zopolrestat and thiazoles

zopolrestat has been researched along with thiazoles in 37 studies

Research

Studies (37)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's25 (67.57)18.2507
2000's12 (32.43)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aldinger, CE; Beyer, TA; Dee, MF; Mylari, BL; Scott, PJ; Siegel, TW; Zembrowski, WJ1
Inskeep, PB; Reed, AE; Ronfeld, RA1
Aldinger, CE; Beyer, TA; Dee, MF; Larson, ER; Mylari, BL; Siegel, TW; Singleton, DH; Zembrowski, WJ1
Chang, K; Corbett, JA; Currie, MG; Hasan, KS; McDaniel, ML; Misko, TP; Moore, WM; Petrash, JM; Smith, SR; Tilton, RG1
Gerber, N; Inskeep, PB; Peterson, MJ; Ronfeld, RA1
Petrash, JM; Quiocho, FA; Tarle, I; Wilson, DK1
Cohen, RA; Gupta, S; Oates, PJ; Ruderman, NB; Tesfamariam, B1
Nakano, T; Petrash, JM1
Beyer-Mears, A; Cruz, E; Diecke, FP; Mistry, K2
Oates, PJ; Ramasamy, R; Schaefer, S1
Ishii, A; Konishi, Y; Kotani, T; Nagaki, Y; Okamoto, K; Okukado, N; Suehiro, S; Yago, H1
Nakano, T; Petrash, JM; Quiocho, FA; Wilson, DK1
Eichberg, J; Kuruvilla, R1
Ramasamy, R; Trueblood, N1
Ramasamy, R; Schaefer, S; Trueblood, N1
Carper, DA; El-Kabbani, O; Hohman, TC; Lai, K; Malamas, MS; McGowan, MH; Putilina, T; Wane, YQ1
Fouda, HG; Inskeep, PB; Schneider, RP1
Davenport, CJ; Hoffmaster, KA; Inskeep, PB; Schneider, RP1
Cussac, M; Fresneau, P; Leclerc, G; Morand, JM; Szymonski, B; Tranqui, D1
Beaudet, LN; Dorsey, DA; Ido, Y; Plurad, SB; Schmidt, RE; Williamson, JR1
Goronzy, JJ; Hafner, V; Klimiuk, PA; Rittner, HL; Szweda, LI; Weyand, CM1
Liu, H; Oates, PJ; Ramasamy, R; Schaefer, S1
Arezzo, JC1
Flynn, TG; Hyndman, D; Jia, Z; Li, X; Ye, Q1
Kim, JY; Lee, SH; Moon, CH; Woo, HG1
Carper, DA; Hohman, TC; Kitchen, D; Malamas, MS; Nilakantan, R; Singh, SB1
Ellery, CA; Knight, DR; MacAndrew, JT; Magee, WP; Oates, PJ; Smith, AH; Tracey, WR1
Barth, P; Chung, RP; El-Kabbani, O; Fletcher, EV; Podjarny, A; Rogniaux, H; Van Dorsselaer, A1
Bakr, S; Hwang, YC; Oates, PJ; Ramasamy, R; Sato, S; Tsai, JY; Yan, S; Zhang, H1
Chough, E; Daley, J; Gupta, S; Keaney, JF; Oates, P; Ruderman, NB; Tornheim, K1
Bartlett, T; Demaine, AG; Hodgkinson, AD; Millward, BA; Oates, PJ1
Alexander, GD; Isales, CM; Marrero, MB; Redd, H; Shaw, S; Wang, X1
Chyun, DA; Johnson, BF; Law, G; Nesto, RW; Pfeifer, MA; Slater, WR; Vinik, AI; Wackers, FJ; Young, LH1
Chung, SK; Chung, SS; Dan, Q; Lam, KS; Wong, R1
Aberra, M; Aten, J; Deira, G; Dragt, CA; Krediet, RT; van Westrhenen, R1
Che, Q; Jiang, T; Li, H; Lin, Y; Zhang, N1

Reviews

1 review(s) available for zopolrestat and thiazoles

ArticleYear
New developments in the diagnosis of diabetic neuropathy.
    The American journal of medicine, 1999, Aug-30, Volume: 107, Issue:2B

    Topics: Aldehyde Reductase; Axons; Benzothiazoles; Biopsy; Controlled Clinical Trials as Topic; Diabetic Neuropathies; Diagnosis, Differential; Electrophysiology; Enzyme Inhibitors; Humans; Immunohistochemistry; Neural Conduction; Peripheral Nerves; Phthalazines; Skin; Thiazoles

