Page last updated: 2024-08-21

acridines and Malaria

acridines has been researched along with Malaria in 40 studies

Research

Studies (40)

TimeframeStudies, this research(%)All Research%
pre-199028 (70.00)18.7374
1990's3 (7.50)18.2507
2000's3 (7.50)29.6817
2010's5 (12.50)24.3611
2020's1 (2.50)2.80

Authors

AuthorsStudies
Awasthi, SK; Sharma, B; Singh, AK; Singh, P1
Cross, RM; Kyle, DE; Lacrue, AN; Maignan, JR; Manetsch, R; Sáenz, FE; Udenze, KO1
Auparakkitanon, S; Denny, WA; Rattanajak, R; Sereekhajornjaru, N; Somboon, C; Wilairat, P1
Bhardwaj, TR; Goyal, S; Kumar, S; Patial, B; Singh, RK1
ALBERT, A; MARSHALL, PB1
SARGENT, LJ; SMALL, L2
DOBSON, J; KERMACK, WO1
SOLODOVNIKOVA, OI1
STEPHEN, JM; TONKIN, IM; WALKER, J1
MOHANTY, JK1
BHATTACHARYA, BK; NATARAHAN, S1
D'Accorso, N; Docampo, M; Fascio, M; Fernández-Calienes, A; Gille, L; Maes, L; Mendiola, J; Monzote, L; Pellón, R; Rojas, L1
Ojha, PK; Roy, K1
COATNEY, GR; COOPER, WC; EDDY, NB; GREENBERG, J1
Rathore, D1
COOPER, WC; RUHE, DS1
COATNEY, HR; COOPER, WC1
Altarelli, M; Basilico, N; Borriello, M; Brindisi, M; Butini, S; Campiani, G; Croft, S; Fattorusso, C; Fattorusso, E; Gemma, S; Kukreja, G; Nacci, V; Novellino, E; Parapini, S; Persico, M; Romano, MP; Ros, S; Savini, L; Taramelli, D; Yardley, V1
Berry, N; Biagini, GA; Bonar-Law, R; Bray, PG; Fisher, N; Meunier, B; O'Neill, PM; Owen, A; Stocks, PA; Ward, SA; Williams, DP1
Mehlhorn, H; Raether, W1
Fink, E; Raether, W2
Abdel-Rasoul, S; Königk, E; Mirtsch, S; Putfarken, B1
Chao, HT; Chookruvong, S; Hall, LA; Minigh, HL; Muth, CW1
Loiseau, PM; Nguyen, DX1
Schmidt, LH1
Fisher, FM; Jackson, PR; Kimzey, SL; Winkler, DG1
Degnan, MJ; Hung, J; Kesten, SJ; McNamara, DJ; Ortwine, DF; Uhlendorf, SE; Werbel, LM1
Fujimura, K; Fujioka, H; Fujita, M; Kato, N; Nishiyama, Y1
Fujioka, H; Furukawa, H; Kumada, N; Nishiyama, Y1
Enders, B; Hänel, H; Hofmann, J; Raether, W; Schwannecke, U; Seidenath, H; Uphoff, M1
Newman, MS1
Seitz, HM1
Shute, GT; Sodeman, TM1
Hunter, DT; Janis, B; Richards, DF2
Biel, JH; Stein, RG1
Pinder, RM1
Elslager, EF; Tendick, FH; Werbel, LM; Worth, DF1

Reviews

3 review(s) available for acridines and Malaria

ArticleYear
Advancement of chimeric hybrid drugs to cure malaria infection: An overview with special emphasis on endoperoxide pharmacophores.
    European journal of medicinal chemistry, 2021, Jul-05, Volume: 219

    Topics: Acridines; Antimalarials; Artemisinins; Drug Design; Half-Life; Humans; Malaria; Quinolines; Tetraoxanes

2021
Recent advances in novel heterocyclic scaffolds for the treatment of drug-resistant malaria.
    Journal of enzyme inhibition and medicinal chemistry, 2016, Volume: 31, Issue:2

