Page last updated: 2024-08-21

alpha-aminopyridine and Malaria

alpha-aminopyridine has been researched along with Malaria in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19902 (28.57)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's5 (71.43)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Abraham, TS; Angulo-Barturen, I; Bantscheff, M; Basak, R; Birkholtz, LM; Blagborough, AM; Bodenreider, C; Botha, M; Burrows, J; Cabrera, DG; Campo, B; Charman, SA; Chibale, K; Dechering, KJ; Delves, MJ; Donini, C; Drewes, G; Ferrer, S; Fidock, DA; Gamo, FJ; Ghidelli-Disse, S; Hanson, KK; Henrich, PP; Jiménez-Díaz, MB; Kocken, CHM; Lafuente-Monasterio, MJ; Le Manach, C; Lee, MCS; Leroy, D; Lim, CS; Mannila, J; Marsh, KC; Martínez, MS; Morizzi, J; Paquet, T; Reader, J; Rochford, R; Ruecker, A; Sanz, LM; Sauerwein, RW; Scheurer, C; Shackleford, DM; Solapure, SM; Street, LJ; Tungtaeng, A; Vanachayangkul, P; Waterson, D; White, KL; Wittlin, S; Witty, MJ; Younis, Y; Zakutansky, SE; Zeeman, AM1
Chibale, K; Egan, TJ; Hunter, R; Joshi, MC; Ndove, J; Nsumiwa, S; Okombo, J; Taylor, D; Wiesner, L1
Achar, V; Angulo-Barturen, I; Avery, VM; Awasthy, D; Bharath, S; Coburn-Flynn, O; Duffy, S; Ferrer, S; Fidock, DA; Gamo, FJ; Hameed P, S; Hosagrahara, V; Iyer, PS; Jiménez-Díaz, MB; Kavanagh, S; Lee, MC; Martínez, MS; Menasinakai, S; Morayya, S; Nanduri, R; Narayanan, S; Panduga, V; Prabhakar, KR; Raichurkar, A; Ramachandran, S; Rautela, N; Reddy, J; Sambandamurthy, VK; Sanz, LM; Saralaya, R; Shanbhag, G; Srivastava, A; Waterson, D1
Avery, V; Bashyam, S; Bhamidipati, R; Charman, SA; Chibale, K; Douelle, F; Duffy, S; Feng, TS; González Cabrera, D; Hardick, D; Joseph, JT; Katneni, K; Le Manach, C; Mannila, J; Morizzi, J; Nchinda, AT; Shackleford, DM; Waterson, D; White, KL; Wittlin, S; Witty, MJ; Younis, Y; Zabiulla, KM1
Bashyam, S; Charman, SA; Chibale, K; Douelle, F; Feng, TS; González Cabrera, D; Joseph, JT; Kamber, J; Katneni, K; Le Manach, C; Montagnat, OD; Nchinda, AT; Ryan, E; Scheurer, C; Street, LJ; Waterson, D; White, KL; Wittlin, S; Witty, MJ; Younis, Y; Zabiulla, KM1
Deng, RX; Ding, DB; Zhang, S; Zhang, ZX1
Chen, L; Dai, ZR; Zhang, XJ; Zhang, XP; Zheng, XH1

Other Studies

7 other study(ies) available for alpha-aminopyridine and Malaria

ArticleYear
Antimalarial efficacy of MMV390048, an inhibitor of
    Science translational medicine, 2017, 04-26, Volume: 9, Issue:387

    Topics: 1-Phosphatidylinositol 4-Kinase; Aminopyridines; Animals; Antimalarials; Female; Malaria; Male; Mice; Mice, SCID; Parasitic Sensitivity Tests; Plasmodium; Sulfones

2017
4-Aminoquinoline Antimalarials Containing a Benzylmethylpyridylmethylamine Group Are Active against Drug Resistant Plasmodium falciparum and Exhibit Oral Activity in Mice.
    Journal of medicinal chemistry, 2017, 12-28, Volume: 60, Issue:24

    Topics: Administration, Oral; Aminopyridines; Aminoquinolines; Animals; Antimalarials; Cell Membrane Permeability; Chloroquine; CHO Cells; Cricetulus; Drug Evaluation, Preclinical; Drug Resistance, Microbial; ERG1 Potassium Channel; Hemeproteins; Humans; Malaria; Male; Mice, Inbred BALB C; Plasmodium berghei; Plasmodium falciparum; Solubility; Structure-Activity Relationship

2017
N-aryl-2-aminobenzimidazoles: novel, efficacious, antimalarial lead compounds.
    Journal of medicinal chemistry, 2014, Aug-14, Volume: 57, Issue:15

    Topics: Aminopyridines; Animals; Antimalarials; Benzimidazoles; Hepatocytes; Humans; Malaria; Mice, SCID; Microsomes, Liver; Plasmodium berghei; Plasmodium falciparum; Rats; Structure-Activity Relationship

2014
3,5-Diaryl-2-aminopyridines as a novel class of orally active antimalarials demonstrating single dose cure in mice and clinical candidate potential.
    Journal of medicinal chemistry, 2012, Apr-12, Volume: 55, Issue:7

    Topics: Administration, Oral; Aminopyridines; Animals; Antimalarials; Biological Availability; Cell Line; Chloroquine; Cytochrome P-450 Enzyme Inhibitors; Drug Resistance; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Female; Humans; Isoenzymes; Malaria; Mice; Microsomes, Liver; Plasmodium berghei; Plasmodium falciparum; Rabbits; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship

2012
Structure-activity relationship studies of orally active antimalarial 3,5-substituted 2-aminopyridines.
    Journal of medicinal chemistry, 2012, Dec-27, Volume: 55, Issue:24

    Topics: Administration, Oral; Aminopyridines; Animals; Antimalarials; Drug Resistance, Multiple; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Humans; Malaria; Mice; Microsomes, Liver; Plasmodium berghei; Plasmodium falciparum; Solubility; Structure-Activity Relationship

2012
[Studies on antimalarials. III. Synthesis of 2-(substituted styryl)-4-amino pyridines].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1983, Volume: 18, Issue:4

    Topics: Aminopyridines; Animals; Antimalarials; Malaria; Mice

1983
[Studies on antimalarials. I. Synthesis and antimalarial activities of some derivatives of 2,4-diamino-5-substituted amino pyrimidines and 2,4-diamino-6-methyl-5-substituted amino pyrimidines (author's transl)].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1980, Volume: 15, Issue:12

    Topics: Aminopyridines; Animals; Antimalarials; Malaria; Mice

1980