Page last updated: 2024-08-23

acarbose and Diabetes Mellitus, Type 2

acarbose has been researched along with Diabetes Mellitus, Type 2 in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (6.67)29.6817
2010's11 (73.33)24.3611
2020's3 (20.00)2.80

Authors

AuthorsStudies
Ashraf, M; Bajda, M; Hussain, S; Khan, IU; Mustafa, G; Mutahir, S; Rehman, TU; Riaz, S; Shaukat, A; Yar, M1
Al-Rashida, M; Ashraf, M; Asif, N; Chaudhry, F; Huma, R; Khan, MA; Munawar, MA; Naureen, S; Shaukat, A1
Chigurupati, S; Imran, S; Irshad, M; Ismail, NH; Khan, KM; Nawaz, F; Rahim, F; Selvaraj, M; Taha, M1
Ananthakrishnan, R; Jayamurthy, P; Krishnan, SL; Madhukrishnan, M; Manojkumar, TK; Neethu, S; Prabha, B; Radhakrishnan, KV; Rameshkumar, KB; Sherin, DR1
Adib, M; Bijanzadeh, HR; Faramarzi, MA; Imanparast, S; Jahani, M; Larijani, B; Mahdavi, M; Mahernia, S; Mohammadi-Khanaposhtani, M; Peytam, F; Rahmanian-Jazi, M1
Agarwal, R; Luthra, T; Naga Lalitha, K; Sen, S; Uma, A1
Athrey, G; Jayaprakasha, GK; Patil, BS; Perera, WH; Perez, JL; Shivanagoudra, SR; Sun, Y; Wu, CS1
Athipornchai, A; Chaidam, S; Saeeng, R; Saehlim, N; Sirion, U1
Babkov, DA; Bezsonova, EN; Dubar, M; Klochkov, VG; Lozinskaya, NA; Melekhina, DD; Spasov, AA; Temnov, VV; Zaryanova, EV1
Bnouham, M; Cherfi, M; Daoudi, NE; Harit, T; Malek, F; Oulous, A1
Washburn, WN1
Brindis, F; Bye, R; González-Andrade, M; Mata, R; Rodríguez, R1
Adachi, I; Imahori, T; Kato, A; Murakami, K; Nakagawa, S; Natori, Y; Takahata, H; Yoshimura, Y1
Dhumaskar, KL; Ghadi, SC; Meena, SN; Tilve, SG1
Ahmed, M; Alam, U; Ashraf, M; Bajda, M; Khan, AF; Khan, IU; Shahzad, SA; Shahzadi, L; Yar, M1

Reviews

1 review(s) available for acarbose and Diabetes Mellitus, Type 2

ArticleYear
Development of the renal glucose reabsorption inhibitors: a new mechanism for the pharmacotherapy of diabetes mellitus type 2.
    Journal of medicinal chemistry, 2009, Apr-09, Volume: 52, Issue:7

    Topics: Animals; Clinical Trials as Topic; Diabetes Mellitus, Type 2; Drug Evaluation, Preclinical; Glucose; Glucosides; Humans; Hypoglycemic Agents; Kidney; Sodium-Glucose Transporter 2 Inhibitors

2009

Other Studies

14 other study(ies) available for acarbose and Diabetes Mellitus, Type 2

ArticleYear
Pyridine sulfonamide as a small key organic molecule for the potential treatment of type-II diabetes mellitus and Alzheimer's disease: In vitro studies against yeast α-glucosidase, acetylcholinesterase and butyrylcholinesterase.
    Bioorganic chemistry, 2015, Volume: 63

    Topics: Acetylcholinesterase; alpha-Glucosidases; Alzheimer Disease; Butyrylcholinesterase; Cholinesterase Inhibitors; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Glycoside Hydrolase Inhibitors; Humans; Hypoglycemic Agents; Molecular Docking Simulation; Molecular Structure; Pyridines; Saccharomyces cerevisiae; Structure-Activity Relationship; Sulfonamides

2015
In search of new α-glucosidase inhibitors: Imidazolylpyrazole derivatives.
    Bioorganic chemistry, 2017, Volume: 71

    Topics: alpha-Glucosidases; Diabetes Mellitus, Type 2; Glycoside Hydrolase Inhibitors; Humans; Molecular Docking Simulation; Pyrazoles; Saccharomyces cerevisiae; Structure-Activity Relationship

2017
Synthesis of piperazine sulfonamide analogs as diabetic-II inhibitors and their molecular docking study.
    European journal of medicinal chemistry, 2017, Dec-01, Volume: 141

    Topics: alpha-Amylases; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; Hypoglycemic Agents; Molecular Docking Simulation; Molecular Structure; Piperazine; Piperazines; Structure-Activity Relationship; Sulfonamides

2017
Antidiabetic potential of phytochemicals isolated from the stem bark of Myristica fatua Houtt. var. magnifica (Bedd.) Sinclair.
    Bioorganic & medicinal chemistry, 2018, 07-23, Volume: 26, Issue:12

