocyte Count; Cobicistat; Double-Blind Method; Emtricitabine; HIV Infections; Humans; Middle Aged; Quinolones; Tenofovir; Treatment Outcome; United States

2017
Phase III trial begins for elvitegravir.
    AIDS patient care and STDs, 2008, Volume: 22, Issue:9

    Topics: Double-Blind Method; HIV Infections; HIV Integrase Inhibitors; Humans; Quinolones; Viral Load

2008
Activity of elvitegravir, a once-daily integrase inhibitor, against resistant HIV Type 1: results of a phase 2, randomized, controlled, dose-ranging clinical trial.
    The Journal of infectious diseases, 2010, Mar-15, Volume: 201, Issue:6

    Topics: Adolescent; Adult; Aged; CD4 Lymphocyte Count; Darunavir; Drug Resistance, Viral; Drug Therapy, Combination; Female; HIV Infections; HIV Integrase Inhibitors; HIV Protease Inhibitors; HIV-1; Humans; Male; Middle Aged; Pyridines; Pyrones; Quinolones; Ritonavir; RNA, Viral; Sulfonamides; Treatment Outcome; Young Adult

2010
Pharmacokinetics and bioavailability of an integrase and novel pharmacoenhancer-containing single-tablet fixed-dose combination regimen for the treatment of HIV.
    Journal of acquired immune deficiency syndromes (1999), 2010, Volume: 55, Issue:3

    Topics: Adenine; Administration, Oral; Adult; Anti-HIV Agents; Biological Availability; Deoxycytidine; Drug Combinations; Emtricitabine; Female; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; Humans; Male; Organophosphonates; Plasma; Quinolones; Tablets; Tenofovir

2010
Randomized, phase 2 evaluation of two single-tablet regimens elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate versus efavirenz/emtricitabine/tenofovir disoproxil fumarate for the initial treatment of HIV infection.
    AIDS (London, England), 2011, Mar-27, Volume: 25, Issue:6

    Topics: Adenine; Adult; Alkynes; Anti-HIV Agents; Benzoxazines; Carbamates; CD4 Lymphocyte Count; Cobicistat; Cyclopropanes; Deoxycytidine; Drug Combinations; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Organophosphonates; Patient Compliance; Patient Selection; Quinolones; Tenofovir; Thiazoles; Treatment Outcome

2011
Efficacy and safety of once daily elvitegravir versus twice daily raltegravir in treatment-experienced patients with HIV-1 receiving a ritonavir-boosted protease inhibitor: randomised, double-blind, phase 3, non-inferiority study.
    The Lancet. Infectious diseases, 2012, Volume: 12, Issue:1

    Topics: Adult; Alanine Transaminase; Anti-Retroviral Agents; Aspartate Aminotransferases; Atazanavir Sulfate; CD4 Lymphocyte Count; Diarrhea; Double-Blind Method; Drug Therapy, Combination; Female; HIV Infections; HIV Integrase Inhibitors; HIV Protease Inhibitors; HIV-1; Humans; Lopinavir; Male; Middle Aged; Oligopeptides; Pyridines; Pyrrolidinones; Quinolones; Raltegravir Potassium; Ritonavir; RNA, Viral; Treatment Outcome; Viral Load

2012
Co-formulated elvitegravir, cobicistat, emtricitabine, and tenofovir disoproxil fumarate versus ritonavir-boosted atazanavir plus co-formulated emtricitabine and tenofovir disoproxil fumarate for initial treatment of HIV-1 infection: a randomised, double-
    Lancet (London, England), 2012, Jun-30, Volume: 379, Issue:9835

    Topics: Adenine; Adult; Anti-HIV Agents; Atazanavir Sulfate; Carbamates; Cobicistat; Deoxycytidine; Double-Blind Method; Drug Combinations; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Middle Aged; Oligopeptides; Organophosphonates; Pyridines; Quinolones; Ritonavir; Tenofovir; Thiazoles

2012
Co-formulated elvitegravir, cobicistat, emtricitabine, and tenofovir versus co-formulated efavirenz, emtricitabine, and tenofovir for initial treatment of HIV-1 infection: a randomised, double-blind, phase 3 trial, analysis of results after 48 weeks.
    Lancet (London, England), 2012, Jun-30, Volume: 379, Issue:9835

    Topics: Adenine; Adult; Alkynes; Anti-HIV Agents; Benzoxazines; Carbamates; Cobicistat; Cyclopropanes; Deoxycytidine; Double-Blind Method; Drug Combinations; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Middle Aged; Organophosphonates; Quinolones; Tenofovir; Thiazoles

2012
A randomized, double-blind comparison of coformulated elvitegravir/cobicistat/emtricitabine/tenofovir DF vs ritonavir-boosted atazanavir plus coformulated emtricitabine and tenofovir DF for initial treatment of HIV-1 infection: analysis of week 96 results
    Journal of acquired immune deficiency syndromes (1999), 2013, Apr-15, Volume: 62, Issue:5

    Topics: Adenine; Adult; Alanine Transaminase; Anti-HIV Agents; Aspartate Aminotransferases; Atazanavir Sulfate; Bilirubin; Bone Density; Carbamates; Cobicistat; Confidence Intervals; Creatinine; Deoxycytidine; Double-Blind Method; Drug Combinations; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Oligopeptides; Organophosphonates; Pyridines; Quinolones; Ritonavir; RNA, Viral; Tenofovir; Thiazoles; Triglycerides

2013
A randomized double-blind comparison of coformulated elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate versus efavirenz/emtricitabine/tenofovir disoproxil fumarate for initial treatment of HIV-1 infection: analysis of week 96 results.
    Journal of acquired immune deficiency syndromes (1999), 2013, May-01, Volume: 63, Issue:1

    Topics: Adenine; Adult; Anti-HIV Agents; Carbamates; Creatinine; Deoxycytidine; Double-Blind Method; Drug Combinations; Efavirenz, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; Female; HIV Infections; HIV-1; Humans; Male; Organophosphonates; Oxazines; Quinolones; RNA, Viral; Thiazoles; Treatment Outcome; Young Adult

2013
Antiviral activity, pharmacokinetics, and dose response of the HIV-1 integrase inhibitor GS-9137 (JTK-303) in treatment-naive and treatment-experienced patients.
    Journal of acquired immune deficiency syndromes (1999), 2006, Volume: 43, Issue:1

    Topics: Acquired Immunodeficiency Syndrome; Anti-HIV Agents; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Enzyme Inhibitors; HIV Infections; HIV Integrase; Humans; Quinolones

2006

Other Studies

157 other study(ies) available for carbostyril and HIV Coinfection

ArticleYear
Durability of Integrase STrand Inhibitor (InSTI)-based regimen in geriatric people living with HIV in the GEPPO cohort.
    PloS one, 2021, Volume: 16, Issue:10

    Topics: Aged; Amides; Anti-Retroviral Agents; Drug Therapy, Combination; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Longitudinal Studies; Male; Medication Adherence; Oxazines; Piperazines; Polypharmacy; Proportional Hazards Models; Prospective Studies; Pyridones; Quinolones; Raltegravir Potassium; Treatment Outcome

2021
Switching from efavirenz to elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide reduces central nervous system symptoms in people living with HIV.
    Chinese medical journal, 2021, Oct-13, Volume: 134, Issue:23

    Topics: Adenine; Adult; Alanine; Alkynes; Anti-HIV Agents; Benzoxazines; Central Nervous System; Cobicistat; Cyclopropanes; Drug Combinations; Emtricitabine; Female; HIV Infections; Humans; Male; Prospective Studies; Quality of Life; Quinolones; Sleep Quality; Tenofovir

2021
Incidence of low-level viremia and its impact on virologic failure among people living with HIV-1 who switched to elvitegravir-based antiretroviral therapy.
    Journal of global antimicrobial resistance, 2022, Volume: 29

    Topics: Anti-HIV Agents; Emtricitabine; HIV Infections; HIV-1; Humans; Incidence; Quinolones; Raltegravir Potassium; Retrospective Studies; Viremia

2022
Effectiveness and safety of elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate single-tablet combination among HIV-infected patients in Turkey: results from a real world setting.
    African health sciences, 2021, Volume: 21, Issue:4

    Topics: Adult; Anti-HIV Agents; Cobicistat; Drug Combinations; Emtricitabine; HIV Infections; Homosexuality, Male; Humans; Male; Quinolones; Retrospective Studies; Tablets; Tenofovir; Turkey

2021
A 28-Year-Old Man With Diffuse Bilateral Pulmonary Nodules.
    Chest, 2022, Volume: 162, Issue:1

    Topics: Adult; Anti-HIV Agents; Child; Cobicistat; Drug Combinations; Emtricitabine; HIV Infections; Humans; Male; Quinolones; Tenofovir

2022
High-level dolutegravir resistance can emerge rapidly from few variants and spread by recombination: implications for integrase strand transfer inhibitor salvage therapy.
    AIDS (London, England), 2022, 11-01, Volume: 36, Issue:13

    Topics: Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Mutation; Oxazines; Piperazines; Pyridones; Quinolones; Recombination, Genetic; Salvage Therapy

2022
Dolutegravir in Pregnancy as Compared with Current HIV Regimens in the United States.
    The New England journal of medicine, 2022, 09-01, Volume: 387, Issue:9

    Topics: Adult; Anti-HIV Agents; Atazanavir Sulfate; Cobicistat; Cohort Studies; Darunavir; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Protease Inhibitors; HIV-1; Humans; Infant, Newborn; Oxazines; Piperazines; Pregnancy; Premature Birth; Pyridones; Quinolones; Raltegravir Potassium; Rilpivirine; Ritonavir; United States

