Page last updated: 2024-09-04

atazanavir sulfate and Bilirubinemia

atazanavir sulfate has been researched along with Bilirubinemia in 45 studies

Research

Studies (45)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's15 (33.33)29.6817
2010's28 (62.22)24.3611
2020's2 (4.44)2.80

Authors

AuthorsStudies
Chan, WW; Li, M; Zucker, SD1
Agide, FD; Mohraz, M; Nikfar, S; Tigabu, BM1
Culley, CL; Ensom, MH; Gilchrist, SE; Kiang, TK1
Back, D; Boffito, M; Else, L; Gazzard, B; Jackson, A; Karolia, Z; Moyle, G; Ringner-Nackter, L; Seymour, N; Yapa, MH1
Chang, JH; Cheong, J; Ho, Q; Lin, M; Plise, E1
Bertz, R; Botes, M; Conradie, F; Eley, T; Hardy, H; Huang, SP; Josipovic, D; McGrath, D; Osiyemi, O; Zorrilla, CD1
Baril, JG; Dufresne, S; Laprise, C; Trottier, H1
Bow, DA; Chiou, WJ; de Morais, SM; Kikuchi, R; Li, X; Voorman, RL1
Atrio, JM; Chen, KT; Posada, R; Rodriguez Caprio, G; Sperling, RS1
Bernardino, JI; Carton, JA; Curran, A; Domingo, P; Ferrer, E; Gatell, JM; Gonzalez-Cordon, A; Gutierrez, F; Martinez, E; Murillas, J; Negredo, E; Peraire, J; Perez, I; Pich, J; Podzamczer, D; Portilla, J; Santos, I1
Antoniadou, A; Detsika, M; Hatzakis, A; Katsarolis, I; Panagopoulos, P; Papadopoulos, A; Paraskevis, D; Petrikkos, G; Protopapas, K; Sypsa, V1
Daar, ES; Haas, DW; Johnson, DH; McLaren, PJ; Morse, GD; Ritchie, MD; Venuto, C1
Bourgeois-Moine, A; Bourse, P; Calvez, V; Damond, F; Descamps, D; Dommergues, M; Duro, D; Faucher, P; Ichou, H; Landman, R; Lariven, S; Lê, MP; Legac, S; Mandelbrot, L; Matheron, S; Meier, F; Mortier, E; Peytavin, G; Soulié, C; Tubiana, R; Valantin, MA1
Avihingsanon, A; Gorowara, M; Kerr, SJ; Punyawudho, B; Ruxrungtham, K; Shotelersuk, V; Suphapeetiporn, K; Tongkobpetch, S1
Cattaneo, D; Charbe, N; Clementi, E; Cozzi, V; Ferraris, L; Galli, M; Gervasoni, C; Landonio, S; Meraviglia, P; Minisci, D; Molinari, L; Riva, A; Rizzardini, G1
Alvarellos, M; Brummel, SS; Caudle, KE; Court, MH; Gammal, RS; Gaur, AH; Guillemette, C; Haas, DW; Haidar, CE; Iwuchukwu, OF; Klein, TE; Lennox, JL; Ratain, MJ; Schackman, BR; Whirl-Carrillo, M1
Chang, SC; Chang, SY; Hung, CC; Kuo, CH; Lin, SW; Liu, WC; Su, YC; Sun, HY; Tang, SY; Tsai, MS; Wu, BR1
