btm 1042 has been researched along with Muscle Contraction in 3 studies
*Muscle Contraction: A process leading to shortening and/or development of tension in muscle tissue. Muscle contraction occurs by a sliding filament mechanism whereby actin filaments slide inward among the myosin filaments. [MeSH]
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 2 (66.67) | 18.7374 |
1990's | 1 (33.33) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Kizawa, Y; Nakazo, K; Takayanagi, I | 1 |
Jackson, KN; Kachur, JF; Lowe, VC; Noronha-Blob, L; Sturm, BL | 1 |
Boer, R; Eltze, M; Lambrecht, G; Mutschler, E | 1 |
3 other study(ies) available for btm 1042 and Muscle Contraction
Article | Year |
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Possible mechanisms of a new type of antispasmodic drug, BTM-1042(cis-(--)-2,3-dihydro-3-(4-methyl-piperazinyl)methyl-2-phenyl-1,5-benzothiazepin-4(5H)-one dihydrochloride).
Topics: Animals; Binding Sites; Colon; Diaphragm; Drug Interactions; Electric Stimulation; Guinea Pigs; Ileum; Male; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Rabbits; Rats; Thiazepines; Trachea; Urinary Bladder; Vas Deferens | 1980 |
In vitro and in vivo antimuscarinic effects of (-)cis 2,3-dihydro-3-(4-methylpiperazinylmethyl)-2-phenyl-1,5 benzothiazepin-4-(5H)one HCl (BTM-1086) in guinea pig peripheral tissues.
Topics: Animals; Atropine; Calcium; Female; Guinea Pigs; Heart Atria; Ileum; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Neurons; Parasympatholytics; Piperidines; Pirenzepine; Structure-Activity Relationship; Thiazepines; Tumor Cells, Cultured; Urinary Bladder; Vas Deferens | 1990 |
Affinity profiles of BTM-1086 and BTM-1041 at muscarinic receptor subtypes and at H1- and alpha 1-receptors.
Topics: Adrenergic alpha-Antagonists; Animals; Cerebral Cortex; Female; Guinea Pigs; Heart; Histamine H1 Antagonists; Ileum; In Vitro Techniques; Male; Muscle Contraction; Myocardium; Parasympatholytics; Rabbits; Rats; Receptors, Adrenergic, alpha; Stereoisomerism; Thiazepines | 1989 |