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bupranolol and Muscle Relaxation

bupranolol has been researched along with Muscle Relaxation in 26 studies

Bupranolol: An adrenergic-beta-2 antagonist that has been used for cardiac arrhythmia, angina pectoris, hypertension, glaucoma, and as an antithrombotic.

Muscle Relaxation: That phase of a muscle twitch during which a muscle returns to a resting position.

Research Excerpts

ExcerptRelevanceReference
"(+)-Pindolol was less potent as antagonist of the relaxant effects of (-)-noradrenaline on trachea than against those of (-)-adrenaline, (-)-isoprenaline and (+/-)-salbutamol."1.27Stimulant and blocking effects of optical isomers of pindolol on the sinoatrial node and trachea of guinea pig. Role of beta-adrenoceptor subtypes in the dissociation between blockade and stimulation. ( Kaumann, AJ; Lemoine, H; Walter, M, 1984)

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-19902 (7.69)18.7374
1990's10 (38.46)18.2507
2000's14 (53.85)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Akimoto, Y1
Horinouchi, T17
Tanaka, Y2
Koike, K18
Doheny, HC1
Lynch, CM1
Smith, TJ1
Morrison, JJ1
Yamashita, Y1
Michikawa, H1
Clouse, AK1
Riedel, E1
Hieble, JP1
Westfall, TD1
Walter, M1
Lemoine, H2
Kaumann, AJ2
Takayanagi, I3
Ichino, T1
Koshikawa, H2
Nagatomo, T1
Geyer, O1
Bar-Ilan, A1
Nachman, R1
Lazar, M1
Oron, Y1
Igawa, Y1
Yamazaki, Y1
Takeda, H1
Akahane, M1
Ajisawa, Y1
Yoneyama, T1
Nishizawa, O1
Tsujitani, M1
Brawley, L1
Shaw, AM1
MacDonald, A1
Yamamoto, Y1
Nakagawa, Y1
Wakabayashi, M1
Satoh, H1
Endoh, M1

Other Studies

26 other studies available for bupranolol and Muscle Relaxation

ArticleYear
The beta2- and beta3-adrenoceptor-mediated relaxation induced by fenoterol in guinea pig taenia caecum.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2002, Volume: 38, Issue:4-5

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Butoxamine; Cecum; Dose-

2002
Functional coupling of beta3-adrenoceptors and large conductance calcium-activated potassium channels in human uterine myocytes.
    The Journal of clinical endocrinology and metabolism, 2005, Volume: 90, Issue:10

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Bupranolol; Dose-Response Relationship, Drug;

2005
Pharmacological characterization of the beta-adrenoceptor that mediates the relaxant response to noradrenaline in guinea-pig tracheal smooth muscle.
    Naunyn-Schmiedeberg's archives of pharmacology, 2007, Volume: 375, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Antagonists; A

2007
The effects and selectivity of beta-adrenoceptor agonists in rat myometrium and urinary bladder.
    European journal of pharmacology, 2007, Nov-14, Volume: 573, Issue:1-3

    Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-3 Recep

2007
Stimulant and blocking effects of optical isomers of pindolol on the sinoatrial node and trachea of guinea pig. Role of beta-adrenoceptor subtypes in the dissociation between blockade and stimulation.
    Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 327, Issue:2

    Topics: Animals; Bupranolol; Cimetidine; Female; Guinea Pigs; Heart Rate; In Vitro Techniques; Isoproterenol

1984
A model for the interaction of competitive antagonists with two receptor-subtypes characterized by a Schild-plot with apparent slope unity. Agonist-dependent enantiomeric affinity ratios for bupranolol in tracheae but not in right atria of guinea pigs.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 322, Issue:2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Dose-Response Relationsh

1983
Possible mechanisms of beta-adrenoceptor-mediated relaxation induced by noradrenaline in guinea pig taenia caecum.
    European journal of pharmacology, 1995, Jun-12, Volume: 279, Issue:2-3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Cecum; Cyclic AMP; Guine

1995
Effect of bupranolol on CGP 12177-induced relaxation and cAMP accumulation in the guinea pig taenia caecum.
    General pharmacology, 1995, Volume: 26, Issue:8

    Topics: Adrenergic beta-Antagonists; Animals; Bupranolol; Cyclic AMP; Dose-Response Relationship, Drug; Guin

1995
Beta3-adrenoceptors mediate relaxation of guinea pig taenia caecum by BRL37344A and BRL35135A.
    European journal of pharmacology, 1997, Sep-10, Volume: 334, Issue:2-3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Cecum; Dose-Response Rel

