3,5-bis(trifluoromethyl)benzyl n-acetyltryptophan has been researched along with Muscle Contraction in 9 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 7 (77.78) | 29.6817 |
2010's | 2 (22.22) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Davis, P; Hruby, VJ; Lai, J; Ma, SW; Moye, S; Nair, P; Navratilova, E; Porreca, F; Tumati, S; Vanderah, TW; Yamamoto, T; Yamamura, HI | 1 |
Davis, P; Hruby, VJ; Lai, J; Largent-Milnes, T; Ma, SW; Moye, S; Nair, P; Navratilova, E; Porreca, F; Tumati, S; Vagner, J; Vanderah, TW; Yamamoto, T; Yamamura, HI | 1 |
Davis, P; Hruby, VJ; Jacobsen, NE; Kulkarni, V; Lai, J; Ma, SW; Nair, P; Navratilova, E; Porreca, F; Vagner, J; Vanderah, TW; Yamamoto, T; Yamamura, HI | 1 |
Hayashi, H; Nishimoto, S; Oh-ishi, T; Onaga, T; Shimoda, T | 1 |
Hayashi, H; Oh-ishi, T; Onaga, T; Shimoda, T | 1 |
El-Mahmoudy, A; Khalifa, M; Matsuyama, H; Shimizu, Y; Takewaki, T | 1 |
Hiyama, Y; Ishimura, M; Kataoka, S; Maeda, T; Suda, M | 1 |
Boudaka, A; Kobayashi, H; Neuhuber, WL; Shiina, T; Shimizu, Y; Takewaki, T; Wörl, J | 1 |
Arreola, JL; Chávez, J; Flores-Soto, E; Montaño, LM; Segura, P; Vargas, MH | 1 |
9 other study(ies) available for 3,5-bis(trifluoromethyl)benzyl n-acetyltryptophan and Muscle Contraction
Article | Year |
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Design, synthesis, and biological evaluation of novel bifunctional C-terminal-modified peptides for delta/mu opioid receptor agonists and neurokinin-1 receptor antagonists.
Topics: Analgesics; Animals; Cell Line; Drug Design; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Ligands; Male; Mice; Mice, Inbred ICR; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Oligopeptides; Radioligand Assay; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu; Structure-Activity Relationship; Vas Deferens | 2007 |
A structure-activity relationship study and combinatorial synthetic approach of C-terminal modified bifunctional peptides that are delta/mu opioid receptor agonists and neurokinin 1 receptor antagonists.
Topics: Animals; Cell Line; Cell Line, Tumor; Combinatorial Chemistry Techniques; Cricetinae; Cricetulus; Electric Stimulation; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Oligopeptides; Radioligand Assay; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu; Structure-Activity Relationship; Vas Deferens | 2008 |
Improving metabolic stability by glycosylation: bifunctional peptide derivatives that are opioid receptor agonists and neurokinin 1 receptor antagonists.
Topics: Analgesics; Animals; Cell Line; Cell Membrane; Cricetinae; Cricetulus; Glycosylation; Guinea Pigs; Hydrogen Bonding; Ileum; Ligands; Magnetic Resonance Spectroscopy; Male; Mice; Models, Molecular; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Oligopeptides; Protein Structure, Secondary; Radioligand Assay; Rats; Receptors, Neurokinin-1; Receptors, Opioid, delta; Receptors, Opioid, mu; Structure-Activity Relationship; Vas Deferens | 2009 |
Role of tachykinin and neurokinin receptors in the regulation of ovine omasal contractions.
Topics: Animals; Atropine; Electric Stimulation; Gene Expression; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Omasum; Organ Specificity; Piperidines; Protein Precursors; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Sheep; Tachykinins; Tryptophan | 2012 |
Role of tachykinins and neurokinin receptor subtypes in the regulation of motility of the forestomach and abomasum in conscious sheep.
Topics: Abomasum; Animals; Benzamides; Gastrointestinal Motility; Injections, Intravenous; Kinetics; Male; Muscle Contraction; Neurokinin A; Omasum; Piperidines; Receptors, Neurokinin-2; Rumen; Sheep; Substance P; Tachykinins; Tryptophan | 2013 |
Tachykinins mediate non-adrenergic, non-cholinergic excitatory neurotransmission to the hamster ileum via NK1 and NK2 receptors.
Topics: Animals; Autonomic Agents; Benzamides; Cricetinae; Dose-Response Relationship, Drug; Electric Stimulation; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neuromuscular Junction; NG-Nitroarginine Methyl Ester; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Synaptic Transmission; Tryptophan | 2003 |
Effects of KP-496, a novel dual antagonist for leukotriene D4 and thromboxane A2 receptors, on contractions induced by various agonists in the guinea pig trachea.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetates; Acetylcholine; Albuterol; Animals; Atropine; Benzoquinones; Carbachol; Chromones; Cyclopropanes; Dinoprost; Drug Evaluation, Preclinical; Guinea Pigs; Heptanoic Acids; Histamine; In Vitro Techniques; Indoles; Indomethacin; Ketanserin; Ketotifen; Leukotriene Antagonists; Leukotriene D4; Male; Muscle Contraction; Muscle, Smooth; Phenylcarbamates; Powders; Procaterol; Prostaglandin Antagonists; Prostaglandin D2; Quinolines; Receptors, Thromboxane A2, Prostaglandin H2; Serotonin; Substance P; Sulfides; Sulfonamides; Tosyl Compounds; Trachea; Tryptophan | 2006 |
Involvement of TRPV1-dependent and -independent components in the regulation of vagally induced contractions in the mouse esophagus.
Topics: Alkaloids; Anilides; Animals; Benzodioxoles; Capsaicin; Cinnamates; Cricetinae; Enzyme Inhibitors; Esophagus; Female; Male; Mesocricetus; Mice; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptors, Tachykinin; Species Specificity; TRPV Cation Channels; Tryptophan; Vagus Nerve | 2007 |
Paradoxical effect of salbutamol in a model of acute organophosphates intoxication in guinea pigs: role of substance P release.
Topics: Albuterol; Animals; Calcium; Cholinesterase Inhibitors; Colforsin; Diamines; Guinea Pigs; Lung; Male; Muscle Contraction; omega-Conotoxins; Parathion; Physostigmine; Pirenzepine; Plethysmography, Whole Body; Substance P; Tetrodotoxin; Tryptophan | 2007 |