Page last updated: 2024-08-21

acridines and Malignant Melanoma

acridines has been researched along with Malignant Melanoma in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-199010 (45.45)18.7374
1990's5 (22.73)18.2507
2000's4 (18.18)29.6817
2010's3 (13.64)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cichorek, M; Deptuła, M; Dzierzbicka, K; Gensicka-Kowalewska, M; Klejbor, I; Ronowska, A1
Gately, S; Goodall, ML; Kauffman, AL; Kortus, MG; MacKeigan, JP; Martin, KR; Trent, JM; Wang, T1
Henderson, CJ; MacLeod, AK; McLaughlin, LA; Wolf, CR1
Amodei, S; Antonelli, A; Benassi, B; Biroccio, A; D'Angelo, C; D'Incalci, M; Elli, R; Leonetti, C; Rizzo, A; Stevens, MF; Zupi, G1
Jordan, RT; Pardini, RS1
Baguley, BC; Marshall, E; Zhuang, L1
Baguley, BC; Finlay, GJ; Marshall, E; Matthews, JH; Paull, KD1
Boratyński, J; Duś, D; Kuśnierczyk, H; Paprocka, M; Radzikowski, C1
Charlton, PA; Cree, IA; Neale, MH1
Aboagye, EO; Baguley, BC; Brady, F; Brown, GD; Denny, WA; Gamage, SA; Luthra, SK; Myers, R; Osman, S; Price, PM; Rowlinson-Busza, G1
Miller, DM; Stewart, DA; Thomas, SD; Xu, X1
Kohen, C; Kohen, E; Leising, HB; Marty, A; Salmon, JM; Schachtschabel, DO; Thorell, B; Viallet, P1
Cysyk, RL; Legha, SS; Shoemaker, DD1
Benjamin, RS; Bodey, GP; Burgess, MA; Gutterman, JU; Hall, SW; Legha, SS; Valdivieso, M1
Baguley, BC; Finlay, GJ1
Kapp, A; Komann, A; Schöpf, E1
Balda, BR; Birkmayer, GD3
Balda, BR; Birkmayer, G1
Auersperg, N; Tan, P1
Atwell, GJ; Cain, BF1

Other Studies

22 other study(ies) available for acridines and Malignant Melanoma

ArticleYear
Synthesis and Biological Evaluation of Acridine/Acridone Analogs as Potential Anticancer Agents.
    Medicinal chemistry (Shariqah (United Arab Emirates)), 2019, Volume: 15, Issue:7

    Topics: Acridines; Acridones; Antineoplastic Agents; Apoptosis; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Melanoma; Molecular Structure; Structure-Activity Relationship

2019
Development of potent autophagy inhibitors that sensitize oncogenic BRAF V600E mutant melanoma tumor cells to vemurafenib.
    Autophagy, 2014, Volume: 10, Issue:6

    Topics: Acridines; Animals; Antimalarials; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Autophagy; Cell Line, Tumor; Chloroquine; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Humans; Indoles; Lysosomes; Melanoma; Mice; Mutation; Proto-Oncogene Proteins B-raf; Structure-Activity Relationship; Sulfonamides; Translational Research, Biomedical; Tumor Stem Cell Assay; Vemurafenib

2014
Activation status of the pregnane X receptor influences vemurafenib availability in humanized mouse models.
    Cancer research, 2015, Nov-01, Volume: 75, Issue:21

    Topics: Acridines; Animals; Biological Availability; Biological Transport; Cell Line, Tumor; Constitutive Androstane Receptor; Cytochrome P-450 CYP3A; Female; Indoles; Male; Melanoma; Mice; Mice, Knockout; Pregnane X Receptor; Receptors, Cytoplasmic and Nuclear; Receptors, Steroid; Sulfonamides; Tetrahydroisoquinolines; Vemurafenib

2015
Biological activity of the G-quadruplex ligand RHPS4 (3,11-difluoro-6,8,13-trimethyl-8H-quino[4,3,2-kl]acridinium methosulfate) is associated with telomere capping alteration.
    Molecular pharmacology, 2004, Volume: 66, Issue:5

    Topics: Acridines; Apoptosis; Cell Cycle; Cellular Senescence; Humans; Ligands; Melanoma; Telomere; Tumor Cells, Cultured

2004
Anti-neoplastic activity of C205: a new topical anti-cancer formulation.
    Cancer letters, 1984, Volume: 23, Issue:3

    Topics: Acridines; Administration, Topical; Animals; Antineoplastic Agents; Drug Evaluation, Preclinical; Lung Neoplasms; Melanoma; Mice; Mice, Inbred C57BL; Neoplasm Transplantation; Skin Neoplasms

1984
Experimental solid tumour activity of N-[2-(dimethylamino)ethyl]-acridine-4-carboxamide.
    Cancer chemotherapy and pharmacology, 1995, Volume: 36, Issue:3