1999

Trials

2 trial(s) available for zopolrestat and thiazoles

ArticleYear
Pharmacokinetics of the aldose reductase inhibitor, zopolrestat, in humans.
    Journal of clinical pharmacology, 1994, Volume: 34, Issue:7

    Topics: Administration, Oral; Adolescent; Adult; Aldehyde Reductase; Benzothiazoles; Double-Blind Method; Drug Administration Schedule; Half-Life; Humans; Hypoglycemic Agents; Male; Metabolic Clearance Rate; Phthalazines; Thiazoles

1994
Cardiac abnormalities in diabetic patients with neuropathy: effects of aldose reductase inhibitor administration.
    Diabetes care, 2004, Volume: 27, Issue:2

    Topics: Aldehyde Reductase; Benzothiazoles; Cardiac Output; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Diabetic Neuropathies; Double-Blind Method; Enzyme Inhibitors; Exercise Test; Female; Heart; Heart Conduction System; Heart Rate; Humans; Male; Middle Aged; Phthalazines; Placebos; Stroke Volume; Thiazoles; Ventricular Function, Left

2004

Other Studies

34 other study(ies) available for zopolrestat and thiazoles

ArticleYear
Potent, orally active aldose reductase inhibitors related to zopolrestat: surrogates for benzothiazole side chain.
    Journal of medicinal chemistry, 1992, Feb-07, Volume: 35, Issue:3

    Topics: Administration, Oral; Aldehyde Reductase; Animals; Benzothiazoles; Humans; Hypoglycemic Agents; Phthalazines; Rats; Structure-Activity Relationship; Thiazoles

1992
Pharmacokinetics of zopolrestat, a carboxylic acid aldose reductase inhibitor, in normal and diabetic rats.
    Pharmaceutical research, 1991, Volume: 8, Issue:12

    Topics: Administration, Oral; Aldehyde Reductase; Animals; Benzothiazoles; Blood Proteins; Diabetes Mellitus, Experimental; Drug Administration Schedule; Hypoglycemic Agents; Injections, Intravenous; Male; Phthalazines; Protein Binding; Rats; Rats, Inbred Strains; Thiazoles

1991
Novel, potent aldose reductase inhibitors: 3,4-dihydro-4-oxo-3-[[5-(trifluoromethyl)-2-benzothiazolyl] methyl]-1-phthalazineacetic acid (zopolrestat) and congeners.
    Journal of medicinal chemistry, 1991, Volume: 34, Issue:1

    Topics: Aldehyde Reductase; Animals; Benzothiazoles; Enzyme Inhibitors; Female; Humans; Indicators and Reagents; Kinetics; Lens, Crystalline; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Structure; Phthalazines; Placenta; Pregnancy; Rats; Structure-Activity Relationship; Thiazoles; X-Ray Diffraction

1991
Prevention of diabetic vascular dysfunction by guanidines. Inhibition of nitric oxide synthase versus advanced glycation end-product formation.
    Diabetes, 1993, Volume: 42, Issue:2

    Topics: Aldehyde Reductase; Amino Acid Oxidoreductases; Animals; Arginine; Benzothiazoles; Blood Pressure; Body Weight; Capillary Permeability; Citrulline; Diabetes Mellitus, Experimental; Diabetic Angiopathies; Glycation End Products, Advanced; Guanidines; Imidazoles; Imidazolidines; Inositol; Iodine Radioisotopes; Male; Methylguanidine; Naphthalenes; Nitric Oxide Synthase; omega-N-Methylarginine; Phthalazines; Rats; Rats, Sprague-Dawley; Retina; Sciatic Nerve; Serum Albumin, Bovine; Sorbitol; Thiazoles; Uvea

1993
Refined 1.8 A structure of human aldose reductase complexed with the potent inhibitor zopolrestat.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Nov-01, Volume: 90, Issue:21

    Topics: Aldehyde Reductase; Amino Acid Sequence; Benzothiazoles; Binding Sites; Humans; Models, Molecular; Molecular Structure; NADP; Phthalazines; Protein Conformation; Protein Structure, Secondary; Recombinant Proteins; Thiazoles; X-Ray Diffraction