    Topics: alpha-Glucosidases; Binding Sites; Cell Line; Cell Survival; Diabetes Mellitus, Type 2; Glycoside Hydrolase Inhibitors; Humans; Hypoglycemic Agents; Molecular Dynamics Simulation; Muscle Cells; Myristicaceae; Phytochemicals; Plant Bark; Plant Extracts; Plant Stems; Protein Structure, Tertiary; Resorcinols

2018
New 6-amino-pyrido[2,3-d]pyrimidine-2,4-diones as novel agents to treat type 2 diabetes: A simple and efficient synthesis, α-glucosidase inhibition, molecular modeling and kinetic study.
    European journal of medicinal chemistry, 2018, Jul-15, Volume: 155

    Topics: alpha-Glucosidases; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Glycoside Hydrolase Inhibitors; Humans; Hypoglycemic Agents; Kinetics; Models, Molecular; Molecular Structure; Pyridines; Pyrimidines; Structure-Activity Relationship

2018
Design, synthesis and in vitro study of densely functionalized oxindoles as potent α-glucosidase inhibitors.
    Bioorganic & medicinal chemistry, 2018, 10-01, Volume: 26, Issue:18

    Topics: alpha-Glucosidases; Diabetes Mellitus, Type 2; Drug Design; Glycoside Hydrolase Inhibitors; Humans; Inhibitory Concentration 50; Kinetics; Molecular Docking Simulation; Oxindoles; Structure-Activity Relationship; Yeasts

2018
In vitro and in silico elucidation of antidiabetic and anti-inflammatory activities of bioactive compounds from Momordica charantia L.
    Bioorganic & medicinal chemistry, 2019, 07-15, Volume: 27, Issue:14

    Topics: Anti-Inflammatory Agents; Computer Simulation; Diabetes Mellitus, Type 2; Hypoglycemic Agents; Inflammation; Momordica charantia

2019
Synthesis and biological evaluation of 1,6-bis-triazole-2,3,4-tri-O-benzyl-α-d-glucopyranosides as a novel α-glucosidase inhibitor in the treatment of Type 2 diabetes.
    Bioorganic & medicinal chemistry letters, 2021, 10-15, Volume: 50

    Topics: alpha-Glucosidases; Diabetes Mellitus, Type 2; Glucans; Glycoside Hydrolase Inhibitors; Humans; Hypoglycemic Agents; Models, Molecular; Molecular Docking Simulation; Molecular Structure; Protein Binding; Protein Conformation

2021
Towards multi-target antidiabetic agents: In vitro and in vivo evaluation of 3,5-disubstituted indolin-2-one derivatives as novel α-glucosidase inhibitors.
    Bioorganic & medicinal chemistry letters, 2022, 01-01, Volume: 55

    Topics: alpha-Glucosidases; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Glycoside Hydrolase Inhibitors; Humans; Hypoglycemic Agents; Indoles; Models, Molecular; Molecular Structure; Structure-Activity Relationship

2022
New pyrazole-tetrazole hybrid compounds as potent α-amylase and non-enzymatic glycation inhibitors.
    Bioorganic & medicinal chemistry letters, 2022, 08-01, Volume: 69

    Topics: alpha-Amylases; Diabetes Mellitus, Type 2; Humans; Pyrazoles; Pyridines; Tetrazoles

2022
(Z)-3-butylidenephthalide from Ligusticum porteri , an α-glucosidase inhibitor.
    Journal of natural products, 2011, Mar-25, Volume: 74, Issue:3

    Topics: Acarbose; Administration, Oral; Animals; Blood Glucose; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 2; Glycoside Hydrolase Inhibitors; Hypoglycemic Agents; Insulin; Insulin Secretion; Ligusticum; Medicine, Traditional; Mexico; Mice; Phthalic Anhydrides; Stereoisomerism; Streptozocin

2011
The synthesis and biological evaluation of 1-C-alkyl-L-arabinoiminofuranoses, a novel class of α-glucosidase inhibitors.
    Bioorganic & medicinal chemistry letters, 2011, Jan-15, Volume: 21, Issue:2

    Topics: alpha-Glucosidases; Animals; Diabetes Mellitus, Type 2; Enzyme Inhibitors; Glycoside Hydrolase Inhibitors; Humans; Hypoglycemic Agents; Imino Furanoses; Rats

2011
Graphite catalyzed solvent free synthesis of dihydropyrimidin-2(1H)-ones/thiones and their antidiabetic activity.
    Bioorganic & medicinal chemistry letters, 2014, Jul-01, Volume: 24, Issue:13

    Topics: alpha-Amylases; Catalysis; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Enzyme Inhibitors; Graphite; Humans; Hypoglycemic Agents; Molecular Structure; Pyrimidines; Structure-Activity Relationship; Thiones

2014
Novel synthesis of dihydropyrimidines for α-glucosidase inhibition to treat type 2 diabetes: in vitro biological evaluation and in silico docking.
    Bioorganic chemistry, 2014, Volume: 54

    Topics: alpha-Glucosidases; Amino Acid Sequence; Crystallography, X-Ray; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Glycoside Hydrolase Inhibitors; Molecular Docking Simulation; Molecular Sequence Data; Molecular Structure; Pyrimidines; Saccharomyces cerevisiae; Sequence Alignment; Structure-Activity Relationship

2014