Page last updated: 2024-08-25

artemisinin and Disease Models, Animal

artemisinin has been researched along with Disease Models, Animal in 48 studies

Research

Studies (48)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (6.25)18.2507
2000's5 (10.42)29.6817
2010's27 (56.25)24.3611
2020's13 (27.08)2.80

Authors

AuthorsStudies
Avery, VM; Baragaña, B; Campbell, SF; Delves, MJ; Duffy, S; Fairlamb, AH; Frearson, JA; Gilbert, IH; Gray, DW; Grimaldi, R; Hallyburton, I; Meister, S; Norcross, NR; Norval, S; Osuna-Cabello, M; Porzelle, A; Read, KD; Riley, J; Simeons, FR; Sinden, RE; Stojanovski, L; Waterson, D; Willis, P; Wilson, C; Winzeler, EA; Wittlin, S; Wyatt, PG1
Avery, VM; Baell, JB; Bullen, HE; Cowman, AF; Crabb, BS; Curtis, JM; Di Rago, AE; Duffy, S; Gilson, PR; Hutton, CA; Jarman, KE; Jousset Subroux, H; Lowes, KN; Nguyen, W; Prinz, B; Sleebs, BE; Tan, C1
Bordignon, A; Cieckiewicz, E; Di Giovanni, N; Frédérich, M; Hoareau, F; Illien, B; Jansen, O; Ledoux, A; Marvilliers, A; Pendeville, H; Quetin-Leclercq, J; St-Gelais, A1
Adah, D; Chen, X; Dai, L; Goldberg, DE; Guan, J; Leng, F; Li, X; Liu, J; Liu, X; Liu, Z; Lu, Y; Ma, H; McNitt, SA; Meyers, MJ; Nasamu, AS; Polino, AJ; Qin, L; Tortorella, MD; Tu, Z; Xu, J; Zhao, S1
Faist, J; Hochegger, P; Kaiser, M; Mäser, P; Saf, R; Seebacher, W; Weis, R1
Abrams, RPM; Bachani, M; Balasubramanian, A; Brimacombe, K; Dorjsuren, D; Eastman, RT; Hall, MD; Jadhav, A; Lee, MH; Li, W; Malik, N; Nath, A; Padmanabhan, R; Simeonov, A; Steiner, JP; Teramoto, T; Yasgar, A; Zakharov, AV1
Amanzougaghene, N; Ashraf, K; Azas, N; Benoit-Vical, F; Bosson-Vanga, H; Cohen, A; Dereuddre-Bosquet, N; Donnette, M; Franetich, JF; Gomez, L; Hutter, S; Lagardère, P; Lavazec, C; Le Grand, R; Lisowski, V; Malzert-Fréon, A; Masurier, N; Mazier, D; Mustière, R; Nguyen, M; Paloque, L; Primas, N; Rault, S; Roques, P; Snounou, G; Soulard, V; Suzanne, P; Tajeri, S; Tefit, M; Vanelle, P; Verhaeghe, P1
Chen, G; Kaplan, D; Li, G; Liu, P; Wang, X; Wu, Q; Xie, M; Yu, J; Zheng, Z1
Chen, L; He, SJ; Tong, X; Zuo, JP1
Hajebrahimi, Z; Noureddini, M; Poorgholam, P; Yaghmaei, P1