Cattaneo, D; Clementi, E; Gervasoni, C; Milazzo, L; Riva, A1
Listowsky, I; Roy-Chowdhury, J; Roy-Chowdhury, N; Wolkoff, AW1
Roca, B1
Barreiro, P; González, M; Gonzalez-Lahoz, J; González-Pardo, G; Jiménez-Nácher, I; Morello, J; Rodríguez-Nóvoa, S; Soriano, V; Vispo, E1
Antinori, A; Antonucci, F; Carosi, G; Castelnuovo, F; De Luca, A; Di Perri, G; Esposito, R; Lapadula, G; Lazzarin, A; Maggiolo, F; Maserati, R; Migliorino, G; Paraninfo, G; Quirino, T; Rizzardini, G; Torti, C1
Cauda, R; Colafigli, M; De Luca, A; Di Giambenedetto, S; Fabbiani, M; Navarra, P; Prosperi, M; Ragazzoni, E1
López-Cortés, LF1
Gatell, JM; Zamora, L1
González, M; Palacios, R; Ruiz, J; Santos, J1
Camacho, A; Pérez-Camacho, I; Rivero, A; Torre-Cisneros, J1
Curran, A; Ribera Pascuet, E1
Choe, KW; Choe, PG; Jeon, JH; Kim, HB; Kim, NJ; Oh, MD; Park, SW; Park, WB; Song, KH1
Choe, PG; Kim, HB; Kim, NH; Kim, NJ; Oh, MD; Park, SW; Park, WB; Song, JS; Song, KH1
Bellón, JM; González, MI; José, MI; Larru, B; Mellado, MJ; Muñoz-Fernández, MÁ; Navarro, ML; Nso Roca, AP; Nso, AP; Ramos, JT1
Agnes, G; Basso, RP; de Almeida, S; Kuhmmer, R; Lazzaretti, RK; Mattevi, VS; Pinheiro, CA; Ribeiro, JP; Silveira, JM; Silveira, MF; Sprinz, E; Turatti, L1
Blanton, LS; East, J1
Aubry, C; Badens, C; Javelle, E; Oliver, M; Savini, H; Simon, F1
Butcher, D; Farajallah, A; Hu, W; Juethner, S; McDonald, C; McGrath, D; Moyle, G; Uy, J; Wirtz, V1
Baker, P; Bradbeer, C; George, M; Ngwenya, S1
Bissio, E; Espinola, L; Gadano, A; Gallego, P; Lopardo, G; Stambullian, M1
Bissio, E; Lopardo, GD1
Laurence, J1
Sulkowski, MS1
Barreiro, P; Barrios, A; Corral, A; González-Lahoz, J; Jiménez-Nacher, I; Rendón, A; Rodríguez Nóvoa, S; Soriano, V1
Behrens, G; Lankisch, TO; Manns, MP; Moebius, U; Schmidt, RE; Strassburg, CP; Wehmeier, M1
Barreiro, P; González-Lahoz, J; González-Pardo, G; Jiménez-Nácher, I; Martín-Carbonero, L; Rodríguez-Nóvoa, S; Soriano, V1
De Marez, T; De Paepe, E; De Pauw, M; Hoetelmans, RM; Lefebvre, E; Sekar, VJ; Spinosa-Guzman, S; Vangeneugden, T1
Battegay, M; Bodmer, M; Elzi, L; Haschke, M; Krähenbühl, S; Kummer, O; Mossdorf, E1

