Page last updated: 2024-10-28

1-(5-isoquinolinesulfonyl)-2-methylpiperazine and Infarct

1-(5-isoquinolinesulfonyl)-2-methylpiperazine has been researched along with Infarct in 1 studies

1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine: A specific protein kinase C inhibitor, which inhibits superoxide release from human neutrophils (PMN) stimulated with phorbol myristate acetate or synthetic diacylglycerol.
1-(5-isoquinolinesulfonyl)-2-methylpiperazine : A member of the class of N-sulfonylpiperazines that is 2-methylpiperazine substituted at position 1 by a 5-isoquinolinesulfonyl group.

Research Excerpts

ExcerptRelevanceReference
"The study concluded that the typical gel formulation (liposomal Fasudil dispersed in hydroxypropyl methylcellulose solution, which is added to blank poloxamer 407) had been shown to have significantly anti-anginal properties, including easy administration, its application on the infarct area percentage and subsequently its pharmacological effect on the cardiac tissue."4.31Study on development and tissue permeation of different formulations of Fasudil. ( Alanazi, MG; Alshammari, AH; Alshammari, HS; Bandar, N; Elamine, BA; Gangireddy, R; Jandrajupalli, SB; Khalifa, NE; Khojali, WMA; Mohamed, OA; Osman, ME; Unnisa, A, 2023)

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's1 (100.00)2.80

Authors

AuthorsStudies
Unnisa, A1
Khalifa, NE1
Khojali, WMA1
Osman, ME1
Alshammari, AH1
Alshammari, HS1
Alanazi, MG1
Bandar, N1
Jandrajupalli, SB1
Elamine, BA1
Mohamed, OA1
Gangireddy, R1

Other Studies

1 other study available for 1-(5-isoquinolinesulfonyl)-2-methylpiperazine and Infarct

ArticleYear
Study on development and tissue permeation of different formulations of Fasudil.
    European review for medical and pharmacological sciences, 2023, Volume: 27, Issue:13

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Infarction; Liposomes; Rats; Rats, Sprague-D

2023