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amodiaquine hydrochloride and Infections, Plasmodium

amodiaquine hydrochloride has been researched along with Infections, Plasmodium in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19903 (20.00)18.7374
1990's1 (6.67)18.2507
2000's7 (46.67)29.6817
2010's4 (26.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Johnson, J; Kesten, SJ; Werbel, LM1
Cook, PD; Elslager, EF; Hung, JH; Johnson, JL; Kesten, SJ; McNamara, DJ; Ortwine, DF; Werbel, LM; Worth, DF1
Go, ML; Ngiam, TL; Wan, AS1
O'Neill, PM; Park, BK; Raynes, KJ; Stocks, PA; Ward, SA1
Debreu-Fontaine, MA; Delarue, S; Girault, S; Grellier, P; Labaeïd, M; Maes, L; Sergheraert, C1
Bickley, JF; Bray, PG; Hindley, S; Hughes, RH; Maggs, JL; Mukhtar, A; O'Neil, IA; O'Neill, PM; Park, BK; Randle, LE; Stocks, PA; Storr, RC; Ward, SA; Winstanley, PA1
Delarue-Cochin, S; Grellier, P; Maes, L; Melnyk, P; Mouray, E; Sergheraert, C1
Becker, K; Davioud-Charvet, E; Friebolin, W; Furrer, J; Jannack, B; Lanzer, M; Oeser, T; Sanchez, CP; Wenzel, N; Yardley, V1
Adrián, F; Anderson, P; Brinker, A; Caldwell, JS; Chatterjee, A; Gray, NS; Henson, K; Janes, J; Kato, N; Kuhen, K; Matzen, JT; McNamara, C; Nagle, A; Nam, TG; Plouffe, D; Schultz, PG; Trager, R; Winzeler, EA; Yan, SF; Zhou, Y1
Bambal, RB; Bates, M; Berry, N; Biagini, GA; Bonar-Law, R; Bray, PG; Brigandi, RA; Davis, CB; Gargallo, DV; Gibbons, P; Gomez-delas-Heras, FM; Gresham, SL; Hart, TK; Hindley, S; Lawrence, RM; Maggs, JL; Mukhtar, A; O'Neill, PM; Park, BK; Roberts, P; Shone, AE; Stocks, PA; Ward, SA; Winstanley, PA1
Asadollahy, E; Bambal, RB; Bates, M; Berry, N; Biagini, G; Bray, PG; Brigandi, RA; Davies, J; Davis, CB; Gargallo, DV; Gomez-de-Las-Heras, FM; Gresham, SL; Hall, C; Hindley, S; Lander, H; Maggs, JL; Nixon, G; O'Neill, PM; Parapini, S; Park, BK; Rimmer, K; Roberts, P; Shone, AE; Stanford, D; Stocks, PA; Taramelli, D; Vivas, L; Ward, SA; Winstanley, PA1
Ba, EH; Cairns, M; Cames, C; Cisse, B; Gaye, O; Greenwood, BM; Milligan, PJ; Simondon, K; Sokhna, C; Trape, JF1
Anstey, NM; Chalfein, F; Ebsworth, EP; Kenangalem, E; Marfurt, J; Piera, KA; Prasetyorini, B; Price, RN; Ratcliff, A; Russell, B; Siswantoro, H; Tjitra, E; Wuwung, M1
Chandrashekar, G; Chatterji, D; Meng, L; Robinson, K; Zhu, S1
Biamonte, MA; Le Roch, KG; Wanner, J1

Reviews

1 review(s) available for amodiaquine hydrochloride and Infections, Plasmodium

ArticleYear
Recent advances in malaria drug discovery.
    Bioorganic & medicinal chemistry letters, 2013, May-15, Volume: 23, Issue:10

    Topics: Animals; Antimalarials; Drug Discovery; Humans; Liver; Liver Transplantation; Malaria; Molecular Structure

2013

Trials

1 trial(s) available for amodiaquine hydrochloride and Infections, Plasmodium

ArticleYear
Amodiaquine dosage and tolerability for intermittent preventive treatment to prevent malaria in children.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:3

    Topics: Age Factors; Amodiaquine; Antimalarials; Body Weight; Child; Child, Preschool; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Combinations; Drug Therapy, Combination; Humans; Infant; Malaria; Pyrimethamine; Seasons; Sulfadoxine; Treatment Outcome

2010

Other Studies

13 other study(ies) available for amodiaquine hydrochloride and Infections, Plasmodium

ArticleYear
Synthesis and antimalarial effects of 4-[(7-chloro-4-quinolinyl)amino]-2-[(diethylamino)methyl] -6-alkylphenols and their N omega-oxides.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:5

    Topics: Aminoquinolines; Animals; Chemical Phenomena; Chemistry; Cyclic N-Oxides; Malaria; Mice; Phenols; Plasmodium berghei; Structure-Activity Relationship

1987
Synthesis, antimalarial activity, and quantitative structure-activity relationships of tebuquine and a series of related 5-[(7-chloro-4-quinolinyl)amino]-3-[(alkylamino)methyl] [1,1'-biphenyl]-2-ols and N omega-oxides.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:6

    Topics: Aminoquinolines; Animals; Antimalarials; Drug Resistance; Malaria; Mice; Regression Analysis; Structure-Activity Relationship

