Page last updated: 2024-08-21

benzoxazoles and Pain

benzoxazoles has been researched along with Pain in 24 studies

Research

Studies (24)

TimeframeStudies, this research(%)All Research%
pre-19904 (16.67)18.7374
1990's0 (0.00)18.2507
2000's6 (25.00)29.6817
2010's12 (50.00)24.3611
2020's2 (8.33)2.80

Authors

AuthorsStudies
Askari, K; Ghalebandi, S; Haghparast, A; Mousavi, Z; Zareie, F1
Gaikwad, NJ; Gaikwad, SS; Patil, ML1
Cato, MJ; Clements, MK; Daley, CJ; Filzen, T; Finger, EN; Gregan, Y; Henze, DA; Houghton, AK; Jovanovska, A; Kelly, MJ; Klein, R; Kraus, RL; Layton, ME; Lehman, HDGF; Li, Y; Liang, A; Majercak, JM; Mulhearn, JJ; Panigel, J; Pero, JE; Rossi, MA; Urban, MO; Wang, J; Wang, YH; Wolkenberg, SE1
Aoki, T; Hiyama, H; Kiso, T; Murai, N; Oka, H; Sekizawa, T; Watabiki, T1
Boccella, S; de Novellis, V; Farina, A; Guida, F; Iannotta, M; Luongo, L; Maione, S; Marabese, I; Palazzo, E; Serra, N1
Fazli-Tabaei, S; Haghparast, A; Karimi-Haghighi, S; Rezaee, L1
Alam, MS; Alam, P; Ali, Y; Bano, S; Dhulap, A; Haider, S; Hamid, H; Hussain, F; Kharbanda, C; Nazreen, S; Pasha, MA; Shafi, S; Umar, S1
Ali Reza, M; Azizi, H; Mirnajafi-Zadeh, J; Mohammad-Pour Kargar, H; Semnanian, S1
Babapour, V; Ezzatpanah, S; Haghparast, A1
Esmaeili, MH; Ezzatpanah, S; Haghparast, A; Reisi, Z1
Bradshaw, E; Broom, DC; Buck, ME; Coombs, S; Cortright, DN; Ford, KK; Krause, JE; Matchett, M; Matson, DJ; Meade, R; Ochoa, R; Sun, SH; Wustrow, DJ; Yu, W; Yuan, J1
Erdogan, H; Kelekci, NG; Koksal, M; Mercanoglu, GO1
Chen, XW; Ge, L; Huang, W; Song, B; Yan, JA; Yu, ZP1
Aktay, G; Erdoğan, H; Gökhan-Kelekçi, N; Köksal, M; Unüvar, S1
Holden, JE; Jeong, Y1
Alcin, E; Ayar, A; Kelestimur, H; Ozcan, M; Sahin, Z; Serhatlioglu, I1
Baghdoyan, HA; Lydic, R; Watson, CJ; Watson, SL1
Chiou, LC; Fu, SY; Ho, YC; Lee, HJ; Liao, HT; Liao, YY; Mackie, K; Teng, SF; Tung, LW1
Fun, HK; Isloor, AM; Shetty, P; Sundershan, S; Vijesh, AM1
Bacon, PA; Davies, J; Ring, FJ1
Lightfoot, RW1
Caliş, U; Erdoğan, H; Gökhan, N1
Miller, AR1
Vernon, WG1

Trials

4 trial(s) available for benzoxazoles and Pain

ArticleYear
Benoxaprofen--dose-range studies using quantitative thermography.
    The Journal of rheumatology. Supplement, 1980, Volume: 6

    Topics: Anti-Inflammatory Agents; Arthritis, Rheumatoid; Benzoxazoles; Clinical Trials as Topic; Dose-Response Relationship, Drug; Double-Blind Method; Humans; Indomethacin; Inflammation; Pain; Propionates; Thermography; Time Factors

1980
Benoxaprofen administered once a day: determination of optimum dosage schedule.
    The Journal of rheumatology. Supplement, 1980, Volume: 6