Ciapała, K; Ciechanowska, A; Mika, J; Pawlik, K; Rojewska, E1
Chen, Z; Li, T; Zhu, X1
Anderson, TJC; Button-Simons, K; Cheeseman, IH; Emrich, S; Ferdig, MT; Haile, M; Kappe, SHI; Kumar, S; Li, X; McDew-White, M; Nosten, F; Vaughan, AM1
Cao, Q; Du, H; Duan, N; Fu, X; Li, X; Liu, C1
Li, S; Liu, L; Silva, M; Xing, X; Zhao, X; Zheng, W1
Gille, L; Machín, L; Monzote, L; Nápoles, R1
Ge, W; Huai, M; Zeng, J1
Bao, Y; Chen, L; Dai, F; Li, Z; Liu, Z; Ma, Y; Peng, Y1
Çavuş, İ; Kaya, T; Nuraydın, A; Özbilgin, A1
Dawre, S; Devarajan, PV; Pathak, S; Sharma, S1
Chookajorn, T1
Brewer, JM; Lee, RS; Waters, AP1
Mu, X; Wang, C1
Cao, Y; Feng, YH; Gao, LW; Jin, F; Jin, QX; Li, XY; Lu, SL; Wang, YY; Wei, MJ; Xu, YY1
Cao, Q; Du, H; Fu, X; Jiang, Y; Li, X; Liu, X1
Benoit-Vical, F; Claparols, C; Robert, A; Witkowski, B1
Bakshi, RP; Nenortas, E; Shapiro, TA; Sullivan, DJ; Tripathi, AK1
Conyers, RC; Mazzone, JR; Posner, GH; Sullivan, DJ; Tripathi, AK1
Bhakuni, RS; Chauhan, A; Dhawan, OP; Dhawan, S; Khan, F; Qidwai, T; Sharma, P; Yadav, DK1
Chatterjee, S; Nodiff, EA; Tanabe, K1
Chen, J; Dong, L; Duan, W; Qiao, C; Sun, H; Xia, CM1
Cabral, L; Cristiano, ML; Lobo, L; Nogueira, F; Sousa, Bd1
Alexander, GR; Chatuverdi, NK; Chen, X; Coulter, DW; Dong, Y; Gray, S; Joshi, SS; McGuire, TR; McIntyre, EM; Sharp, JG; Vennerstrom, JL; Wang, X1
He, SJ; Lin, ZM; Tang, W; Yang, XQ; Zhu, FH; Zuo, JP1
Anderson, M; Bayih, AG; Eagon, S; Folefoc, A; Mohon, AN; Pillai, DR1
Atemnkeng, MA; Chimanuka, B; Dejaegher, B; Heyden, YV; Plaizier-Vercammen, J1
Gautam, N; Gupta, RC; Sabarinath, S; Singh, RP; Singh, SK1
Chatterjee, M; Ganguly, S; Saha, P; Sen, R1
Gros, P; Min-Oo, G1
An, P; Qiao, CL; Shi, XM; Sun, WS; Wang, Z; Wu, XL; Zhang, WG1
Bai, SF; Chen, H; Gao, Y; Li, T; Liu, DL; Liu, XG; Mei, X; Wei, N; Zhang, S; Zhou, YX1
An, P; Qiao, CL; Shi, XM; Sun, WS; Wang, Z; Wu, XL1
Bell, A1
Efferth, T1
Ager, A; Andersen, SL; Berman, J; Ellis, W; Kuschner, R; McGreevy, P; Ohrt, C; Rossan, R; Schuster, BG; Wesche, D1
Lederman, J; Rosenbaum, GS; Tanowitz, HB; Weiss, LM; Wittner, M1
Meshnick, SR1
Jain, GK; Pandey, VC; Puri, SK; Singh, S; Srivastava, P1

