Page last updated: 2024-09-04

canertinib and Breast Neoplasms

canertinib has been researched along with Breast Neoplasms in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (55.56)29.6817
2010's4 (44.44)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Grunt, TW; Gschwantler-Kaulich, D; Kölbl, H; Muhr, D; Singer, CF; Wagner, R1
Arun, BK; Franco, SX; Johnston, SR; Letrent, SP; Martin, M; Rixe, O; Rugo, HS; Yardley, DA1
Benjaminsen, RV; Christiansen, IJ; Emdal, KB; Frogne, T; Kirkegaard, T; Lykkesfeldt, AE; Norrie, IC; Sonne-Hansen, K1
Amir, E; Ocaña, A1
Berger, W; Brünner-Kubath, C; Grunt, TW; Grusch, M; Marian, B; Saferding, V; Shabbir, W; Singer, CF; Valent, P; Wagner, R; Zielinski, CC1
Pandiella, A; Sánchez-Martín, M1
Allen, LF; Eiseman, IA; Elliott, WL; Fry, DW; Lenehan, PF1
Allen, LF; Eiseman, IA; Fry, DW; Lenehan, PF1
Brose, MS; Flaherty, KT1

Reviews

4 review(s) available for canertinib and Breast Neoplasms

ArticleYear
Irreversible pan-ErbB tyrosine kinase inhibitors and breast cancer: current status and future directions.
    Cancer treatment reviews, 2009, Volume: 35, Issue:8

    Topics: Afatinib; Aminoquinolines; Aniline Compounds; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Biomarkers, Tumor; Breast Neoplasms; Drug Resistance, Neoplasm; ErbB Receptors; Female; Forecasting; Gene Expression Regulation, Neoplastic; Humans; Lapatinib; Morpholines; Prognosis; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Quinazolines; Quinolines; Trastuzumab; Up-Regulation

2009
Potential benefits of the irreversible pan-erbB inhibitor, CI-1033, in the treatment of breast cancer.
    Seminars in oncology, 2002, Volume: 29, Issue:3 Suppl 11

    Topics: Animals; Antineoplastic Agents; Breast Neoplasms; ErbB Receptors; Female; Humans; Mice; Morpholines; Protein-Tyrosine Kinases; Receptor, ErbB-2; Receptor, ErbB-3; Signal Transduction

2002
CI-1033, an irreversible pan-erbB receptor inhibitor and its potential application for the treatment of breast cancer.
    Seminars in oncology, 2003, Volume: 30, Issue:5 Suppl 16

    Topics: Animals; Antineoplastic Agents; Breast Neoplasms; Clinical Trials, Phase I as Topic; Drug Screening Assays, Antitumor; Humans; Ligands; Morpholines; Neoplasms; Receptor Protein-Tyrosine Kinases; Signal Transduction

2003
Her-2 targeted therapy: beyond breast cancer and trastuzumab.
    Current oncology reports, 2006, Volume: 8, Issue:2

    Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Breast Neoplasms; Colorectal Neoplasms; Female; Humans; Lapatinib; Morpholines; Neoplasms; Ovarian Neoplasms; Protein Kinase Inhibitors; Quinazolines; Receptor, ErbB-2; Signal Transduction; Trastuzumab

2006

Trials

1 trial(s) available for canertinib and Breast Neoplasms

ArticleYear
A randomized, phase II, dose-finding study of the pan-ErbB receptor tyrosine-kinase inhibitor CI-1033 in patients with pretreated metastatic breast cancer.
    Cancer chemotherapy and pharmacology, 2009, Volume: 64, Issue:6

    Topics: Adult; Aged; Breast Neoplasms; Disease-Free Survival; ErbB Receptors; Female; Humans; Kaplan-Meier Estimate; Middle Aged; Morpholines; Neoplasm Metastasis; Receptor, ErbB-2; Receptor, ErbB-3; Receptor, ErbB-4; Receptors, Estrogen; Treatment Outcome

2009

Other Studies

4 other study(ies) available for canertinib and Breast Neoplasms

ArticleYear
HER Specific TKIs Exert Their Antineoplastic Effects on Breast Cancer Cell Lines through the Involvement of STAT5 and JNK.
    PloS one, 2016, Volume: 11, Issue:1

    Topics: Afatinib; Antineoplastic Agents; Apoptosis; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; ErbB Receptors; Female; Humans; Inhibitory Concentration 50; JNK Mitogen-Activated Protein Kinases; Lapatinib; MAP Kinase Signaling System; Morpholines; Phosphorylation; Protein Kinase Inhibitors; Protein Processing, Post-Translational; Quinazolines; STAT5 Transcription Factor

2016
Breast cancer cells can switch between estrogen receptor alpha and ErbB signaling and combined treatment against both signaling pathways postpones development of resistance.
    Breast cancer research and treatment, 2010, Volume: 121, Issue:3

    Topics: Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Cell Line, Tumor; Drug Resistance, Neoplasm; Estradiol; Estrogen Receptor alpha; Female; Fulvestrant; Humans; Morpholines; Oncogene Proteins v-erbB; Signal Transduction

2010
The PI3 kinase/mTOR blocker NVP-BEZ235 overrides resistance against irreversible ErbB inhibitors in breast cancer cells.
    Breast cancer research and treatment, 2011, Volume: 129, Issue:2

    Topics: Aminoquinolines; Aniline Compounds; Antineoplastic Agents; Blotting, Western; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Enzyme Activation; ErbB Receptors; Female; Humans; Imidazoles; Molecular Targeted Therapy; Morpholines; Ovarian Neoplasms; Phosphatidylinositol 3-Kinase; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Quinolines; Signal Transduction; Time Factors; TOR Serine-Threonine Kinases; Transfection

2011
Differential action of small molecule HER kinase inhibitors on receptor heterodimerization: therapeutic implications.
    International journal of cancer, 2012, Jul-01, Volume: 131, Issue:1

    Topics: Aminoquinolines; Aniline Compounds; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; ErbB Receptors; Erlotinib Hydrochloride; Female; Gefitinib; Humans; Lapatinib; Morpholines; Protein Kinase Inhibitors; Protein Multimerization; Quinazolines; Quinolines; Receptor, ErbB-2; Trastuzumab

2012