1993
Reduced Na(+)-K+ pump activity in diabetic rabbit carotid artery: reversal by aldose reductase inhibition.
    The American journal of physiology, 1993, Volume: 265, Issue:4 Pt 2

    Topics: Aldehyde Reductase; Animals; Benzothiazoles; Carotid Arteries; Diabetes Mellitus, Experimental; In Vitro Techniques; Male; Ouabain; Phthalazines; Potassium; Rabbits; Rubidium; Sodium-Potassium-Exchanging ATPase; Thiazoles; Vasoconstriction; Vasodilation

1993
Kinetic and spectroscopic evidence for active site inhibition of human aldose reductase.
    Biochemistry, 1996, Aug-27, Volume: 35, Issue:34

    Topics: Aldehyde Reductase; Benzothiazoles; Binding Sites; Enzyme Inhibitors; Glyceraldehyde; Humans; Hydantoins; Imidazoles; Imidazolidines; Kinetics; Phthalazines; Protein Binding; Recombinant Proteins; Spectrometry, Fluorescence; Thermodynamics; Thiazoles

1996
Zopolrestat prevention of proteinuria, albuminuria and cataractogenesis in diabetes mellitus.
    Pharmacology, 1996, Volume: 52, Issue:5

    Topics: Albuminuria; Aldehyde Reductase; Animals; Benzothiazoles; Cataract; Chromatography, Gas; Diabetes Mellitus, Experimental; Enzyme Inhibitors; Eye; Glucose; Lens, Crystalline; Male; Ouabain; Phthalazines; Potassium; Proteinuria; Rats; Rats, Sprague-Dawley; Rubidium; Sodium-Potassium-Exchanging ATPase; Thiazoles

1996
Aldose reductase inhibition protects diabetic and nondiabetic rat hearts from ischemic injury.
    Diabetes, 1997, Volume: 46, Issue:2

    Topics: Adenosine Triphosphate; Aldehyde Reductase; Animals; Benzothiazoles; Blood Glucose; Diabetes Mellitus, Type 1; Energy Metabolism; Enzyme Inhibitors; Fructose; Hydrogen-Ion Concentration; Lactates; Magnetic Resonance Spectroscopy; Myocardial Ischemia; Myocardium; NAD; Phthalazines; Pyruvates; Rats; Rats, Inbred BB; Reperfusion Injury; Sorbitol; Thiazoles

1997
Highly selective aldose reductase inhibitors. 3. Structural diversity of 3-(arylmethyl)-2,4,5-trioxoimidazolidine-1-acetic acids.
    Journal of medicinal chemistry, 1997, Feb-28, Volume: 40, Issue:5

    Topics: Acetates; Aldehyde Reductase; Animals; Benzothiazoles; Diabetes Complications; Enzyme Inhibitors; Humans; Imidazoles; Kidney; Lens, Crystalline; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Structure; Phthalazines; Pyrimidinones; Rats; Sorbitol; Structure-Activity Relationship; Thiazoles

1997
Structural studies of aldo-keto reductase inhibition.
    Advances in experimental medicine and biology, 1997, Volume: 414

    Topics: Aldehyde Reductase; Benzothiazoles; Binding Sites; Crystallography, X-Ray; Enzyme Inhibitors; Humans; Models, Structural; NADP; Phthalazines; Protein Structure, Secondary; Recombinant Proteins; Thiazoles

1997
Comparison of the effects of Zopolrestat and Sorbinil on lens myo-inositol influx.
    Pharmacology, 1997, Volume: 54, Issue:2

    Topics: Aldehyde Reductase; Animals; Benzothiazoles; Carbohydrate Metabolism; Carbohydrates; Culture Media; Enzyme Inhibitors; Galactose; Glucose; Imidazoles; Imidazolidines; In Vitro Techniques; Inositol; Lens, Crystalline; Male; Phthalazines; Polymers; Rats; Rats, Sprague-Dawley; Sorbitol; Thiazoles

1997
Depletion of phospholipid arachidonoyl-containing molecular species in a human Schwann cell line grown in elevated glucose and their restoration by an aldose reductase inhibitor.
    Journal of neurochemistry, 1998, Volume: 71, Issue:2

    Topics: Aldehyde Reductase; Arachidonic Acid; Benzothiazoles; Cell Division; Culture Media; Enzyme Inhibitors; Fructose; Glucose; Humans; Imidazoles; Imidazolidines; L-Iditol 2-Dehydrogenase; Mannitol; Neurofibroma; Organic Chemicals; Phospholipids; Phthalazines; Piperazines; Pyrimidines; Schwann Cells; Sorbitol; Thiazoles; Tumor Cells, Cultured