    Topics: Adult; Aged; Anti-Inflammatory Agents; Arthritis, Rheumatoid; Benzoxazoles; Clinical Trials as Topic; Double-Blind Method; Drug Administration Schedule; Female; Humans; Male; Middle Aged; Osteoarthritis; Pain; Propionates

1980
A comparative study of Parafon Forte tablets and soma compound in the treatment of painful skeletal muscle conditions.
    Current therapeutic research, clinical and experimental, 1976, Volume: 19, Issue:4

    Topics: Acetaminophen; Adolescent; Adult; Benzoxazoles; Carisoprodol; Chlorzoxazone; Drug Combinations; Female; Humans; Male; Middle Aged; Muscular Diseases; Pain; Spasm

1976
A double-blind evaluation of Parafon Forte in the treatment of musculo-skeletal back conditions.
    Current therapeutic research, clinical and experimental, 1972, Volume: 14, Issue:12

    Topics: Acetaminophen; Adolescent; Adult; Back; Benzoxazoles; Bone Diseases; Chlorzoxazone; Clinical Trials as Topic; Drug Combinations; Humans; Male; Middle Aged; Muscle Relaxants, Central; Muscular Diseases; Pain; Placebos; Spasm

1972

Other Studies

20 other study(ies) available for benzoxazoles and Pain

ArticleYear
Orexin receptors in the CA1 region of hippocampus modulate the stress-induced antinociceptive responses in an animal model of persistent inflammatory pain.
    Peptides, 2022, Volume: 147

    Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Benzoxazoles; CA1 Region, Hippocampal; Cyclophosphamide; Disease Models, Animal; Doxorubicin; Etoposide; Inflammation; Isoquinolines; Male; Microinjections; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Pain; Pain Measurement; Prednisone; Pyridines; Rats, Wistar; Stress, Psychological; Urea; Vincristine

2022
Anti-nociceptive and Anti-inflammatory Activity of Synthesized Novel Benzoxazole Derivatives.
    Anti-inflammatory & anti-allergy agents in medicinal chemistry, 2021, Volume: 20, Issue:4

    Topics: Analgesics; Animals; Anti-Inflammatory Agents; Benzoxazoles; Carrageenan; Disease Models, Animal; Edema; Male; Mice; Nociception; Pain; Plant Extracts

2021
Benzoxazolinone aryl sulfonamides as potent, selective Na
    Bioorganic & medicinal chemistry letters, 2017, 06-15, Volume: 27, Issue:12

    Topics: Administration, Oral; Analgesics; Animals; Benzoxazoles; Biological Availability; Disease Models, Animal; Dose-Response Relationship, Drug; Formaldehyde; Humans; Mice; Molecular Structure; Myocytes, Smooth Muscle; NAV1.7 Voltage-Gated Sodium Channel; Pain; Rats; Structure-Activity Relationship; Sulfonamides

2017
Analgesic effects of novel lysophosphatidic acid receptor 5 antagonist AS2717638 in rodents.
    Neuropharmacology, 2017, Volume: 126

    Topics: Analgesics; Animals; Benzoxazoles; Cells, Cultured; Cyclic AMP; Female; Hyperalgesia; Inflammation; Injections, Spinal; Isoquinolines; Lysophospholipids; Male; Mice, Inbred C57BL; Mice, Knockout; Neuralgia; Pain; Pain Threshold; Piperidines; Polyisoprenyl Phosphates; Rats, Inbred Lew; Rats, Sprague-Dawley; Receptors, Lysophosphatidic Acid

2017
Metabotropic glutamate receptor subtype 7 in the dorsal striatum oppositely modulates pain in sham and neuropathic rats.
    Neuropharmacology, 2018, Volume: 135

    Topics: Animals; Benzhydryl Compounds; Benzoxazoles; Corpus Striatum; Glutamic Acid; Hyperalgesia; Lidocaine; Male; Medulla Oblongata; Microinjections; Neuralgia; Neurons; Neuroprotective Agents; Pain; Rats; Receptors, Metabotropic Glutamate; Reticular Formation; Sciatic Nerve; Subthalamic Nucleus