    Topics: Acridines; Adenocarcinoma; Animals; Antineoplastic Agents; Cell Division; Cell Line; Colonic Neoplasms; Humans; Intercalating Agents; Lung Neoplasms; Melanoma; Mice; Mice, Inbred C3H; Mice, Inbred C57BL; Mice, Inbred DBA; Mice, Nude; Regression Analysis; Time Factors; Transplantation, Heterologous

1995
In vitro assessment of N-[2-(dimethylamino)ethyl]acridine-4-carboxamide, a DNA-intercalating antitumour drug with reduced sensitivity to multidrug resistance.
    Cancer chemotherapy and pharmacology, 1993, Volume: 31, Issue:5

    Topics: Acridines; Aminoacridines; Antineoplastic Agents; DNA Topoisomerases, Type I; Drug Resistance; Drug Screening Assays, Antitumor; Humans; Intercalating Agents; Leukemia; Melanoma; Tumor Cells, Cultured

1993
Conjugation of the monoclonal antibody 17-1A with the nitroacridine compound C921 with the poly-L-lysine as an intermediate agent.
    Archivum immunologiae et therapiae experimentalis, 1997, Volume: 45, Issue:4

    Topics: Acridines; Adenocarcinoma; Antibodies, Monoclonal; Antibody Specificity; Colonic Neoplasms; Flow Cytometry; Humans; Immunotoxins; Melanoma; Polylysine; Tumor Cells, Cultured

1997
Ex vivo activity of XR5000 against solid tumors.
    Anti-cancer drugs, 2000, Volume: 11, Issue:6

    Topics: Acridines; Adenosine Triphosphate; Adult; Aged; Antineoplastic Agents; DNA, Neoplasm; Dose-Response Relationship, Drug; Female; Humans; Luminescent Measurements; Male; Melanoma; Middle Aged; Ovarian Neoplasms; Skin Neoplasms; Topoisomerase I Inhibitors; Topoisomerase II Inhibitors; Tumor Cells, Cultured

2000
Comparative biodistribution and metabolism of carbon-11-labeled N-[2-(dimethylamino)ethyl]acridine-4-carboxamide and DNA-intercalating analogues.
    Cancer research, 2001, Apr-01, Volume: 61, Issue:7

    Topics: Acridines; Animals; Antineoplastic Agents; Carbon Radioisotopes; Female; Glioma; HT29 Cells; Humans; Inhibitory Concentration 50; Intercalating Agents; Isotope Labeling; Melanoma; Mice; Mice, Inbred ICR; Mice, Nude; Tissue Distribution; Tomography, Emission-Computed; Tumor Cells, Cultured; Xenograft Model Antitumor Assays

2001
Acridine-modified, clamp-forming antisense oligonucleotides synergize with cisplatin to inhibit c-Myc expression and B16-F0 tumor progression.
    Nucleic acids research, 2002, Jun-01, Volume: 30, Issue:11

    Topics: Acridines; Animals; Apoptosis; Base Sequence; Blotting, Western; Cell Division; Cisplatin; Disease Progression; Drug Synergism; Fluorescent Antibody Technique; Gene Expression Regulation, Neoplastic; Genes, myc; In Situ Nick-End Labeling; Melanoma; Mice; Mice, Inbred C57BL; Oligonucleotides, Antisense; Proliferating Cell Nuclear Antigen; Proto-Oncogene Proteins c-myc; Tumor Cells, Cultured

2002
The effect of atebrine and an acridine analog (BCMA) on the coenzyme fluorescence spectra of cultured melanoma and Ehrlich ascites (EL2) cells.
    Histochemistry, 1978, Sep-15, Volume: 57, Issue:3

    Topics: Acridines; Animals; Carcinoma, Ehrlich Tumor; Cell Division; Cell Line; DNA, Neoplasm; Melanoma; NAD; NADP; Neoplasm Proteins; Quinacrine; Spectrometry, Fluorescence

1978
Selective localization of 4'-(9-acridinylamino)-methanesulfon-m-anisidide in B 16 melanoma.
    Pharmacology, 1978, Volume: 16, Issue:4

    Topics: Acridines; Animals; Antineoplastic Agents; Chemical Phenomena; Chemistry; Drug Evaluation, Preclinical; Male; Melanoma; Mesylates; Mice; Neoplasms, Experimental; Time Factors

1978
Phase 1 clinical investigation of 4'-(9-acridinylamino)methanesulfon-m-anisidide (NSC 249992), a new acridine derivative.
    Cancer research, 1978, Volume: 38, Issue:11 Pt 1

    Topics: Acridines; Adenocarcinoma; Adult; Aged; Antineoplastic Agents; Bone Marrow; Drug Administration Schedule; Drug Evaluation; Female; Humans; Injections, Intravenous; Leukemia, Myeloid, Acute; Lung Neoplasms; Male; Melanoma; Middle Aged; Neoplasms; Phenylenediamines; Remission, Spontaneous

