azacitidine has been researched along with Leukemia L 1210 in 65 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 57 (87.69) | 18.7374 |
1990's | 4 (6.15) | 18.2507 |
2000's | 3 (4.62) | 29.6817 |
2010's | 1 (1.54) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Abbasi, MM; Beisler, JA; Driscoll, JS; Kelley, JA | 1 |
Beisler, JA | 1 |
Abbasi, MM; Beisler, JA; Driscoll, JS | 3 |
Hansch, C; Khwaja, TA; Selassie, CD | 1 |
Cook, PD; McNamara, DJ | 1 |
Charbonneau, M; Momparler, LF; Momparler, RL; Raynal, NJ | 1 |
Momparler, LF; Momparler, RL; Raynal, NJ; Rivard, GE | 1 |
Bernstein, ML; Lemaire, M; Marquez, VE; Momparler, LF; Momparler, RL | 1 |
Huang, TH; Liu, JC; Plass, C; Potter, D; Smith, LT; Wang, SH; Wu, J; Wu, YZ | 1 |
Momparler, LF; Momparler, RL; Samson, J | 2 |
Covey, JM; Zaharko, DS | 4 |
Lee, MH; Sartorelli, AC | 1 |
Abbasi, MM; Beisler, JA; Glazer, RI; Peale, AL | 1 |
Glazer, RI; Hartman, KD | 1 |
Cihák, A; Veselý, J | 3 |
Cadman, E; Grant, S; Jakubowski, A; Rauscher, F | 1 |
Darzynkiewicz, Z; Melamed, MR; Staiano-Coico, L; Traganos, F | 1 |
Coulter, D; Presant, CA; Valeriote, F; Vietti, TJ | 1 |
Coulter, DM; Presant, CA; Valeriote, F; Vietti, TJ | 1 |
Cadman, E; Grant, S; Margolin, J; Rauscher, F | 1 |
Veselý, J | 2 |
Jones, PA; Momparler, RL; Wilson, VL | 1 |
Campbell, J; Li, ZR; Rustum, YM | 1 |
Blowers, CL; Buskirk, HH; Hanka, LJ; Li, LH; Neil, GL | 1 |
Pískala, A; Veselý, J | 2 |
Lu, LJ; Randerath, K | 1 |
Glazier, RI; Minford, J; Nichols, M; Shackney, S; Zwelling, LA | 1 |
Chabot, GG; Momparler, RL | 2 |
Jacquemin-Sablon, A; Segal-Bendirdjian, E | 2 |
Fabianowska-Majewska, K; Wyczechowska, D | 1 |
Presant, CA; Valeriote, F; Vietti, T | 1 |
Berger, AE; Bhuyan, BK; DeSante, DC; Neil, GL | 1 |
Muggia, FM; Slavik, M; Von Hoff, DD | 1 |
Carter, SK; Slavik, M | 1 |
Presant, CA; Valeriote, F; Vietti, TJ | 1 |
Abbasi, MM; Beisler, JA; Voytek, P; Wolpert-DeFilippes, MK | 1 |
Gonzales, FA; Momparier, RL | 1 |
Gaudio, L; Kelly, CJ; Schoenemann, PT; Wodinsky, I; Yesair, DW | 1 |
Covey, JM; D'Incalci, M; Kohn, KW; Zaharko, DS | 1 |
Zaharko, DS | 1 |
Driscoll, JS; Johns, DG; Plowman, J | 1 |
Covey, JM; D'Incalci, M; Kohn, KW; Tilchen, EJ; Zaharko, DS | 1 |
Colombo, T; D'Incalci, M; Rossi, C | 1 |
Allegrucci, M; Borri Voltattorni, C; Dominici, P; Fioretti, MC; Puccetti, P; Romani, L | 1 |
Avramis, VI; Powell, WC | 1 |
Fioretti, MC; Fuschiotti, P; Puccetti, P; Romani, L | 1 |
Momparler, LF; Momparler, RL | 1 |
Covey, JM; Muneses, CC; Zaharko, DS | 1 |
Oliverio, VT | 1 |
Carter, SK | 1 |
Heby, O; Russell, DH | 1 |
Gang, M; Kline, I; Sirica, AE; Venditti, JM; Woodman, RJ | 1 |
Dulmadge, EA; Lloyd, HH; Wilkoff, LJ | 1 |
5 review(s) available for azacitidine and Leukemia L 1210
Article | Year |
---|---|
[Cisplatin resistance in a murine leukemia cell line associated with defect of apoptosis].
