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1h-imidazo(4,5-b)pyridine and Malaria

1h-imidazo(4,5-b)pyridine has been researched along with Malaria in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (60.00)24.3611
2020's2 (40.00)2.80

Authors

AuthorsStudies
Ansell, KH; Baker, DA; Birchall, K; Bouloc, NS; Bowyer, PW; Coombs, PJ; Kettleborough, CA; Large, JM; Merritt, AT; Osborne, SA; Smiljanic-Hurley, E; Stewart, LB; Tsagris, DJ; Whalley, D; Wheldon, MC1
Andrijevic, A; Basarab, GS; Birkholtz, LM; Brunschwig, C; Chibale, K; Dam, J; de Sousa, ACC; Duffy, J; Egan, TJ; Fish, PV; Gibhard, L; Horatscheck, A; Khonde, LP; Lawrence, N; Le Manach, C; Maepa, K; Nchinda, AT; Njoroge, M; Okombo, J; Paquet, T; Pawar, K; Reader, J; Street, LJ; Taylor, D; van der Watt, M; Wicht, K; Wittlin, S1
Beteck, RM; Legoabe, LJ; Moolman, C; Sluis, RV1
Angulo-Barturén, I; Ansell, KH; Baker, DA; Birchall, K; Bouloc, NS; Bousema, T; Bowyer, PW; Coombs, PJ; Croft, SL; Dechering, KJ; Dessens, JT; El Bakkouri, M; Ferrer, SB; Gamo, FJ; Gutteridge, WE; Harding, DJ; Hui, R; Jiménez-Díaz, MB; Kettleborough, CA; Lafuente, MJ; Large, JM; Merritt, AT; Osborne, SA; Sanz, LM; Smiljanic-Hurley, E; Stewart, LB; Walker, EM; Whalley, D; Wheldon, MC1
Abay, E; Angulo-Barturen, I; Brunschwig, C; Burrows, J; Chibale, K; Duffy, J; Ferrer, S; Gonzàlez Cabrera, D; Jiménez-Díaz, MB; Lafuente-Monasterio, MJ; Lawrence, N; Le Manach, C; Nchinda, AT; Njoroge, M; Paquet, T; Santos Martínez, M; Street, LJ; Taylor, D; Wicht, KJ; Wittlin, S1

Reviews

1 review(s) available for 1h-imidazo(4,5-b)pyridine and Malaria

ArticleYear
An Update on Development of Small-Molecule Plasmodial Kinase Inhibitors.
    Molecules (Basel, Switzerland), 2020, Nov-07, Volume: 25, Issue:21

    Topics: Animals; Antimalarials; Calcium; Casein Kinase I; Culicidae; Drug Design; Drug Discovery; Drug Resistance; Glycogen Synthase Kinase 3; Humans; Imidazoles; Inhibitory Concentration 50; Life Cycle Stages; Malaria; MAP Kinase Signaling System; Phosphotransferases; Plasmodium; Protein Kinase Inhibitors; Pyridines

2020

Other Studies

4 other study(ies) available for 1h-imidazo(4,5-b)pyridine and Malaria

ArticleYear
Potent bicyclic inhibitors of malarial cGMP-dependent protein kinase: approaches to combining improvements in cell potency, selectivity and structural novelty.
    Bioorganic & medicinal chemistry letters, 2019, 10-01, Volume: 29, Issue:19

    Topics: Bridged Bicyclo Compounds, Heterocyclic; Cyclic GMP-Dependent Protein Kinases; Humans; Imidazoles; Malaria; Models, Molecular; Molecular Docking Simulation; Plasmodium falciparum; Protein Conformation; Protein Kinase Inhibitors; Pyridines

2019
Identification of 2,4-Disubstituted Imidazopyridines as Hemozoin Formation Inhibitors with Fast-Killing Kinetics and
    Journal of medicinal chemistry, 2020, 11-12, Volume: 63, Issue:21

    Topics: Animals; Antimalarials; Disease Models, Animal; Half-Life; Hemeproteins; Imidazoles; Life Cycle Stages; Malaria; Mice; Mice, Inbred BALB C; Mice, Inbred NOD; Mice, SCID; Microsomes, Liver; Plasmodium falciparum; Protozoan Proteins; Pyridines; Structure-Activity Relationship

2020
A potent series targeting the malarial cGMP-dependent protein kinase clears infection and blocks transmission.
    Nature communications, 2017, 09-05, Volume: 8, Issue:1

    Topics: Animals; Cell Line; Crystallography, X-Ray; Culicidae; Cyclic GMP-Dependent Protein Kinases; Disease Models, Animal; Female; Humans; Imidazoles; Life Cycle Stages; Malaria; Mice, Inbred BALB C; Models, Molecular; Plasmodium chabaudi; Plasmodium falciparum; Protein Kinase Inhibitors; Pyridines; Treatment Outcome

2017
Identification of Fast-Acting 2,6-Disubstituted Imidazopyridines That Are Efficacious in the in Vivo Humanized Plasmodium falciparum NODscidIL2Rγ
    Journal of medicinal chemistry, 2018, 05-10, Volume: 61, Issue:9

    Topics: Animals; Disease Models, Animal; Drug Discovery; Drug Stability; ERG1 Potassium Channel; Humans; Imidazoles; Malaria; Mice; Plasmodium falciparum; Pyridines; Solubility; Structure-Activity Relationship; Tissue Distribution; Water

2018