1978
Potentiation by phenylbisbenzimidazoles of cytotoxicity of anticancer drugs directed against topoisomerase II.
    European journal of cancer (Oxford, England : 1990), 1990, Volume: 26, Issue:5

    Topics: Acridines; Amsacrine; Animals; Antineoplastic Agents; Benzimidazoles; Bisbenzimidazole; Colonic Neoplasms; Doxorubicin; Drug Synergism; Etoposide; Fluorescent Dyes; Leukemia L1210; Lung Neoplasms; Melanoma; Mice; Topoisomerase II Inhibitors; Tumor Cells, Cultured; Tumor Stem Cell Assay

1990
Effect of tumour necrosis factor alpha in vivo on human granulocyte oxidative metabolism.
    Archives of dermatological research, 1991, Volume: 283, Issue:6

    Topics: Acridines; Amino Acid Sequence; Granulocyte-Macrophage Colony-Stimulating Factor; Humans; Luminescent Measurements; Lymphotoxin-alpha; Melanoma; Molecular Sequence Data; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Oxidation-Reduction; Recombinant Proteins; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha; Zymosan

1991
Drug effects in melanoma: tumor-specific interactions of proflavine and ethidiumbromide.
    The Yale journal of biology and medicine, 1973, Volume: 46, Issue:5

    Topics: Acridines; Animals; Antineoplastic Agents; Cell Transformation, Neoplastic; Centrifugation, Density Gradient; Coloring Agents; Cricetinae; Depression, Chemical; Diamines; DNA, Neoplasm; Ethidium; Melanoma; Neoplasm Transplantation; Neoplasms, Experimental; Oncogenic Viruses; Reverse Transcriptase Inhibitors; RNA; RNA Viruses; RNA, Neoplasm; Templates, Genetic; Tritium; Uridine

1973
[Nucleic acid and protein synthesis in hamster melanoma under the influence of drugs. I. In vivo studies of DNA synthesis in hamster melanoma].
    Naunyn-Schmiedebergs Archiv fur Pharmakologie, 1970, Volume: 266, Issue:4

    Topics: Acridines; Animals; Cell Nucleus; Cricetinae; DNA, Neoplasm; Melanoma; Mitochondria; Neoplasm Proteins; Neoplasms, Experimental; Thymidine; Tritium

1970
[Nucleic acid and protein synthesis in hamster melanoma under the action of drugs. II. In vivo studies of protein synthesis in hamster melanoma following treatment with proflavin, chloramphenicol and D-penicillamine].
    Naunyn-Schmiedebergs Archiv fur Pharmakologie, 1970, Volume: 266, Issue:4

    Topics: Acridines; Animals; Cell Nucleus; Chloramphenicol; Cricetinae; Melanoma; Mitochondria; Neoplasm Proteins; Neoplasms, Experimental; Penicillamine; Phenylalanine; Ribosomes; Stereoisomerism; Tritium

1970
Effects of the antineoplastic alkaloid acronycine on the ultrastructure and growth patterns of cultured cells.
    Cancer research, 1973, Volume: 33, Issue:10

    Topics: Acridines; Alkaloids; Animals; Antineoplastic Agents; Cell Adhesion; Cell Division; Cell Line; Cell Nucleus; Cells, Cultured; Cyclic AMP; Cytochalasin B; Female; Golgi Apparatus; Humans; Leukemia, Experimental; Leukemia, Lymphoid; Melanoma; Mice; Microscopy, Electron; Mitochondria; Mitosis; Simian virus 40; Time Factors; Tumor Virus Infections; Uterine Cervical Neoplasms

1973
The experimental antitumour properties of three congeners of the acridylmethanesulphonanilide (AMSA) series.
    European journal of cancer, 1974, Volume: 10, Issue:8

    Topics: Acridines; Animals; Anisoles; Antineoplastic Agents; Chemical Phenomena; Chemistry, Physical; Cytarabine; Dose-Response Relationship, Drug; Injections, Intradermal; Injections, Intraperitoneal; Injections, Intravenous; Injections, Subcutaneous; Leukemia L1210; Leukemia, Experimental; Mammary Neoplasms, Experimental; Melanoma; Mice; Mice, Inbred Strains; Neoplasms, Experimental; Phenylenediamines; Skin Neoplasms; Structure-Activity Relationship; Sulfones

1974
[Effects of proflavine on DNA metabolism in hamster melanoma].
    Archiv fur klinische und experimentelle Dermatologie, 1970, Volume: 239, Issue:2

    Topics: Acridines; Animals; Antimetabolites; Cell Nucleus; Cricetinae; DNA, Neoplasm; Female; Liver; Melanoma; Mitochondria; Mitochondria, Liver; Thymidine; Tritium

1970