Reviews

10 review(s) available for atazanavir sulfate and Bilirubinemia

ArticleYear
Atazanavir / ritonavir versus Lopinavir / ritonavir-based combined antiretroviral therapy (cART) for HIV-1 infection: a systematic review and meta-analysis.
    African health sciences, 2020, Volume: 20, Issue:1

    Topics: Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; HIV Infections; HIV Protease Inhibitors; HIV-1; Humans; Hyperbilirubinemia; Lopinavir; Ritonavir; Treatment Outcome; Viral Load

2020
Effect of the UGT1A1*28 allele on unconjugated hyperbilirubinemia in HIV-positive patients receiving Atazanavir: a systematic review.
    The Annals of pharmacotherapy, 2013, Volume: 47, Issue:4

    Topics: Alleles; Anti-HIV Agents; Atazanavir Sulfate; Glucuronosyltransferase; HIV Infections; Homozygote; Humans; Hyperbilirubinemia; Oligopeptides; Polymorphism, Genetic; Prospective Studies; Pyridines; Retrospective Studies

2013
Clinical Pharmacogenetics Implementation Consortium (CPIC) Guideline for UGT1A1 and Atazanavir Prescribing.
    Clinical pharmacology and therapeutics, 2016, Volume: 99, Issue:4

    Topics: Atazanavir Sulfate; Genetic Predisposition to Disease; Genotype; Glucuronosyltransferase; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Jaundice; Liver; Pharmacogenetics; Phenotype; Risk Assessment; Risk Factors

2016
Pharmacogenomics of antiretrovirals.
    Recent patents on anti-infective drug discovery, 2008, Volume: 3, Issue:2

    Topics: Alkynes; Anti-Retroviral Agents; Aryl Hydrocarbon Hydroxylases; Atazanavir Sulfate; Benzoxazines; Central Nervous System Diseases; Cyclopropanes; Cytochrome P-450 CYP2B6; Dideoxynucleosides; Drug Hypersensitivity; Drug Resistance, Viral; Dyslipidemias; Genetic Predisposition to Disease; Genetic Testing; Glucuronosyltransferase; HLA Antigens; Humans; Hyperbilirubinemia; Nevirapine; Oligopeptides; Oxidoreductases, N-Demethylating; Patents as Topic; Patient Selection; Pharmacogenetics; Pyridines; Ritonavir

2008
[Pharmacology, pharmacokinetic features and interactions of atazanavir].
    Enfermedades infecciosas y microbiologia clinica, 2008, Volume: 26 Suppl 17

    Topics: Anti-HIV Agents; Atazanavir Sulfate; Biological Availability; Biotransformation; Blood Proteins; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Drug Interactions; Drug Therapy, Combination; Female; Fetal Blood; Glucuronosyltransferase; HIV Infections; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Infant, Newborn; Kidney Diseases; Liver Diseases; Maternal-Fetal Exchange; Metabolic Clearance Rate; Molecular Structure; Oligopeptides; Pregnancy; Pregnancy Complications, Infectious; Pyridines

2008
[Efficacy of atazanavir in simplification regimens].
    Enfermedades infecciosas y microbiologia clinica, 2008, Volume: 26 Suppl 17

    Topics: Adult; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; Clinical Trials as Topic; Drug Administration Schedule; Drug Therapy, Combination; Dyslipidemias; Female; Gastrointestinal Diseases; HIV Infections; HIV Protease Inhibitors; HIV-1; Humans; Hyperbilirubinemia; Lipids; Male; Middle Aged; Multicenter Studies as Topic; Oligopeptides; Pyridines; Ritonavir; Salvage Therapy; Treatment Outcome

2008
[Adverse effects of atazanavir].
    Enfermedades infecciosas y microbiologia clinica, 2008, Volume: 26 Suppl 17

    Topics: Anti-HIV Agents; Atazanavir Sulfate; Carbohydrate Metabolism; Clinical Trials as Topic; Drug Interactions; Drug Therapy, Combination; Dyslipidemias; Gastrointestinal Diseases; Glucose; HIV Infections; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Hyperinsulinism; Insulin Resistance; Oligopeptides; Pyridines; Urolithiasis

2008
[Safety of atazanavir in patients with HIV and hepatitis B and/or C virus coinfection].
    Enfermedades infecciosas y microbiologia clinica, 2008, Volume: 26 Suppl 17

    Topics: Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; Chemical and Drug Induced Liver Injury; Clinical Trials as Topic; Cohort Studies; Disease Progression; Drug Therapy, Combination; Hepatitis B, Chronic; Hepatitis C, Chronic; Hepatitis D, Chronic; HIV Infections; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Insulin Resistance; Liver; Liver Cirrhosis; Multicenter Studies as Topic; Oligopeptides; Pyridines

2008
[Clinical utility of atazanavir].
    Enfermedades infecciosas y microbiologia clinica, 2008, Volume: 26 Suppl 17

    Topics: Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; Clinical Trials as Topic; Cohort Studies; Comorbidity; Drug Interactions; Drug Resistance, Viral; HIV Infections; HIV Protease Inhibitors; HIV-1; Humans; Hyperbilirubinemia; Insulin Resistance; Oligopeptides; Patient Acceptance of Health Care; Pyridines; Ritonavir; Salvage Therapy; Treatment Outcome; Viral Load

