Page last updated: 2024-09-05

asimadoline and Pain

asimadoline has been researched along with Pain in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (28.57)18.2507
2000's4 (57.14)29.6817
2010's0 (0.00)24.3611
2020's1 (14.29)2.80

Authors

AuthorsStudies
Ford, NC; Gao, X; Guan, Y; Guo, R; He, SQ; Huang, Q; Liu, S; Ma, D; Raja, SN; Zhang, C1
Burton, DD; Camilleri, M; Chial, HJ; Delgado-Aros, S; Ferber, I; Jacob, J; McKinzie, S; Szarka, LA; Weber, FT; Zinsmeister, AR1
Beck, A; Bouzamondo, H; Delvaux, M; Frexinos, J; Jacob, J; Weber, FT1
Averbeck, B; Guthmann, C; Kress, M; Reeh, PW1
Daubert, JD; Dehaven, R; Machelska, H; Pflüger, M; Piranvisseh-Völk, M; Stein, C; Weber, W1
Gebhart, GF; Ozaki, N; Sengupta, JN1
Gebhart, GF; Joshi, SK; Porreca, F; Su, X1

Trials

3 trial(s) available for asimadoline and Pain

ArticleYear
Effects of a kappa-opioid agonist, asimadoline, on satiation and GI motor and sensory functions in humans.
    American journal of physiology. Gastrointestinal and liver physiology, 2003, Volume: 284, Issue:4

    Topics: Acetamides; Adolescent; Adult; Colon; Compliance; Double-Blind Method; Female; Flatulence; Gastrointestinal Motility; Humans; Male; Middle Aged; Pain; Postprandial Period; Pyrrolidines; Receptors, Opioid, kappa; Satiation; Sensation; Stomach; Visceral Afferents

2003
Effect of asimadoline, a kappa opioid agonist, on pain induced by colonic distension in patients with irritable bowel syndrome.
    Alimentary pharmacology & therapeutics, 2004, Jul-15, Volume: 20, Issue:2

    Topics: Acetamides; Administration, Oral; Adolescent; Adult; Aged; Dilatation; Double-Blind Method; Female; Humans; Irritable Bowel Syndrome; Middle Aged; Narcotic Antagonists; Pain; Pain Measurement; Pain Threshold; Pressure; Pyrrolidines

2004
Peripheral effects of the kappa-opioid agonist EMD 61753 on pain and inflammation in rats and humans.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:1

    Topics: Acetamides; Adult; Analgesics, Opioid; Animals; Arthritis, Experimental; Arthroscopy; Behavior, Animal; CHO Cells; Cricetinae; Double-Blind Method; Female; Humans; Inflammation; Knee Joint; Male; Pain; Pain Measurement; Pain Threshold; Pain, Postoperative; Pyrrolidines; Rats; Rats, Wistar; Receptors, Opioid, kappa

1999

Other Studies

4 other study(ies) available for asimadoline and Pain

ArticleYear
The Utility of Peripherally Restricted Kappa-Opioid Receptor Agonists for Inhibiting Below-Level Pain After Spinal Cord Injury in Mice.
    Neuroscience, 2023, 09-01, Volume: 527

    Topics: Animals; Ganglia, Spinal; Mice; Pain; Pyrrolidines; Receptors, Opioid; Spinal Cord; Spinal Cord Injuries

2023
Calcitonin gene-related peptide and prostaglandin E2 but not substance P release induced by antidromic nerve stimulation from rat skin in vitro.
    Neuroscience, 1999, Volume: 89, Issue:1

    Topics: Acetamides; Analgesics, Opioid; Animals; Calcitonin Gene-Related Peptide; Dinoprostone; Electric Stimulation; Female; In Vitro Techniques; Male; Membrane Potentials; Nerve Fibers; Neurogenic Inflammation; Nociceptors; Pain; Pyrrolidines; Rats; Rats, Wistar; Receptors, Opioid, kappa; Skin; Stimulation, Chemical; Substance P; Vasodilation

1999
Differential effects of mu-, delta-, and kappa-opioid receptor agonists on mechanosensitive gastric vagal afferent fibers in the rat.
    Journal of neurophysiology, 2000, Volume: 83, Issue:4

    Topics: Acetamides; Analgesics; Analgesics, Opioid; Animals; Benzamides; Catheterization; Electric Stimulation; Male; Mechanoreceptors; Morphine; Naloxone; Narcotic Antagonists; Nerve Fibers; Neurons, Afferent; Pain; Piperazines; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Stomach; Vagus Nerve

2000
kappa -opioid receptor agonists modulate visceral nociception at a novel, peripheral site of action.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Aug-01, Volume: 20, Issue:15

    Topics: Acetamides; Analgesics, Opioid; Animals; Colon; Disinfectants; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Formaldehyde; Ganglia, Spinal; Male; Nociceptors; Oligonucleotides, Antisense; Oligopeptides; Pain; Physical Stimulation; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Rectum; Visceral Afferents

2000