Topics: Alkaloids; Animals; Antimetabolites, Antineoplastic; Apoptosis; Azacitidine; Cell Division; Cisplatin; Clone Cells; DNA, Neoplasm; Drug Resistance, Neoplasm; Endonucleases; Leukemia L1210; Mice; Protein Kinase C; Staurosporine; Tumor Cells, Cultured | 1996 |
5-Azacytidine. A new anticancer drug with effectiveness in acute myelogenous leukemia.
Topics: Animals; Azacitidine; Breast Neoplasms; Chemical and Drug Induced Liver Injury; Chemical Phenomena; Chemistry; Europe; Female; Humans; Kinetics; Leukemia L1210; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Leukopenia; Liver; Nausea; Neoplasms, Experimental; Neuromuscular Diseases; RNA, Messenger; United States; Vomiting | 1976 |
Investigational drugs under study by the United States National Cancer Institute.
Topics: Acrylates; Alkylating Agents; Ancitabine; Animals; Antibiotics, Antineoplastic; Antimetabolites, Antineoplastic; Antineoplastic Agents; Azacitidine; Chemical Phenomena; Chemistry; Chromomycins; Cisplatin; DNA, Neoplasm; Drug Evaluation, Preclinical; Etoposide; Humans; Ifosfamide; Leukemia L1210; Mice; Mitosis; National Institutes of Health (U.S.); Neoplasms; Neoplasms, Experimental; Razoxane; Tegafur; Teniposide; United States | 1976 |
[Possibilities for the clinical use of 5-azacytidine].
Topics: Adult; Animals; Azacitidine; Biopharmaceutics; Chemical Phenomena; Chemistry; Child; Clinical Trials as Topic; Drug Evaluation; Drug Evaluation, Preclinical; Humans; In Vitro Techniques; Leukemia L1210; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Mice; Mice, Inbred AKR; Molecular Conformation | 1977 |
Current status of new agents.
Topics: Alopecia; Animals; Antibiotics, Antineoplastic; Antineoplastic Agents; Azacitidine; Azaguanine; Carmustine; Cyclohexanes; Drug Combinations; Heart; Humans; Leukemia L1210; Nitrosourea Compounds; Platinum; Prednisone; Remission, Spontaneous | 1972 |
1 trial(s) available for azacitidine and Leukemia L 1210
Article | Year |
---|---|
[Possibilities for the clinical use of 5-azacytidine].
Topics: Adult; Animals; Azacitidine; Biopharmaceutics; Chemical Phenomena; Chemistry; Child; Clinical Trials as Topic; Drug Evaluation; Drug Evaluation, Preclinical; Humans; In Vitro Techniques; Leukemia L1210; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Mice; Mice, Inbred AKR; Molecular Conformation | 1977 |
60 other study(ies) available for azacitidine and Leukemia L 1210
Article | Year |
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Synthesis and antitumor activity of dihydro-5-azacytidine, a hydrolytically stable analogue of 5-azacytidine.
Topics: Animals; Antineoplastic Agents; Azacitidine; Hydrolysis; Leukemia L1210; Leukemia, Experimental; Melanoma; Mice; Neoplasms, Experimental | 1977 |
Isolation, characterization, and properties of a labile hydrolysis product of the antitumor nucleoside, 5-azacytidine.
Topics: Animals; Azacitidine; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Stability; Hydrolysis; Leukemia L1210; Mice; Solutions; Time Factors | 1978 |
Synthesis and antitumor activity of 5-azacytosine arabinoside.