2022
Higher Risk of Dyslipidemia With Coformulated Elvitegravir, Cobicistat, Emtricitabine, and Tenofovir Alafenamide than Efavirenz, Lamivudine, and Tenofovir Disoproxil Fumarate Among Antiretroviral-Naive People Living With HIV in China.
    Journal of acquired immune deficiency syndromes (1999), 2022, 10-01, Volume: 91, Issue:S1

    Topics: Adenine; Alanine; Alkynes; Anti-HIV Agents; Anti-Retroviral Agents; Benzoxazines; Cholesterol, LDL; Cobicistat; Cyclopropanes; Emtricitabine; HIV Infections; HIV-1; Humans; Hypercholesterolemia; Hypertriglyceridemia; Lamivudine; Lipoproteins, HDL; Quinolones; Retrospective Studies; Tenofovir

2022
Switching to Tenofovir Alafenamide in Elvitegravir-Based Regimens: Pharmacokinetics and Antiviral Activity in Cerebrospinal Fluid.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2020, 08-14, Volume: 71, Issue:4

    Topics: Adenine; Adult; Alanine; Anti-HIV Agents; Emtricitabine; HIV Infections; Humans; Quinolones; Tenofovir

2020
Switching antiretrovirals in older patients.
    The lancet. HIV, 2019, Volume: 6, Issue:10

    Topics: Adenine; Aged; Alanine; Bone Density; Cobicistat; Emtricitabine; HIV Infections; HIV-1; Humans; Middle Aged; Quinolones; Tablets; Tenofovir

2019
Impact of NRTI resistance mutations on virological effectiveness of antiretroviral regimens containing elvitegravir: a multi-cohort study.
    The Journal of antimicrobial chemotherapy, 2020, 01-01, Volume: 75, Issue:1

    Topics: Adult; Anti-Retroviral Agents; Antiretroviral Therapy, Highly Active; Cohort Studies; Databases, Factual; Drug Resistance, Viral; Drug Therapy, Combination; Female; HIV Infections; HIV-1; Humans; Italy; Male; Middle Aged; Mutation; Quinolones; Treatment Outcome; Viral Load

2020
Comparable
    Antimicrobial agents and chemotherapy, 2019, 12-20, Volume: 64, Issue:1

    Topics: Amides; Heterocyclic Compounds, 3-Ring; Heterocyclic Compounds, 4 or More Rings; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Mutation; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium

2019
Fevers and Night Sweats in a 35-year-old Man With Recent Travel to Southeast Asia.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2019, 10-15, Volume: 69, Issue:9

    Topics: Adenine; Adult; Alanine; Anti-HIV Agents; Asia, Southeastern; Cobicistat; Emtricitabine; HIV Infections; Humans; Laos; Male; Quinolones; Sweating; Tenofovir; Thailand; Travel; United States

2019
The impact of integrase inhibitor-based regimens on markers of inflammation among HIV naïve patients.
    Cytokine, 2020, Volume: 126

    Topics: Adult; Anti-HIV Agents; Atazanavir Sulfate; Cytokines; Drug Therapy, Combination; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Inflammation; Male; Middle Aged; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium

2020
Brief Report: Integrase Strand Transfer Inhibitors Are Associated With Lower Risk of Incident Cardiovascular Disease in People Living With HIV.
    Journal of acquired immune deficiency syndromes (1999), 2020, 08-01, Volume: 84, Issue:4

    Topics: Adult; Anti-Retroviral Agents; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Ischemic Stroke; Male; Middle Aged; Myocardial Infarction; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Retrospective Studies

2020
Clinically Significant Lower Elvitegravir Exposure During the Third Trimester of Pregnant Patients Living With Human Immunodeficiency Virus: Data From the Pharmacokinetics of ANtiretroviral agents in HIV-infected pregNAnt women (PANNA) Network.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2020, 12-17, Volume: 71, Issue:10

    Topics: Anti-HIV Agents; Anti-Retroviral Agents; Female; HIV Infections; Humans; Pregnancy; Pregnancy Complications, Infectious; Pregnancy Trimester, Third; Pregnant Women; Quinolones

2020
Molecular dynamic simulations to investigate the structural impact of known drug resistance mutations on HIV-1C Integrase-Dolutegravir binding.
    PloS one, 2020, Volume: 15, Issue:5

    Topics: Amino Acid Sequence; Catalytic Domain; Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Molecular Dynamics Simulation; Mutation; Oxazines; Piperazines; Protein Binding; Protein Stability; Pyridones; Quinolones; Raltegravir Potassium; South Africa; Virus Replication

2020
Design, synthesis and SAR study of bridged tricyclic pyrimidinone carboxamides as HIV-1 integrase inhibitors.
    Bioorganic & medicinal chemistry, 2020, 07-01, Volume: 28, Issue:13

    Topics: Antiviral Agents; Drug Resistance, Viral; Drug Therapy, Combination; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Imidazoles; Mutation; Pyrrolidinones; Quinolones; Raltegravir Potassium; Structure-Activity Relationship

2020
An Elvitegravir Nanoformulation Crosses the Blood-Brain Barrier and Suppresses HIV-1 Replication in Microglia.
    Viruses, 2020, 05-20, Volume: 12, Issue:5

    Topics: Animals; Anti-HIV Agents; Anti-Retroviral Agents; Blood-Brain Barrier; Disease Models, Animal; Drug Carriers; Drug Delivery Systems; HIV Infections; HIV-1; Integrase Inhibitors; Macrophages; Male; Mice; Mice, Inbred NOD; Microglia; Nanoparticles; Pilot Projects; Plasma; Quinolones; Viral Load; Virus Replication

2020
Susceptibility to HIV-1 integrase strand transfer inhibitors (INSTIs) in highly treatment-experienced patients who failed an INSTI-based regimen.
    International journal of antimicrobial agents, 2020, Volume: 56, Issue:1

    Topics: Amides; Drug Resistance, Multiple, Viral; Female; Heterocyclic Compounds, 3-Ring; Heterocyclic Compounds, 4 or More Rings; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Male; Middle Aged; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Treatment Outcome

2020
Effectiveness of the combination elvitegravir/cobicistat/tenofovir/emtricitabine (EVG/COB/TFV/FTC) plus darunavir among treatment-experienced patients in clinical practice: a multicentre cohort study.
    AIDS research and therapy, 2020, 07-20, Volume: 17, Issue:1

    Topics: Adult; Anti-HIV Agents; Cobicistat; Darunavir; Drug Therapy, Combination; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Middle Aged; Quinolones; Spain; Tenofovir; Treatment Outcome; Viral Load

2020
Single oral dose for HIV pre or post-exposure prophylaxis: user desirability and biological efficacy in macaques.
    EBioMedicine, 2020, Volume: 58

    Topics: Adenine; Administration, Oral; Animals; Cross-Sectional Studies; Drug Combinations; Emtricitabine; HIV Infections; Homosexuality, Male; Humans; Macaca; Male; Patient Compliance; Pre-Exposure Prophylaxis; Quinolones; Rectum; Surveys and Questionnaires; Tenofovir

2020
Impact of archived M184V/I mutation on the effectiveness of switch to co-formulated elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide among virally suppressed people living with HIV.
    The Journal of antimicrobial chemotherapy, 2020, 10-01, Volume: 75, Issue:10

    Topics: Adenine; Adult; Alanine; Anti-HIV Agents; Cobicistat; Emtricitabine; HIV Infections; HIV-1; Humans; Mutation; Quinolones; Retrospective Studies; Tenofovir

2020
Structural Comparison of Diverse HIV-1 Subtypes using Molecular Modelling and Docking Analyses of Integrase Inhibitors.
    Viruses, 2020, 08-26, Volume: 12, Issue:9

    Topics: Amides; Binding Sites; Heterocyclic Compounds, 3-Ring; Heterocyclic Compounds, 4 or More Rings; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Linear Models; Models, Molecular; Molecular Docking Simulation; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Sequence Alignment

2020
Differential effects of integrase strand transfer inhibitors, elvitegravir and raltegravir, on oligodendrocyte maturation: A role for the integrated stress response.
    Glia, 2021, Volume: 69, Issue:2

    Topics: Animals; Cell Differentiation; Cuprizone; HIV Infections; Humans; Integrases; Mice; Mice, Inbred C57BL; Myelin Sheath; Oligodendroglia; Quinolones; Raltegravir Potassium; Rats

2021
Second-generation integrase strand inhibitors can be effective against elvitegravir-derived multiple integrase gene substitutions.
    AIDS (London, England), 2020, 11-15, Volume: 34, Issue:14

    Topics: Adult; Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Integrases; Male; Pyridones; Quinolones; Raltegravir Potassium

2020
Changes in neurocognitive assessment scores after initiating dolutegravir- versus elvitegravir-based antiretroviral therapy.
    AIDS care, 2021, Volume: 33, Issue:11

    Topics: Adult; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Male; Middle Aged; Oxazines; Piperazines; Prospective Studies; Pyridones; Quinolones

2021
Elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide discontinuation and return to normal weight.
    International journal of STD & AIDS, 2021, Volume: 32, Issue:1

    Topics: Adult; Alanine; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Cobicistat; Drug Combinations; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Quinolones; Tenofovir; Weight Gain

2021
Efficacy and Safety of Elvitegravir/Cobicistat/Emtricitabine/Tenofovir Alafenamide as Maintenance Treatment in HIV/HBV-Coinfected Patients.
    Journal of acquired immune deficiency syndromes (1999), 2021, 04-01, Volume: 86, Issue:4

    Topics: Adult; Alanine; Anti-HIV Agents; Cobicistat; Cohort Studies; Drug Combinations; Drug Substitution; Emtricitabine; Female; Hepatitis B, Chronic; HIV Infections; HIV-1; Humans; Male; Middle Aged; Prospective Studies; Quinolones; Taiwan; Tenofovir

2021
Preoperative rapid suppression of viral load by elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide regimen in human immunodeficiency virus-positive fracture patients significantly reduces postoperative complications.
    Chinese medical journal, 2020, Dec-05, Volume: 133, Issue:23