1997
Beta3-adrenergic relaxation of bovine iris sphincter.
    FEBS letters, 1998, Jun-16, Volume: 429, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Bupranolol; Cattle; Colfo

1998
Possible beta 3-adrenoceptor-mediated relaxation of the human detrusor.
    Acta physiologica Scandinavica, 1998, Volume: 164, Issue:1

    Topics: Adrenergic Antagonists; Adrenergic beta-Agonists; Adult; Aged; Bupranolol; Dobutamine; Dose-Response

1998
Characterization of atypical beta-adrenoceptors in the guinea pig duodenum.
    European journal of pharmacology, 1999, Jul-02, Volume: 376, Issue:1-2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Catecholamines; Duodenum

1999
Effect of bupranolol for BRL37344 and noradrenaline-induced relaxations mediating atypical beta/beta3-adrenoceptor in rat oesophageal muscularis mucosae.
    General pharmacology, 1999, Volume: 33, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolo

1999
Pharmacological analysis of atypical beta-adrenoceptors in the guinea pig gastric fundus using the beta(3)-adrenoceptor antagonist bupranolol.
    Pharmacology, 1999, Volume: 59, Issue:6

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atenolol; Bupranolol; Butoxamine; Ca

1999
[Pharmacological analysis of atypical beta-adrenoceptors in the guinea pig gastrointestinal tissue systems].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1999, Volume: 114 Suppl 1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Digestive System; Duoden

1999
Beta 1-, beta 2- and atypical beta-adrenoceptor-mediated relaxation in rat isolated aorta.
    British journal of pharmacology, 2000, Volume: 129, Issue:4

    Topics: Acetylcholine; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Ani

2000
Partial agonist activity of carteolol on atypical beta-adrenoceptors in the guinea pig duodenum.
    European journal of pharmacology, 2000, Sep-01, Volume: 403, Issue:1-2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Carteolol; Dose-Response

2000
The beta3-adrenoceptor-mediated relaxation induced by epinephrine in guinea pig taenia caecum.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2000, Volume: 36, Issue:3

    Topics: Animals; Bupranolol; Cecum; Cyclic AMP; Epinephrine; Guinea Pigs; In Vitro Techniques; Male; Muscle

2000
Partial agonistic effects of carteolol on atypical beta-adrenoceptors in the guinea pig gastric fundus.
    Japanese journal of pharmacology, 2000, Volume: 84, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Carteolol; Gastric Fundu

2000
(+/-)-Pindolol acts as a partial agonist at atypical beta-adrenoceptors in the guinea pig duodenum.
    Japanese journal of pharmacology, 2001, Volume: 85, Issue:1

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Recep

2001
Functional identification of beta3-adrenoceptors in the guinea-pig ileum using the non-selective beta-adrenoceptor antagonist (+/-)-bupranolol.
    Journal of autonomic pharmacology, 2000, Volume: 20, Issue:4

    Topics: Adipocytes; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Catecholamin

2000
Functional properties of atypical beta-adrenoceptors on the guinea pig duodenum.
    European journal of pharmacology, 2001, Mar-23, Volume: 416, Issue:1-2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Alprenolol; Animals; Bupranolol; C

2001
Agonistic activity of SR59230A at atypical beta-adrenoceptors in guinea pig gastric fundus and duodenum.
    European journal of pharmacology, 2001, Mar-23, Volume: 416, Issue:1-2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Dose-Response Relationsh

2001
Further evidence that (+/-)-carteolol-induced relaxation is mediated by beta2-adrenoceptors but not by beta3-adrenoceptors in the guinea pig taenia caecum.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2000, Volume: 36, Issue:5

    Topics: Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-3 Receptor Antagonists; Adrenergic beta-Anta

2000
Structure-activity relationship studies of (+/-)-terbutaline and (+/-)-fenoterol on beta3-adrenoceptors in the guinea pig gastric fundus.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2001, Volume: 37, Issue:3-4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atenolol; Bupranolol; Butoxamine; Fe

2001
Effects of a new cardiotonic agent 1,2-dihydro-6-methyl-2-oxo-5-[imidazo (1,2-a) pyridin-6-yl]-3-pyridine carbonitrile hydrochloride monohydrate (E-1020) on contractile force and cyclic AMP metabolism in canine ventricular muscle.
    Japanese journal of pharmacology, 1990, Volume: 52, Issue:2

    Topics: Amrinone; Animals; Bupranolol; Carbachol; Cardiotonic Agents; Cyclic AMP; Dogs; Female; Heart; Heart

1990