Topics: Animals; Antineoplastic Agents; Azacitidine; Chemical Phenomena; Chemistry; Leukemia L1210; Mice; Stereoisomerism | 1979 |
Structure-activity relationships of antineoplastic agents in multidrug resistance.
Topics: Animals; Antineoplastic Agents; Cell Line; Cell Survival; Cricetinae; Dactinomycin; Drug Resistance; Leukemia L1210; Mice; Regression Analysis; Structure-Activity Relationship; Tumor Cells, Cultured | 1990 |
Synthesis and antitumor activity of fluorine-substituted 4-amino-2(1H)-pyridinones and their nucleosides. 3-Deazacytosines.
Topics: Animals; Antimetabolites, Antineoplastic; Cytosine; Drug Evaluation, Preclinical; Indicators and Reagents; Leukemia L1210; Magnetic Resonance Spectroscopy; Mass Spectrometry; Mice; Spectrophotometry; Structure-Activity Relationship | 1987 |
Synergistic effect of 5-Aza-2'-deoxycytidine and genistein in combination against leukemia.
Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Azacitidine; Cyclin-Dependent Kinase Inhibitor p57; Decitabine; DNA Methylation; DNA, Neoplasm; Drug Synergism; Genistein; HL-60 Cells; Humans; Leukemia; Leukemia L1210; Male; Mice; Promoter Regions, Genetic | 2008 |
3-Deazauridine enhances the antileukemic action of 5-aza-2'-deoxycytidine and targets drug-resistance due to deficiency in deoxycytidine kinase.
Topics: 3-Deazauridine; Animals; Azacitidine; Cell Line, Tumor; Decitabine; Deoxycytidine Kinase; Drug Resistance, Neoplasm; Drug Synergism; Humans; Leukemia L1210; Male; Mice; Reverse Transcriptase Polymerase Chain Reaction | 2011 |
Enhancement of antineoplastic action of 5-aza-2'-deoxycytidine by zebularine on L1210 leukemia.
Topics: Animals; Antimetabolites, Antineoplastic; Azacitidine; Cell Line, Tumor; Cytidine; Cytidine Deaminase; Decitabine; DNA Methylation; Dose-Response Relationship, Drug; Drug Interactions; Humans; Leukemia L1210; Male; Mice; Pyrimidine Nucleosides; Reverse Transcriptase Polymerase Chain Reaction; Tumor Stem Cell Assay | 2005 |
Diverse histone modifications on histone 3 lysine 9 and their relation to DNA methylation in specifying gene silencing.
Topics: Acetylation; Animals; Azacitidine; Cell Line, Tumor; Chromatin Immunoprecipitation; CpG Islands; Decitabine; DNA Methylation; DNA Modification Methylases; Gene Expression Regulation; Gene Silencing; Histones; Hydroxamic Acids; Leukemia L1210; Lysine; Methylation; Mice; Mice, Inbred DBA; Oligonucleotide Array Sequence Analysis; Protein Processing, Post-Translational | 2007 |
Comparison of the antileukemic activity of 5-AZA-2'-deoxycytidine, 1-beta-D-arabinofuranosylcytosine and 5-azacytidine against L1210 leukemia.
Topics: Animals; Antineoplastic Agents; Azacitidine; Cytarabine; Decitabine; DNA, Neoplasm; Leukemia L1210; Male; Methylation; Mice; Mice, Inbred BALB C; Mice, Inbred DBA | 1984 |
Effects of 5-aza-2'-deoxycytidine in combination with the biochemical modulator thymidine or the immune modulator pyran copolymer on L1210 leukemia-bearing mice.
Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Azacitidine; Body Weight; Decitabine; Leukemia L1210; Male; Mice; Polymers; Pyran Copolymer; Thymidine; Time Factors | 1984 |
Combination chemotherapy with Clostridium perfringens phospholipase C and cytosine antimetabolites: complementary inhibition directed at membrane lipids.