    Topics: Adenine; Alanine; Anti-HIV Agents; Cobicistat; Drug Combinations; Emtricitabine; HIV; HIV Infections; Humans; Postoperative Complications; Quinolones; Tenofovir; Viral Load

2020
Switching to Elvitegravir/Cobicistat/Emtricitabine/Tenofovir Alafenamide in Adults With HIV and M184V/I Mutation.
    Journal of acquired immune deficiency syndromes (1999), 2021, 04-01, Volume: 86, Issue:4

    Topics: Adult; Aged; Alanine; Anti-HIV Agents; Cobicistat; Drug Combinations; Drug Resistance, Viral; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Middle Aged; Mutation; Quinolones; Tenofovir; Young Adult

2021
Integrase Strand Transfer Inhibitor Start or Switch Impacts Learning in Women With HIV.
    Journal of acquired immune deficiency syndromes (1999), 2021, 04-15, Volume: 86, Issue:5

    Topics: Adult; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; Humans; Integrases; Middle Aged; Oxazines; Piperazines; Prospective Studies; Pyridones; Quinolones; Raltegravir Potassium; Reverse Transcriptase Inhibitors; United States

2021
Hepatic Steatosis Associated With Exposure to Elvitegravir and Raltegravir.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2021, 08-02, Volume: 73, Issue:3

    Topics: HIV Infections; Humans; Prospective Studies; Quinolones; Raltegravir Potassium

2021
Tolerability of integrase inhibitors in a real-life setting.
    The Journal of antimicrobial chemotherapy, 2017, 06-01, Volume: 72, Issue:6

    Topics: Adult; Cohort Studies; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Life Style; Male; Medication Adherence; Middle Aged; Oxazines; Piperazines; Proportional Hazards Models; Pyridones; Quinolones; Raltegravir Potassium; Retrospective Studies

2017
Efficacy of elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate as treatment for primary or recent HIV infection-authors' response.
    The Journal of antimicrobial chemotherapy, 2017, 05-01, Volume: 72, Issue:5

    Topics: Adenine; Anti-HIV Agents; Cobicistat; Deoxycytidine; Emtricitabine; HIV Infections; Humans; Organophosphonates; Quinolones; Tenofovir

2017
Right hip and bilateral shoulder capsulitis in an HIV-infected individual treated with elvitegravir and cobicistat.
    AIDS (London, England), 2017, May-15, Volume: 31, Issue:8

    Topics: Anti-HIV Agents; Bursitis; Cobicistat; Hip Joint; HIV Infections; Humans; Male; Middle Aged; Quinolones; Radionuclide Imaging; Shoulder Joint

2017
HIV-1 integrase inhibitor resistance among treatment naïve patients in the West of Scotland.
    Journal of clinical virology : the official publication of the Pan American Society for Clinical Virology, 2017, Volume: 92

    Topics: Adult; Aged; Drug Resistance, Viral; Female; Genotype; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Male; Middle Aged; Mutation; Quinolones; Scotland; Treatment Outcome; Viral Load; Young Adult

2017
Free and total plasma concentrations of elvitegravir/cobicistat during pregnancy and postpartum: a case report.
    British journal of clinical pharmacology, 2017, Volume: 83, Issue:12

    Topics: Adult; Anti-HIV Agents; Cobicistat; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; Female; HIV Infections; Humans; Postpartum Period; Pregnancy; Quinolones

2017
High decay of blood HIV reservoir when tenofovir/emtricitabine/elvitegravir/cobicistat is initiated during the acute primary HIV infection.
    The Journal of antimicrobial chemotherapy, 2017, 09-01, Volume: 72, Issue:9

    Topics: Adult; Anti-HIV Agents; Blood; Cobicistat; Emtricitabine; HIV Infections; HIV-1; Humans; Male; Middle Aged; Quinolones; Secondary Prevention; Tenofovir; Treatment Outcome; Viral Load

2017
Clinical Experience with the Integrase Inhibitors Dolutegravir and Elvitegravir in HIV-infected Patients: Efficacy, Safety and Tolerance.
    Basic & clinical pharmacology & toxicology, 2017, Volume: 121, Issue:5

    Topics: Adult; Aged; Aged, 80 and over; Cobicistat; Dideoxynucleosides; Drug Combinations; Female; Follow-Up Studies; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Lamivudine; Male; Middle Aged; Oxazines; Piperazines; Pyridones; Quinolones; Retrospective Studies; Risk Factors; Spain; Treatment Outcome; Young Adult

2017
Safety and tolerability of Elvitegravir/Cobicistat/Emtricitabine/Tenofovir Disoproxil fumarate in a real life setting: Data from surveillance cohort long-term toxicity antiretrovirals/antivirals (SCOLTA) project.
    PloS one, 2017, Volume: 12, Issue:6

    Topics: Adult; Anti-HIV Agents; Cobicistat; Drug Combinations; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Maximum Tolerated Dose; Middle Aged; Quinolones; Safety; Tenofovir

2017
Prevalence of drug-drug interactions in the era of HIV integrase inhibitors: a retrospective clinical study.
    The Netherlands journal of medicine, 2017, Volume: 75, Issue:6

    Topics: Adult; Anti-Retroviral Agents; Databases, Factual; Drug Interactions; Drug-Related Side Effects and Adverse Reactions; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Male; Middle Aged; Oxazines; Piperazines; Prevalence; Pyridones; Quinolones; Retrospective Studies; Risk Factors

2017
Degradable bioadhesive nanoparticles for prolonged intravaginal delivery and retention of elvitegravir.
    Biomaterials, 2017, Volume: 144

    Topics: Administration, Intravaginal; Animals; Anti-HIV Agents; Delayed-Action Preparations; Female; HIV; HIV Infections; Humans; Mice, Inbred C57BL; Nanoparticles; Quinolones; Vagina

2017
HIV-1 non-group M phenotypic susceptibility to integrase strand transfer inhibitors.
    The Journal of antimicrobial chemotherapy, 2017, 09-01, Volume: 72, Issue:9

    Topics: Amino Acid Substitution; Drug Resistance, Viral; Genotype; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Inhibitory Concentration 50; Mutation; Oxazines; Phenotype; Phylogeny; Piperazines; Polymorphism, Genetic; Pyridones; Quinolones; Raltegravir Potassium

2017
Mutations Located outside the Integrase Gene Can Confer Resistance to HIV-1 Integrase Strand Transfer Inhibitors.
    mBio, 2017, 09-26, Volume: 8, Issue:5

    Topics: Amino Acid Substitution; Cell Line; Drug Resistance, Viral; Genes, nef; Heterocyclic Compounds, 3-Ring; High-Throughput Nucleotide Sequencing; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Mutation; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Virus Integration; Virus Replication; Zidovudine

2017
Effect of Cobicistat on Tenofovir Disoproxil Fumarate (TDF): What Is True for TAF May Also Be True for TDF.
    Journal of acquired immune deficiency syndromes (1999), 2018, 01-01, Volume: 77, Issue:1

    Topics: Adenine; Adult; Aged; Alanine; Anti-HIV Agents; Cobicistat; Drug Combinations; Drug Interactions; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; Humans; Kaplan-Meier Estimate; Male; Middle Aged; Oxazines; Piperazines; Proportional Hazards Models; Pyridones; Quinolones; Raltegravir Potassium; Ritonavir; Tenofovir; Treatment Outcome

2018
Adverse drug reactions to integrase strand transfer inhibitors.
    AIDS (London, England), 2018, 04-24, Volume: 32, Issue:7

    Topics: Adult; British Columbia; Cobicistat; Drug-Related Side Effects and Adverse Reactions; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Male; Middle Aged; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Retrospective Studies

2018
Reciprocal Effects of Antiretroviral Drugs Used To Treat HIV Infection on the Fibroblast Growth Factor 21/β-Klotho System.
    Antimicrobial agents and chemotherapy, 2018, Volume: 62, Issue:6

    Topics: Adipose Tissue; Alkynes; Anti-Retroviral Agents; Benzoxazines; Cyclopropanes; Diabetes Mellitus, Type 2; Drug Combinations; Endoplasmic Reticulum Stress; Fibroblast Growth Factors; Hep G2 Cells; HIV Infections; HIV Integrase Inhibitors; Humans; Klotho Proteins; Liver; Lopinavir; Maraviroc; Membrane Proteins; Muscle, Skeletal; Obesity; Oxidative Stress; Protease Inhibitors; Quinolones; Reverse Transcriptase Inhibitors; Ritonavir; Thapsigargin; Tunicamycin

2018
2018 update to the HIV-TRePS system: the development of new computational models to predict HIV treatment outcomes, with or without a genotype, with enhanced usability for low-income settings.
    The Journal of antimicrobial chemotherapy, 2018, 08-01, Volume: 73, Issue:8

    Topics: Adult; Anti-HIV Agents; Computer Simulation; Developing Countries; Drug Substitution; Female; HIV Infections; Humans; Male; Maraviroc; Pyridines; Pyrones; Quinolones; Sulfonamides; Sustained Virologic Response; Treatment Outcome

2018
Dolutegravir (DTG)-containing regimens after receiving raltegravir (RAL) or elvitegravir (EVG): Durability and virological response in a large Italian HIV drug resistance network (ARCA).
    Journal of clinical virology : the official publication of the Pan American Society for Clinical Virology, 2018, Volume: 105

    Topics: Adult; Anti-HIV Agents; Cohort Studies; Drug Resistance, Multiple, Viral; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV-1; Humans; Male; Middle Aged; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Retrospective Studies; RNA, Viral; Sustained Virologic Response; Young Adult

2018
Selective resistance profiles emerging in patient-derived clinical isolates with cabotegravir, bictegravir, dolutegravir, and elvitegravir.
    Retrovirology, 2018, 08-17, Volume: 15, Issue:1