1998
Aldose reductase inhibition improves altered glucose metabolism of isolated diabetic rat hearts.
    The American journal of physiology, 1998, Volume: 275, Issue:1

    Topics: Aldehyde Reductase; Animals; Benzothiazoles; Blood Pressure; Citric Acid Cycle; Diabetes Mellitus, Type 1; Enzyme Inhibitors; Glucose; Glyceraldehyde 3-Phosphate; Glycolysis; Heart; Heart Rate; In Vitro Techniques; Models, Chemical; Myocardium; Phthalazines; Rats; Rats, Inbred BB; Reference Values; Thiazoles

1998
Metabolic effects of aldose reductase inhibition during low-flow ischemia and reperfusion.
    The American journal of physiology, 1998, Volume: 275, Issue:1

    Topics: Aldehyde Reductase; Animals; Benzothiazoles; Cytosol; Diabetes Mellitus, Type 1; Enzyme Inhibitors; Glycolysis; Heart; Hydrogen-Ion Concentration; In Vitro Techniques; Lactates; Male; Myocardial Ischemia; Myocardial Reperfusion; Myocardium; Oxidation-Reduction; Phthalazines; Pyruvates; Rats; Rats, Inbred BB; Reference Values; Sorbitol; Thiazoles; Ventricular Function, Left

1998
Probing the inhibitor-binding site of aldose reductase with site-directed mutagenesis.
    European journal of biochemistry, 1998, Sep-01, Volume: 256, Issue:2

    Topics: Aldehyde Reductase; Benzothiazoles; Binding Sites; Computer Simulation; Enzyme Inhibitors; Humans; Imidazoles; Imidazolidines; Kinetics; Models, Molecular; Molecular Structure; Mutagenesis, Site-Directed; NADP; Naphthalenes; Phthalazines; Recombinant Proteins; Thiazoles

1998
Tissue distribution and biotransformation of zopolrestat, an aldose reductase inhibitor, in rats.
    Drug metabolism and disposition: the biological fate of chemicals, 1998, Volume: 26, Issue:11

    Topics: Administration, Oral; Aldehyde Reductase; Animals; Benzothiazoles; Bile Ducts; Biotransformation; Chromatography, High Pressure Liquid; Enzyme Inhibitors; Female; Half-Life; Hypoglycemic Agents; Male; Mass Spectrometry; Phthalazines; Rats; Rats, Long-Evans; Thiazoles; Tissue Distribution

1998
Bioavailability, multiple-dose pharmacokinetics, and biotransformation of the aldose reductase inhibitor zopolrestat in dogs.
    Drug metabolism and disposition: the biological fate of chemicals, 1998, Volume: 26, Issue:11

    Topics: Administration, Oral; Aldehyde Reductase; Animals; Benzothiazoles; Biological Availability; Biotransformation; Dogs; Drug Administration Schedule; Enzyme Inhibitors; Female; Half-Life; Hypoglycemic Agents; Male; Mass Spectrometry; Phthalazines; Thiazoles

1998
Synthesis, activity, and molecular modeling of new 2, 4-dioxo-5-(naphthylmethylene)-3-thiazolidineacetic acids and 2-thioxo analogues as potent aldose reductase inhibitors.
    Journal of medicinal chemistry, 1998, Nov-19, Volume: 41, Issue:24

    Topics: Acetates; Aldehyde Reductase; Animals; Benzothiazoles; Cattle; Crystallography, X-Ray; Enzyme Inhibitors; Lens, Crystalline; Models, Molecular; Phthalazines; Structure-Activity Relationship; Thiazoles

1998
Effect of sorbitol dehydrogenase inhibition on experimental diabetic autonomic neuropathy.
    Journal of neuropathology and experimental neurology, 1998, Volume: 57, Issue:12

    Topics: Animals; Autonomic Nervous System Diseases; Benzothiazoles; Diabetic Neuropathies; Drug Evaluation, Preclinical; Enzyme Inhibitors; Ganglia, Sympathetic; L-Iditol 2-Dehydrogenase; Male; Mesentery; Neuroaxonal Dystrophies; Phthalazines; Piperazines; Pyrimidines; Rats; Rats, Sprague-Dawley; Thiazoles