Reviews

6 review(s) available for artemisinin and Disease Models, Animal

ArticleYear
Artemisinin derivative SM934 in the treatment of autoimmune and inflammatory diseases: therapeutic effects and molecular mechanisms.
    Acta pharmacologica Sinica, 2022, Volume: 43, Issue:12

    Topics: Animals; Artemisinins; Autoimmune Diseases; Biological Products; Disease Models, Animal; Water

2022
Artemisinins-a Promising New Treatment for Systemic Lupus Erythematosus: a Descriptive Review.
    Current rheumatology reports, 2018, 07-28, Volume: 20, Issue:9

    Topics: Animals; Artemisinins; Artesunate; Disease Models, Animal; Humans; Immunosuppressive Agents; Lupus Erythematosus, Systemic; Mice

2018
Genetic analysis in mice identifies cysteamine as a novel partner for artemisinin in the treatment of malaria.
    Mammalian genome : official journal of the International Mammalian Genome Society, 2011, Volume: 22, Issue:7-8

    Topics: Amidohydrolases; Animals; Artemisinins; Cysteamine; Disease Models, Animal; Drug Therapy, Combination; GPI-Linked Proteins; Humans; Malaria; Mice; Plasmodium

2011
Antimalarial drug synergism and antagonism: mechanistic and clinical significance.
    FEMS microbiology letters, 2005, Dec-15, Volume: 253, Issue:2

    Topics: Animals; Antimalarials; Artemisinins; Disease Models, Animal; Drug Synergism; Drug Therapy, Combination; Folic Acid Antagonists; Humans; Malaria; Plasmodium berghei; Plasmodium falciparum; Protease Inhibitors; Quinolines; Sesquiterpenes

2005
Willmar Schwabe Award 2006: antiplasmodial and antitumor activity of artemisinin--from bench to bedside.
    Planta medica, 2007, Volume: 73, Issue:4

    Topics: Animals; Antimalarials; Antineoplastic Agents, Phytogenic; Artemisia annua; Artemisinins; Awards and Prizes; Disease Models, Animal; Drug Resistance, Multiple; Humans; Pharmacogenetics; Phytotherapy; Sesquiterpenes

2007
Artemisinin antimalarials: mechanisms of action and resistance.
    Medecine tropicale : revue du Corps de sante colonial, 1998, Volume: 58, Issue:3 Suppl

    Topics: Animals; Antimalarials; Artemisinins; Disease Models, Animal; Drug Evaluation, Preclinical; Drug Resistance; Humans; Malaria, Falciparum; Mice; Plasmodium falciparum; Protozoan Proteins; Sesquiterpenes

1998

Other Studies

42 other study(ies) available for artemisinin and Disease Models, Animal

ArticleYear
Discovery of a Quinoline-4-carboxamide Derivative with a Novel Mechanism of Action, Multistage Antimalarial Activity, and Potent in Vivo Efficacy.
    Journal of medicinal chemistry, 2016, 11-10, Volume: 59, Issue:21

    Topics: Animals; Antimalarials; Disease Models, Animal; Drug Discovery; Malaria; Mice; Molecular Structure; Plasmodium falciparum; Quinolines; Structure-Activity Relationship

2016
Optimization of 2-Anilino 4-Amino Substituted Quinazolines into Potent Antimalarial Agents with Oral in Vivo Activity.
    Journal of medicinal chemistry, 2017, 02-09, Volume: 60, Issue:3

    Topics: Administration, Oral; Animals; Antimalarials; Disease Models, Animal; Mice; Plasmodium falciparum; Quinazolines; Structure-Activity Relationship

2017
Antimalarial Activities of Alkyl Cyclohexenone Derivatives Isolated from the Leaves of Poupartia borbonica.
    Journal of natural products, 2017, 06-23, Volume: 80, Issue:6

    Topics: Anacardiaceae; Animals; Antimalarials; Belgium; Cyclohexanones; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Female; Flavonoids; HeLa Cells; Humans; Inhibitory Concentration 50; Malaria; Mice; Molecular Structure; Nuclear Magnetic Resonance, Biomolecular; Parasitic Sensitivity Tests; Plant Leaves; Plasmodium berghei; Plasmodium falciparum; Quercetin; Zebrafish

2017
4-Aryl Pyrrolidines as a Novel Class of Orally Efficacious Antimalarial Agents. Part 1: Evaluation of 4-Aryl- N-benzylpyrrolidine-3-carboxamides.
    Journal of medicinal chemistry, 2019, 04-11, Volume: 62, Issue:7

    Topics: Administration, Oral; Animals; Antimalarials; Biological Availability; Disease Models, Animal; Drug Evaluation, Preclinical; Malaria; Mice; Microsomes, Liver; Pyrrolidines; Structure-Activity Relationship

2019
Synthesis and structure-activity relationships for new 6-fluoroquinoline derivatives with antiplasmodial activity.
    Bioorganic & medicinal chemistry, 2019, 05-15, Volume: 27, Issue:10