    Topics: Acridines; Aminoquinolines; Antimalarials; Biological Products; Clinical Trials as Topic; Drug Resistance, Microbial; Ferrous Compounds; Heterocyclic Compounds; Humans; Malaria; Metallocenes; Pyridones; Pyrimidines

2016
Recent advances in the chemotherapy of malaria.
    Progress in medicinal chemistry, 1971, Volume: 8, Issue:2

    Topics: Acridines; Animals; Anti-Bacterial Agents; Antimalarials; Antineoplastic Agents; Cinchona; Culture Media; Humans; Malaria; Microbial Sensitivity Tests; Naphthoquinones; Phytotherapy; Plants, Medicinal; Plasmodium; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Proguanil; Pyrimethamine; Quinacrine; Quinolines; Sulfonamides; Sulfones

1971

Other Studies

37 other study(ies) available for acridines and Malaria

ArticleYear
4-(1H)-Quinolones and 1,2,3,4-Tetrahydroacridin-9(10H)-ones prevent the transmission of Plasmodium falciparum to Anopheles freeborni.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:12

    Topics: Acridines; Animals; Anopheles; Antimalarials; Female; Humans; Insect Vectors; Life Cycle Stages; Malaria; Malaria, Falciparum; Male; Mice; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Quinolones; Salivary Glands; Structure-Activity Relationship

2013
Comparison of hematin-targeting properties of pynacrine, an acridine analog of the benzonaphthyridine antimalarial pyronaridine.
    Acta tropica, 2014, Volume: 140

    Topics: Acridines; Antimalarials; Erythrocytes; Hemeproteins; Humans; Malaria; Naphthyridines; Plasmodium falciparum

2014
Absence of correlation between respiratory inhibition of plasmodia by acridines and antimalarial action.
    Nature, 1948, Jun-26, Volume: 161, Issue:4104

    Topics: Acridines; Antimalarials; Humans; Malaria; Nervous System Diseases; Plasmodium; Respiratory Insufficiency

1948
Attempts to find new antimalarials; studies in the acridine series; dialkylaminoalkylamines derived from 9-chloro-1,2,3,4-tetrahydroacridine.
    The Journal of organic chemistry, 1946, Volume: 11, Issue:4

    Topics: Acridines; Antimalarials; Malaria

1946
Attempts to find new antimalarials; derivatives of 3:4:2':3'-pyridoacridine and 1:2:2':3'-pyridoacridine.
    Journal of the Chemical Society, 1946

    Topics: Acridines; Antimalarials; Malaria; Phenanthrolines

1946
[Action of acridine no. 8 and acriquin on the infection of A. maculipennis sacharovi with parasites of malaria tropica].
    Meditsinskaia parazitologiia i parazitarnye bolezni, 1945, Volume: 14, Issue:1

    Topics: Acridines; Animals; Coloring Agents; Culicidae; Humans; Malaria; Parasites

1945
Antimalarial activity in tetrahydroacridones and related substances.
    Nature, 1945, Volume: 156

    Topics: Acridines; Antimalarials; Coloring Agents; Malaria

1945
Atebrine brand of amyl-acridine derivative in human malaria.
    The Antiseptic, 1945, Volume: 42

    Topics: Acridines; Malaria; Quinacrine

1945
Attempts to find new antimalarials; studies in the acridine series; 9-N-heterocyclic acridines and 9-acridylsulfanilamides.
    The Journal of organic chemistry, 1946, Volume: 11

    Topics: Acridines; Antimalarials; Coloring Agents; Malaria

1946
Chemotherapy of some acridine derivatives in fowl malaria.
    Current science, 1946, Volume: 15

    Topics: Acridines; Animals; Coloring Agents; Malaria; Malaria, Avian

1946
Antimalarial activity of new acridinone derivatives.
    Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, 2011, Volume: 65, Issue:3