    Topics: Amides; Anti-HIV Agents; Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; Heterocyclic Compounds, 4 or More Rings; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Mutation; Oxazines; Piperazines; Pyridones; Quinolones; Virus Replication

2018
Overdose of elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide in an HIV-1-infected subject with attempted suicide.
    Infection, 2019, Volume: 47, Issue:1

    Topics: Adenine; Alanine; Anti-HIV Agents; Cobicistat; Drug Combinations; Drug Overdose; Emtricitabine; HIV Infections; Humans; Male; Middle Aged; Quinolones; Renal Insufficiency; Suicide, Attempted; Tenofovir

2019
Optimizing concentrations of concomitant antiretrovirals by reducing etravirine doses: two case reports of complex drug-drug interactions.
    Antiviral therapy, 2019, Volume: 24, Issue:1

    Topics: Anti-Retroviral Agents; Darunavir; Drug Interactions; Drug Monitoring; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV-1; Humans; Male; Middle Aged; Nitriles; Oxazines; Piperazines; Pyridazines; Pyridones; Pyrimidines; Quinolones

2019
Efficacy and safety of switching to dolutegravir plus emtricitabine/tenofovir disoproxil fumarate (TDF) or elvitegravir/cobicistat/emtricitabine/TDF in virologically suppressed HIV-infected patients in clinical practice: results from a multicentre, observ
    HIV medicine, 2019, Volume: 20, Issue:2

    Topics: Adult; Cobicistat; Drug Therapy, Combination; Emtricitabine; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV-1; Humans; Male; Middle Aged; Oxazines; Piperazines; Pyridones; Quinolones; Retrospective Studies; RNA, Viral; Tenofovir; Viral Load

2019
Prevalence and determinants of resistance mutations in HIV-1-infected patients exposed to integrase inhibitors in a large Italian cohort.
    HIV medicine, 2019, Volume: 20, Issue:2

    Topics: Adult; Drug Resistance, Viral; Female; Genotype; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Italy; Logistic Models; Male; Middle Aged; Mutation; Oxazines; Piperazines; Prevalence; Pyridones; Quinolones; Raltegravir Potassium

2019
Abnormal elevation of international normalized ratio in a patient during the coadministration of elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide and warfarin: a case report.
    AIDS (London, England), 2019, 02-01, Volume: 33, Issue:2

    Topics: Adenine; Alanine; Cobicistat; Emtricitabine; HIV Infections; Humans; International Normalized Ratio; Quinolones; Tenofovir; Warfarin

2019
Brief Report: Surveillance of Congenital Anomalies After Exposure to Raltegravir or Elvitegravir During Pregnancy in the United Kingdom and Ireland, 2008-2018.
    Journal of acquired immune deficiency syndromes (1999), 2019, 03-01, Volume: 80, Issue:3

    Topics: Abnormalities, Drug-Induced; Adult; Female; HIV Infections; Humans; Infectious Disease Transmission, Vertical; Ireland; Pregnancy; Pregnancy Complications, Infectious; Quinolones; Raltegravir Potassium; Stillbirth; United Kingdom

2019
Integrase strand transfer inhibitors and neuropsychiatric adverse events in a large prospective cohort.
    The Journal of antimicrobial chemotherapy, 2019, 03-01, Volume: 74, Issue:3

    Topics: Antiretroviral Therapy, Highly Active; CD4 Lymphocyte Count; Cohort Studies; Female; France; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Male; Mental Disorders; Nervous System Diseases; Oxazines; Piperazines; Prospective Studies; Public Health Surveillance; Pyridones; Quinolones; Raltegravir Potassium; Viral Load

2019
Barrier to Resistance of Dolutegravir in Two-Drug Combinations.
    Antimicrobial agents and chemotherapy, 2019, Volume: 63, Issue:3

    Topics: Anti-HIV Agents; Cell Line; Drug Resistance, Viral; Drug Therapy, Combination; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Lamivudine; Oxazines; Piperazines; Pyridones; Quinolones; Rilpivirine

2019
HIV Integrase Inhibitor Pharmacogenetics: An Exploratory Study.
    Clinical drug investigation, 2019, Volume: 39, Issue:3

    Topics: Adult; Female; Genotype; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Male; Middle Aged; Oxazines; Pharmacogenetics; Piperazines; Pyridones; Quinolones; Raltegravir Potassium

2019
Discontinuation of dolutegravir, elvitegravir/cobicistat and raltegravir because of toxicity in a prospective cohort.
    HIV medicine, 2019, Volume: 20, Issue:3

    Topics: Adult; CD4 Lymphocyte Count; Cobicistat; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; Humans; Male; Middle Aged; Oxazines; Piperazines; Proportional Hazards Models; Prospective Studies; Pyridones; Quinolones; Raltegravir Potassium; Spain

2019
Durability of first-line regimens including integrase strand transfer inhibitors (INSTIs): data from a real-life setting.
    The Journal of antimicrobial chemotherapy, 2019, 05-01, Volume: 74, Issue:5

    Topics: Adult; CD4 Lymphocyte Count; Cobicistat; Cohort Studies; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; HIV Seropositivity; Humans; Italy; Male; Middle Aged; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Regression Analysis; Survival Analysis; Treatment Failure

2019
Severe rhabdomyolysis-induced acute kidney injury following concomitant use of Genvoya® (EVG/COBI/FTC/TAF) and simvastatin; a case report.
    BMC nephrology, 2019, 02-26, Volume: 20, Issue:1

    Topics: Acute Kidney Injury; Anti-HIV Agents; Cobicistat; Drug Combinations; Drug Interactions; Dyslipidemias; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; Emtricitabine; Hepatitis A; Hepatitis C; HIV Infections; Humans; Hypolipidemic Agents; Liver Function Tests; Male; Middle Aged; Quinolones; Renal Dialysis; Rhabdomyolysis; Simvastatin; Tenofovir; Treatment Outcome

2019
Antiretroviral Hydrophobic Core Graft-Copolymer Nanoparticles: The Effectiveness against Mutant HIV-1 Strains and in Vivo Distribution after Topical Application.
    Pharmaceutical research, 2019, Mar-27, Volume: 36, Issue:5

    Topics: Alkynes; Animals; Anti-HIV Agents; Benzoxazines; Cell Line; Cyclopropanes; Drug Carriers; Drug Combinations; Drug Liberation; Drug Resistance, Viral; Female; HIV Infections; HIV Integrase Inhibitors; HIV-1; Hydrophobic and Hydrophilic Interactions; Molecular Dynamics Simulation; Mutation; Nanoparticles; Polyethylene Glycols; Polylysine; Quinolones; Rats; Reverse Transcriptase Inhibitors; Tissue Distribution

2019
Paediatric Integrase Inhibitor Use in a Real-Life Setting: A Single-Centre Cohort Experience 2009-2018.
    Clinical drug investigation, 2019, Volume: 39, Issue:6

    Topics: Adolescent; Child; Child, Preschool; Cohort Studies; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Male; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Retrospective Studies; Viral Load

2019
Effects of guggulsterones-containing thermogenic complex on elvitegravir plasma concentrations: a case report.
    European journal of clinical pharmacology, 2019, Volume: 75, Issue:8

    Topics: Anti-HIV Agents; CD4-Positive T-Lymphocytes; Cytochrome P-450 CYP3A; Drug Interactions; HIV Infections; Humans; Lymphocyte Count; Male; Middle Aged; Pregnenediones; Quinolones; RNA, Viral

2019
Is There a Safety Signal for Dolutegravir and Integrase Inhibitors During Pregnancy?
    Journal of acquired immune deficiency syndromes (1999), 2019, 08-01, Volume: 81, Issue:4

    Topics: Adult; Anti-Retroviral Agents; Cohort Studies; Congenital Abnormalities; Drug Resistance, Viral; Female; France; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Neural Tube Defects; Oxazines; Pharmacovigilance; Piperazines; Pregnancy; Pyridones; Quinolones; Raltegravir Potassium; Treatment Outcome; Young Adult

2019
Resistance to HIV integrase strand transfer inhibitors in Argentina: first interim survey.
    Revista espanola de quimioterapia : publicacion oficial de la Sociedad Espanola de Quimioterapia, 2019, Volume: 32, Issue:3

    Topics: Adult; Argentina; Drug Resistance, Viral; Female; Heterocyclic Compounds, 3-Ring; HIV; HIV Infections; HIV Integrase Inhibitors; Humans; Male; Middle Aged; Oxazines; Pilot Projects; Piperazines; Prevalence; Pyridones; Quinolones; Raltegravir Potassium; Retrospective Studies; Surveys and Questionnaires; Urban Population; Viral Load; Young Adult

2019
E157Q integrase strand-transfer inhibitor substitution in patients with acute/recent HIV infection.
    AIDS (London, England), 2019, 08-01, Volume: 33, Issue:10

    Topics: Adult; Amino Acid Substitution; Disease Transmission, Infectious; Drug Resistance, Viral; Female; Gene Frequency; Genotype; Genotyping Techniques; High-Throughput Nucleotide Sequencing; HIV; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; Humans; Male; Molecular Epidemiology; Mutation, Missense; Phylogeny; Prevalence; Prospective Studies; Quinolones; Raltegravir Potassium; Sexual and Gender Minorities; Viral Load

2019
Sustained HIV virologic suppression with crushed combination tablets containing elvitegravir, cobicistat, emtricitabine, and tenofovir alafenamide.
    American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists, 2019, 08-01, Volume: 76, Issue:16

    Topics: Adenine; Alanine; Anti-HIV Agents; Cobicistat; Drug Therapy, Combination; Emtricitabine; Enteral Nutrition; Gastrostomy; HIV Infections; HIV-1; Humans; Male; Middle Aged; Quinolones; Sustained Virologic Response; Tablets; Tenofovir

