Page last updated: 2024-08-21

acridines and Cancer of Prostate

acridines has been researched along with Cancer of Prostate in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19901 (6.67)18.7374
1990's4 (26.67)18.2507
2000's5 (33.33)29.6817
2010's4 (26.67)24.3611
2020's1 (6.67)2.80

Authors

AuthorsStudies
Augustin, E; Bujak, P; Kasprzak, A; Kowalczyk, A; Kowalik, P; Nowicka, AM; Paluszkiewicz, E; Pilch, J1
Chao, SW; Guh, JH; Hsu, JL; Huang, WJ; Li, TK; Liu, SP; Pan, SL; Yang, YC; Yu, CC1
Ho, HY; Su, TL; Wu, YC; Yen, WY; Yih, LH1
Bolger, GB; De Souza, PL; Fujimori, M; Khoo, KS; Lim, R; North, S; Phillips, J; Spiridonidis, H1
Corcoran, C; Devery, A; Dowling, C; Fan, Y; Fitzpatrick, JM; Gallagher, WM; Mulrane, L; O'Connor, D; O'Connor, R; O'Driscoll, L; O'Neill, AJ; Prencipe, M; Rani, S; Watson, RW1
Dzierzbicka, K; Kołodziejczyk, AM1
Bailly, C; Chackal, S; Facompré, M; Goossens, JF; Hénichart, JP; Houssin, R; Pommery, N1
Chackal, S; Henichart, JP; Houssin, R; Pommery, N1
Incles, CM; Kelland, LR; Kempski, H; Koehler, H; Neidle, S; Schultes, CM1
Amantini, C; Antonini, I; Lucciarini, R; Magnano, A; Santoni, G; Sparapani, S1
Gambertoglio, JG; Jayewardene, AL; Santoro, JE1
Ashizawa, T; Gomi, K; Okabe, M; Shimizu, M1
Fippin, LJ; Small, EJ; Whisenant, SP1
Adelstein, SJ; Fayad, F; Kassis, AI; Kinsey, BM; Venkateshan, CN1
Nilsson, S; Trulson, A; Venge, P1

Trials

3 trial(s) available for acridines and Cancer of Prostate

ArticleYear
A phase II trial of weekly i.v. KW-2170 in advanced castrate-resistant prostate cancer.
    Asia-Pacific journal of clinical oncology, 2010, Volume: 6, Issue:4

    Topics: Acridines; Adenocarcinoma; Adult; Aged; Antineoplastic Agents; Castration; Follow-Up Studies; Humans; Male; Middle Aged; Neoplasms, Hormone-Dependent; Prostatic Neoplasms; Pyrazoles; Quality of Life; Survival Rate; Treatment Outcome

2010
High-performance liquid chromatographic determination of pyrazoloacridine, a nitro-9-methoxyacridine anticancer agent, in human plasma.
    Journal of chromatography. B, Biomedical sciences and applications, 1997, Nov-21, Volume: 702, Issue:1-2

    Topics: Acridines; Antineoplastic Agents; Chromatography, High Pressure Liquid; Circadian Rhythm; Drug Stability; Freezing; Humans; Infusions, Intravenous; Male; Osmolar Concentration; Prostatic Neoplasms; Pyrazoles; Reproducibility of Results; Sensitivity and Specificity; Temperature; Time Factors

1997
Pyrazoloacridine for the treatment of hormone-refractory prostate cancer.
    Cancer investigation, 1998, Volume: 16, Issue:7

    Topics: Acridines; Aged; Antineoplastic Agents; Drug Administration Schedule; Drug Resistance, Neoplasm; Humans; Male; Middle Aged; Prostate-Specific Antigen; Prostatic Neoplasms; Pyrazoles; Survival Analysis

1998

Other Studies

12 other study(ies) available for acridines and Cancer of Prostate

ArticleYear
Foliate-Targeting Quantum Dots-
    International journal of molecular sciences, 2022, Jan-23, Volume: 23, Issue:3

    Topics: Acridines; Antineoplastic Agents; beta-Cyclodextrins; Cell Line, Tumor; Drug Carriers; Drug Delivery Systems; Folic Acid; Humans; Lung; Lung Neoplasms; Male; Nanoconjugates; Nanostructures; Prostate; Prostatic Neoplasms; Quantum Dots

2022
A novel small molecule hybrid of vorinostat and DACA displays anticancer activity against human hormone-refractory metastatic prostate cancer through dual inhibition of histone deacetylase and topoisomerase I.
    Biochemical pharmacology, 2014, Aug-01, Volume: 90, Issue:3

    Topics: Acridines; Animals; Antineoplastic Agents; Cell Cycle; Cell Line, Tumor; Cells, Cultured; DNA Damage; DNA Repair; DNA Topoisomerases, Type I; Drug Resistance, Neoplasm; Drugs, Investigational; Histone Deacetylase 6; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; Hydroxamic Acids; Male; Mice, Nude; Neoplasm Proteins; Prostate; Prostatic Neoplasms; Topoisomerase I Inhibitors; Topoisomerase II Inhibitors; Tumor Burden; Vorinostat; Xenograft Model Antitumor Assays

2014
Glyfoline induces mitotic catastrophe and apoptosis in cancer cells.
    International journal of cancer, 2010, Feb-15, Volume: 126, Issue:4