2008
HIV therapeutics, continued: another HIV protease inhibitor approved.
    The AIDS reader, 2003, Volume: 13, Issue:8

    Topics: Acquired Immunodeficiency Syndrome; Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; CD4 Lymphocyte Count; Drug Approval; Drug Resistance, Viral; Headache; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Hypercholesterolemia; Nausea; Oligopeptides; Patient Selection; Pyridines; Treatment Outcome; United States; United States Food and Drug Administration; Viral Load

2003

Trials

7 trial(s) available for atazanavir sulfate and Bilirubinemia

ArticleYear
Coadministration of atazanavir-ritonavir and zinc sulfate: impact on hyperbilirubinemia and pharmacokinetics.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:8

    Topics: Adolescent; Adult; Aged; Anti-HIV Agents; Area Under Curve; Atazanavir Sulfate; Bilirubin; Confidence Intervals; Cross-Over Studies; Drug Administration Schedule; Drug Therapy, Combination; Drug Tolerance; Female; HIV Infections; HIV-1; Humans; Hyperbilirubinemia; Male; Middle Aged; Oligopeptides; Pyridines; Ritonavir; Young Adult; Zinc Sulfate

2013
Clinical and pharmacogenetic factors affecting neonatal bilirubinemia following atazanavir treatment of mothers during pregnancy.
    AIDS research and human retroviruses, 2013, Volume: 29, Issue:10

    Topics: Adult; Anti-HIV Agents; Atazanavir Sulfate; Bilirubin; Female; Glucuronosyltransferase; HIV Infections; Humans; Hyperbilirubinemia; Infant, Newborn; Oligopeptides; Plasma; Pregnancy; Pregnancy Complications, Infectious; Prospective Studies; Pyridines; Ritonavir

2013
Early lipid changes with atazanavir/ritonavir or darunavir/ritonavir.
    HIV medicine, 2014, Volume: 15, Issue:6

    Topics: Adult; Atazanavir Sulfate; Bilirubin; CD4 Lymphocyte Count; CD8-Positive T-Lymphocytes; Darunavir; Drug Therapy, Combination; Female; Glomerular Filtration Rate; HIV Infections; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Lipids; Male; Middle Aged; Oligopeptides; Prospective Studies; Pyridines; Ritonavir; RNA, Viral; Spain; Sulfonamides

2014
Genomewide association study of atazanavir pharmacokinetics and hyperbilirubinemia in AIDS Clinical Trials Group protocol A5202.
    Pharmacogenetics and genomics, 2014, Volume: 24, Issue:4

    Topics: Acquired Immunodeficiency Syndrome; Adult; Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; Bilirubin; Female; Genome-Wide Association Study; Glucuronosyltransferase; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Male; Middle Aged; Multivariate Analysis; Oligopeptides; Polymorphism, Single Nucleotide; Prospective Studies; Pyridines; Ritonavir

2014
Clinical significance of hyperbilirubinemia among HIV-1-infected patients treated with atazanavir/ritonavir through 96 weeks in the CASTLE study.
    AIDS patient care and STDs, 2012, Volume: 26, Issue:5

    Topics: Acquired Immunodeficiency Syndrome; Adult; Anti-HIV Agents; Atazanavir Sulfate; Female; HIV-1; Humans; Hyperbilirubinemia; Lopinavir; Male; Medication Adherence; Oligopeptides; Pyridines; Quality of Life; Ritonavir; Surveys and Questionnaires

2012
Short communication: fasting increases serum concentrations of bilirubin in patients receiving atazanavir: results from a pilot study.
    AIDS research and human retroviruses, 2013, Volume: 29, Issue:3

    Topics: Adult; Anti-HIV Agents; Atazanavir Sulfate; Bilirubin; Fasting; Female; HIV Infections; Humans; Hyperbilirubinemia; Male; Middle Aged; Oligopeptides; Pyridines; Serum

2013
Pharmacokinetics of darunavir (TMC114) and atazanavir during coadministration in HIV-negative, healthy volunteers.
    Drugs in R&D, 2007, Volume: 8, Issue:4