Topics: Animals; Azacitidine; Cell Line; Choline; Clostridium; Cytarabine; Leukemia L1210; Membrane Lipids; Mice; Microscopy, Electron, Scanning; Sarcoma 180; Type C Phospholipases | 1983 |
The effect of 5-azacytidine and dihydro-5-azacytidine on nuclear ribosomal RNA and poly(A) RNA synthesis in L1210 cells in vitro.
Topics: Adenosine; Animals; Azacitidine; Cells, Cultured; Depression, Chemical; Dose-Response Relationship, Drug; Leukemia L1210; Methionine; Methylation; Mice; Poly A; RNA; RNA, Heterogeneous Nuclear; RNA, Messenger; RNA, Ribosomal; Uridine | 1980 |
The comparative effects of 5-azacytidine and dihydro-5-azacytidine on 4 S and 5 S nuclear RNA.
Topics: Animals; Azacitidine; Chromatography, Thin Layer; Electrophoresis, Polyacrylamide Gel; Leukemia L1210; Methylation; Mice; Molecular Weight; RNA, Neoplasm | 1980 |
Kinetics of 5-aza-2'-deoxycytidine phosphorylation in mouse spleen and L1210 leukemic cell extracts.
Topics: Animals; Azacitidine; Binding, Competitive; Cell-Free System; Decitabine; Deoxycytidine Kinase; Deoxyribonucleosides; Kinetics; Leukemia L1210; Mice; Nucleosides; Phosphorylation; Spleen | 1980 |
Effect of N-(phosphonacetyl)-L-aspartate on 5-azacytidine metabolism in P388 and L1210 cells.
Topics: Animals; Aspartate Carbamoyltransferase; Aspartic Acid; Azacitidine; Cell Division; Cytidine; DNA, Neoplasm; Leukemia L1210; Leukemia, Experimental; Mice; Neoplasm Proteins; Organophosphorus Compounds; Phosphonoacetic Acid; RNA, Neoplasm; Uridine | 1981 |
Effects of dihydro-5-azacytidine on cell survival and cell cycle progression of cultured mammalian cells.
Topics: Animals; Azacitidine; Cell Cycle; Cell Survival; Cells, Cultured; Cricetinae; Cricetulus; Female; Humans; Leukemia L1210; Leukemia, Experimental; Lymphocyte Activation; Mice; Ovary; Phytohemagglutinins; RNA | 1981 |
Contrasting cytotoxicity kinetics of 5-azacytidine and dihydro-5-azacytidine hydrochloride in L1210 leukemia in mice.
Topics: Animals; Azacitidine; Bone Marrow; Cell Survival; Colony-Forming Units Assay; Dose-Response Relationship, Drug; Hematopoietic Stem Cells; Kinetics; Lethal Dose 50; Leukemia L1210; Male; Mice; Spleen | 1981 |
Chemotherapy of L1210 leukemia with 5-azacytidine in combination with vincristine, adriamycin, or beta-cytosine arabinoside.
Topics: Animals; Azacitidine; Colony-Forming Units Assay; Cytarabine; Doxorubicin; Drug Administration Schedule; Drug Interactions; Drug Therapy, Combination; Leukemia L1210; Mice; Mice, Inbred BALB C; Mice, Inbred DBA; Vincristine | 1981 |
Dose- and schedule-dependent activation and drug synergism between thymidine and 5-aza-2'-deoxycytidine in a human promyelocytic leukemia cell line.
Topics: Animals; Antineoplastic Agents; Azacitidine; Biological Transport; Cell Line; Cell Survival; Chromatography, High Pressure Liquid; Decitabine; DNA; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Synergism; Humans; Leukemia L1210; Leukemia, Myeloid, Acute; Mice; Thymidine; Time Factors | 1982 |
Synergistic effect of cis-dichlorodiammineplatinum and 5-aza-2'-deoxycytidine on mouse leukemic cells in vivo and in vitro.