1998
Aldose reductase functions as a detoxification system for lipid peroxidation products in vasculitis.
    The Journal of clinical investigation, 1999, Volume: 103, Issue:7

    Topics: Aldehyde Reductase; Aldehydes; Animals; Apoptosis; Benzothiazoles; Chimera; Enzyme Inhibitors; Free Radical Scavengers; Giant Cell Arteritis; Humans; Imidazoles; Imidazolidines; Lipid Peroxidation; Mice; Mice, SCID; Phthalazines; RNA, Messenger; Temporal Arteries; Thiazoles; Up-Regulation; Vasculitis

1999
Attenuation of ischemia induced increases in sodium and calcium by the aldose reductase inhibitor zopolrestat.
    Cardiovascular research, 1999, Volume: 42, Issue:1

    Topics: Aldehyde Reductase; Analysis of Variance; Animals; Benzothiazoles; Calcium; Diabetes Mellitus, Type 2; Enzyme Inhibitors; Intracellular Fluid; Magnetic Resonance Spectroscopy; Metals; Myocardial Ischemia; Myocardial Reperfusion; Myocardium; Perfusion; Phthalazines; Rats; Rats, Inbred BB; Sodium; Sodium-Potassium-Exchanging ATPase; Thiazoles; Time Factors

1999
Crystal structure of CHO reductase, a member of the aldo-keto reductase superfamily.
    Proteins, 2000, Jan-01, Volume: 38, Issue:1

    Topics: Alcohol Oxidoreductases; Amino Acid Sequence; Animals; Benzothiazoles; Catalytic Domain; CHO Cells; Cricetinae; Crystallography, X-Ray; Enzyme Inhibitors; Humans; Models, Molecular; Molecular Sequence Data; NADP; Phthalazines; Protein Conformation; Sequence Homology, Amino Acid; Thiazoles

2000
Augmentation effects of high glucose on endotoxin-induced nitric oxide production in murine macrophages.
    Advances in experimental medicine and biology, 1999, Volume: 469

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Aldehyde Reductase; Animals; Benzothiazoles; Cell Line; Drug Synergism; Enzyme Inhibitors; Glucose; Lipopolysaccharides; Macrophages; Mice; NAD; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Phthalazines; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate; Thiazoles

1999
Molecular modeling of the aldose reductase-inhibitor complex based on the X-ray crystal structure and studies with single-site-directed mutants.
    Journal of medicinal chemistry, 2000, Mar-23, Volume: 43, Issue:6

    Topics: Aldehyde Reductase; Benzothiazoles; Binding Sites; Crystallography, X-Ray; Enzyme Inhibitors; Humans; Models, Molecular; Mutagenesis, Site-Directed; Phthalazines; Recombinant Proteins; Structure-Activity Relationship; Thiazoles

2000
Aldose reductase inhibition alone or combined with an adenosine A(3) agonist reduces ischemic myocardial injury.
    American journal of physiology. Heart and circulatory physiology, 2000, Volume: 279, Issue:4

    Topics: Adenosine; Aldehyde Reductase; Animals; Benzothiazoles; Dose-Response Relationship, Drug; Enzyme Inhibitors; In Vitro Techniques; Male; Myocardial Ischemia; Myocardium; Phthalazines; Purinergic P1 Receptor Agonists; Rabbits; Receptor, Adenosine A3; Sorbitol; Thiazoles

2000
Aldose and aldehyde reductases: correlation of molecular modeling and mass spectrometric studies on the binding of inhibitors to the active site.
    Proteins, 2000, Nov-15, Volume: 41, Issue:3

    Topics: Aldehyde Reductase; Animals; Benzothiazoles; Binding Sites; Crystallography, X-Ray; Enzyme Inhibitors; Humans; Imidazoles; Imidazolidines; Inhibitory Concentration 50; Models, Molecular; Naphthalenes; Phthalazines; Spectrometry, Mass, Electrospray Ionization; Swine; Thiazoles

2000
Aldose reductase activation is a key component of myocardial response to ischemia.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2002, Volume: 16, Issue:2

    Topics: Aldehyde Reductase; Animals; Benzothiazoles; Enzyme Inhibitors; Glucose; Myocardial Ischemia; Myocardium; Nitric Oxide; Nitric Oxide Donors; Penicillamine; Phthalazines; Rats; Thiazoles

2002
Hyperglycemia increases endothelial superoxide that impairs smooth muscle cell Na+-K+-ATPase activity.
    American journal of physiology. Cell physiology, 2002, Volume: 282, Issue:3