    Topics: Adolescent; Adult; Area Under Curve; Atazanavir Sulfate; Chromatography, Liquid; Cross-Over Studies; Darunavir; Dose-Response Relationship, Drug; Drug Interactions; Female; Half-Life; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Male; Middle Aged; Nausea; Oligopeptides; Pyridines; Sulfonamides; Tandem Mass Spectrometry; Time Factors; Vomiting

2007

Other Studies

28 other study(ies) available for atazanavir sulfate and Bilirubinemia

ArticleYear
Association Between Atazanavir-Induced Hyperbilirubinemia and Cardiovascular Disease in Patients Infected with HIV.
    Journal of the American Heart Association, 2020, 10-20, Volume: 9, Issue:19

    Topics: Atazanavir Sulfate; Bilirubin; Cardiovascular Diseases; Darunavir; Female; HIV Infections; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Ischemic Stroke; Kaplan-Meier Estimate; Male; Middle Aged; Myocardial Infarction; Proportional Hazards Models; Retrospective Studies; Time Factors

2020
Evaluating the in vitro inhibition of UGT1A1, OATP1B1, OATP1B3, MRP2, and BSEP in predicting drug-induced hyperbilirubinemia.
    Molecular pharmaceutics, 2013, Aug-05, Volume: 10, Issue:8

    Topics: Atazanavir Sulfate; Bilirubin; Cell Line; Glucuronosyltransferase; Humans; Hyperbilirubinemia; Indinavir; Liver-Specific Organic Anion Transporter 1; Models, Biological; Oligopeptides; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Pyridines; Solute Carrier Organic Anion Transporter Family Member 1B3

2013
Atazanavir and other determinants of hyperbilirubinemia in a cohort of 1150 HIV-positive patients: results from 9 years of follow-up.
    AIDS patient care and STDs, 2013, Volume: 27, Issue:7

    Topics: Adult; Anti-HIV Agents; Atazanavir Sulfate; Female; Follow-Up Studies; HIV Infections; Humans; Hyperbilirubinemia; Incidence; Kaplan-Meier Estimate; Male; Middle Aged; Oligopeptides; Proportional Hazards Models; Prospective Studies; Pyridines; Treatment Outcome

2013
In vitro OATP1B1 and OATP1B3 inhibition is associated with observations of benign clinical unconjugated hyperbilirubinemia.
    Xenobiotica; the fate of foreign compounds in biological systems, 2014, Volume: 44, Issue:3

    Topics: Antirheumatic Agents; Atazanavir Sulfate; Bilirubin; Carbamates; Cyclosporine; Furans; Glucuronosyltransferase; HIV Protease Inhibitors; Hyperbilirubinemia; In Vitro Techniques; Indinavir; Liver-Specific Organic Anion Transporter 1; Oligopeptides; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Pyridines; Rifampin; Rifamycins; Saquinavir; Solute Carrier Organic Anion Transporter Family Member 1B3; Sulfonamides

2014
Maternal atazanavir usage in HIV-infected pregnant women and the risk of maternal and neonatal hyperbilirubinemia.
    Journal of acquired immune deficiency syndromes (1999), 2013, Aug-15, Volume: 63, Issue:5

    Topics: Anti-HIV Agents; Atazanavir Sulfate; Female; HIV Infections; Humans; Hyperbilirubinemia; Infant, Newborn; Oligopeptides; Pregnancy; Pregnancy Complications, Infectious; Pregnant Women; Prevalence; Pyridines; Risk Assessment

2013
High prevalence of the UGT1A1*28 variant in HIV-infected individuals in Greece.
    International journal of STD & AIDS, 2014, Volume: 25, Issue:12

    Topics: Adult; Aged; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; Bilirubin; Cross-Sectional Studies; Glucuronosyltransferase; Greece; HIV Infections; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Middle Aged; Oligopeptides; Pharmacogenetics; Polymorphism, Genetic; Prevalence; Pyridines; Ritonavir

2014
Pharmacokinetics, safety and efficacy of ritonavir-boosted atazanavir (300/100 mg once daily) in HIV-1-infected pregnant women.
    Antiviral therapy, 2015, Volume: 20, Issue:5