2019
Evaluation of HIV-1 integrase resistance emergence and evolution in patients treated with integrase inhibitors.
    Journal of global antimicrobial resistance, 2020, Volume: 20

    Topics: Adult; Drug Resistance, Viral; Evolution, Molecular; Female; Genotype; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Logistic Models; Male; Middle Aged; Mutation; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium

2020
Brief Report: Urine Emtricitabine and Tenofovir Concentrations Provide Markers of Recent Antiretroviral Drug Exposure Among HIV-Negative Men Who Have Sex With Men.
    Journal of acquired immune deficiency syndromes (1999), 2019, 11-01, Volume: 82, Issue:3

    Topics: Adenine; Administration, Oral; Adolescent; Adult; Alanine; Anti-HIV Agents; Anti-Retroviral Agents; Biomarkers; Cobicistat; Emtricitabine; HIV Infections; Homosexuality, Male; Humans; Male; Middle Aged; Quinolones; Sexual and Gender Minorities; Tenofovir; Time Factors; Young Adult

2019
Antiviral activity of HIV-1 integrase strand-transfer inhibitors against mutants with integrase resistance-associated mutations and their frequency in treatment-naïve individuals.
    Journal of medical virology, 2019, Volume: 91, Issue:12

    Topics: Amides; Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; Heterocyclic Compounds, 4 or More Rings; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Mutation; Oxazines; Piperazines; Polymorphism, Genetic; Pyridones; Quinolones

2019
Impact of primary elvitegravir resistance-associated mutations in HIV-1 integrase on drug susceptibility and viral replication fitness.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:6

    Topics: Cell Line; Drug Resistance, Viral; Genotype; HEK293 Cells; HIV Infections; HIV Integrase; HIV-1; Humans; Microbial Sensitivity Tests; Mutation; Quinolones; Virus Replication

2013
The pharmacokinetic and pharmacodynamic interactions between buprenorphine/naloxone and elvitegravir/cobicistat in subjects receiving chronic buprenorphine/naloxone treatment.
    Journal of acquired immune deficiency syndromes (1999), 2013, Aug-01, Volume: 63, Issue:4

    Topics: Adult; Anti-Retroviral Agents; Area Under Curve; Buprenorphine; Carbamates; Cobicistat; Drug Interactions; Female; HIV Infections; HIV Seronegativity; Humans; Male; Middle Aged; Naloxone; Narcotic Antagonists; Opioid-Related Disorders; Quinolones; Thiazoles

2013
A validated assay by liquid chromatography-tandem mass spectrometry for the simultaneous quantification of elvitegravir and rilpivirine in HIV positive patients.
    Journal of mass spectrometry : JMS, 2013, Volume: 48, Issue:5

    Topics: Anti-Retroviral Agents; Chromatography, Liquid; Drug Stability; HIV Infections; Humans; Nitriles; Pyrimidines; Quinolones; Reproducibility of Results; Rilpivirine; Sensitivity and Specificity; Tandem Mass Spectrometry

2013
Multiple genetic pathways involving amino acid position 143 of HIV-1 integrase are preferentially associated with specific secondary amino acid substitutions and confer resistance to raltegravir and cross-resistance to elvitegravir.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:9

    Topics: Amino Acid Substitution; Drug Resistance, Viral; Genes, Reporter; HEK293 Cells; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Luciferases; Mutagenesis, Site-Directed; Pyrrolidinones; Quinolones; Raltegravir Potassium; Tyrosine

2013
In vitro phenotypes to elvitegravir and dolutegravir in primary macrophages and lymphocytes of clonal recombinant viral variants selected in patients failing raltegravir.
    The Journal of antimicrobial chemotherapy, 2013, Volume: 68, Issue:11

    Topics: Anti-HIV Agents; Cells, Cultured; Cloning, Molecular; Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV-1; Humans; Lymphocytes; Macrophages; Oxazines; Piperazines; Pyridones; Pyrrolidinones; Quinolones; Raltegravir Potassium; Recombination, Genetic; Reverse Transcriptase Polymerase Chain Reaction; RNA, Viral; Sequence Analysis, DNA

2013
[ First integrase inhibitor based single tablet regimen].
    MMW Fortschritte der Medizin, 2013, Jun-13, Volume: 155 Suppl 1

    Topics: Adenine; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Carbamates; Cobicistat; Deoxycytidine; Drug Approval; Drug Combinations; Emtricitabine; HIV Infections; HIV Integrase Inhibitors; Humans; Organophosphonates; Quinolones; Tenofovir; Thiazoles; Treatment Outcome

2013
Discovery of a small molecule agonist of phosphatidylinositol 3-kinase p110α that reactivates latent HIV-1.
    PloS one, 2014, Volume: 9, Issue:1

    Topics: Anti-HIV Agents; CD4-Positive T-Lymphocytes; CD8-Positive T-Lymphocytes; Cell Line; Class Ia Phosphatidylinositol 3-Kinase; Drug Discovery; Drug Therapy, Combination; Enzyme Activation; Gene Expression; Heterocyclic Compounds, 4 or More Rings; Histone Deacetylase Inhibitors; HIV Infections; HIV-1; Humans; Hydroxamic Acids; Lymphocyte Activation; Lymphocyte Depletion; Proto-Oncogene Proteins c-akt; Quinolones; Signal Transduction; Virus Activation; Virus Latency; Vorinostat

2014
Examining structural analogs of elvitegravir as potential inhibitors of HIV-1 integrase.
    Archives of virology, 2014, Volume: 159, Issue:8

    Topics: Amino Acid Motifs; Amino Acid Sequence; Drug Resistance, Viral; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Molecular Docking Simulation; Molecular Structure; Quinolones

2014
Single-tablet, once-daily treatment regimens for HIV.
    The Lancet. Infectious diseases, 2014, Volume: 14, Issue:4

    Topics: Adenine; Alkynes; Anti-HIV Agents; Benzoxazines; Carbamates; Cobicistat; Cyclopropanes; Cytochrome P-450 CYP3A Inhibitors; Deoxycytidine; Drug Combinations; Emtricitabine; HIV Infections; HIV Integrase Inhibitors; HIV Reverse Transcriptase; Humans; Nitriles; Organophosphonates; Pyrimidines; Quinolones; Reverse Transcriptase Inhibitors; Rilpivirine; Tenofovir; Thiazoles

2014
Elvitegravir for the treatment of HIV infection.
    Drugs of today (Barcelona, Spain : 1998), 2014, Volume: 50, Issue:3

    Topics: Animals; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Drug Administration Schedule; Drug Interactions; Drug Resistance, Viral; Drug Therapy, Combination; Half-Life; HIV Infections; HIV Integrase Inhibitors; Humans; Quinolones; Ritonavir

2014
New raltegravir resistance pathways induce broad cross-resistance to all currently used integrase inhibitors.
    The Journal of antimicrobial chemotherapy, 2014, Volume: 69, Issue:8

    Topics: Amino Acid Substitution; Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Mutation; Oxazines; Piperazines; Protein Binding; Pyridones; Pyrrolidinones; Quinolones; Raltegravir Potassium; Treatment Failure

2014
Sustained virological response after taking crushed elvitegravir-cobicistat-emtricitabine-tenofovir tablets.
    American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists, 2014, May-15, Volume: 71, Issue:10

    Topics: Adenine; Adult; Antiretroviral Therapy, Highly Active; Carbamates; Cobicistat; Deoxycytidine; Emtricitabine; Female; HIV; HIV Infections; Humans; Organophosphonates; Powders; Quinolones; Tablets; Tenofovir; Thiazoles; Viral Load

2014
Lack of resistance to integrase inhibitors among antiretroviral-naive subjects with primary HIV-1 infection, 2007-2013.
    Antiviral therapy, 2015, Volume: 20, Issue:1

    Topics: Adult; Drug Resistance, Viral; Genotype; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Male; Mutation; Quinolones; Raltegravir Potassium; Retrospective Studies; Sequence Analysis, RNA

2015
Switching STRATEGIES in HIV treatment.
    The Lancet. Infectious diseases, 2014, Volume: 14, Issue:7

    Topics: Adenine; Anti-HIV Agents; Carbamates; Cobicistat; Deoxycytidine; Emtricitabine; Female; HIV; HIV Infections; Humans; Male; Organophosphonates; Protease Inhibitors; Quinolones; Reverse Transcriptase Inhibitors; Ritonavir; Tenofovir; Thiazoles

2014
Virological and immunological outcomes of elvitegravir-based regimen in a treatment-naïve HIV-2-infected patient.
    AIDS (London, England), 2014, Sep-24, Volume: 28, Issue:15

    Topics: Anti-HIV Agents; CD4 Lymphocyte Count; HIV Infections; HIV-2; Humans; Male; Middle Aged; Quinolones; Time Factors; Treatment Outcome; Viral Load

2014
Suppression of Foxo1 activity and down-modulation of CD62L (L-selectin) in HIV-1 infected resting CD4 T cells.
    PloS one, 2014, Volume: 9, Issue:10

    Topics: CD4-Positive T-Lymphocytes; Forkhead Box Protein O1; Forkhead Transcription Factors; Gene Expression Regulation; HIV Infections; HIV-1; Humans; Kruppel-Like Transcription Factors; L-Selectin; Lymphocyte Activation; Lymphoid Tissue; Quinolones; Receptors, Interleukin-7; Virus Replication

2014
Antiviral characteristics of GSK1265744, an HIV integrase inhibitor dosed orally or by long-acting injection.
    Antimicrobial agents and chemotherapy, 2015, Volume: 59, Issue:1

    Topics: Anti-HIV Agents; Cell Line; Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Microbial Sensitivity Tests; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Virus Replication

2015
Elvitegravir/cobicistat/emtricitabine/tenofovir DF in HIV-infected patients with mild-to-moderate renal impairment.
    Journal of acquired immune deficiency syndromes (1999), 2015, Mar-01, Volume: 68, Issue:3