    Topics: Animals; Antimalarials; Cell Line; Cell Survival; Disease Models, Animal; Drug Resistance; Malaria; Mice; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Quinolines; Structure-Activity Relationship

2019
Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors.
    Proceedings of the National Academy of Sciences of the United States of America, 2020, 12-08, Volume: 117, Issue:49

    Topics: Animals; Antiviral Agents; Artificial Intelligence; Chlorocebus aethiops; Disease Models, Animal; Drug Evaluation, Preclinical; High-Throughput Screening Assays; Immunocompetence; Inhibitory Concentration 50; Methacycline; Mice, Inbred C57BL; Protease Inhibitors; Quantitative Structure-Activity Relationship; Small Molecule Libraries; Vero Cells; Zika Virus; Zika Virus Infection

2020
A New Thienopyrimidinone Chemotype Shows Multistage Activity against Plasmodium falciparum, Including Artemisinin-Resistant Parasites.
    Microbiology spectrum, 2021, 10-31, Volume: 9, Issue:2

    Topics: Animals; Antimalarials; Artemisinins; Cell Line, Tumor; Disease Models, Animal; Dogs; Drug Resistance; Female; Hep G2 Cells; Humans; Liver; Macaca fascicularis; Madin Darby Canine Kidney Cells; Malaria, Falciparum; Male; Mice; Mice, Inbred BALB C; Plasmodium cynomolgi; Plasmodium falciparum; Plasmodium yoelii; Pyrimidinones

2021
Sustainable Antibacterial and Anti-Inflammatory Silk Suture with Surface Modification of Combined-Therapy Drugs for Surgical Site Infection.
    ACS applied materials & interfaces, 2022, Mar-09, Volume: 14, Issue:9

    Topics: Animals; Anti-Bacterial Agents; Anti-Inflammatory Agents; Artemisinins; Berberine; Cell Line; Cell Survival; Coated Materials, Biocompatible; Disease Models, Animal; Drug Liberation; Drug Therapy, Combination; Escherichia coli; Hemolysis; Humans; Male; Physical Phenomena; Rats, Sprague-Dawley; Silk; Staphylococcus aureus; Surgical Wound Infection; Sutures

2022
Artemisin and human endometrial-derived stem cells improve cognitive function and synaptic plasticity in a rat model of Alzheimer disease and diabetes.
    Metabolic brain disease, 2023, Volume: 38, Issue:6

    Topics: Alzheimer Disease; Animals; Artemisinins; Cognition; Diabetes Mellitus; Disease Models, Animal; Hippocampus; Humans; Long-Term Potentiation; Maze Learning; Neurodegenerative Diseases; Neuronal Plasticity; Rats; Streptozocin; Thrombospondin 1

2023
Analgesic Effects of Fisetin, Peimine, Astaxanthin, Artemisinin, Bardoxolone Methyl and 740 Y-P and Their Influence on Opioid Analgesia in a Mouse Model of Neuropathic Pain.
    International journal of molecular sciences, 2023, May-19, Volume: 24, Issue:10

    Topics: Analgesia; Analgesics; Analgesics, Opioid; Animals; Artemisinins; Disease Models, Animal; Hyperalgesia; Male; Mice; Morphine; Neuralgia; NF-E2-Related Factor 2; NF-kappa B; Oxycodone; Phosphatidylinositol 3-Kinases

2023
[Oral administration of artemisinin nanospheres alleviates inflammation in mice with spontaneous ulcerative colitis].
    Xi bao yu fen zi mian yi xue za zhi = Chinese journal of cellular and molecular immunology, 2023, Volume: 39, Issue:9

    Topics: Administration, Oral; Animals; Artemisinins; Colitis, Ulcerative; Disease Models, Animal; Inflammation; Mice; Nanospheres; RNA, Messenger

2023
Genetic mapping of fitness determinants across the malaria parasite Plasmodium falciparum life cycle.
    PLoS genetics, 2019, Volume: 15, Issue:10

