bremazocine and Ache

bremazocine has been researched along with Ache in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19902 (18.18)18.7374
1990's3 (27.27)18.2507
2000's5 (45.45)29.6817
2010's1 (9.09)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Duarte, ID; Pacheco, CM; Pacheco, Dda F1
Amarante, LH; Duarte, ID1
Folk, JE; Linsenmayer, DC; Negus, SS; Rice, KC; Stevenson, GW1
Aceto, MD; Breeden, S; Broadbear, J; Grundt, P; Husbands, SM; Lewis, JW; Neilan, CL; Traynor, JR; Woods, JH1
Dortch-Carnes, J; Potter, DE1
da Fonseca Pacheco, CM; da Fonseca Pacheco, D; de Castro Perez, A; de Francischi, JN; Duarte, ID; Klein, A1
Iwamoto, ET; Martin, WR1
Angel, F; Chevalier, E; Dahl, SG; Friese, N; Junien, JL; Pascaud, X; Riviere, PJ1
Mamede Rosa, ML; Prado, WA1
Millan, MJ; Morris, BJ2

Reviews

2 review(s) available for bremazocine and Ache

ArticleYear
Bremazocine: a kappa-opioid agonist with potent analgesic and other pharmacologic properties.
    CNS drug reviews, 2005,Summer, Volume: 11, Issue:2

    Topics: Analgesics; Animals; Benzomorphans; Cardiovascular System; Disease Models, Animal; Diuresis; Humans; Motor Activity; Pain; Receptors, Opioid, kappa; Respiration; Signal Transduction; Synaptic Transmission

2005
Multiple opioid receptors.
    Medicinal research reviews, 1981,Winter, Volume: 1, Issue:4

    Topics: Analgesics; Animals; Behavior, Animal; Benzomorphans; Cyclazocine; Discrimination Learning; Dogs; Dopamine; Drug Tolerance; Electroencephalography; Humans; Macaca mulatta; Mice; Morphine; Morphine Dependence; Motor Activity; Nalorphine; Pain; Rabbits; Rats; Receptors, Dopamine; Receptors, Opioid; Receptors, Opioid, kappa; Seizures; Temperature

1981

Other Studies

9 other study(ies) available for bremazocine and Ache

ArticleYear
δ-Opioid receptor agonist SNC80 induces central antinociception mediated by Ca2+ -activated Cl- channels.
    The Journal of pharmacy and pharmacology, 2012, Volume: 64, Issue:8

    Topics: Analgesics, Opioid; Animals; Benzamides; Benzomorphans; Calcium; Cations; Chloride Channels; Enkephalins; Hot Temperature; Male; Mice; Mice, Inbred Strains; Niflumic Acid; Pain; Pain Threshold; Piperazines; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

2012
The kappa-opioid agonist (+/-)-bremazocine elicits peripheral antinociception by activation of the L-arginine/nitric oxide/cyclic GMP pathway.
    European journal of pharmacology, 2002, Nov-01, Volume: 454, Issue:1

    Topics: Analgesics; Animals; Arginine; Benzomorphans; Cyclic GMP; Guanylate Cyclase; Hyperalgesia; Male; Methylene Blue; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Pain; Phosphodiesterase Inhibitors; Purinones; Rats; Rats, Wistar; Receptors, Opioid, kappa

2002
Opioid interactions in rhesus monkeys: effects of delta + mu and delta + kappa agonists on schedule-controlled responding and thermal nociception.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 307, Issue:3

    Topics: Analgesics, Opioid; Animals; Benzamides; Benzeneacetamides; Benzomorphans; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Hot Temperature; Macaca mulatta; Male; Naltrexone; Narcotic Antagonists; Pain; Piperazines; Pyrrolidines; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reinforcement Schedule

2003
BU74, a complex oripavine derivative with potent kappa opioid receptor agonism and delayed opioid antagonism.
    European journal of pharmacology, 2005, Feb-21, Volume: 509, Issue:2-3

    Topics: Acetic Acid; Analgesics; Animals; Benzomorphans; Binding, Competitive; Bridged-Ring Compounds; Cell Line, Tumor; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Hot Temperature; Ileum; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Morphinans; Narcotic Antagonists; Pain; Pain Measurement; Radioligand Assay; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sulfur Radioisotopes; Vas Deferens

2005
The mu-opioid receptor agonist morphine, but not agonists at delta- or kappa-opioid receptors, induces peripheral antinociception mediated by cannabinoid receptors.
    British journal of pharmacology, 2008, Volume: 154, Issue:5

    Topics: Amidohydrolases; Analgesics, Opioid; Animals; Arachidonic Acids; Benzamides; Benzomorphans; Cannabinoid Receptor Modulators; Dinoprostone; Disease Models, Animal; Dose-Response Relationship, Drug; Enzyme Inhibitors; Hyperalgesia; Indoles; Male; Morphine; Organophosphonates; Pain; Pain Measurement; Piperazines; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

2008
Reversal by kappa-agonists of peritoneal irritation-induced ileus and visceral pain in rats.
    Life sciences, 1997, Volume: 60, Issue:9

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acetic Acid; Analgesics; Animals; Benzofurans; Benzomorphans; Cyclazocine; Fentanyl; Gastric Emptying; Intestinal Pseudo-Obstruction; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Pain; Peritoneum; Pyrroles; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Receptors, Opioid, mu; Thiophenes

1997
Antinociception induced by opioid or 5-HT agonists microinjected into the anterior pretectal nucleus of the rat.
    Brain research, 1997, May-16, Volume: 757, Issue:1

    Topics: Analgesics; Animals; Benzomorphans; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Male; Microinjections; Pain; Phenazocine; Piperazines; Quinoxalines; Rats; Rats, Wistar; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Serotonin; Serotonin Receptor Agonists

1997
Inability of an opioid antagonist lacking negative intrinsic activity to induce opioid receptor up-regulation in vivo.
    British journal of pharmacology, 1991, Volume: 102, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzomorphans; Binding, Competitive; Drinking; Eating; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Male; Narcotic Antagonists; Pain; Pain Measurement; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Sensory Thresholds; Up-Regulation

1991
Long-term blockade of mu-opioid receptors suggests a role in control of ingestive behaviour, body weight and core temperature in the rat.
    Brain research, 1988, May-31, Volume: 450, Issue:1-2

    Topics: Animals; Benzomorphans; Body Temperature Regulation; Body Weight; Circadian Rhythm; Drinking Behavior; Feeding Behavior; Fentanyl; Male; Naloxone; Pain; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, mu; Sufentanil

1988