    Topics: Adult; Atazanavir Sulfate; CD4 Lymphocyte Count; Cross-Sectional Studies; Drug Administration Schedule; Drug Combinations; Female; HIV Protease Inhibitors; HIV-1; Humans; Hyperbilirubinemia; Infant, Newborn; Pregnancy; Pregnancy Complications, Infectious; Ritonavir; Viral Load

2015
Pharmacogenetic testing can identify patients taking atazanavir at risk for hyperbilirubinemia.
    Journal of acquired immune deficiency syndromes (1999), 2015, May-01, Volume: 69, Issue:1

    Topics: Adult; Anti-HIV Agents; Atazanavir Sulfate; Female; Genetic Testing; Glucuronosyltransferase; Humans; Hyperbilirubinemia; Male; Middle Aged; Oligopeptides; Pharmacogenetics; Pyridines

2015
Metabolic and kidney disorders correlate with high atazanavir concentrations in HIV-infected patients: is it time to revise atazanavir dosages?
    PloS one, 2015, Volume: 10, Issue:4

    Topics: Adult; Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; Drug Administration Schedule; Drug Dosage Calculations; Drug Monitoring; Dyslipidemias; Female; HIV Infections; HIV Protease Inhibitors; HIV-1; Humans; Hyperbilirubinemia; Male; Middle Aged; Nephrolithiasis; Ritonavir; Viral Load

2015
Treatment response to unboosted atazanavir in combination with tenofovir disoproxil fumarate and lamivudine in human immunodeficiency virus-1-infected patients who have achieved virological suppression: A therapeutic drug monitoring and pharmacogenetic st
    Journal of microbiology, immunology, and infection = Wei mian yu gan ran za zhi, 2017, Volume: 50, Issue:6

    Topics: Adult; Aged; Atazanavir Sulfate; ATP Binding Cassette Transporter, Subfamily B; Drug Combinations; Drug Monitoring; Female; Glucuronosyltransferase; HIV Infections; HIV Protease Inhibitors; HIV-1; Humans; Hyperbilirubinemia; Lamivudine; Male; Middle Aged; Peroxisome-Targeting Signal 1 Receptor; Pharmacogenomic Testing; Polymorphism, Single Nucleotide; Retrospective Studies; Reverse Transcriptase Inhibitors; Tenofovir; Treatment Failure; Viral Load; Young Adult

2017
Severe Hyperbilirubinemia in an HIV-HCV-Coinfected Patient Starting the 3D Regimen That Resolved After TDM-Guided Atazanavir Dose Reduction.
    Therapeutic drug monitoring, 2016, Volume: 38, Issue:3

    Topics: 2-Naphthylamine; Anilides; Antiviral Agents; Atazanavir Sulfate; Carbamates; Coinfection; Cyclopropanes; Dose-Response Relationship, Drug; Drug Interactions; Drug Monitoring; Drug Therapy, Combination; Female; Follow-Up Studies; Hepatitis C; HIV Infections; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Lactams, Macrocyclic; Macrocyclic Compounds; Middle Aged; Proline; Ritonavir; Sulfonamides; Uracil; Valine

2016
Drug- and Drug Abuse-Associated Hyperbilirubinemia: Experience With Atazanavir.
    Clinical pharmacology in drug development, 2017, Volume: 6, Issue:2

    Topics: Animals; Atazanavir Sulfate; Bilirubin; Cells, Cultured; Female; Glucuronosyltransferase; Glutathione Transferase; Hepatocytes; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Male; Rats, Wistar; Ritonavir; Substance-Related Disorders

2017
Increase in serum bilirubin in HIV/hepatitis-C virus-coinfected patients on atazanavir therapy following initiation of pegylated-interferon and ribavirin.
    AIDS (London, England), 2008, Nov-30, Volume: 22, Issue:18

    Topics: Adult; Antiviral Agents; Atazanavir Sulfate; Bilirubin; Drug Interactions; Female; Glucuronosyltransferase; Hepacivirus; HIV Infections; HIV Protease Inhibitors; HIV-1; Humans; Hyperbilirubinemia; Male; Middle Aged; Oligopeptides; Pyridines; Ribavirin