    Topics: Animals; Anopheles; Antimalarials; Artemisinins; Chromosome Mapping; Disease Models, Animal; Drug Resistance; Female; Gene Frequency; Genetic Loci; Host-Parasite Interactions; Humans; Life Cycle Stages; Malaria, Falciparum; Male; Mice; Mosquito Vectors; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Plasmodium falciparum; Polymorphism, Single Nucleotide; Protozoan Proteins; Ribosomal Proteins; Selection, Genetic; Transplantation Chimera

2019
Artemisinin Attenuated Atherosclerosis in High-Fat Diet-Fed ApoE-/- Mice by Promoting Macrophage Autophagy Through the AMPK/mTOR/ULK1 Pathway.
    Journal of cardiovascular pharmacology, 2020, Volume: 75, Issue:4

    Topics: AMP-Activated Protein Kinases; Animals; Anti-Inflammatory Agents; Aorta; Aortic Diseases; Artemisinins; Atherosclerosis; Autophagy; Autophagy-Related Protein-1 Homolog; Diet, High-Fat; Disease Models, Animal; Foam Cells; Lipoproteins, LDL; Male; Mice; Mice, Inbred C57BL; Mice, Knockout, ApoE; Microtubule-Associated Proteins; Phosphorylation; Plaque, Atherosclerotic; RAW 264.7 Cells; Sequestosome-1 Protein; Signal Transduction; TOR Serine-Threonine Kinases

2020
Artemisinin protects motoneurons against axotomy-induced apoptosis through activation of the PKA-Akt signaling pathway and promotes neural stem/progenitor cells differentiation into NeuN
    Pharmacological research, 2020, Volume: 159

    Topics: Animals; Apoptosis; Artemisinins; Axotomy; Behavior, Animal; Brachial Plexus; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Disease Models, Animal; DNA-Binding Proteins; Mice, Inbred C57BL; Motor Neurons; Nerve Tissue Proteins; Neural Stem Cells; Neurogenesis; Neuroprotective Agents; Peripheral Nerve Injuries; Phosphorylation; Proto-Oncogene Proteins c-akt; Recovery of Function; Signal Transduction; Spinal Cord

2020
Leishmania amazonensis response to artemisinin and derivatives.
    Parasitology international, 2021, Volume: 80

    Topics: Animals; Artemether; Artemisinins; Artesunate; Disease Models, Animal; Female; Leishmania mexicana; Mice; Mice, Inbred BALB C; Parasite Load; Trypanocidal Agents

2021
Artemisinin ameliorates intestinal inflammation by skewing macrophages to the M2 phenotype and inhibiting epithelial-mesenchymal transition.
    International immunopharmacology, 2021, Volume: 91

    Topics: Animals; Anti-Inflammatory Agents; Artemisinins; Colitis; Colon; Crohn Disease; Cytokines; Dextran Sulfate; Disease Models, Animal; Epithelial-Mesenchymal Transition; Female; Humans; Inflammation Mediators; Macrophages; Mice; Mice, Inbred C57BL; Phenotype; RAW 264.7 Cells; Signal Transduction; Tissue Culture Techniques

2021
Electrospun PLGA/SF/artemisinin composite nanofibrous membranes for wound dressing.
    International journal of biological macromolecules, 2021, Jul-31, Volume: 183

    Topics: Animals; Anti-Infective Agents; Artemisinins; Bandages; Cytokines; Delayed-Action Preparations; Disease Models, Animal; Drug Carriers; Drug Compounding; Drug Liberation; Fibroins; Macrophages; Male; Membranes, Artificial; Mice; Nanofibers; Polylactic Acid-Polyglycolic Acid Copolymer; Rats, Sprague-Dawley; RAW 264.7 Cells; Skin; Wound Healing; Wounds, Penetrating

2021
In vivo and in vitro Models for Scanning Drug Substances in Malaria: Prestudy.
    Turkiye parazitolojii dergisi, 2017, Volume: 41, Issue:3

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; Disease Models, Animal; Drug Evaluation, Preclinical; In Vitro Techniques; Malaria; Male; Mice; Mice, Inbred BALB C; Plant Extracts; Plasmodium berghei; Tetracycline