    Topics: Acridines; Animals; Antimalarials; Cattle; Cell Line; Drug Resistance, Microbial; Hemeproteins; Humans; Malaria; Plasmodium falciparum; Yeasts

2011
First report on exploring structural requirements of 1,2,3,4- tetrahydroacridin-9(10H)-one analogs as antimalarials using multiple QSAR approaches: descriptor-based QSAR, CoMFA-CoMSIA 3DQSAR, HQSAR and G-QSAR approaches.
    Combinatorial chemistry & high throughput screening, 2013, Volume: 16, Issue:1

    Topics: Acridines; Antimalarials; Computer Simulation; Drug Design; Humans; Malaria; Models, Biological; Models, Molecular; Plasmodium; Quantitative Structure-Activity Relationship

2013
Survey of antimalarial agents: chemotherapy of Plasmodium gallinaceum infections; toxicity; correlation of structure and action.
    Public health monograph, 1953, Volume: 9

    Topics: Acridines; Amines; Amino Alcohols; Anti-Bacterial Agents; Antimalarials; Benzene; Benzene Derivatives; Biphenyl Compounds; Coloring Agents; Cyclohexanes; Malaria; Methane; Naphthalenes; Phenanthrenes; Plasmodium gallinaceum; Quinolines; Sulfonamides

1953
American Society of Tropical Medicine and Hygiene--55th Annual Meeting. 12-16 November 2006, Atlanta, GA, USA.
    IDrugs : the investigational drugs journal, 2007, Volume: 10, Issue:2

    Topics: Acridines; Aminoquinolines; Antigens, Protozoan; Antimalarials; Dengue Vaccines; Drug Design; Drug Industry; Humans; Hygiene; Malaria; Mefloquine; Tropical Medicine; Vaccines, Attenuated

2007
Studies in human malaria; the protective and therapeutic action of quinacrine against St. Elizabeth strain vivax malaria.
    American journal of hygiene, 1949, Volume: 49, Issue:1

    Topics: Acridines; Coloring Agents; Malaria; Malaria, Vivax; Quinacrine; Sprains and Strains

1949
Studies in human malaria; trials of quinacrine, colchicine (SN 12,080) and quinine against Chesson strain vivax malaria.
    American journal of hygiene, 1949, Volume: 50, Issue:2

    Topics: Acridines; Colchicine; Coloring Agents; Humans; Malaria; Malaria, Vivax; Quinacrine; Quinine; Sprains and Strains

1949
Design, synthesis, and structure-activity relationship studies of 4-quinolinyl- and 9-acrydinylhydrazones as potent antimalarial agents.
    Journal of medicinal chemistry, 2008, Mar-13, Volume: 51, Issue:5

    Topics: Acridines; Animals; Antimalarials; Chloroquine; Drug Design; Drug Resistance; Hemeproteins; Humans; Hydrazones; KB Cells; Malaria; Mice; Mice, Inbred BALB C; Models, Molecular; Molecular Conformation; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Quinolines; Structure-Activity Relationship

2008
Acridinediones: selective and potent inhibitors of the malaria parasite mitochondrial bc1 complex.
    Molecular pharmacology, 2008, Volume: 73, Issue:5

    Topics: Acridines; Animals; Antimalarials; Atovaquone; Cattle; Drug Synergism; Electron Transport Complex III; Heme; Hemeproteins; Humans; Malaria; Male; Membrane Potential, Mitochondrial; Mitochondria; Oxidation-Reduction; Parasitic Sensitivity Tests; Plasmodium falciparum; Rats; Rats, Wistar; Saccharomyces cerevisiae

2008
Action of a new floxacrine derivative (S 82 5455) on asexual stages of Plasmodium berghei: a light and electron microscopical study.
    Zentralblatt fur Bakteriologie, Mikrobiologie, und Hygiene. Series A, Medical microbiology, infectious diseases, virology, parasitology, 1984, Volume: 256, Issue:3