2018
Effects of intrathecal administration of orexin-1 receptor antagonist on antinociceptive responses induced by chemical stimulation of lateral hypothalamus in an animal model of tonic nociception.
    Neuropeptides, 2018, Volume: 69

    Topics: Analgesics; Animals; Benzoxazoles; Hypothalamic Area, Lateral; Injections, Spinal; Male; Naphthyridines; Nociception; Orexin Receptor Antagonists; Orexin Receptors; Pain; Pain Measurement; Rats, Wistar; Spinal Cord; Urea

2018
Synthesis of novel 2-mercaptobenzoxazole based 1,2,3-triazoles as inhibitors of proinflammatory cytokines and suppressors of COX-2 gene expression.
    European journal of medicinal chemistry, 2014, Jun-23, Volume: 81

    Topics: Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzoxazoles; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cytokines; Edema; Gene Expression Regulation, Enzymologic; HeLa Cells; Humans; Inflammation; Mice; Models, Molecular; Pain; Rats; Rats, Wistar; Sulfhydryl Compounds; Triazoles; Tumor Cells, Cultured

2014
Microinjection of orexin-A into the rat locus coeruleus nucleus induces analgesia via cannabinoid type-1 receptors.
    Brain research, 2015, Oct-22, Volume: 1624

    Topics: Analgesics; Analysis of Variance; Animals; Benzoxazoles; Carrier Proteins; Dose-Response Relationship, Drug; Formaldehyde; Locus Coeruleus; Male; Microinjections; Naphthyridines; Orexins; Pain; Pain Measurement; Piperidines; Pyrazoles; Rats; Rats, Wistar; Urea

2015
Differential contribution of orexin receptors within the ventral tegmental area to modulation of persistent inflammatory pain.
    European journal of pain (London, England), 2016, Volume: 20, Issue:7

    Topics: Animals; Benzoxazoles; Carbachol; Hypothalamic Area, Lateral; Isoquinolines; Male; Naphthyridines; Nociception; Orexin Receptor Antagonists; Orexin Receptors; Pain; Pain Measurement; Pyridines; Rats; Rats, Wistar; Urea; Ventral Tegmental Area

2016
Functional interaction between orexin-1 and CB1 receptors in the periaqueductal gray matter during antinociception induced by chemical stimulation of the lateral hypothalamus in rats.
    European journal of pain (London, England), 2016, Volume: 20, Issue:10

    Topics: Animals; Benzoxazoles; Carbachol; Disease Models, Animal; Hypothalamic Area, Lateral; Male; Microinjections; Naphthyridines; Orexin Receptors; Orexins; Pain; Pain Measurement; Periaqueductal Gray; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Stimulation, Chemical; Urea

2016
Characterization of N-(adamantan-1-ylmethyl)-5-[(3R-amino-pyrrolidin-1-yl)methyl]-2-chloro-benzamide, a P2X7 antagonist in animal models of pain and inflammation.
    The Journal of pharmacology and experimental therapeutics, 2008, Volume: 327, Issue:3

    Topics: Adamantane; Animals; Anti-Inflammatory Agents, Non-Steroidal; Arthritis; Benzamides; Benzoxazoles; Calcium; Disease Models, Animal; Humans; Inflammation; Inhibitory Concentration 50; Pain; Purinergic P2 Receptor Antagonists; Quinolinium Compounds; Rats; Receptors, Purinergic P2X7

2008
Synthesis and evaluation of analgesic, anti-inflammatory and antioxidant activities of new 6-acyl-3-alkyl-5-methyl-2(3H)-benzoxazolones.
    Arzneimittel-Forschung, 2008, Volume: 58, Issue:8

    Topics: Analgesics, Non-Narcotic; Animals; Anti-Inflammatory Agents, Non-Steroidal; Antioxidants; Benzoxazoles; Carrageenan; Chemical Phenomena; Chemistry, Physical; Edema; Indicators and Reagents; Male; Mice; Pain; Stomach Ulcer

2008
Orexin affects dorsal root ganglion neurons: a mechanism for regulating the spinal nociceptive processing.
    Physiological research, 2008, Volume: 57, Issue:5