Topics: Animals; Azacitidine; Cell Division; Cisplatin; Decitabine; DNA, Neoplasm; Drug Synergism; In Vitro Techniques; Leucine; Leukemia L1210; Leukemia, Experimental; Male; Mice; Mice, Inbred Strains; RNA, Neoplasm | 1982 |
Combinational chemotherapy of L1210 and L1210/ARA-C leukemia with 5-AZA-2'-deoxycytidine and beta-2'-deoxythioguanosine.
Topics: Animals; Antineoplastic Agents; Azacitidine; Decitabine; Deoxyguanosine; Drug Evaluation; Drug Therapy, Combination; Leukemia L1210; Male; Mice; Thionucleosides | 1982 |
Inhibition of DNA methylation in L1210 leukemic cells by 5-aza-2'-deoxycytidine as a possible mechanism of chemotherapeutic action.
Topics: 5-Methylcytosine; Animals; Antineoplastic Agents; Azacitidine; Cytosine; Decitabine; DNA; DNA (Cytosine-5-)-Methyltransferases; Dose-Response Relationship, Drug; Leukemia L1210; Male; Methylation; Mice | 1983 |
Effect of 3-deazauridine on the metabolism, toxicity, and antitumor activity of azacitidine in mice bearing L1210 leukemia sensitive and resistant to cytarabine.
Topics: 3-Deazauridine; Animals; Azacitidine; Chromatography, High Pressure Liquid; Cytarabine; Drug Therapy, Combination; Lethal Dose 50; Leukemia L1210; Mice; Mice, Inbred DBA; Purine Nucleotides; Pyrimidine Nucleotides; Uridine | 1983 |
Biological evaluation of stability of 5-azacytidine.
Topics: Animals; Azacitidine; Drug Stability; Escherichia coli; Leukemia L1210; Mice; Temperature | 1984 |
Effects of the alpha-D-anomer of 5-aza-2'-deoxycytidine on L1210 mouse leukemic cells in vitro and in vivo.
Topics: Animals; Azacitidine; Cell Division; Decitabine; Deoxycytidine Kinase; DNA Replication; Drug Evaluation, Preclinical; Isomerism; Leukemia L1210; Mice; Transcription, Genetic | 1984 |
Long term instability and molecular mechanism of 5-azacytidine-induced DNA hypomethylation in normal and neoplastic tissues in vivo.
Topics: Animals; Azacitidine; DNA; DNA (Cytosine-5-)-Methyltransferases; DNA, Neoplasm; Kinetics; Leukemia L1210; Liver; Liver Regeneration; Male; Methylation; Methyltransferases; Mice; Mice, Inbred BALB C; Mice, Inbred DBA | 1984 |
Enhancement of intercalator-induced deoxyribonucleic acid scission and cytotoxicity in murine leukemia cells treated with 5-azacytidine.
Topics: Animals; Azacitidine; Cell Survival; DNA Replication; DNA, Neoplasm; Intercalating Agents; Leukemia L1210; Mice | 1984 |
Effects of dose and duration of exposure on 5-aza-2'-deoxycytidine cytotoxicity for L1210 leukemia in vitro.
Topics: Animals; Azacitidine; Cell Division; Cell Survival; Clone Cells; Decitabine; Kinetics; Leukemia L1210; Mice; Time Factors | 1984 |
Antileukemic activity of 5-aza-2'-deoxycytidine and cytarabine against intracerebral L1210 murine leukemia.
Topics: Animals; Azacitidine; Brain Neoplasms; Cytarabine; Decitabine; Dose-Response Relationship, Drug; Kinetics; Leukemia L1210; Male; Mice; Mice, Inbred Strains | 1984 |
Cisplatin resistance in a murine leukemia cell line is associated with a defective apoptotic process.
Topics: Alkaloids; Animals; Apoptosis; Azacitidine; Cell Division; Cell Nucleus; Cisplatin; Clone Cells; Cycloheximide; DNA, Neoplasm; Drug Resistance; Endonucleases; Leukemia L1210; Mice; Microscopy, Confocal; Microscopy, Electron; Protein Kinase C; Staurosporine; Tumor Cells, Cultured | 1995 |
Does 2-chlorodeoxyadenosine contribute to alteration of DNA methyltransferase activity?
