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7-chloro-4-aminoquinoline and Malaria, Falciparum

7-chloro-4-aminoquinoline has been researched along with Malaria, Falciparum in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's4 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chibale, K; Egan, TJ; Kuter, D; Nsumiwa, S; Wittlin, S1
Miller, ME; Nelson, SW; Parrott, EE; Singh, R1
Agarwal, P; Ahmad, H; Dola, VR; Dwivedi, AK; Haq, W; Katti, SB; Puri, SK; Raju, KS; Rashid, M; Soni, A; Srivastava, K; Wahajuddin, M1
Barteselli, A; Basilico, N; Casagrande, M; Parapini, S; Sparatore, A; Taramelli, D1

Other Studies

4 other study(ies) available for 7-chloro-4-aminoquinoline and Malaria, Falciparum

ArticleYear
Structure-activity relationships for ferriprotoporphyrin IX association and β-hematin inhibition by 4-aminoquinolines using experimental and ab initio methods.
    Bioorganic & medicinal chemistry, 2013, Jul-01, Volume: 21, Issue:13

    Topics: Aminoquinolines; Antimalarials; Hemeproteins; Hemin; Humans; Malaria, Falciparum; Models, Molecular; Plasmodium falciparum; Structure-Activity Relationship

2013
A High-Throughput Assay to Identify Inhibitors of the Apicoplast DNA Polymerase from Plasmodium falciparum.
    Journal of biomolecular screening, 2014, Volume: 19, Issue:6

    Topics: Antimalarials; Apicoplasts; Chloroplasts; DNA; DNA-Directed DNA Polymerase; Drug Discovery; Exonucleases; Humans; Kinetics; Malaria, Falciparum; Mitochondria; Multienzyme Complexes; Nucleic Acid Synthesis Inhibitors; Peptide Library; Plasmodium falciparum; Protozoan Proteins; Spectrometry, Fluorescence

2014
Synthesis and Evaluation of Chirally Defined Side Chain Variants of 7-Chloro-4-Aminoquinoline To Overcome Drug Resistance in Malaria Chemotherapy.
    Antimicrobial agents and chemotherapy, 2017, Volume: 61, Issue:3

    Topics: Administration, Oral; Aminoquinolines; Animals; Antimalarials; Chlorocebus aethiops; Chloroquine; Drug Resistance; Erythrocytes; Heme; Hemin; Inhibitory Concentration 50; Macaca mulatta; Malaria; Malaria, Falciparum; Parasitic Sensitivity Tests; Plasmodium cynomolgi; Plasmodium falciparum; Plasmodium yoelii; Structure-Activity Relationship; Vero Cells

2017
Synthesis and antiplasmodial activity of new heteroaryl derivatives of 7-chloro-4-aminoquinoline.
    Bioorganic & medicinal chemistry, 2012, Oct-01, Volume: 20, Issue:19

    Topics: Aminoquinolines; Antimalarials; Cell Line; Cell Survival; Humans; Malaria, Falciparum; Plasmodium falciparum

2012