2008
Hyperbilirubinemia during atazanavir treatment in 2,404 patients in the Italian atazanavir expanded access program and MASTER Cohorts.
    Infection, 2009, Volume: 37, Issue:3

    Topics: Adult; Alanine Transaminase; Analysis of Variance; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; CD4 Lymphocyte Count; Cohort Studies; Female; Hepatitis C; HIV Infections; Humans; Hyperbilirubinemia; Liver; Male; Multivariate Analysis; Oligopeptides; Prevalence; Proportional Hazards Models; Pyridines; Risk Factors; Ritonavir; Severity of Illness Index

2009
Mid-dosing interval concentration of atazanavir and virological outcome in patients treated for HIV-1 infection.
    HIV medicine, 2010, Volume: 11, Issue:5

    Topics: Adult; Atazanavir Sulfate; Bilirubin; Drug Administration Schedule; Drug Interactions; Drug Monitoring; Drug Resistance, Viral; Drug Therapy, Combination; Female; HIV Infections; HIV Protease Inhibitors; HIV-1; Humans; Hyperbilirubinemia; Male; Middle Aged; Multivariate Analysis; Oligopeptides; Pyridines; Retrospective Studies; Ritonavir; Treatment Outcome; Viral Load

2010
Genetic factors influencing severe atazanavir-associated hyperbilirubinemia in a population with low UDP-glucuronosyltransferase 1A1*28 allele frequency.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2010, Jul-01, Volume: 51, Issue:1

    Topics: Adult; Anti-HIV Agents; Atazanavir Sulfate; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bilirubin; Female; Gene Frequency; Genes, MDR; Glucuronosyltransferase; HIV Infections; Humans; Hyperbilirubinemia; Korea; Logistic Models; Male; Middle Aged; Multivariate Analysis; Oligopeptides; Polymorphism, Genetic; Pyridines; Risk Factors; Sequence Analysis, DNA; Severity of Illness Index

2010
Incidence of atazanavir-associated hyperbilirubinemia in Korean HIV patients: 30 months follow-up results in a population with low UDP-glucuronosyltransferase1A1*28 allele frequency.
    Journal of Korean medical science, 2010, Volume: 25, Issue:10

    Topics: Adult; Alleles; Anti-HIV Agents; Asian People; Atazanavir Sulfate; Female; Follow-Up Studies; Gene Frequency; Glucuronosyltransferase; HIV Infections; Humans; Hyperbilirubinemia; Incidence; Male; Middle Aged; Oligopeptides; Promoter Regions, Genetic; Pyridines; Republic of Korea

2010
HIV-infected adolescents: relationship between atazanavir plasma levels and bilirubin concentrations.
    The Journal of adolescent health : official publication of the Society for Adolescent Medicine, 2011, Volume: 48, Issue:1

    Topics: Adolescent; Adolescent Health Services; Anti-HIV Agents; Atazanavir Sulfate; Bilirubin; Child; Drug Administration Schedule; Drug Monitoring; Female; HIV Infections; Humans; Hyperbilirubinemia; Male; Oligopeptides; Pyridines; Spain

2011
Short communication: UGT1A1*28 variant allele is a predictor of severe hyperbilirubinemia in HIV-infected patients on HAART in southern Brazil.
    AIDS research and human retroviruses, 2012, Volume: 28, Issue:9

    Topics: Acquired Immunodeficiency Syndrome; Adult; Alleles; Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; Bilirubin; Brazil; Cross-Sectional Studies; Female; Genotype; Glucuronosyltransferase; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Indinavir; Male; Oligopeptides; Predictive Value of Tests; Pyridines; Risk Factors; Severity of Illness Index

2012
Symptomatic hyperbilirubinemia secondary to dapsone-induced hemolysis and atazanavir therapy.
    Antimicrobial agents and chemotherapy, 2012, Volume: 56, Issue:2