Topics: Adenosylhomocysteinase; Animals; Antimetabolites, Antineoplastic; Antineoplastic Agents; Azacitidine; Cladribine; Decitabine; DNA (Cytosine-5-)-Methyltransferases; Hydrolases; Kinetics; Leukemia L1210; Mice; Tumor Cells, Cultured; Vidarabine | 1998 |
Kinetics of both leukemic and normal cell population reduction following 5-azacytidine.
Topics: Animals; Azacitidine; Bone Marrow; Bone Marrow Cells; Dose-Response Relationship, Drug; Femur; Hematopoietic Stem Cells; Kinetics; Leukemia L1210; Mice; Mice, Inbred BALB C; Mice, Inbred DBA; Time Factors | 1975 |
Combination chemotherapy of L1210 leukemia with 1-beta-D-arabinofuranosylcytosine and 5-azacytidine.
Topics: Animals; Azacitidine; Body Weight; Cells, Cultured; DNA Replication; Dose-Response Relationship, Drug; Drug Therapy, Combination; Female; Leukemia L1210; Mice | 1976 |
Biological characterization of a prolonged antileukemic effect of 5-azacytidine.
Topics: Animals; Azacitidine; Bone Marrow; Bone Marrow Cells; Cell Division; Cell Survival; Cytidine; Dose-Response Relationship, Drug; Immunity; Leukemia L1210; Mice; Mice, Inbred DBA; Neoplasm Transplantation; Thymidine; Time Factors; Transplantation, Isogeneic | 1977 |
Dihydro-5-azacytidine hydrochloride, a biologically active and chemically stable analog of 5-azacytidine.
Topics: Animals; Azacitidine; Leukemia L1210; Mice | 1976 |
Comparative studies of the cytostatic action and metabolism of 5-azacytidine and 5,6-dihydro-5-azacytidine.
Topics: Animals; Azacitidine; Cell Division; Cells, Cultured; Cytidine; Cytidine Deaminase; Deoxycytidine; Drug Synergism; Kinetics; Leukemia L1210; Oxidative Phosphorylation; Tetrahydrouridine; Thymidine; Uridine | 1977 |
Incorporation of a potent antileukemic agent, 5-aza-2'-deoxycytidine, into DNA of cells from leukemic mice.
Topics: Animals; Azacitidine; Deoxycytidine; Epithelium; Female; Leukemia L1210; Leukemia, Experimental; Liver; Lymph Nodes; Mice; Mice, Inbred AKR; Mice, Inbred BALB C; Mice, Inbred DBA; Precancerous Conditions; Thymidine | 1977 |
The synthesis and antitumor activity of arabinosyl-5-azacytosine.
Topics: Animals; Antineoplastic Agents; Azacitidine; Cytarabine; Leukemia L1210; Mice | 1977 |
Effect of intravenous infusion of 5-aza-2'-deoxycytidine on survival time of mice with L1210 leukemia.
Topics: Animals; Azacitidine; Cell Survival; Deoxycytidine; In Vitro Techniques; Infusions, Parenteral; Leukemia L1210; Male; Mice; Mice, Inbred Strains; Time Factors | 1978 |
Pharmacokinetic considerations in evaluating the effects of tetrahydrouridine on 5-azacytidine chemotherapy in L1210 leukemic mice.
Topics: Animals; Azacitidine; Drug Therapy, Combination; Female; Infusions, Parenteral; Injections, Intraperitoneal; Leukemia L1210; Mice; Tetrahydrouridine; Uridine | 1978 |
DNA alkali-labile sites induced by incorporation of 5-aza-2'-deoxycytidine into DNA of mouse leukemia L1210 cells.