    Topics: Acridines; Animals; Antiprotozoal Agents; Blood; Chemical Phenomena; Chemistry; Female; Malaria; Male; Mice; Mice, Inbred Strains; Microscopy, Electron; Plasmodium berghei; Rats; Rats, Inbred Strains

1984
Antimalarial activity of floxacrine (HOE 991) II: Studies on causal prophylactic and blood schizontocidal action of floxacrine and related dihydroacridinediones against Plasmodium yoelii and P. berghei.
    Annals of tropical medicine and parasitology, 1982, Volume: 76, Issue:5

    Topics: Acridines; Animals; Antimalarials; Female; Malaria; Male; Mice; Mice, Inbred Strains; Plasmodium; Plasmodium berghei

1982
Plasmodium chabaudi-infection of mice: effects of chloroquine and mefloquine. Inhibition of ornithine decarboxylase activity.
    Tropenmedizin und Parasitologie, 1981, Volume: 32, Issue:2

    Topics: Acridines; Animals; Antimalarials; Carboxy-Lyases; Chloroquine; Enzyme Repression; Erythrocyte Membrane; Malaria; Mefloquine; Mice; Ornithine Decarboxylase Inhibitors; Piperidines; Plasmodium; Primaquine; Quinolines

1981
Syntheses of 9-acridine- and 2-phenanthridinemethanols as potential antimalarials.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:8

    Topics: Acridines; Animals; Antimalarials; Drug Evaluation, Preclinical; Malaria; Mice; Phenanthridines; Plasmodium berghei

1981
Plasmodium berghei mouse model: antimalarial activity of new alkaloid salts and of thiosemicarbazone and acridine derivatives.
    Tropical medicine & international health : TM & IH, 1996, Volume: 1, Issue:3

    Topics: Acridines; Alkaloids; Animals; Antimalarials; Cinchona Alkaloids; Disease Models, Animal; Female; Malaria; Mice; Mice, Inbred Strains; Plasmodium berghei; Quinine; Resorcinols; Thiosemicarbazones

1996
Antimalarial properties of floxacrine, a dihydroacridinedione derivative.
    Antimicrobial agents and chemotherapy, 1979, Volume: 16, Issue:4

    Topics: Acridines; Animals; Antimalarials; Chloroquine; Haplorhini; Macaca mulatta; Malaria; Plasmodium falciparum; Plasmodium malariae

1979
Antimalarial activity of Floxacrine (HOE 991) I. Studies on blood schizontocidal action of Floxacrine against Plasmodium berghei, P. vinckei and P. cynomolgi.
    Annals of tropical medicine and parasitology, 1979, Volume: 73, Issue:6

    Topics: 4-Aminobenzoic Acid; Acridines; Animals; Antimalarials; Blood; Cricetinae; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Resistance, Microbial; Drug Tolerance; Female; Folic Acid; Haplorhini; Macaca mulatta; Malaria; Male; Mesocricetus; Mice; Plasmodium; Plasmodium berghei; Rats

1979
Cytofluorograf detection of Plasmodium yoelii, Trypanosoma gambiense, and Trypanosoma equiperdum by laser excited fluorescence of stained rodent blood.
    The Journal of parasitology, 1977, Volume: 63, Issue:4

    Topics: Acridines; Animals; Blood; Ethidium; Fluorescent Dyes; Lasers; Malaria; Male; Mice; Plasmodium; Trypanosoma; Trypanosoma brucei gambiense; Trypanosomiasis

1977
Synthesis and antimalarial properties of 1-imino derivatives of 7-chloro-3-substituted-3,4-dihydro-1,9(2H,10H)-acridinediones and related structures.
    Journal of medicinal chemistry, 1992, Sep-18, Volume: 35, Issue:19

    Topics: Acridines; Animals; Antimalarials; Haplorhini; Malaria; Mice; Plasmodium berghei; Structure-Activity Relationship

1992
Activities of new acridone alkaloid derivatives against Plasmodium yoelii in vitro.
    Arzneimittel-Forschung, 1990, Volume: 40, Issue:9