    Topics: Action Potentials; Animals; Benzoxazoles; Calcium Signaling; Ganglia, Spinal; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neurons; Neuropeptides; Orexin Receptors; Orexins; Pain; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Synaptic Transmission; Urea

2008
Synthesis and characterization of some new 2(3H)-benzoxazolones with analgesic and antiinflammatory activities.
    Journal of enzyme inhibition and medicinal chemistry, 2009, Volume: 24, Issue:1

    Topics: Analgesics; Animals; Anti-Inflammatory Agents; Benzoxazoles; Drug Evaluation, Preclinical; Edema; Mice; Pain; Structure-Activity Relationship

2009
The role of spinal orexin-1 receptors in posterior hypothalamic modulation of neuropathic pain.
    Neuroscience, 2009, Apr-10, Volume: 159, Issue:4

    Topics: Analgesics; Animals; Benzoxazoles; Carbachol; Cholinergic Agonists; Dose-Response Relationship, Drug; Female; Hypothalamus; Naphthyridines; Neurons; Orexin Receptors; Pain; Pain Measurement; Posterior Horn Cells; Random Allocation; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sciatic Neuropathy; Spinal Cord; Urea

2009
Orexins activates protein kinase C-mediated Ca(2+) signaling in isolated rat primary sensory neurons.
    Physiological research, 2010, Volume: 59, Issue:2

    Topics: Animals; Benzoxazoles; Calcium Signaling; Cells, Cultured; Ganglia, Spinal; Intracellular Signaling Peptides and Proteins; Naphthyridines; Neuropeptides; Neurotransmitter Agents; Nociceptors; Orexins; Pain; Protein Kinase C; Rats; Rats, Wistar; Sensory Receptor Cells; Urea

2010
Thermal nociception is decreased by hypocretin-1 and an adenosine A1 receptor agonist microinjected into the pontine reticular formation of Sprague Dawley rat.
    The journal of pain, 2010, Volume: 11, Issue:6

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Aging; Animals; Benzoxazoles; Hot Temperature; Intracellular Signaling Peptides and Proteins; Male; Microinjections; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Pain; Pain Measurement; Pons; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reticular Formation; Time Factors; Urea

2010
Activation of orexin 1 receptors in the periaqueductal gray of male rats leads to antinociception via retrograde endocannabinoid (2-arachidonoylglycerol)-induced disinhibition.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Oct-12, Volume: 31, Issue:41

    Topics: Analysis of Variance; Animals; Animals, Newborn; Arachidonic Acids; Benzoxazines; Benzoxazoles; Biphenyl Compounds; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Disease Models, Animal; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Estrenes; gamma-Aminobutyric Acid; Glycerides; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Intracellular Signaling Peptides and Proteins; Lactones; Male; Morpholines; Naphthalenes; Naphthyridines; Neural Inhibition; Neural Pathways; Neuropeptides; Orexin Receptors; Orexins; Orlistat; Pain; Pain Measurement; Patch-Clamp Techniques; Periaqueductal Gray; Piperidines; Pyrazoles; Pyrrolidinones; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea

2011
New pyrazole derivatives containing 1,2,4-triazoles and benzoxazoles as potent antimicrobial and analgesic agents.
    European journal of medicinal chemistry, 2013, Volume: 62

    Topics: Analgesics; Animals; Anti-Bacterial Agents; Antifungal Agents; Bacteria; Benzoxazoles; Dose-Response Relationship, Drug; Fungi; Microbial Sensitivity Tests; Molecular Structure; Pain; Pain Measurement; Pyrazoles; Rats; Rats, Wistar; Structure-Activity Relationship; Triazoles

2013
Synthesis of some novel 3-methyl-6-(2-substituted propanoyl/propyl)-2-benzoxazolinone derivatives and anti-nociceptive activity.
    Farmaco (Societa chimica italiana : 1989), 2001, Volume: 56, Issue:9

    Topics: Analgesics; Animals; Benzoxazoles; Female; Mice; Pain

2001