    Topics: Adenine; Adult; Anti-HIV Agents; Carbamates; Cobicistat; Cohort Studies; Deoxycytidine; Emtricitabine; Female; HIV Infections; Humans; Male; Middle Aged; Organophosphonates; Quinolones; Renal Insufficiency; Tenofovir; Thiazoles; Treatment Outcome

2015
Cross-resistance to elvitegravir and dolutegravir in 502 patients failing on raltegravir: a French national study of raltegravir-experienced HIV-1-infected patients.
    The Journal of antimicrobial chemotherapy, 2015, Volume: 70, Issue:5

    Topics: Adult; Anti-HIV Agents; Drug Resistance, Viral; Female; France; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Protease; HIV Reverse Transcriptase; HIV-1; Humans; Male; Middle Aged; Mutant Proteins; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Sequence Analysis, DNA

2015
Tenofovir alafenamide for HIV infection: is less more?
    Lancet (London, England), 2015, Jun-27, Volume: 385, Issue:9987

    Topics: Adenine; Alanine; Anti-HIV Agents; Carbamates; Cobicistat; Deoxycytidine; Emtricitabine; Female; HIV Infections; Humans; Male; Organophosphonates; Quinolones; Tenofovir; Thiazoles

2015
An unexpected interaction between warfarin and cobicistat-boosted elvitegravir.
    AIDS (London, England), 2015, May-15, Volume: 29, Issue:8

    Topics: Adult; Anti-HIV Agents; Cobicistat; Drug Interactions; HIV Infections; Humans; Male; Quinolones; Warfarin

2015
Infectious disease: New HIV-1 prodrug shows promise in phase III trials.
    Nature reviews. Urology, 2015, Volume: 12, Issue:6

    Topics: Adenine; Anti-HIV Agents; Carbamates; Deoxycytidine; Female; HIV Infections; Humans; Male; Organophosphonates; Quinolones; Thiazoles

2015
Rapid regression of Kaposi's sarcoma of the hard palate under therapy with boosted elvitegravir-containing fixdose antiretroviral combination therapy.
    Infection, 2016, Volume: 44, Issue:1

    Topics: Adult; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; HIV Infections; Humans; Male; Palatal Neoplasms; Palate, Hard; Quinolones; Sarcoma, Kaposi; Treatment Outcome

2016
N-Substituted Quinolinonyl Diketo Acid Derivatives as HIV Integrase Strand Transfer Inhibitors and Their Activity against RNase H Function of Reverse Transcriptase.
    Journal of medicinal chemistry, 2015, Jun-11, Volume: 58, Issue:11

    Topics: Catalytic Domain; HeLa Cells; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Keto Acids; Models, Molecular; Molecular Structure; Quinolones; Ribonuclease H; RNA-Directed DNA Polymerase; Structure-Activity Relationship; Virus Replication

2015
The Combination of the R263K and T66I Resistance Substitutions in HIV-1 Integrase Is Incompatible with High-Level Viral Replication and the Development of High-Level Drug Resistance.
    Journal of virology, 2015, Volume: 89, Issue:22

    Topics: Amino Acid Substitution; Cell Line, Tumor; Drug Resistance, Viral; HEK293 Cells; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium; Virus Replication

2015
Deep analysis of HIV-1 natural variability across HIV-1 variants at residues associated with integrase inhibitor (INI) resistance in INI-naive individuals.
    The Journal of antimicrobial chemotherapy, 2016, Volume: 71, Issue:2

    Topics: Amino Acid Substitution; Computational Biology; Drug Resistance, Viral; Genetic Variation; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium

2016
Elvitegravir (Vitekta) for HIV.
    The Medical letter on drugs and therapeutics, 2016, Jan-18, Volume: 58, Issue:1486

    Topics: Animals; Drug Interactions; Female; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Pregnancy; Quinolones; Risk Factors; Treatment Outcome

2016
Genvoya--a new 4-drug combination for HIV.
    The Medical letter on drugs and therapeutics, 2016, Feb-15, Volume: 58, Issue:1488

    Topics: Cobicistat; Drug Combinations; Drug Interactions; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; Emtricitabine; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Quinolones; Randomized Controlled Trials as Topic; Tenofovir; Treatment Outcome

2016
First reported use of elvitegravir and cobicistat during pregnancy.
    AIDS (London, England), 2016, Mar-13, Volume: 30, Issue:5

    Topics: Adult; Anti-HIV Agents; Cobicistat; Female; HIV Infections; Humans; Plasma; Pregnancy; Pregnancy Complications, Infectious; Quinolones

2016
Elvitegravir/Cobicistat/Tenofovir/Emtricitabine Penetration in the Cerebrospinal Fluid of Three HIV-Positive Patients.
    AIDS research and human retroviruses, 2016, Volume: 32, Issue:5

    Topics: Adult; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Cobicistat; Emtricitabine; Female; HIV Infections; Humans; Male; Middle Aged; Quinolones; Tenofovir

2016
Q148N, a Novel Integrase Inhibitor Resistance Mutation Associated with Low-Level Reduction in Elvitegravir Susceptibility.
    AIDS research and human retroviruses, 2016, Volume: 32, Issue:7

    Topics: Amino Acid Substitution; Drug Resistance, Viral; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Male; Microbial Sensitivity Tests; Middle Aged; Mutation, Missense; Quinolones

2016
HIV-infected CD4+ T Cells Use T-bet-dependent Pathway for Production of IL-10 Upon Antigen Recognition.
    Scandinavian journal of immunology, 2016, Volume: 83, Issue:4

    Topics: Adult; CD4 Lymphocyte Count; CD4-Positive T-Lymphocytes; Cells, Cultured; Cyclosporine; Extracellular Signal-Regulated MAP Kinases; Female; Flavonoids; Forkhead Transcription Factors; HIV Core Protein p24; HIV Infections; Humans; Interferon-gamma; Interleukin-10; Lymphocyte Activation; Male; Middle Aged; Quinolones; T-Box Domain Proteins; Young Adult

2016
Population pharmacokinetic analysis of elvitegravir and cobicistat in HIV-1-infected individuals.
    The Journal of antimicrobial chemotherapy, 2016, Volume: 71, Issue:7

    Topics: Adolescent; Adult; Aged; Anti-HIV Agents; Area Under Curve; Cobicistat; Cohort Studies; Computer Simulation; Drug Interactions; Female; HIV Infections; HIV-1; Humans; Male; Middle Aged; Models, Statistical; Quinolones; Young Adult

2016
The development and application of a novel LC-MS/MS method for the measurement of Dolutegravir, Elvitegravir and Cobicistat in human plasma.
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2016, Aug-01, Volume: 1027

    Topics: Anti-HIV Agents; Chromatography, High Pressure Liquid; Cobicistat; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; Humans; Limit of Detection; Liquid-Liquid Extraction; Oxazines; Piperazines; Pyridones; Quinolones; Tandem Mass Spectrometry

2016
Elvitegravir/cobicistat-associated toxic optical neuropathy in an HIV-infected patient: a call for caution?
    Antiviral therapy, 2017, Volume: 22, Issue:5

    Topics: Antiretroviral Therapy, Highly Active; CD4 Lymphocyte Count; Cobicistat; HIV Infections; HIV-1; Humans; Male; Middle Aged; Optic Nerve Diseases; Quinolones; Viral Load

2017
Simultaneous quantification of tenofovir, emtricitabine, rilpivirine, elvitegravir and dolutegravir in mouse biological matrices by LC-MS/MS and its application to a pharmacokinetic study.
    Journal of pharmaceutical and biomedical analysis, 2016, Sep-10, Volume: 129

    Topics: Animals; Anti-Retroviral Agents; Chromatography, Liquid; Emtricitabine; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; Mice; Oxazines; Piperazines; Pyridones; Quinolones; Rilpivirine; Solid Phase Extraction; Tandem Mass Spectrometry; Tenofovir

2016
Development of a phenotypic susceptibility assay for HIV-1 integrase inhibitors.
    Journal of virological methods, 2016, Volume: 238

    Topics: Drug Resistance, Viral; Genotype; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Mutation; Oxazines; Phenotype; Piperazines; Pyridones; Quinolones; Raltegravir Potassium

2016
Efficacy of elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate as treatment for primary or recent HIV infection.
    The Journal of antimicrobial chemotherapy, 2017, Volume: 72, Issue:2

    Topics: Adult; Anti-HIV Agents; CD4 Lymphocyte Count; Cobicistat; Emtricitabine; HIV; HIV Infections; Humans; Male; Middle Aged; Quinolones; Retrospective Studies; Tenofovir; Treatment Outcome; Viral Load

2017
Pharmacokinetic interactions between cobicistat-boosted elvitegravir and darunavir in HIV-infected patients.
    The Journal of antimicrobial chemotherapy, 2017, 03-01, Volume: 72, Issue:3

    Topics: Adult; Aged; Aged, 80 and over; Anti-HIV Agents; Cobicistat; Darunavir; Drug Combinations; Drug Interactions; Female; HIV Infections; HIV-1; Humans; Male; Middle Aged; Quinolones; Young Adult

2017
Unravelling the dynamics of selection of multiresistant variants to integrase inhibitors in an HIV-1-infected child using ultra-deep sequencing.
    The Journal of antimicrobial chemotherapy, 2017, 03-01, Volume: 72, Issue:3

    Topics: Child; Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; High-Throughput Nucleotide Sequencing; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Mutation; Oxazines; Piperazines; Pyridones; Pyrrolidinones; Quinolones; Raltegravir Potassium; RNA, Viral; Selection, Genetic

2017
Tenofovir alafenamide, emtricitabine, elvitegravir, and cobicistat combination therapy for the treatment of HIV.
    Expert review of anti-infective therapy, 2017, Volume: 15, Issue:3

    Topics: Anti-HIV Agents; Clinical Trials, Phase I as Topic; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Cobicistat; Drug Combinations; Drug Interactions; Emtricitabine; HIV Infections; Humans; Quinolones; Tenofovir

