Page last updated: 2024-10-22

am 251 and Cocaine Abuse

am 251 has been researched along with Cocaine Abuse in 6 studies

AM 251: an analog of SR141716A; structure given in first source
AM-251 : A carbohydrazide obtained by formal condensation of the carboxy group of 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-1H-pyrazole-3-carboxylic acid with the amino group of 1-aminopiperidine. An antagonist at the CB1 cannabinoid receptor.

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (33.33)29.6817
2010's4 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
McReynolds, JR2
Doncheck, EM2
Li, Y1
Vranjkovic, O2
Graf, EN1
Ogasawara, D1
Cravatt, BF1
Baker, DA2
Liu, QS1
Hillard, CJ2
Mantsch, JR2
Ganzman, GS1
Adamczyk, P1
Miszkiel, J1
McCreary, AC1
Filip, M1
Papp, M1
Przegaliński, E1
Kupferschmidt, DA1
Klas, PG1
Erb, S1
Xi, ZX1
Gilbert, JG1
Peng, XQ1
Pak, AC1
Li, X1
Gardner, EL1
Corbillé, AG1
Valjent, E1
Marsicano, G1
Ledent, C1
Lutz, B1
Hervé, D1
Girault, JA1

Other Studies

6 other studies available for am 251 and Cocaine Abuse

ArticleYear
Stress Promotes Drug Seeking Through Glucocorticoid-Dependent Endocannabinoid Mobilization in the Prelimbic Cortex.
    Biological psychiatry, 2018, 07-15, Volume: 84, Issue:2

    Topics: Animals; Arachidonic Acids; Cocaine; Cocaine-Related Disorders; Drug-Seeking Behavior; Endocannabino

2018
CB1 receptor antagonism blocks stress-potentiated reinstatement of cocaine seeking in rats.
    Psychopharmacology, 2016, Volume: 233, Issue:1

    Topics: Animals; Arachidonic Acids; Behavior, Addictive; Cocaine; Cocaine-Related Disorders; Endocannabinoid

2016
The effects of cannabinoid CB1, CB2 and vanilloid TRPV1 receptor antagonists on cocaine addictive behavior in rats.
    Brain research, 2012, Mar-20, Volume: 1444

    Topics: Analysis of Variance; Anilides; Animals; Behavior, Addictive; Camphanes; Cinnamates; Cocaine-Related

2012
Cannabinoid CB1 receptors mediate the effects of corticotropin-releasing factor on the reinstatement of cocaine seeking and expression of cocaine-induced behavioural sensitization.
    British journal of pharmacology, 2012, Volume: 167, Issue:1

    Topics: Animals; Behavior, Animal; Cannabinoid Receptor Antagonists; Cocaine; Cocaine-Related Disorders; Cor

2012
Cannabinoid CB1 receptor antagonist AM251 inhibits cocaine-primed relapse in rats: role of glutamate in the nucleus accumbens.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2006, Aug-16, Volume: 26, Issue:33

    Topics: Animals; Behavior, Animal; Cocaine; Cocaine-Related Disorders; Dopamine; Extracellular Space; gamma-

2006
Role of cannabinoid type 1 receptors in locomotor activity and striatal signaling in response to psychostimulants.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2007, Jun-27, Volume: 27, Issue:26

    Topics: Animals; Central Nervous System Stimulants; Cocaine; Cocaine-Related Disorders; Corpus Striatum; Dos

2007