Page last updated: 2024-09-05

zm 241385 and morphine

zm 241385 has been researched along with morphine in 1 studies

Compound Research Comparison

Studies
(zm 241385)
Trials
(zm 241385)
Recent Studies (post-2010)
(zm 241385)
Studies
(morphine)
Trials
(morphine)
Recent Studies (post-2010) (morphine)
401312444,2705,2008,695

Protein Interaction Comparison

ProteinTaxonomyzm 241385 (IC50)morphine (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.2939
Delta-type opioid receptorRattus norvegicus (Norway rat)0.2278
Kappa-type opioid receptorMus musculus (house mouse)0.0828
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0385
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0545
Mu-type opioid receptorHomo sapiens (human)0.122
Delta-type opioid receptorHomo sapiens (human)0.1199
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.9308
Kappa-type opioid receptorHomo sapiens (human)0.655
Mu-type opioid receptorMus musculus (house mouse)0.3305
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.202
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.25

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Betti, M; Borea, PA; Catarzi, D; Colotta, V; Falsini, M; Ravani, A; Varani, K; Varano, F; Vincenzi, F1

Other Studies

1 other study(ies) available for zm 241385 and morphine

ArticleYear
Design, Synthesis, and Pharmacological Characterization of 2-(2-Furanyl)thiazolo[5,4-d]pyrimidine-5,7-diamine Derivatives: New Highly Potent A
    Journal of medicinal chemistry, 2016, 12-08, Volume: 59, Issue:23

    Topics: Acetic Acid; Adenosine A2 Receptor Agonists; Analgesics; Animals; CHO Cells; Cricetulus; Cyclic AMP; Diamines; Dose-Response Relationship, Drug; Drug Design; Female; Humans; Mice; Molecular Structure; Pain; Pyrimidines; Receptor, Adenosine A2A; Structure-Activity Relationship; Thiazoles

2016