2017
Tenofovir alafenamide and elvitegravir loaded nanoparticles for long-acting prevention of HIV-1 vaginal transmission.
    AIDS (London, England), 2017, 02-20, Volume: 31, Issue:4

    Topics: Adenine; Alanine; Animals; Delayed-Action Preparations; Disease Transmission, Infectious; Female; HIV Infections; Injections, Subcutaneous; Mice; Mice, SCID; Nanoparticles; Plasma; Quinolones; Tenofovir; Treatment Outcome; Vagina; Viral Load

2017
Comment on: Efficacy of elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate as treatment for primary or recent HIV infection.
    The Journal of antimicrobial chemotherapy, 2017, 05-01, Volume: 72, Issue:5

    Topics: Adenine; Anti-HIV Agents; Cobicistat; Deoxycytidine; Emtricitabine; HIV Infections; Humans; Organophosphonates; Quinolones; Tenofovir

2017
Alterations in cellular pharmacokinetics and pharmacodynamics of elvitegravir in response to ethanol exposure in HIV-1 infected monocytic (U1) cells.
    PloS one, 2017, Volume: 12, Issue:2

    Topics: Anti-HIV Agents; Cell Line; Drug Interactions; Ethanol; HIV Infections; HIV-1; Humans; Monocytes; Quinolones

2017
Structure-activity relationship study on anti-HIV 6-desfluoroquinolones.
    Journal of medicinal chemistry, 2008, Sep-11, Volume: 51, Issue:17

    Topics: Anti-HIV Agents; Cells, Cultured; HIV Infections; HIV-1; Humans; Quinolines; Quinolones; Structure-Activity Relationship

2008
HIV-2 integrase gene polymorphism and phenotypic susceptibility of HIV-2 clinical isolates to the integrase inhibitors raltegravir and elvitegravir in vitro.
    The Journal of antimicrobial chemotherapy, 2008, Volume: 62, Issue:5

    Topics: Amino Acid Sequence; Amino Acid Substitution; Catalytic Domain; Codon, Nonsense; Cohort Studies; Conserved Sequence; Drug Resistance, Viral; France; HIV Infections; HIV Integrase; HIV-1; HIV-2; Humans; Inhibitory Concentration 50; Integrase Inhibitors; Microbial Sensitivity Tests; Molecular Sequence Data; Mutation, Missense; Polymorphism, Genetic; Pyrrolidinones; Quinolones; Raltegravir Potassium

2008
Clade-specific HIV-1 integrase polymorphisms do not reduce raltegravir and elvitegravir phenotypic susceptibility.
    AIDS (London, England), 2008, Sep-12, Volume: 22, Issue:14

    Topics: Drug Resistance, Viral; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Polymorphism, Genetic; Pyrrolidinones; Quinolones; Raltegravir Potassium

2008
Elvitegravir, an oral HIV integrase inhibitor, for the potential treatment of HIV infection.
    Current opinion in investigational drugs (London, England : 2000), 2009, Volume: 10, Issue:2

    Topics: Biological Availability; Clinical Trials as Topic; Dose-Response Relationship, Drug; Drug Administration Routes; Drug Administration Schedule; Drug Combinations; Drug Evaluation, Preclinical; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Molecular Structure; Quinolones; Ritonavir

2009
Genetic barriers for integrase inhibitor drug resistance in HIV type-1 B and CRF02_AG subtypes.
    Antiviral therapy, 2009, Volume: 14, Issue:1

    Topics: DNA, Viral; Drug Resistance, Viral; Genetic Variation; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Mutation; Pyrrolidinones; Quinolones; Raltegravir Potassium; Sequence Analysis, DNA

2009
Treatment of delusional parasitosis with aripiprazole.
    Archives of dermatology, 2009, Volume: 145, Issue:4

    Topics: Adult; Antipsychotic Agents; Aripiprazole; Delusions; Female; HIV Infections; Humans; Lupus Erythematosus, Systemic; Male; Middle Aged; Piperazines; Quinolones; Skin Diseases, Parasitic

2009
A combined genotypic and phenotypic human immunodeficiency virus type 1 recombinant virus assay for the reverse transcriptase and integrase genes.
    Journal of virological methods, 2009, Volume: 161, Issue:2

    Topics: Drug Resistance, Multiple, Viral; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV Reverse Transcriptase; HIV-1; Humans; Microbial Sensitivity Tests; Polymorphism, Genetic; Pyrrolidinones; Quinolones; Raltegravir Potassium; Reproducibility of Results; Ribonuclease H, Human Immunodeficiency Virus; RNA, Viral; Sensitivity and Specificity; Sequence Analysis, DNA

2009
Synthesis, antiviral activity and molecular modeling of oxoquinoline derivatives.
    Bioorganic & medicinal chemistry, 2009, Aug-01, Volume: 17, Issue:15

    Topics: Animals; Anti-HIV Agents; Cell Survival; Chlorocebus aethiops; HIV Infections; HIV-1; Humans; Leukocytes, Mononuclear; Models, Molecular; Molecular Structure; Quinolones; Structure-Activity Relationship; Vero Cells

2009
[New antiretroviral drug classes in HIV therapy].
    MMW Fortschritte der Medizin, 2009, Apr-30, Volume: 151, Issue:18

    Topics: Anti-HIV Agents; CCR5 Receptor Antagonists; Cyclohexanes; HIV Fusion Inhibitors; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Maraviroc; Piperazines; Pyrimidines; Pyrrolidinones; Quinolones; Raltegravir Potassium; Succinates; Triazoles; Triterpenes; Viral Load

2009
Single-tablet Quad regimen achieves high rate of virologic suppression.
    AIDS patient care and STDs, 2010, Volume: 24, Issue:3

    Topics: Adenine; Anti-HIV Agents; Atazanavir Sulfate; CD4 Lymphocyte Count; Clinical Trials, Phase II as Topic; Cytochrome P-450 CYP3A Inhibitors; Deoxycytidine; Double-Blind Method; Drug Combinations; Drug Therapy, Combination; Efavirenz, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV Infections; HIV-1; Humans; Multicenter Studies as Topic; Oligopeptides; Organophosphonates; Organophosphorus Compounds; Oxazines; Pyridines; Quinolones; Randomized Controlled Trials as Topic; Ritonavir; Treatment Outcome; Viral Load

2010
Natural polymorphisms of integrase among HIV type 1-infected South African patients.
    AIDS research and human retroviruses, 2010, Volume: 26, Issue:4

    Topics: Amino Acid Sequence; Drug Resistance, Multiple, Viral; Genetic Variation; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Molecular Sequence Data; Phylogeny; Polymorphism, Single Nucleotide; Pyrrolidinones; Quinolones; Raltegravir Potassium; RNA, Viral; South Africa

2010
HIV-1 resistance patterns to integrase inhibitors in antiretroviral-experienced patients with virological failure on raltegravir-containing regimens.
    The Journal of antimicrobial chemotherapy, 2010, Volume: 65, Issue:6

    Topics: Amino Acid Substitution; Drug Resistance, Viral; Genotype; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Microbial Sensitivity Tests; Mutation, Missense; Prospective Studies; Pyrrolidinones; Quinolones; Raltegravir Potassium; RNA, Viral; Sequence Analysis, DNA; Treatment Failure; Viral Load

2010
Studies of anti-HIV transcription inhibitor quinolones: identification of potent N1-vinyl derivatives.
    ChemMedChem, 2010, Nov-08, Volume: 5, Issue:11

    Topics: Anti-HIV Agents; Cell Line; HIV Infections; Humans; Quinolones; Structure-Activity Relationship; Transcription, Genetic; Vinyl Compounds; Virus Replication

2010
Increased aripiprazole concentrations in an HIV-positive male concurrently taking duloxetine, darunavir, and ritonavir.
    The Annals of pharmacotherapy, 2010, Volume: 44, Issue:11

    Topics: Adult; Antidepressive Agents; Antipsychotic Agents; Anxiety; Aripiprazole; Cytochrome P-450 Enzyme Inhibitors; Darunavir; Depression; Dose-Response Relationship, Drug; Duloxetine Hydrochloride; HIV Infections; HIV Protease Inhibitors; Humans; Male; Piperazines; Quinolones; Ritonavir; Sulfonamides; Thiophenes

2010
Structural modifications of quinolone-3-carboxylic acids with anti-HIV activity.
    Bioorganic & medicinal chemistry, 2011, Aug-15, Volume: 19, Issue:16

    Topics: Anti-HIV Agents; Carboxylic Acids; Cell Line, Tumor; Cell Survival; HIV Infections; HIV Seropositivity; HIV-1; Humans; Models, Molecular; Quinolones; Structure-Activity Relationship

2011
Microwave assisted organic synthesis (MAOS) of small molecules as potential HIV-1 integrase inhibitors.
    Molecules (Basel, Switzerland), 2011, Aug-11, Volume: 16, Issue:8

    Topics: Green Chemistry Technology; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Indoles; Kinetics; Magnetic Resonance Spectroscopy; Microwaves; Models, Molecular; Molecular Structure; Pyrrolidinones; Quinolones; Raltegravir Potassium; Small Molecule Libraries; Structure-Activity Relationship

2011
Elvitegravir: a once daily alternative to raltegravir.
    The Lancet. Infectious diseases, 2012, Volume: 12, Issue:1

    Topics: Anti-Retroviral Agents; Female; HIV Infections; HIV-1; Humans; Male; Pyrrolidinones; Quinolones; Raltegravir Potassium

2012
Molecular dynamics approaches estimate the binding energy of HIV-1 integrase inhibitors and correlate with in vitro activity.
    Antimicrobial agents and chemotherapy, 2012, Volume: 56, Issue:1