1986
Synthesis of some novel amodiaquine analogues as potential antimalarial and antifilarial compounds.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:12

    Topics: Amodiaquine; Animals; Anthelmintics; Antimalarials; Chemical Phenomena; Chemistry; Filariasis; Filaricides; Malaria; Mice; Plasmodium berghei

1981
New 4-aminoquinoline Mannich base antimalarials. 1. Effect of an alkyl substituent in the 5'-position of the 4'-hydroxyanilino side chain.
    Journal of medicinal chemistry, 1999, Jul-29, Volume: 42, Issue:15

    Topics: Aniline Compounds; Animals; Antimalarials; Inhibitory Concentration 50; Malaria; Male; Mannich Bases; Mice; Plasmodium berghei; Plasmodium falciparum; Quinolines; Structure-Activity Relationship

1999
Synthesis and in vitro and in vivo antimalarial activity of new 4-anilinoquinolines.
    Journal of medicinal chemistry, 2001, Aug-16, Volume: 44, Issue:17

    Topics: Aniline Compounds; Animals; Antimalarials; Cells, Cultured; Drug Resistance; Female; Humans; Macrophages, Peritoneal; Malaria; Mice; Plasmodium berghei; Plasmodium falciparum; Quinolines; Structure-Activity Relationship

2001
Isoquine and related amodiaquine analogues: a new generation of improved 4-aminoquinoline antimalarials.
    Journal of medicinal chemistry, 2003, Nov-06, Volume: 46, Issue:23

    Topics: Aminoquinolines; Amodiaquine; Animals; Antimalarials; Crystallography, X-Ray; Malaria; Male; Plasmodium falciparum; Plasmodium yoelii; Rats; Rats, Wistar; Structure-Activity Relationship

2003
Synthesis and antimalarial activity of carbamate and amide derivatives of 4-anilinoquinoline.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:10

    Topics: Amides; Animals; Antimalarials; Carbamates; Cell Line; Female; Humans; Malaria; Mice; Plasmodium falciparum; Quinolines; Structure-Activity Relationship

2008
Antimalarial dual drugs based on potent inhibitors of glutathione reductase from Plasmodium falciparum.
    Journal of medicinal chemistry, 2008, Mar-13, Volume: 51, Issue:5

    Topics: Animals; Antimalarials; Biological Transport; Cell Line, Tumor; Chloroquine; Drug Resistance; Drug Therapy, Combination; Glutathione Reductase; Humans; In Vitro Techniques; Malaria; Mice; Mice, Inbred BALB C; Naphthalenes; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Structure-Activity Relationship

2008
In silico activity profiling reveals the mechanism of action of antimalarials discovered in a high-throughput screen.
    Proceedings of the National Academy of Sciences of the United States of America, 2008, Jul-01, Volume: 105, Issue:26

    Topics: Animals; Antimalarials; Cluster Analysis; Computational Biology; Drug Evaluation, Preclinical; Drug Resistance; Folic Acid Antagonists; Malaria; Models, Molecular; Parasites; Plasmodium falciparum; Reproducibility of Results; Structure-Activity Relationship; Tetrahydrofolate Dehydrogenase

2008
Candidate selection and preclinical evaluation of N-tert-butyl isoquine (GSK369796), an affordable and effective 4-aminoquinoline antimalarial for the 21st century.
    Journal of medicinal chemistry, 2009, Mar-12, Volume: 52, Issue:5

    Topics: Aminoquinolines; Amodiaquine; Animals; Antimalarials; Benzylamines; Cytochrome P-450 Enzyme Inhibitors; Dogs; Drug Evaluation, Preclinical; Drug Resistance; Female; Haplorhini; Heme; Humans; Malaria; Mice; Models, Molecular; Plasmodium berghei; Plasmodium falciparum; Plasmodium yoelii; Rats; Structure-Activity Relationship

2009
Synthesis, antimalarial activity, and preclinical pharmacology of a novel series of 4'-fluoro and 4'-chloro analogues of amodiaquine. Identification of a suitable "back-up" compound for N-tert-butyl isoquine.
    Journal of medicinal chemistry, 2009, Apr-09, Volume: 52, Issue:7

    Topics: Aminoquinolines; Amodiaquine; Animals; Antimalarials; Cell Survival; Chloroquine; Dogs; Drug Resistance; Female; Haplorhini; Hepatocytes; Humans; In Vitro Techniques; Malaria; Male; Mice; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Plasmodium yoelii; Rats; Rats, Wistar; Structure-Activity Relationship

2009
In vivo and in vitro efficacy of chloroquine against Plasmodium malariae and P. ovale in Papua, Indonesia.
    Antimicrobial agents and chemotherapy, 2011, Volume: 55, Issue:1

    Topics: Adolescent; Adult; Antimalarials; Child; Child, Preschool; Chloroquine; Female; Humans; Indonesia; Malaria; Male; Middle Aged; Plasmodium malariae; Plasmodium ovale; Treatment Outcome; Young Adult

2011
Febrifugine analogue compounds: synthesis and antimalarial evaluation.
    Bioorganic & medicinal chemistry, 2012, Jan-15, Volume: 20, Issue:2

    Topics: Animals; Antimalarials; Aotus trivirgatus; Drug Evaluation, Preclinical; Malaria; Piperidines; Plasmodium falciparum; Quinazolines

2012