Topics: Alkalies; Animals; Antineoplastic Agents; Azacitidine; Cells, Cultured; Decitabine; DNA, Neoplasm; Hydrogen-Ion Concentration; Leukemia L1210; Mice | 1985 |
Immunological concepts and the combination of cyclophosphamide with 5-aza-2'-deoxycytidine on L1210 in vivo.
Topics: Animals; Antineoplastic Agents; Azacitidine; Cell Survival; Cyclophosphamide; Decitabine; Drug Synergism; Drug Therapy, Combination; Leukemia L1210; Male; Mice; Mice, Inbred Strains; T-Lymphocytes, Regulatory | 1985 |
Arabinosyl-5-azacytosine: plasma kinetics and therapeutic response (L1210) in vitro and in vivo in mice.
Topics: Animals; Antineoplastic Agents; Azacitidine; Cells, Cultured; Decitabine; Kinetics; Leukemia L1210; Male; Mice; Mice, Inbred Strains | 1985 |
Comparison of the activity of arabinosyl-5-azacytosine, arabinosyl cytosine, and 5-azacytidine against intracerebrally implanted L1210 leukemia.
Topics: Animals; Antineoplastic Agents; Azacitidine; Brain Neoplasms; Carmustine; Cytarabine; Leukemia L1210; Mice; Mice, Inbred Strains; Neoplasm Transplantation | 1985 |
Mechanism of action of 1-beta-D-arabinofuranosyl-5-azacytosine and its effects in L1210 mouse leukemia cells.
Topics: Animals; Antineoplastic Agents; Azacitidine; Bone Marrow; Bone Marrow Cells; Cell Division; Cell Line; Cell Survival; Cytarabine; Decitabine; Drug Evaluation, Preclinical; Kinetics; Leukemia L1210; Leukocyte Count; Male; Mice; Mice, Inbred DBA; Nucleosides; Phosphorylation; Thymidine | 1986 |
Effects of 5-aza-2'-deoxycytidine on survival and cell cycle progression of L1210 leukemia cells.
Topics: Animals; Antineoplastic Agents; Azacitidine; Cell Cycle; Cell Survival; Cells, Cultured; Decitabine; DNA, Neoplasm; Leukemia L1210; Mice; Thymidine | 1986 |
Differences in DNA damage produced by incorporation of 5-aza-2'-deoxycytidine or 5,6-dihydro-5-azacytidine into DNA of mammalian cells.
Topics: Animals; Azacitidine; Cell Cycle; Cell Line; Decitabine; DNA; DNA Damage; DNA Replication; Humans; Hydrogen-Ion Concentration; Leukemia L1210; Lymphocytes; Mice | 1986 |
Antagonism of 5-aza-2'-deoxycytidine antileukemic activity by concomitant treatment with cytarabine.
Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Azacitidine; Cytarabine; Decitabine; Drug Interactions; Leukemia L1210; Male; Mice; Statistics as Topic | 1986 |
DNA methylating activity in murine lymphoma cells treated with xenogenizing chemicals.
Topics: Animals; Azacitidine; Carmustine; DNA, Neoplasm; Leukemia L1210; Male; Methylation; Mice; Mice, Inbred Strains; Neoplasm Transplantation; Triazenes | 1987 |
High degree of resistance to 5-aza-2'-deoxycytidine in L1210 cells in vitro associated with almost complete loss of deoxycytidine kinase activity.
Topics: 5-Methylcytosine; Animals; Azacitidine; Cell Line; Cells, Cultured; Cytosine; Decitabine; Deoxycytidine; Deoxycytidine Kinase; DNA (Cytosine-5-)-Methyltransferases; Drug Resistance; Leukemia L1210; Mice; Phosphorylation; Phosphotransferases | 1987 |
Biochemical pharmacology of 5,6-dihydro-5-azacytidine (DHAC) and DNA hypomethylation in tumor (L1210)-bearing mice.