    Topics: Amino Acid Substitution; Binding Sites; DNA, Viral; Drug Design; Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Molecular Dynamics Simulation; Mutation; Oxazines; Piperazines; Protein Binding; Pyridones; Pyrrolidinones; Quantitative Structure-Activity Relationship; Quinolones; Raltegravir Potassium; Spumavirus; Thermodynamics

2012
In vitro resistance selections using elvitegravir, raltegravir, and two metabolites of elvitegravir M1 and M4.
    Antiviral research, 2012, Volume: 93, Issue:2

    Topics: Cell Line; Drug Resistance, Viral; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Mutation; Pyrrolidinones; Quinolones; Raltegravir Potassium

2012
Broad phenotypic cross-resistance to elvitegravir in HIV-infected patients failing on raltegravir-containing regimens.
    Antimicrobial agents and chemotherapy, 2012, Volume: 56, Issue:6

    Topics: Drug Resistance, Viral; Genotype; HIV Infections; HIV Integrase Inhibitors; Humans; Molecular Sequence Data; Pyrrolidinones; Quinolones; Raltegravir Potassium

2012
Genetic barrier to the development of resistance to integrase inhibitors in HIV-1 subtypes CRF01_AE and B.
    Intervirology, 2012, Volume: 55, Issue:4

    Topics: Amino Acid Substitution; Drug Resistance, Viral; Genotype; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Mutant Proteins; Mutation, Missense; Oxazines; Piperazines; Pyridones; Pyrrolidinones; Quinolones; Raltegravir Potassium; RNA, Viral; Sequence Analysis, DNA

2012
The elvitegravir Quad pill: the first once-daily dual-target anti-HIV tablet.
    Expert opinion on investigational drugs, 2012, Volume: 21, Issue:7

    Topics: Adenine; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Carbamates; Clinical Trials as Topic; Deoxycytidine; Drug Administration Schedule; Drug Combinations; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV Infections; Humans; Organophosphonates; Quinolones; Tablets; Thiazoles

2012
[A single tablet against HIV: new combination preparation improves therapy].
    Deutsche medizinische Wochenschrift (1946), 2012, Volume: 137, Issue:34-35

    Topics: Adenine; Alkynes; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; Benzoxazines; Carbamates; CD4 Lymphocyte Count; Clinical Trials, Phase III as Topic; Cobicistat; Cyclopropanes; Deoxycytidine; Double-Blind Method; Drug Combinations; Drug Resistance, Viral; Emtricitabine; Glomerular Filtration Rate; HIV Infections; Humans; Oligopeptides; Organophosphonates; Pyridines; Quinolones; Randomized Controlled Trials as Topic; Ritonavir; Tenofovir; Thiazoles; Viral Load

2012
FDA approves new 4-drug once-a-day HIV treatment.
    AIDS policy & law, 2012, Volume: 27, Issue:11

    Topics: Adenine; Carbamates; Cobicistat; Deoxycytidine; Drug Administration Schedule; Drug Approval; Drug Combinations; Emtricitabine; HIV Infections; Humans; Organophosphonates; Quinolones; Tenofovir; Thiazoles; United States; United States Food and Drug Administration

2012
A 4-drug combination (Stribild) for HIV.
    The Medical letter on drugs and therapeutics, 2012, Nov-26, Volume: 54, Issue:1404

    Topics: Adenine; Anti-HIV Agents; Carbamates; Clinical Trials as Topic; Cobicistat; Deoxycytidine; Double-Blind Method; Drug Approval; Drug Combinations; Drug Interactions; Drug Resistance, Multiple, Viral; Emtricitabine; HIV; HIV Infections; Humans; Organophosphonates; Quinolones; Randomized Controlled Trials as Topic; Tenofovir; Thiazoles; United States; United States Food and Drug Administration

2012
Elvitegravir/cobicistat, mirabegron, and linaclotide.
    Journal of the American Pharmacists Association : JAPhA, 2012, Volume: 52, Issue:6

    Topics: Acetanilides; Adenine; Anti-Retroviral Agents; Carbamates; Constipation; Deoxycytidine; Drug Combinations; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV Infections; HIV-1; Humans; Organophosphonates; Peptides; Quinolones; Thiazoles; Urinary Bladder, Overactive

2012
Novel HIV-1 treatment Stribild™ gains regulatory approval.
    Expert review of clinical pharmacology, 2012, Volume: 5, Issue:6

    Topics: Adenine; Anti-HIV Agents; Carbamates; Deoxycytidine; Drug Approval; Drug Combinations; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV; HIV Infections; Humans; Organophosphonates; Quinolones; Thiazoles

2012
Improved adherence expected with new HIV combo treatment.
    Managed care (Langhorne, Pa.), 2012, Volume: 21, Issue:11

    Topics: Adenine; Aged; Aged, 80 and over; Anti-HIV Agents; Carbamates; Deoxycytidine; Drug Combinations; Drug Labeling; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV Infections; Humans; Medication Adherence; Middle Aged; Organophosphonates; Quinolones; Randomized Controlled Trials as Topic; Thiazoles; United States

2012
Multiple choices for HIV therapy with integrase strand transfer inhibitors.
    Retrovirology, 2012, Dec-19, Volume: 9

    Topics: Clinical Trials as Topic; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; HIV-1; Humans; Oxazines; Piperazines; Pyridones; Pyrrolidinones; Quinolones; Raltegravir Potassium

2012
A review of rilpivirine and elvitegravir resistance features and implications for treatment sequencing.
    HIV clinician, 2012,Autumn, Volume: 24, Issue:4

    Topics: Drug Administration Schedule; Drug Resistance, Viral; Drug Therapy, Combination; HIV Infections; HIV Integrase Inhibitors; Humans; Nitriles; Pyrimidines; Quinolones; Reverse Transcriptase Inhibitors; Rilpivirine

2012
Characterization of pathogenic Escherichia coli in human immunodeficiency virus-related diarrhea in Senegal.
    The Journal of infectious diseases, 2004, Jan-01, Volume: 189, Issue:1

    Topics: Anti-Bacterial Agents; Bacterial Adhesion; Case-Control Studies; Child; Diarrhea; Drug Resistance, Multiple, Bacterial; Escherichia coli; Escherichia coli Infections; Feces; Genes, Bacterial; HIV Infections; HIV-1; HIV-2; Humans; Microbial Sensitivity Tests; Prevalence; Quinolones; Risk Factors; Senegal; Virulence; Virulence Factors

2004
Mitochondrial toxicity associated with HAART following liver transplantation in an HIV-infected recipient.
    Liver transplantation : official publication of the American Association for the Study of Liver Diseases and the International Liver Transplantation Society, 2004, Volume: 10, Issue:5

    Topics: Acidosis, Lactic; Adult; Antiretroviral Therapy, Highly Active; Azepines; Biopsy, Needle; Comorbidity; Fluoroquinolones; Hepatitis C; HIV Infections; Humans; Liver; Liver Transplantation; Male; Mitochondria, Liver; Necrosis; Postoperative Period; Quinolones

2004
Novel in vivo model for the study of human immunodeficiency virus type 1 transcription inhibitors: evaluation of new 6-desfluoroquinolone derivatives.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:4

    Topics: Animals; Anti-HIV Agents; Cell Line; Disease Models, Animal; HIV Infections; HIV-1; Humans; Mice; Mice, SCID; Models, Biological; Quinolones

2007
New results for integrase inhibitor.
    AIDS patient care and STDs, 2007, Volume: 21, Issue:4

    Topics: Drug Administration Schedule; HIV Infections; HIV Integrase Inhibitors; Humans; Quinolones; Randomized Controlled Trials as Topic

2007
Resistance to integrase inhibitors.
    Journal of HIV therapy, 2007, Volume: 12, Issue:4

    Topics: Drug Resistance, Viral; HIV Infections; HIV Integrase Inhibitors; Humans; Quinolones

2007
Prior antimicrobials and staphylococcal bacteremia in HIV-infected patients.
    AIDS (London, England), 1997, Volume: 11, Issue:10

    Topics: Adult; AIDS-Related Opportunistic Infections; Anti-Bacterial Agents; Bacteremia; Case-Control Studies; Cohort Studies; Drug Resistance, Microbial; Female; HIV Infections; Humans; Macrolides; Male; Multivariate Analysis; Pentamidine; Quinolones; Rifabutin; Risk Factors; Staphylococcal Infections; Sulfamethoxazole; Trimethoprim

1997
QSAR study and VolSurf characterization of anti-HIV quinolone library.
    Journal of computer-aided molecular design, 2001, Volume: 15, Issue:3

    Topics: Anti-HIV Agents; Computer-Aided Design; Databases, Factual; Drug Design; HIV; HIV Infections; Humans; Models, Chemical; Multivariate Analysis; Quantitative Structure-Activity Relationship; Quinolones; Software

2001
Campylobacter laridis colitis in a human immunodeficiency virus-positive patient treated with a quinolone.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 1992, Volume: 15, Issue:1

    Topics: Adult; Campylobacter Infections; Colitis; Female; HIV Infections; Humans; Quinolones

1992
[Acute Campylobacter jejuni enterocolitis resistant to quinolones in an HIV-positive patient].
    Enfermedades infecciosas y microbiologia clinica, 1992, Volume: 10, Issue:5

    Topics: Adult; Campylobacter Infections; Campylobacter jejuni; Drug Resistance, Microbial; Enterocolitis; HIV Infections; Humans; Male; Quinolones

1992
[In vitro activity of twenty antibiotics against Rhodococcus equi].
    Pathologie-biologie, 1991, Volume: 39, Issue:5

    Topics: Actinomycetales Infections; Aminoglycosides; Anti-Bacterial Agents; Dose-Response Relationship, Drug; Doxycycline; Drug Resistance, Microbial; HIV Infections; Humans; In Vitro Techniques; Lactams; Macrolides; Opportunistic Infections; Quinolones; Rhodococcus; Rifampin

1991