Page last updated: 2024-08-17

carbostyril and African Sleeping Sickness

carbostyril has been researched along with African Sleeping Sickness in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (75.00)24.3611
2020's1 (25.00)2.80

Authors

AuthorsStudies
Engstler, M; Holzgrabe, U; Kirchner, L; Meinel, L; Weinmann, J1
Al-Momani, E; Berninger, M; Erk, C; Fuß, A; Güntzel, P; Holzgrabe, U; Israel, I; Raschig, M; Samnick, S; Skaf, J1
Biot, C; Dubar, F; Forge, D; Loiseau, PM; Pomel, S1
Braunschweig, H; Damme, A; Engstler, M; Hiltensperger, G; Holzgrabe, U; Jones, NG; Jung, J; Kaiser, M; Meinel, L; Niedermeier, S; Puhl, S; Stich, A1

Other Studies

4 other study(ies) available for carbostyril and African Sleeping Sickness

ArticleYear
Design, synthesis and biological evaluations of quinolone amides against African trypanosomiasis with improved solubility.
    European journal of medicinal chemistry, 2023, Mar-15, Volume: 250

    Topics: Amides; Animals; Humans; Quinolones; Solubility; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2023
Fluorine walk: The impact of fluorine in quinolone amides on their activity against African sleeping sickness.
    European journal of medicinal chemistry, 2018, May-25, Volume: 152

    Topics: Amides; Animals; Cells, Cultured; Dose-Response Relationship, Drug; Fluorine; Humans; Mice; Molecular Structure; Quinolones; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2018
New heterocyclic compounds: Synthesis and antitrypanosomal properties.
    Bioorganic & medicinal chemistry, 2015, Aug-15, Volume: 23, Issue:16

    Topics: Aminoquinolines; Animals; Benzimidazoles; Cell Line; Ferrous Compounds; Halogenation; Heterocyclic Compounds; Humans; Metallocenes; Mice; Quinolines; Quinolones; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2015
Synthesis and structure-activity relationships of new quinolone-type molecules against Trypanosoma brucei.
    Journal of medicinal chemistry, 2012, Mar-22, Volume: 55, Issue:6

    Topics: Acute Disease; Animals; Cell Line; DNA Topoisomerases, Type II; DNA, Kinetoplast; Mice; Microscopy, Fluorescence; Mitochondria; Models, Molecular; Morpholines; Quinolones; Structure-Activity Relationship; Topoisomerase II Inhibitors; Trypanocidal Agents; Trypanosoma brucei gambiense; Trypanosoma brucei rhodesiense; Trypanosomiasis, African

2012