2017
Enhanced antimalalarial activity of a prolonged release in situ gel of arteether-lumefantrine in a murine model.
    European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V, 2018, Volume: 123

    Topics: Animals; Antimalarials; Artemisinins; Chemistry, Pharmaceutical; Delayed-Action Preparations; Disease Models, Animal; Drug Therapy, Combination; Ethanolamines; Fluorenes; Gels; Lumefantrine; Malaria, Falciparum; Male; Mice; Polymers

2018
How to combat emerging artemisinin resistance: Lessons from "The Three Little Pigs".
    PLoS pathogens, 2018, Volume: 14, Issue:4

    Topics: Animals; Antimalarials; Artemisinins; Disease Models, Animal; Drug Resistance; Humans; Malaria, Falciparum; Plasmodium falciparum; Public Health; Swine

2018
A cryptic cycle in haematopoietic niches promotes initiation of malaria transmission and evasion of chemotherapy.
    Nature communications, 2018, 04-27, Volume: 9, Issue:1

    Topics: Animals; Antimalarials; Artemisinins; Disease Models, Animal; Drug Resistance; Female; Gametogenesis; Hematopoietic Stem Cells; Humans; Malaria; Mice; Mice, Inbred BALB C; Plasmodium berghei; Reproduction, Asexual; Reticulocytes; Stem Cell Niche

2018
Artemisinin enhances the anti-tumor immune response in 4T1 breast cancer cells in vitro and in vivo.
    International immunopharmacology, 2019, Volume: 70

    Topics: Animals; Apoptosis; Artemisinins; Breast Neoplasms; CD4-Positive T-Lymphocytes; Cell Line, Tumor; Cell Proliferation; Disease Models, Animal; Female; Humans; Immunity, Cellular; Immunization; Interferon-gamma; Lymphocyte Activation; Medicine, Chinese Traditional; Mice; Mice, Inbred BALB C; T-Box Domain Proteins; T-Lymphocytes, Cytotoxic; T-Lymphocytes, Regulatory

2019
Artemisinin alleviates atherosclerotic lesion by reducing macrophage inflammation via regulation of AMPK/NF-κB/NLRP3 inflammasomes pathway.
    Journal of drug targeting, 2020, Volume: 28, Issue:1

    Topics: AMP-Activated Protein Kinases; Animals; Artemisinins; Atherosclerosis; Cell Culture Techniques; Diet, High-Fat; Disease Models, Animal; Dose-Response Relationship, Drug; Inflammasomes; Inflammation; Inflammation Mediators; Macrophages; Male; Mice; NF-kappa B; NLR Family, Pyrin Domain-Containing 3 Protein

2020
Correlation between Plasmodium yoelii nigeriensis susceptibility to artemisinin and alkylation of heme by the drug.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:8

    Topics: Alkylation; Animals; Antimalarials; Artemisinins; Disease Models, Animal; Drug Evaluation, Preclinical; Drug Resistance; Erythrocytes; Female; Heme; Malaria; Mice; Plasmodium yoelii; Protein Binding; Spleen

2013
Model system to define pharmacokinetic requirements for antimalarial drug efficacy.
    Science translational medicine, 2013, Oct-02, Volume: 5, Issue:205

    Topics: Animals; Antimalarials; Artemisinins; Chloroquine; Disease Models, Animal; Humans; Malaria, Falciparum; Mice; Mice, Inbred C57BL; Models, Biological; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Reproducibility of Results; Treatment Outcome

2013
Antimalarial chemotherapy: artemisinin-derived dimer carbonates and thiocarbonates.
    Bioorganic & medicinal chemistry letters, 2014, Jun-01, Volume: 24, Issue:11

    Topics: Animals; Antimalarials; Artemisinins; Carbonates; Dimerization; Disease Models, Animal; Dose-Response Relationship, Drug; Malaria; Male; Mice; Mice, Inbred C57BL; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium berghei; Structure-Activity Relationship; Sulfhydryl Compounds