Topics: Animals; Azacitidine; Bone Marrow; Brain; Chromatography, High Pressure Liquid; DNA, Neoplasm; Erythrocytes; Intestinal Mucosa; Kidney; Leukemia L1210; Liver; Lung; Male; Methylation; Mice; Muscles; Myocardium; Spleen; Testis; Tissue Distribution; Tumor Cells, Cultured | 1988 |
Lack of correlation between DNA-methylating activity and appearance of the immunogenic phenotype in clones of a murine lymphoma treated with mutagens.
Topics: 5-Methylcytosine; Animals; Antigens, Neoplasm; Azacitidine; Clone Cells; Cytosine; DNA, Neoplasm; Female; Leukemia L1210; Male; Methylation; Methylnitronitrosoguanidine; Mice; Mutagens; Phenotype; Triazenes | 1989 |
Chemotherapy of L1210 and L1210/ARA-C leukemia with 5-aza-2'-deoxycytidine and 3-deazauridine.
Topics: 3-Deazauridine; Animals; Antineoplastic Combined Chemotherapy Protocols; Azacitidine; Cell Line; Cytarabine; Decitabine; Drug Interactions; Drug Resistance; Drug Screening Assays, Antitumor; Leukemia L1210; Male; Mice; Mice, Inbred BALB C; Neoplasm Transplantation; Tumor Cells, Cultured | 1989 |
Comparison of the in vitro cytotoxicity (L1210) of 5-aza-2'-deoxycytidine with its therapeutic and toxic effects in mice.
Topics: Animals; Antineoplastic Agents; Azacitidine; Cell Survival; Cells, Cultured; Decitabine; Dose-Response Relationship, Drug; Kinetics; Leukemia L1210; Mice | 1985 |
Experimental chemotherapy (L1210) with 5-aza-2'-deoxycytidine in combination with pyran copolymer (MVE-4), an immune adjuvant.
Topics: Adjuvants, Immunologic; Animals; Antibody Formation; Antineoplastic Combined Chemotherapy Protocols; Azacitidine; Decitabine; Leukemia L1210; Mice; Mice, Inbred Strains; Pyran Copolymer | 1985 |
Second Joint Working Conference: National Cancer Institute Chemotherapy Program. Working session report: pharmacology.
Topics: Alkaloids; Animals; Antimetabolites; Antineoplastic Agents; Autoradiography; Azacitidine; Carbazoles; Carbon Isotopes; Cell Line; Cells, Cultured; Cricetinae; Cytarabine; DNA; DNA Nucleotidyltransferases; Dogs; Half-Life; Humans; Leukemia L1210; Lung; Pyridines; RNA | 1972 |
Depression of polyamine synthesis in L1210 leukemic mice during treatment with a potent antileukemic agent, 5-azacytidine.
Topics: Animals; Antineoplastic Agents; Azacitidine; Carboxy-Lyases; Cytidine; Depression, Chemical; Enzyme Repression; Injections, Intraperitoneal; Leukemia L1210; Liver; Male; Mice; Mice, Inbred Strains; Neoplasm Transplantation; Organ Size; Ornithine; Polyamines; Putrescine; S-Adenosylmethionine; Spermidine; Spleen; Triazines | 1973 |
The enhanced therapeutic effect of cis-platinum (II) diamminodichloride against L1210 leukemia when combined with cyclophosphamide or 1,2-bis(3,5-dioxopiperazine-1-yl)propane or several other antitumor agents.
Topics: Amines; Animals; Antineoplastic Agents; Azacitidine; Camptothecin; Carmustine; Chlorides; Cyclophosphamide; Cytarabine; Drug Synergism; Emetine; Fluorouracil; Ketones; Leukemia L1210; Male; Methotrexate; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Piperazines; Platinum; Propane; Time Factors | 1973 |
Kinetics of the reduction in viability of cultured L1210 leukemia cells exposed to 5-azacytidine (NSC-102816).
Topics: Animals; Azacitidine; Cell Division; Cell Survival; Cells, Cultured; Chromatography, Paper; Cytidine; Hydrolysis; Kinetics; Leukemia L1210; Mice; Time Factors; Triazines | 1972 |