    Topics: Acridines; Adenocarcinoma; Animals; Antineoplastic Agents; Apoptosis; Cell Division; Cell Line, Tumor; Female; HeLa Cells; Humans; Lung Neoplasms; Male; Mice; Microtubules; Mitosis; Neoplasms; Prostatic Neoplasms; Tubulin

2010
Characterisation and manipulation of docetaxel resistant prostate cancer cell lines.
    Molecular cancer, 2011, Oct-07, Volume: 10

    Topics: Acridines; Antineoplastic Agents; Apoptosis; Apoptosis Regulatory Proteins; ATP Binding Cassette Transporter, Subfamily B, Member 1; beta-Galactosidase; Cell Line, Tumor; Cell Survival; Cellular Senescence; Docetaxel; Drug Resistance, Neoplasm; Gene Expression; Gene Expression Profiling; Genes, Reporter; Humans; Luciferases, Renilla; Male; Molecular Targeted Therapy; NF-kappa B; Nitriles; Prostatic Neoplasms; Sulfones; Taxoids; Tetrahydroisoquinolines

2011
Synthesis and antitumor activity of conjugates of muramyldipeptide or normuramyldipeptide with hydroxyacridine/acridone derivatives.
    Journal of medicinal chemistry, 2003, Jan-02, Volume: 46, Issue:1

    Topics: Acetylmuramyl-Alanyl-Isoglutamine; Acridines; Acridones; Animals; Antineoplastic Agents; Drug Screening Assays, Antitumor; Humans; Lymphoma, AIDS-Related; Male; Mice; Mice, Nude; Neoplasm Transplantation; Prostatic Neoplasms; Structure-Activity Relationship; Tumor Cells, Cultured

2003
Highly cytotoxic benzo[c]pyrido[2,3,4-kl]acridines.
    Bioorganic & medicinal chemistry letters, 2003, Mar-10, Volume: 13, Issue:5

    Topics: Acridines; Animals; Antineoplastic Agents; Cattle; DNA; DNA Topoisomerases; Drug Screening Assays, Antitumor; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Male; Nucleic Acid Conformation; Nucleic Acid Denaturation; Prostatic Neoplasms; Topoisomerase Inhibitors; Tumor Cells, Cultured

2003
Design, synthesis and pharmacological evaluation of new anticancer fused pentacycles.
    Journal of enzyme inhibition and medicinal chemistry, 2003, Volume: 18, Issue:2

    Topics: Acridines; Antineoplastic Agents; Cell Division; Cell Survival; Drug Design; Drug Screening Assays, Antitumor; Humans; Inhibitory Concentration 50; Male; Molecular Structure; Prostatic Neoplasms; Pyridines; Structure-Activity Relationship; Tumor Cells, Cultured

2003
A G-quadruplex telomere targeting agent produces p16-associated senescence and chromosomal fusions in human prostate cancer cells.
    Molecular cancer therapeutics, 2004, Volume: 3, Issue:10

    Topics: 3T3 Cells; Acridines; Animals; Blotting, Western; Catalysis; Cell Line, Tumor; Cell Proliferation; Cellular Senescence; Chromosomes; Cyclin-Dependent Kinase Inhibitor p16; DNA; G-Quadruplexes; Humans; Ligands; Male; Metaphase; Mice; Models, Chemical; Nucleic Acid Conformation; Prostatic Neoplasms; Rhodamines; Telomerase; Telomere; Time Factors; Up-Regulation

2004
Synthesis and biological evaluation of new asymmetrical bisintercalators as potential antitumor drugs.
    Journal of medicinal chemistry, 2006, Nov-30, Volume: 49, Issue:24

    Topics: Acridines; Antineoplastic Agents; Binding, Competitive; Cell Line, Tumor; DNA; Drug Screening Assays, Antitumor; Heterocyclic Compounds, 4 or More Rings; Humans; Intercalating Agents; Male; Prostatic Neoplasms; Solubility; Structure-Activity Relationship

2006
Antitumor activity of KW-2170, a novel pyrazoloacridone derivative.
    Anti-cancer drugs, 1998, Volume: 9, Issue:3

    Topics: Acridines; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Breast Neoplasms; Doxorubicin; Drug Resistance, Multiple; Female; Fibrosarcoma; Gastrointestinal Neoplasms; Humans; Liver Neoplasms; Lung Neoplasms; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Nude; Molecular Structure; Neoplasms; Prostatic Neoplasms; Pyrazoles; Sarcoma 180; Transplantation, Heterologous; Tumor Cells, Cultured

1998
Synthesis and biological activity of the intercalating agent 3-acetamido-5-[123/125I]iodo-6-aminoacridine.
    International journal of radiation applications and instrumentation. Part B, Nuclear medicine and biology, 1990, Volume: 17, Issue:3

    Topics: Acridines; DNA; Humans; In Vitro Techniques; Intercalating Agents; Iodine Radioisotopes; Isotope Labeling; Male; Proflavine; Prostatic Neoplasms

1990
Lucigenin-enhanced chemiluminescence in blood is increased in cancer.
    American journal of clinical pathology, 1989, Volume: 91, Issue:4

    Topics: Acridines; Adult; Aged; Aged, 80 and over; Cell Separation; Female; Humans; Kidney Neoplasms; Leukocyte Count; Luminescent Measurements; Luminol; Male; Middle Aged; Monocytes; Neoplasms; Neutrophils; Prostatic Neoplasms

1989