2014
QSAR and docking based semi-synthesis and in vivo evaluation of artemisinin derivatives for antimalarial activity.
    Current drug targets, 2014, Volume: 15, Issue:8

    Topics: Animals; Antimalarials; Artemisinins; Aspartic Acid Endopeptidases; Binding Sites; Biological Availability; Computer-Aided Design; Disease Models, Animal; Drug Design; Magnetic Resonance Spectroscopy; Malaria; Mice; Molecular Docking Simulation; Plasmodium yoelii; Protozoan Proteins; Quantitative Structure-Activity Relationship

2014
In search of next generation antimalarials.
    Bioorganic & medicinal chemistry letters, 2014, Sep-01, Volume: 24, Issue:17

    Topics: Animals; Antimalarials; Artemisinins; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Discovery; Macaca mulatta; Malaria; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium; Structure-Activity Relationship

2014
An artemisinin derivative of praziquantel as an orally active antischistosomal agent.
    PloS one, 2014, Volume: 9, Issue:11

    Topics: Administration, Oral; Animals; Artemisinins; Disease Models, Animal; Female; Mice; Mice, Inbred ICR; Praziquantel; Schistosomiasis japonica; Schistosomicides

2014
Highly active ozonides selected against drug resistant malaria.
    Memorias do Instituto Oswaldo Cruz, 2016, Jun-07, Volume: 0

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Chloroquine; Disease Models, Animal; Female; Humans; Malaria, Falciparum; Mefloquine; Mice; Parasitemia; Plasmodium falciparum

2016
Treatment of a chemoresistant neuroblastoma cell line with the antimalarial ozonide OZ513.
    BMC cancer, 2016, 11-08, Volume: 16, Issue:1

    Topics: Animals; Antimalarials; Antineoplastic Agents; Apoptosis; Artemisinins; Biomarkers; Caspase 3; Cell Cycle; Cell Line, Tumor; Disease Models, Animal; Drug Resistance, Neoplasm; Heterocyclic Compounds; Humans; Metabolome; Metabolomics; Mice; Neuroblastoma; Xenograft Model Antitumor Assays

2016
Artemisinin analogue SM934 attenuate collagen-induced arthritis by suppressing T follicular helper cells and T helper 17 cells.
    Scientific reports, 2016, 11-29, Volume: 6

    Topics: Animals; Artemisinins; Arthritis, Experimental; Arthritis, Rheumatoid; Cattle; CD4-Positive T-Lymphocytes; Collagen Type II; Disease Models, Animal; Female; Interferon-gamma; Interleukins; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Inbred DBA; Proto-Oncogene Proteins c-bcl-6; STAT3 Transcription Factor; Th17 Cells

2016
In vitro and in vivo anti-malarial activity of novel harmine-analog heat shock protein 90 inhibitors: a possible partner for artemisinin.
    Malaria journal, 2016, Dec-01, Volume: 15, Issue:1

    Topics: Animals; Antimalarials; Artemisinins; Cell Line; Cell Survival; Disease Models, Animal; Drug Synergism; Female; Harmine; HSP90 Heat-Shock Proteins; Humans; Inhibitory Concentration 50; Malaria; Mice, Inbred BALB C; Plasmodium berghei; Plasmodium falciparum; Protein Binding; Protozoan Proteins; Treatment Outcome

2016
Evaluation of Artemisia annua infusion efficacy for the treatment of malaria in Plasmodium chabaudi chabaudi infected mice.
    Experimental parasitology, 2009, Volume: 122, Issue:4

    Topics: Animals; Anti-Infective Agents; Artemisia annua; Artemisinins; Beverages; Chromatography, Thin Layer; Densitometry; Disease Models, Animal; Female; Malaria; Mice; Parasitemia; Phytotherapy; Plant Leaves; Plasmodium chabaudi

2009
Liquid chromatographic tandem mass spectrometric assay for quantification of 97/78 and its metabolite 97/63: a promising trioxane antimalarial in monkey plasma.
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2009, Jul-15, Volume: 877, Issue:22

