alpha-aminopyridine has been researched along with Malaria in 7 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 2 (28.57) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 5 (71.43) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Abraham, TS; Angulo-Barturen, I; Bantscheff, M; Basak, R; Birkholtz, LM; Blagborough, AM; Bodenreider, C; Botha, M; Burrows, J; Cabrera, DG; Campo, B; Charman, SA; Chibale, K; Dechering, KJ; Delves, MJ; Donini, C; Drewes, G; Ferrer, S; Fidock, DA; Gamo, FJ; Ghidelli-Disse, S; Hanson, KK; Henrich, PP; Jiménez-Díaz, MB; Kocken, CHM; Lafuente-Monasterio, MJ; Le Manach, C; Lee, MCS; Leroy, D; Lim, CS; Mannila, J; Marsh, KC; Martínez, MS; Morizzi, J; Paquet, T; Reader, J; Rochford, R; Ruecker, A; Sanz, LM; Sauerwein, RW; Scheurer, C; Shackleford, DM; Solapure, SM; Street, LJ; Tungtaeng, A; Vanachayangkul, P; Waterson, D; White, KL; Wittlin, S; Witty, MJ; Younis, Y; Zakutansky, SE; Zeeman, AM | 1 |
Chibale, K; Egan, TJ; Hunter, R; Joshi, MC; Ndove, J; Nsumiwa, S; Okombo, J; Taylor, D; Wiesner, L | 1 |
Achar, V; Angulo-Barturen, I; Avery, VM; Awasthy, D; Bharath, S; Coburn-Flynn, O; Duffy, S; Ferrer, S; Fidock, DA; Gamo, FJ; Hameed P, S; Hosagrahara, V; Iyer, PS; Jiménez-Díaz, MB; Kavanagh, S; Lee, MC; Martínez, MS; Menasinakai, S; Morayya, S; Nanduri, R; Narayanan, S; Panduga, V; Prabhakar, KR; Raichurkar, A; Ramachandran, S; Rautela, N; Reddy, J; Sambandamurthy, VK; Sanz, LM; Saralaya, R; Shanbhag, G; Srivastava, A; Waterson, D | 1 |
Avery, V; Bashyam, S; Bhamidipati, R; Charman, SA; Chibale, K; Douelle, F; Duffy, S; Feng, TS; González Cabrera, D; Hardick, D; Joseph, JT; Katneni, K; Le Manach, C; Mannila, J; Morizzi, J; Nchinda, AT; Shackleford, DM; Waterson, D; White, KL; Wittlin, S; Witty, MJ; Younis, Y; Zabiulla, KM | 1 |
Bashyam, S; Charman, SA; Chibale, K; Douelle, F; Feng, TS; González Cabrera, D; Joseph, JT; Kamber, J; Katneni, K; Le Manach, C; Montagnat, OD; Nchinda, AT; Ryan, E; Scheurer, C; Street, LJ; Waterson, D; White, KL; Wittlin, S; Witty, MJ; Younis, Y; Zabiulla, KM | 1 |
Deng, RX; Ding, DB; Zhang, S; Zhang, ZX | 1 |
Chen, L; Dai, ZR; Zhang, XJ; Zhang, XP; Zheng, XH | 1 |
7 other study(ies) available for alpha-aminopyridine and Malaria
Article | Year |
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Antimalarial efficacy of MMV390048, an inhibitor of
Topics: 1-Phosphatidylinositol 4-Kinase; Aminopyridines; Animals; Antimalarials; Female; Malaria; Male; Mice; Mice, SCID; Parasitic Sensitivity Tests; Plasmodium; Sulfones | 2017 |
4-Aminoquinoline Antimalarials Containing a Benzylmethylpyridylmethylamine Group Are Active against Drug Resistant Plasmodium falciparum and Exhibit Oral Activity in Mice.
Topics: Administration, Oral; Aminopyridines; Aminoquinolines; Animals; Antimalarials; Cell Membrane Permeability; Chloroquine; CHO Cells; Cricetulus; Drug Evaluation, Preclinical; Drug Resistance, Microbial; ERG1 Potassium Channel; Hemeproteins; Humans; Malaria; Male; Mice, Inbred BALB C; Plasmodium berghei; Plasmodium falciparum; Solubility; Structure-Activity Relationship | 2017 |
N-aryl-2-aminobenzimidazoles: novel, efficacious, antimalarial lead compounds.
Topics: Aminopyridines; Animals; Antimalarials; Benzimidazoles; Hepatocytes; Humans; Malaria; Mice, SCID; Microsomes, Liver; Plasmodium berghei; Plasmodium falciparum; Rats; Structure-Activity Relationship | 2014 |
3,5-Diaryl-2-aminopyridines as a novel class of orally active antimalarials demonstrating single dose cure in mice and clinical candidate potential.
Topics: Administration, Oral; Aminopyridines; Animals; Antimalarials; Biological Availability; Cell Line; Chloroquine; Cytochrome P-450 Enzyme Inhibitors; Drug Resistance; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Female; Humans; Isoenzymes; Malaria; Mice; Microsomes, Liver; Plasmodium berghei; Plasmodium falciparum; Rabbits; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship | 2012 |
Structure-activity relationship studies of orally active antimalarial 3,5-substituted 2-aminopyridines.
Topics: Administration, Oral; Aminopyridines; Animals; Antimalarials; Drug Resistance, Multiple; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Humans; Malaria; Mice; Microsomes, Liver; Plasmodium berghei; Plasmodium falciparum; Solubility; Structure-Activity Relationship | 2012 |
[Studies on antimalarials. III. Synthesis of 2-(substituted styryl)-4-amino pyridines].
Topics: Aminopyridines; Animals; Antimalarials; Malaria; Mice | 1983 |
[Studies on antimalarials. I. Synthesis and antimalarial activities of some derivatives of 2,4-diamino-5-substituted amino pyrimidines and 2,4-diamino-6-methyl-5-substituted amino pyrimidines (author's transl)].
Topics: Aminopyridines; Animals; Antimalarials; Malaria; Mice | 1980 |