    Topics: Aldehyde Reductase; Animals; Aorta; Arginine; Benzothiazoles; Endothelium, Vascular; Enzyme Inhibitors; Free Radical Scavengers; Glucose; Hyperglycemia; In Vitro Techniques; Muscle, Smooth, Vascular; Phthalazines; Pyrogallol; Rabbits; Sodium-Potassium-Exchanging ATPase; Sorbitol; Superoxide Dismutase; Superoxides; Thiazoles

2002
The response of antioxidant genes to hyperglycemia is abnormal in patients with type 1 diabetes and diabetic nephropathy.
    Diabetes, 2003, Volume: 52, Issue:3

    Topics: Adult; Aged; Aldehyde Reductase; Antioxidants; Benzothiazoles; Blood Glucose; Catalase; Cells, Cultured; Diabetes Mellitus, Type 1; Diabetic Nephropathies; Enzyme Inhibitors; Female; Gene Expression; Genetic Predisposition to Disease; Glutathione Peroxidase; Humans; Hyperglycemia; Leukocytes, Mononuclear; Male; Middle Aged; Phthalazines; Polymorphism, Genetic; RNA; RNA, Messenger; Superoxide Dismutase; Thiazoles

2003
High glucose augments the angiotensin II-induced activation of JAK2 in vascular smooth muscle cells via the polyol pathway.
    The Journal of biological chemistry, 2003, Aug-15, Volume: 278, Issue:33

    Topics: Acetophenones; Aldehyde Reductase; Angiotensin II; Animals; Antibodies; Aorta; Benzothiazoles; Cells, Cultured; Drug Synergism; Electroporation; Enzyme Inhibitors; Glucose; Intracellular Signaling Peptides and Proteins; Janus Kinase 2; Muscle, Smooth, Vascular; NADPH Oxidases; Oligonucleotides, Antisense; Phosphoproteins; Phosphorylation; Phthalazines; Polymers; Protein Kinase C; Protein Kinase C beta; Protein Tyrosine Phosphatase, Non-Receptor Type 11; Protein Tyrosine Phosphatase, Non-Receptor Type 6; Protein Tyrosine Phosphatases; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Rats; Reactive Oxygen Species; Thiazoles; Tyrosine; Vasoconstrictor Agents

2003
Interaction between the polyol pathway and non-enzymatic glycation on aortic smooth muscle cell migration and monocyte adhesion.
    Life sciences, 2004, Dec-10, Volume: 76, Issue:4

    Topics: Aldehyde Reductase; Animals; Antigens, CD; Aorta, Thoracic; Benzothiazoles; Blotting, Northern; Cell Adhesion; Cell Adhesion Molecules; Cell Movement; Cells, Cultured; Chemokine CCL2; Enzyme Inhibitors; Female; Glycation End Products, Advanced; Male; Mice; Mice, Transgenic; Monocytes; Muscle, Smooth, Vascular; Nerve Tissue Proteins; Oligoribonucleotides, Antisense; Phthalazines; Polymers; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serum Albumin, Bovine; Thiazoles

2004
Effects of inhibition of the polyol pathway during chronic peritoneal exposure to a dialysis solution.
    Peritoneal dialysis international : journal of the International Society for Peritoneal Dialysis, 2005, Volume: 25 Suppl 3

    Topics: Aldehyde Reductase; Animals; Benzothiazoles; Dialysis Solutions; Enzyme Inhibitors; Fibrosis; Glucose; Infusions, Parenteral; Lactic Acid; Male; Models, Animal; Neovascularization, Pathologic; Peritoneal Dialysis; Peritoneal Diseases; Peritoneum; Phthalazines; Polymers; Rats; Signal Transduction; Thiazoles

2005
Aldose reductase regulates TGF-beta1-induced production of fibronectin and type IV collagen in cultured rat mesangial cells.
    Nephrology (Carlton, Vic.), 2006, Volume: 11, Issue:2

    Topics: Aldehyde Reductase; Animals; Benzothiazoles; Cells, Cultured; Collagen Type IV; Fibronectins; Imidazolidines; MAP Kinase Signaling System; Mesangial Cells; Phthalazines; Rats; Signal Transduction; Smad2 Protein; Thiazoles; Transcription Factor AP-1; Transforming Growth Factor beta; Transforming Growth Factor beta1

2006