    Topics: Animals; Antimalarials; Artemisinins; Chromatography, Liquid; Disease Models, Animal; Humans; Macaca mulatta; Malaria; Male; Tandem Mass Spectrometry

2009
Efficacy of artemisinin in experimental visceral leishmaniasis.
    International journal of antimicrobial agents, 2010, Volume: 36, Issue:1

    Topics: Animals; Antiprotozoal Agents; Artemisinins; Disease Models, Animal; Humans; Inhibitory Concentration 50; Leishmania donovani; Leishmaniasis, Visceral; Macrophages; Mice; Mice, Inbred BALB C; Parasitic Sensitivity Tests; Spleen; Treatment Outcome

2010
Effect of artemisinin combined with glucocorticoid on the expressions of glucocorticoid receptor α mRNA, glucocorticoid receptor β mRNA and P300/CBP protein in lupus nephritis mice.
    Chinese journal of integrative medicine, 2011, Volume: 17, Issue:4

    Topics: Animals; Artemisinins; Base Sequence; Disease Models, Animal; DNA Primers; Electrophoresis, Agar Gel; Female; Lupus Nephritis; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; p300-CBP Transcription Factors; Prednisone; Receptors, Glucocorticoid; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2011
Anti-inflammatory and immunomodulatory mechanisms of artemisinin on contact hypersensitivity.
    International immunopharmacology, 2012, Volume: 12, Issue:1

    Topics: Animals; Anti-Inflammatory Agents; Artemisinins; Concanavalin A; Cytokines; Dermatitis, Contact; Dinitrofluorobenzene; Disease Models, Animal; Female; Immunologic Factors; Irritants; Lymph Nodes; Mice; Mice, Inbred BALB C; Mitogens; Organ Size; Phytotherapy; Spleen; T-Lymphocytes, Regulatory; Th17 Cells

2012
[Effect of artemisinin on the expressions of GRalpha mRNA, GRbeta mRNA and P300/CBP protein in lupus nephritis mice].
    Zhong yao cai = Zhongyaocai = Journal of Chinese medicinal materials, 2012, Volume: 35, Issue:4

    Topics: Animals; Artemisia annua; Artemisinins; Disease Models, Animal; Female; Leukocytes, Mononuclear; Lupus Nephritis; Mice; Mice, Inbred Strains; p300-CBP Transcription Factors; Prednisone; Receptors, Glucocorticoid; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2012
Activity of azithromycin as a blood schizonticide against rodent and human plasmodia in vivo.
    The American journal of tropical medicine and hygiene, 1995, Volume: 52, Issue:2

    Topics: Administration, Oral; Animals; Antimalarials; Aotus trivirgatus; Artemisinins; Azithromycin; Disease Models, Animal; Doxycycline; Drug Therapy, Combination; Humans; Injections, Subcutaneous; Malaria; Malaria, Falciparum; Mice; Parasitemia; Phenanthrenes; Plasmodium berghei; Quinine; Sesquiterpenes

1995
Atovaquone in the treatment of Babesia microti infections in hamsters.
    The American journal of tropical medicine and hygiene, 1996, Volume: 55, Issue:2

    Topics: Animals; Anti-Bacterial Agents; Antimalarials; Antiprotozoal Agents; Artemisinins; Atovaquone; Azithromycin; Babesiosis; Cricetinae; Disease Models, Animal; Drug Therapy, Combination; Naphthoquinones; Parasitemia; Recurrence; Sesquiterpenes

1996
A simple and rapid evaluation of methemoglobin toxicity of 8-aminoquinolines and related compounds.
    Ecotoxicology and environmental safety, 2000, Volume: 45, Issue:3

    Topics: Administration, Cutaneous; Administration, Oral; Aminoquinolines; Animals; Antimalarials; Artemisinins; Cell-Free System; Chloroquine; Cytochrome-B(5) Reductase; Disease Models, Animal; Dogs; Dose-Response Relationship, Drug; Erythrocytes; Macaca mulatta; Methemoglobin; Methemoglobinemia; Muridae; Oxyhemoglobins; Primaquine; Rats; Sesquiterpenes

2000