    Topics: Acridines; Acridones; Alkaloids; Animals; Antimalarials; Cell Survival; Chloroquine; Erythrocytes; In Vitro Techniques; Leukemia L1210; Malaria; Male; Mice; Mice, Inbred ICR; Plasmodium yoelii; Pyrimethamine; Structure-Activity Relationship; Tumor Cells, Cultured

1990
In vitro and in vivo activities of atalaphillinine and related acridone alkaloids against rodent malaria.
    Antimicrobial agents and chemotherapy, 1989, Volume: 33, Issue:1

    Topics: Acridines; Alkaloids; Animals; Antimalarials; Drug Evaluation, Preclinical; Malaria; Male; Mice; Mice, Inbred ICR; Plasmodium; Plasmodium berghei; Plasmodium yoelii

1989
Antimalarial activity of new floxacrine-related acridinedione derivatives: studies on blood schizontocidal action of potential candidates against P. berghei in mice and P. falciparum in vivo and in vitro.
    Parasitology research, 1989, Volume: 75, Issue:8

    Topics: Acridines; Animals; Antimalarials; Cebidae; Chloroquine; Drug Resistance; Female; Malaria; Male; Mice; Microbial Sensitivity Tests; Molecular Structure; Plasmodium berghei; Plasmodium falciparum; Saimiri

1989
Concerning steric effects in antimalarial agents.
    Drug design and delivery, 1987, Volume: 1, Issue:4

    Topics: Acridines; Animals; Antimalarials; Chemical Phenomena; Chemistry; Drug Tolerance; Female; Magnetic Resonance Spectroscopy; Malaria; Male; Mice; Plasmodium berghei; Quinacrine

1987
[Comparative studies on acridine orange and Wright's stain in the diagnosis of malaria].
    Zeitschrift fur Tropenmedizin und Parasitologie, 1971, Volume: 22, Issue:2

    Topics: Acridines; Adolescent; Black People; Child; Child, Preschool; Fluorescent Dyes; Humans; Infant; Malaria; Methods; Microscopy, Fluorescence; Nigeria; Staining and Labeling

1971
Identification of malaria parasites by fluorescence microscopy and acridine orange staining.
    Bulletin of the World Health Organization, 1973, Volume: 48, Issue:5

    Topics: Acridines; Bacteriological Techniques; Blood; Humans; Malaria; Microscopy, Fluorescence; Philippines; Plasmodium falciparum; Plasmodium vivax; Staining and Labeling

1973
Detection of plasmodia by acridine orange stain.
    Technical bulletin of the Registry of Medical Technologists. American Society of Clinical Pathologists. Registry of Medical Technologists, 1969, Volume: 39, Issue:1

    Topics: Acridines; Humans; Malaria; Methods; Microscopy, Fluorescence; Plasmodium; Plasmodium falciparum; Plasmodium vivax; Staining and Labeling

1969
Antimalarials. Some 9-substituted amino-6-chloro-2-methoxyacridines.
    Journal of medicinal chemistry, 1973, Volume: 16, Issue:1

    Topics: Acridines; Amines; Animals; Antimalarials; Dose-Response Relationship, Drug; Malaria; Mice; Plasmodium berghei; Structure-Activity Relationship

1973
A new method for detecting Plasmodia.
    Military medicine, 1971, Volume: 136, Issue:1

    Topics: Acridines; Adult; Fluorescence; Humans; Malaria; Male; Methods; Plasmodium

1971
Antimalarial and antischistosomal effects of proximal hydrazine and hydroxylamine analogs of chloroquine and quinacrine.
    Journal of medicinal chemistry, 1969, Volume: 12, Issue:6

    Topics: Acridines; Animals; Chemical Phenomena; Chemistry; Hydrazines; Hydroxylamines; Malaria; Mice; Plasmodium; Quinine; Quinolines; Schistosomiasis

1969