    Topics: Adult; AIDS-Related Opportunistic Infections; Anemia, Hemolytic; Anti-HIV Agents; Anti-Infective Agents; Atazanavir Sulfate; Dapsone; Drug Therapy, Combination; Female; HIV Infections; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Male; Middle Aged; Oligopeptides; Pneumocystis carinii; Pneumonia, Pneumocystis; Pyridines

2012
Severe atazanavir-associated hyperbilirubinemia revealing Canton G6PD deficiency in an Asian HIV-infected patient.
    AIDS (London, England), 2012, Jan-14, Volume: 26, Issue:2

    Topics: Adult; Anti-HIV Agents; Asian People; Atazanavir Sulfate; Gilbert Disease; Glucosephosphate Dehydrogenase Deficiency; HIV Seropositivity; Humans; Hyperbilirubinemia; Male; Oligopeptides; Pyridines

2012
Atazanavir-related hyperbilirubinaemia is not highlighted in the British National Formulary.
    International journal of STD & AIDS, 2012, Volume: 23, Issue:10

    Topics: Anti-HIV Agents; Atazanavir Sulfate; Delivery of Health Care; Female; Germany; HIV Infections; Humans; Hyperbilirubinemia; Jaundice; Oligopeptides; Pharmacopoeias as Topic; Practice Guidelines as Topic; Pyridines; Referral and Consultation; United Kingdom

2012
Incidence of hyperbilirubinemia and jaundice due to atazanavir in a cohort of Hispanic patients.
    AIDS research and human retroviruses, 2013, Volume: 29, Issue:3

    Topics: Adult; Anti-HIV Agents; Atazanavir Sulfate; Female; Hispanic or Latino; HIV Infections; Humans; Hyperbilirubinemia; Incidence; Jaundice; Male; Middle Aged; Oligopeptides; Pyridines

2013
Drug-induced liver injury associated with antiretroviral therapy that includes HIV-1 protease inhibitors.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2004, Mar-01, Volume: 38 Suppl 2

    Topics: Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; Chemical and Drug Induced Liver Injury; HIV Infections; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Indinavir; Oligopeptides; Pyridines

2004
Plasma levels of atazanavir and the risk of hyperbilirubinemia are predicted by the 3435C-->T polymorphism at the multidrug resistance gene 1.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2006, Jan-15, Volume: 42, Issue:2

    Topics: Adult; Anti-HIV Agents; Atazanavir Sulfate; CD4 Lymphocyte Count; Female; Genes, MDR; Genetic Predisposition to Disease; Genotype; HIV Infections; HIV-1; Humans; Hyperbilirubinemia; Male; Middle Aged; Odds Ratio; Oligopeptides; Polymorphism, Genetic; Pyridines; Risk Factors; RNA, Viral; Viral Load

2006
Gilbert's disease and atazanavir: from phenotype to UDP-glucuronosyltransferase haplotype.
    Hepatology (Baltimore, Md.), 2006, Volume: 44, Issue:5

    Topics: Adult; Aged; Atazanavir Sulfate; Female; Genetic Variation; Gilbert Disease; Glucuronosyltransferase; Haplotypes; HIV Infections; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Male; Middle Aged; Oligopeptides; Polymorphism, Single Nucleotide; Pyridines

2006
Genetic factors influencing atazanavir plasma concentrations and the risk of severe hyperbilirubinemia.
    AIDS (London, England), 2007, Jan-02, Volume: 21, Issue:1

    Topics: Adult; Anti-HIV Agents; Atazanavir Sulfate; Female; Genes, MDR; Genotype; Glucuronosyltransferase; HIV Infections; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Logistic Models; Male; Middle Aged; Oligopeptides; Polymorphism, Genetic; Pyridines; Risk; Ritonavir

2007
Treatment of an atazanivir associated grade 4 hyperbilirubinaemia with efavirenz.
    Gut, 2007, Volume: 56, Issue:10

    Topics: Alkynes; Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; Benzoxazines; Cyclopropanes; HIV Infections; HIV Protease Inhibitors; Humans; Hyperbilirubinemia; Middle Aged; Oligopeptides; Pyridines

2007